NO955112L - Fremgangsmåte for fremstilling av oksazolidinkarboksylsyre samt anvendelse derav for fremstiling av terapeutisk aktive taxoider - Google Patents

Fremgangsmåte for fremstilling av oksazolidinkarboksylsyre samt anvendelse derav for fremstiling av terapeutisk aktive taxoider

Info

Publication number
NO955112L
NO955112L NO955112A NO955112A NO955112L NO 955112 L NO955112 L NO 955112L NO 955112 A NO955112 A NO 955112A NO 955112 A NO955112 A NO 955112A NO 955112 L NO955112 L NO 955112L
Authority
NO
Norway
Prior art keywords
preparation
carboxylic acid
therapeutically active
oxazolidine carboxylic
taxoids
Prior art date
Application number
NO955112A
Other languages
English (en)
Other versions
NO955112D0 (no
Inventor
Jean-Dominique Bourzat
Alain Commercon
Original Assignee
Rhone Poulenc Rorer Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhone Poulenc Rorer Sa filed Critical Rhone Poulenc Rorer Sa
Publication of NO955112L publication Critical patent/NO955112L/no
Publication of NO955112D0 publication Critical patent/NO955112D0/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/04—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Epoxy Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

Frengangsnåte for fremstilling av en oksazolldlnkarboksylsyre ned den generelle formel: .COOR- (D fra en okBazolldlnkarbokfiylsyre med den generelle formel: .coor (U) for fremstilling av terapeutisk aktive taxolder med den generelle formel: R,-NH (III) ; I formlene, (I), (II) og (III) har eubstltuentene K, RI( 83. 83, 84. RS samt R' diverse betydninger.
NO955112A 1993-06-16 1995-12-15 Fremgangsmåte for fremstilling av oksazolidinkarboksylsyre samt anvendelse derav for fremstiling av terapeutisk aktive taxoider NO955112D0 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9307240A FR2706457B1 (fr) 1993-06-16 1993-06-16 Procédé de préparation d'un acide oxazolidinecarboxylique utile pour préparer des taxoïdes thérapeutiquement actifs.
PCT/FR1994/000713 WO1994029284A1 (fr) 1993-06-16 1994-06-15 Procede de preparation d'un acide oxazolidinecarboxylique utile pour preparer des taxoides therapeutiquement actifs

Publications (2)

Publication Number Publication Date
NO955112L true NO955112L (no) 1995-12-15
NO955112D0 NO955112D0 (no) 1995-12-15

Family

ID=9448182

Family Applications (1)

Application Number Title Priority Date Filing Date
NO955112A NO955112D0 (no) 1993-06-16 1995-12-15 Fremgangsmåte for fremstilling av oksazolidinkarboksylsyre samt anvendelse derav for fremstiling av terapeutisk aktive taxoider

Country Status (23)

Country Link
US (2) US6444825B1 (no)
EP (1) EP0703907B1 (no)
JP (1) JPH09500370A (no)
KR (1) KR960703118A (no)
AT (1) ATE156819T1 (no)
AU (1) AU678585B2 (no)
CA (1) CA2165328A1 (no)
CZ (1) CZ284051B6 (no)
DE (1) DE69404991T2 (no)
DK (1) DK0703907T3 (no)
ES (1) ES2107237T3 (no)
FI (1) FI956025A0 (no)
FR (1) FR2706457B1 (no)
GR (1) GR3024534T3 (no)
HU (1) HUT73972A (no)
NO (1) NO955112D0 (no)
NZ (1) NZ268037A (no)
PL (1) PL312212A1 (no)
RU (1) RU2128652C1 (no)
SK (1) SK156995A3 (no)
WO (1) WO1994029284A1 (no)
YU (1) YU37594A (no)
ZA (1) ZA943994B (no)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5973160A (en) 1992-12-23 1999-10-26 Poss; Michael A. Methods for the preparation of novel sidechain-bearing taxanes
CA2170661A1 (en) 1995-03-22 1996-09-23 John K. Thottathil Novel methods for the preparation of taxanes using oaxzolidine intermediates
NZ332475A (en) * 1996-05-08 2000-05-26 Upjohn Co silylated baccatin derivatives, 3-(substituted amino)-3-phenyl-(2R,3S)-isoserinate derivatives, the oxazolidine ester thereof and other immediates used to prepare baccatin derivatives
KR100225535B1 (ko) * 1996-08-27 1999-10-15 정지석 파클리탁셀의 제조방법
MXPA03002494A (es) * 2000-09-22 2004-05-24 Bristol Myers Squibb Co Metodo para reducir toxicidad de quimio terapias combinadas.
WO2006055837A2 (en) * 2004-11-19 2006-05-26 Dr. Reddy's Laboratories Ltd. Process for preparing oxazolidine derivatives
CA2599888C (en) 2005-03-31 2010-06-15 Bioxel Pharma Inc. Preparation of taxanes from 9-dihydro-13-acetylbaccatin iii

