NO960425L - 15,15-dialkyl-substituerte derivater av östradiol - Google Patents

15,15-dialkyl-substituerte derivater av östradiol

Info

Publication number: NO960425L
Authority: NO; Norway
Prior art keywords: carbon atoms; estradiol; dialkyl; group; substituted derivatives
Prior art date: 1993-08-02

Application number

NO960425A

Other languages

English (en)

Norwegian (no)

Other versions

NO960425D0 (no

Inventor

James Ronald Bull

Karl-Heinrich Fritzemeier

Christa Hegele-Hartung

Original Assignee

Schering Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1993-08-02

Filing date

1996-02-01

Publication date

1996-04-02

1996-02-01 Application filed by Schering Ag filed Critical Schering Ag

1996-02-01 Publication of NO960425D0 publication Critical patent/NO960425D0/no

1996-04-02 Publication of NO960425L publication Critical patent/NO960425L/no

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0066—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa
- C07J1/007—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0059—Estrane derivatives substituted in position 17 by a keto group

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Diabetes (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Epidemiology (AREA)
Endocrinology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Steroid Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Saccharide Compounds (AREA)
Silver Salt Photography Or Processing Solution Therefor (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

NO960425A 1993-08-02 1996-02-01 15,15-dialkyl-substituerte derivater av östradiol NO960425L (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE4326240A DE4326240A1 (de)	1993-08-02	1993-08-02	15,15-Dialkyl-substituierte Derivate des Estradiols
PCT/EP1994/002540 WO1995004070A1 (en)	1993-08-02	1994-08-01	15,15-dialkyl-substituted derivatives of estradiol

Publications (2)

Publication Number	Publication Date
NO960425D0 NO960425D0 (no)	1996-02-01
NO960425L true NO960425L (no)	1996-04-02

Family

ID=6494482

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO960425A NO960425L (no)	1993-08-02	1996-02-01	15,15-dialkyl-substituerte derivater av östradiol

Country Status (21)

Country	Link
US (2)	US5587496A (de)
EP (1)	EP0712412B1 (de)
JP (1)	JPH09500891A (de)
KR (1)	KR960703940A (de)
CN (1)	CN1040329C (de)
AT (1)	ATE175418T1 (de)
AU (1)	AU674609B2 (de)
CA (1)	CA2168657A1 (de)
CZ (1)	CZ26796A3 (de)
DE (2)	DE4326240A1 (de)
FI (1)	FI960465A7 (de)
HU (1)	HUT73238A (de)
IL (1)	IL110530A (de)
MY (1)	MY111121A (de)
NO (1)	NO960425L (de)
NZ (1)	NZ271091A (de)
PL (1)	PL312792A1 (de)
RU (1)	RU2147306C1 (de)
SK (1)	SK13596A3 (de)
WO (1)	WO1995004070A1 (de)
ZA (1)	ZA945754B (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE4326240A1 (de) *	1993-08-02	1995-02-09	Schering Ag	15,15-Dialkyl-substituierte Derivate des Estradiols
DE4447401A1 (de)	1994-12-23	1996-07-04	Schering Ag	14,17-C¶2¶-überbrückte Steroide
DE19906159A1 (de) *	1999-02-09	2000-08-10	Schering Ag	16-Hydroxyestratriene als selektiv wirksame Estrogene
DE10151365A1 (de) *	2001-10-17	2003-04-30	Schering Ag	17-Chlor-D-Homosteroide als selektive Estrogenrezeptorantagonisten
MY142989A (en) *	2004-03-10	2011-02-14	Bayer Schering Pharma Ag	Stabilised supersaturated solids of lipophilic drugs
DE602005014227D1 (de) *	2004-03-10	2009-06-10	Bayer Schering Pharma Ag	Zusammensetzungen aus drospirenon in molekularer dispersion
US20050220825A1 (en) *	2004-03-10	2005-10-06	Adrian Funke	Molecular dispersions of drospirenone

