OA10251A - Novel use of histamine h2 and/or h3 receptor agonist for the treatment of erectile disfunction - Google Patents

Novel use of histamine h2 and/or h3 receptor agonist for the treatment of erectile disfunction Download PDF

Info

Publication number: OA10251A
Authority: OA; OAPI
Prior art keywords: agonist; histamine; agent; pyridyl; phentolamine
Prior art date: 1992-08-21

Application number

OA60612A

Other languages

English (en)

Inventor

Cesar Roberto Dias Nahoum

Original Assignee

Cesar Roberto Dias Nahoum

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1992-08-21

Filing date

1995-02-16

Publication date

1997-10-07

1995-02-16 Application filed by Cesar Roberto Dias Nahoum filed Critical Cesar Roberto Dias Nahoum

1997-10-07 Publication of OA10251A publication Critical patent/OA10251A/en

Links

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RYFMWSXOAZQYPI-UHFFFAOYSA-K trisodium phosphate Chemical compound [Na+].[Na+].[Na+].[O-]P([O-])([O-])=O RYFMWSXOAZQYPI-UHFFFAOYSA-K 0.000 description 1
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Classifications

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- A61K9/02—Suppositories; Bougies; Bases therefor; Ovules
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/17—Amides, e.g. hydroxamic acids having the group >N—C(O)—N< or >N—C(S)—N<, e.g. urea, thiourea, carmustine
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Organic Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Endocrinology (AREA)
Gynecology & Obstetrics (AREA)
Reproductive Health (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Steroid Compounds (AREA)
Medicinal Preparation (AREA)

OA60612A 1992-08-21 1995-02-16 Novel use of histamine h2 and/or h3 receptor agonist for the treatment of erectile disfunction OA10251A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
BR929203277A BR9203277A (pt)	1992-08-21	1992-08-21	Utilizaccao de drogas eretogenicas e respectivas metodologias de aplicacao

Publications (1)

Publication Number	Publication Date
OA10251A true OA10251A (en)	1997-10-07

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ID=4054796

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Application Number	Title	Priority Date	Filing Date
OA60612A OA10251A (en)	1992-08-21	1995-02-16	Novel use of histamine h2 and/or h3 receptor agonist for the treatment of erectile disfunction

Country Status (13)

Country	Link
US (1)	US5908853A (de)
EP (1)	EP0655914B1 (de)
JP (1)	JP2002510277A (de)
KR (1)	KR100331754B1 (de)
AT (1)	ATE233091T1 (de)
BR (1)	BR9203277A (de)
CA (1)	CA2142875A1 (de)
DE (1)	DE69332713D1 (de)
NZ (1)	NZ255278A (de)
OA (1)	OA10251A (de)
TW (1)	TW418090B (de)
WO (1)	WO1994004120A2 (de)
ZA (1)	ZA936118B (de)

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US20050065161A1 (en) *	1996-02-02	2005-03-24	Nitromed, Inc.	Nitrosated and nitrosylated alpha-adrenergic receptor antagonist compounds, compositions and their uses
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1992
- 1992-08-21 BR BR929203277A patent/BR9203277A/pt not_active Application Discontinuation
1993
- 1993-08-18 EP EP93918819A patent/EP0655914B1/de not_active Expired - Lifetime
- 1993-08-18 JP JP50569694A patent/JP2002510277A/ja not_active Ceased
- 1993-08-18 WO PCT/BR1993/000027 patent/WO1994004120A2/en not_active Ceased
- 1993-08-18 CA CA002142875A patent/CA2142875A1/en not_active Abandoned
- 1993-08-18 DE DE69332713T patent/DE69332713D1/de not_active Expired - Lifetime
- 1993-08-18 KR KR1019950700672A patent/KR100331754B1/ko not_active Expired - Fee Related
- 1993-08-18 US US08/381,945 patent/US5908853A/en not_active Expired - Fee Related
- 1993-08-18 AT AT93918819T patent/ATE233091T1/de not_active IP Right Cessation
- 1993-08-20 ZA ZA936118A patent/ZA936118B/xx unknown
- 1993-08-20 TW TW082106721A patent/TW418090B/zh not_active IP Right Cessation
1995
- 1995-02-15 NZ NZ255278A patent/NZ255278A/xx unknown
- 1995-02-16 OA OA60612A patent/OA10251A/en unknown

Also Published As

Publication number	Publication date
ATE233091T1 (de)	2003-03-15
ZA936118B (en)	1995-04-20
JP2002510277A (ja)	2002-04-02
KR950702823A (ko)	1995-08-23
AU678996B2 (en)	1997-06-19
EP0655914B1 (de)	2003-02-26
BR9203277A (pt)	1994-03-01
CA2142875A1 (en)	1994-03-03
EP0655914A4 (de)	1998-04-22
TW418090B (en)	2001-01-11
US5908853A (en)	1999-06-01
AU4937193A (en)	1994-03-15
KR100331754B1 (ko)	2002-10-04
EP0655914A1 (de)	1995-06-07
NZ255278A (en)	1999-05-28
DE69332713D1 (de)	2003-04-03
WO1994004120A3 (en)	1994-05-26
WO1994004120A2 (en)	1994-03-03

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EP0618798B1 (de)	1997-03-12	Pyridylguanidine verbindungen zur behandlung von erektionsstörungen
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AU2003273291A1 (en)	2004-03-29	Methods of treatment of male erectile dysfuntion