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4240987A (en) * 1979-10-29 1980-12-23 Xerox Corporation Chemical process
FR2629819B1 (fr) * 1988-04-06 1990-11-16 Rhone Poulenc Sante Procede de preparation de derives de la baccatine iii et de la desacetyl-10 baccatine iii
MX9102128A (es) * 1990-11-23 1992-07-08 Rhone Poulenc Rorer Sa Derivados de taxano,procedimiento para su preparacion y composicion farmaceutica que los contiene
FR2696458B1 (fr) * 1992-10-05 1994-11-10 Rhone Poulenc Rorer Sa Procédé de préparation de dérivés du taxane.
FR2696459B1 (fr) * 1992-10-05 1994-11-25 Rhone Poulenc Rorer Sa Procédé de préparation de dérivés du taxane.
FR2696460B1 (fr) * 1992-10-05 1994-11-25 Rhone Poulenc Rorer Sa Procédé de préparation de dérivés du taxane.
FR2698361B1 (fr) * 1992-11-20 1995-01-13 Rhone Poulenc Rorer Sa Procédé de préparation d'un acide oxazolidine-1,3 carboxylique-5.
FR2698871B1 (fr) * 1992-12-09 1995-02-24 Rhone Poulenc Rorer Sa Nouveau taxoïdes, leur préparation et les compositions pharmaceutiques qui les contiennent.
FR2702212B1 (fr) * 1993-03-02 1995-04-07 Rhone Poulenc Rorer Sa Nouveaux taxoïdes, leur préparation et les compositions pharmaceutiques qui les contiennent.

Also Published As

Publication number Publication date
CZ284051B6 (cs) 1998-07-15
SK156995A3 (en) 1996-06-05
JPH09500370A (ja) 1997-01-14
WO1994029284A1 (fr) 1994-12-22
DE69404991D1 (de) 1997-09-18
US6043375A (en) 2000-03-28
FI956025A7 (fi) 1995-12-14
CZ329295A3 (en) 1996-03-13
HUT73972A (en) 1996-10-28
AU678585B2 (en) 1997-06-05
YU37594A (sh) 1997-03-07
FR2706457A1 (fr) 1994-12-23
FR2706457B1 (fr) 1995-07-28
ZA943994B (en) 1995-02-03
AU7076294A (en) 1995-01-03
CA2165328A1 (fr) 1994-12-22
ATE156819T1 (de) 1997-08-15
KR960703118A (ko) 1996-06-19
EP0703907A1 (fr) 1996-04-03
DE69404991T2 (de) 1998-01-22
RU2128652C1 (ru) 1999-04-10
FI956025A0 (fi) 1995-12-14
NZ268037A (en) 1997-11-24
EP0703907B1 (fr) 1997-08-13
US6444825B1 (en) 2002-09-03
GR3024534T3 (en) 1997-12-31
DK0703907T3 (da) 1998-03-23
ES2107237T3 (es) 1997-11-16
NO955112D0 (no) 1995-12-15
HU9503611D0 (en) 1996-02-28
PL312212A1 (en) 1996-04-01

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