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US2275752A (en) *	1938-11-25	1942-03-10	Ciba Pharm Prod Inc	Cyclic condensation products and process of making same
US3472881A (en) *	1965-05-14	1969-10-14	Merck & Co Inc	3 - hydroxy - 13 - lower alkyl - 15 - carboxyl - 1,3,5(10),8,14 - gonapentaen - 17-ones and intermediates in the production thereof
US3766224A (en) *	1971-06-03	1973-10-16	Sandoz Ag	15-methyl-substituted steroids
DD145919B1 (de) *	1978-06-28	1982-06-30	Kurt Ponsold	Verfahren zur herstellung von 14,1 -methylenderivaten der oestranreihe
DE3628189A1 (de) *	1986-08-20	1988-02-25	Schering Ag	Oestrogen wirksame mittel und 14,17ss-ethano-14ss-estratriene
DE4326240A1 (de) *	1993-08-02	1995-02-09	Schering Ag	15,15-Dialkyl-substituierte Derivate des Estradiols

1993
- 1993-08-02 DE DE4326240A patent/DE4326240A1/de not_active Withdrawn
1994
- 1994-08-01 EP EP94924304A patent/EP0712412B1/de not_active Expired - Lifetime
- 1994-08-01 KR KR1019960700521A patent/KR960703940A/ko not_active Ceased
- 1994-08-01 PL PL94312792A patent/PL312792A1/xx unknown
- 1994-08-01 AT AT94924304T patent/ATE175418T1/de not_active IP Right Cessation
- 1994-08-01 SK SK135-96A patent/SK13596A3/sk unknown
- 1994-08-01 WO PCT/EP1994/002540 patent/WO1995004070A1/en not_active Ceased
- 1994-08-01 IL IL11053094A patent/IL110530A/en not_active IP Right Cessation
- 1994-08-01 NZ NZ271091A patent/NZ271091A/en unknown
- 1994-08-01 JP JP7505581A patent/JPH09500891A/ja not_active Ceased
- 1994-08-01 RU RU96105421A patent/RU2147306C1/ru active
- 1994-08-01 CN CN94192968A patent/CN1040329C/zh not_active Expired - Fee Related
- 1994-08-01 DE DE69415812T patent/DE69415812T2/de not_active Expired - Lifetime
- 1994-08-01 HU HU9600234A patent/HUT73238A/hu unknown
- 1994-08-01 FI FI960465A patent/FI960465A7/fi not_active Application Discontinuation
- 1994-08-01 AU AU74610/94A patent/AU674609B2/en not_active Ceased
- 1994-08-01 CA CA002168657A patent/CA2168657A1/en not_active Abandoned
- 1994-08-01 CZ CZ96267A patent/CZ26796A3/cs unknown
- 1994-08-02 MY MYPI94002013A patent/MY111121A/en unknown
- 1994-08-02 ZA ZA945754A patent/ZA945754B/xx unknown
- 1994-08-02 US US08/284,786 patent/US5587496A/en not_active Expired - Fee Related
1995
- 1995-06-07 US US08/472,722 patent/US5656622A/en not_active Expired - Fee Related
1996
- 1996-02-01 NO NO960425A patent/NO960425L/no unknown

Also Published As

Publication number	Publication date
NO960425D0 (no)	1996-02-01
DE69415812D1 (de)	1999-03-18
EP0712412B1 (de)	1999-01-07
KR960703940A (ko)	1996-08-31
CN1040329C (zh)	1998-10-21
HU9600234D0 (en)	1996-04-29
PL312792A1 (en)	1996-05-13
HUT73238A (en)	1996-07-29
CZ26796A3 (en)	1996-07-17
CN1128031A (zh)	1996-07-31
SK13596A3 (en)	1997-03-05
ATE175418T1 (de)	1999-01-15
MY111121A (en)	1999-08-30
FI960465A0 (fi)	1996-02-01
EP0712412A1 (de)	1996-05-22
AU7461094A (en)	1995-02-28
FI960465L (fi)	1996-02-01
CA2168657A1 (en)	1995-02-09
WO1995004070A1 (en)	1995-02-09
JPH09500891A (ja)	1997-01-28
IL110530A (en)	1998-08-16
FI960465A7 (fi)	1996-02-01
AU674609B2 (en)	1997-01-02
RU2147306C1 (ru)	2000-04-10
US5656622A (en)	1997-08-12
ZA945754B (en)	1995-03-15
NZ271091A (en)	1996-08-27
DE69415812T2 (de)	1999-09-16
US5587496A (en)	1996-12-24
DE4326240A1 (de)	1995-02-09
IL110530A0 (en)	1994-11-11

Similar Documents

Publication	Publication Date	Title
DE3570038D1 (en)	1989-06-15	Steroids for use as immunomodulators
MY103850A (en)	1993-09-30	Phenol substituted gem-diphosphonate derivatives, process for their preparation and pharmaceutical compositions containing them.
IL75337A (en)	1989-02-28	Polyenoic acids omega-substituted by a 4,5-dimethoxy-2-methyl-quinone or a 4,5-dimethoxy-2-methyl-phenyl group,process for the preparation thereof and pharmaceutical compositions containing the same
NO954681L (no)	1995-11-20	Kjemiske forbindelser
IL96636A0 (en)	1991-09-16	Piperidine derivatives and pharmaceutical compositions containing them
IL87657A (en)	1993-02-21	Preparation of methylene derivatives of androsta-1,4-diene-3,17-dione and pharmaceutical compositions containing them
IL88396A (en)	1992-12-01	Preparation of 6-methylene derivatives of androsta-1,4- diene-3,17-diones and pharmaceutical compositions containing them
IL76538A0 (en)	1986-02-28	Alkylpiperazino substituted indane derivatives and methods of preparation and treatment and pharmaceutical compositions containing them
GR1002384B (el)	1996-07-03	Μεθοδος παρασκευης παραγωγων υποκατεστημενου στυρολιου.
NZ224638A (en)	1990-04-26	1-(2',3'-dideoxy-2'-fluoro-beta-d-arabinofuranosyl)- cytosine derivatives and pharmaceutical compositions
EP0158340A3 (en)	1986-05-28	Novel 1,5-benzothiazepine derivative, processes for preparing the same and pharmaceutical compositions
DK186788A (da)	1988-04-06	14,17beta-ethano-14beta-oestratriener og oestratetraener, fremgangsmaader til deres fremstilling og farmaceutiske praeparater indeholdende dem
AU7461094A (en)	1995-02-28	15,15-dialkyl-substituted derivatives of estradiol
AU588315B2 (en)	1989-09-14	Novel isoxazole derivatives, a process for their preparation and pharmaceutical products containing these
DE3572648D1 (en)	1989-10-05	Halogen labeled compounds including estradiol derivatives, their synthetic intermediates and the syntheses thereof
PT86283A (fr)	1988-01-01	Procede de preparation de nouveaux produits steroides comportant en position 23 un radical sulfinyle
US3917833A (en)	1975-11-04	Amino-substituted benzocycloheptenones for inducing sleep
AU7895087A (en)	1988-03-31	Antigestagens for the inhibition of uterine synthesis of prostaglandin
NO855383L (no)	1986-07-14	Fremgangsmaate for fremstilling av piperazin-derivater.
ES8204741A1 (es)	1982-06-01	Procedimiento para la preparacion de 3-desoxi-a15-esteroides
GR3000773T3 (en)	1991-10-10	2,2;6,6-diethylene-3-oxo-17-alpha-pregn-4-ene-21,17-carbolactones, process for their preparation and pharmaceutical compositions containing them
GB1502337A (en)	1978-03-01	6-aminochroman derivatives and a process for their preparation
EP0324184A3 (en)	1990-05-02	2-amino-1,2,3,4-tetrahydroisoquinoline derivatives, method for their preparation and their use as medicines
MY101746A (en)	1992-01-17	1,5-benzothiazepine derivatives, a process for preparing the same, pharmaceutical compositions as well as the use thereof.
BE903194A (fr)	1986-03-06	Nouveaux steroides et leur preparation