OA11225A - 9-Oxime erythromycin derivatives - Google Patents

9-Oxime erythromycin derivatives Download PDF

Info

Publication number: OA11225A
Authority: OA; OAPI
Prior art keywords: carbamate; deoxo; deoxy; hydrazo; desosaminyl
Prior art date: 1997-06-11

Application number

OA9900269A

Other languages

English (en)

Inventor

Yong-Jin Wu

Original Assignee

Pfizer Prod Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1997-06-11

Filing date

1999-12-03

Publication date

2003-07-17

1999-12-03 Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc

2003-07-17 Publication of OA11225A publication Critical patent/OA11225A/en

Links

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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins

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Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Molecular Biology (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
Genetics & Genomics (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Engineering & Computer Science (AREA)
Biochemistry (AREA)
Biotechnology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Tropical Medicine & Parasitology (AREA)
Epidemiology (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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OA9900269A 1997-06-11 1999-12-03 9-Oxime erythromycin derivatives OA11225A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US4934997P	1997-06-11	1997-06-11

Publications (1)

Publication Number	Publication Date
OA11225A true OA11225A (en)	2003-07-17

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ID=21959341

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Application Number	Title	Priority Date	Filing Date
OA9900269A OA11225A (en)	1997-06-11	1999-12-03	9-Oxime erythromycin derivatives

Country Status (31)

Country	Link
EP (1)	EP0988308A1 (is)
JP (1)	JP2000513026A (is)
KR (1)	KR20010013660A (is)
CN (1)	CN1259135A (is)
AP (1)	AP9801253A0 (is)
AR (1)	AR012244A1 (is)
AU (1)	AU7226798A (is)
BG (1)	BG103947A (is)
BR (1)	BR9810021A (is)
CA (1)	CA2293335A1 (is)
CO (1)	CO4940506A1 (is)
CZ (1)	CZ9904388A3 (is)
EA (1)	EA199901016A1 (is)
GT (1)	GT199800074A (is)
HN (1)	HN1998000073A (is)
HR (1)	HRP980316A2 (is)
HU (1)	HUP0002252A3 (is)
ID (1)	ID24529A (is)
IL (1)	IL132767A0 (is)
IS (1)	IS5251A (is)
MA (1)	MA26505A1 (is)
NO (1)	NO996108L (is)
OA (1)	OA11225A (is)
PA (1)	PA8451801A1 (is)
PE (1)	PE79899A1 (is)
PL (1)	PL337606A1 (is)
TN (1)	TNSN98083A1 (is)
TR (1)	TR199902995T2 (is)
TW (1)	TW448174B (is)
WO (1)	WO1998056800A1 (is)
ZA (1)	ZA985018B (is)

Families Citing this family (29)

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Publication number	Priority date	Publication date	Assignee	Title
HN1998000159A (es) *	1997-10-29	1999-02-09	Monsanto Co	Derivados de 9- amino - 3 ceto eritromicina
AU5299499A (en)	1998-09-22	2000-04-10	Pfizer Products Inc.	Carbamate and carbazate ketolide antibiotics
FR2786188B1 (fr) *	1998-11-24	2002-10-31	Hoechst Marion Roussel Inc	Nouveaux derives de l'erythromycine, leur procede de preparation et leur applicaion comme medicaments
US6258785B1 (en)	1998-12-02	2001-07-10	Pfizer Inc.	Crystalline 9-E-(O-methyl)oxime of 11, 12-dideoxy-3-de(2,6-dideoxy-3-C-methyl-3-O-methyl-α-L-ribohexopyranosyloxy)-6-O-methyl-12,11-(iminocarbonyl-(2-(3-(4-(3-pyridinyl)1H-imadazol-1-yl)propyl)hydrazono))-3-oxoerythromycin
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1998
- 1998-05-15 EP EP98919394A patent/EP0988308A1/en not_active Withdrawn
- 1998-05-15 JP JP11501928A patent/JP2000513026A/ja active Pending
- 1998-05-15 ID IDW991570A patent/ID24529A/id unknown
- 1998-05-15 TR TR1999/02995T patent/TR199902995T2/xx unknown
- 1998-05-15 AU AU72267/98A patent/AU7226798A/en not_active Abandoned
- 1998-05-15 HU HU0002252A patent/HUP0002252A3/hu unknown
- 1998-05-15 PL PL98337606A patent/PL337606A1/xx unknown
- 1998-05-15 CA CA002293335A patent/CA2293335A1/en not_active Abandoned
- 1998-05-15 IL IL13276798A patent/IL132767A0/xx unknown
- 1998-05-15 KR KR1019997011672A patent/KR20010013660A/ko not_active Ceased
- 1998-05-15 BR BR9810021-1A patent/BR9810021A/pt not_active IP Right Cessation
- 1998-05-15 EA EA199901016A patent/EA199901016A1/ru unknown
- 1998-05-15 CZ CZ19994388A patent/CZ9904388A3/cs unknown
- 1998-05-15 WO PCT/IB1998/000741 patent/WO1998056800A1/en not_active Ceased
- 1998-05-15 CN CN98805848A patent/CN1259135A/zh active Pending
- 1998-05-19 HN HN1998000073A patent/HN1998000073A/es unknown
- 1998-05-21 PA PA19988451801A patent/PA8451801A1/es unknown
- 1998-06-04 AP APAP/P/1998/001253A patent/AP9801253A0/en unknown
- 1998-06-05 GT GT199800074A patent/GT199800074A/es unknown
- 1998-06-08 PE PE1998000470A patent/PE79899A1/es not_active Application Discontinuation
- 1998-06-08 TW TW087109086A patent/TW448174B/zh active
- 1998-06-09 AR ARP980102703A patent/AR012244A1/es unknown
- 1998-06-10 TN TNTNSN98083A patent/TNSN98083A1/fr unknown
- 1998-06-10 ZA ZA9805018A patent/ZA985018B/xx unknown
- 1998-06-10 MA MA25105A patent/MA26505A1/fr unknown
- 1998-06-11 CO CO98033538A patent/CO4940506A1/es unknown
- 1998-06-11 HR HR60/049,349A patent/HRP980316A2/hr not_active Application Discontinuation
1999
- 1999-11-16 IS IS5251A patent/IS5251A/is unknown
- 1999-12-03 BG BG103947A patent/BG103947A/xx unknown
- 1999-12-03 OA OA9900269A patent/OA11225A/en unknown
- 1999-12-10 NO NO996108A patent/NO996108L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
TNSN98083A1 (fr)	2005-03-15
JP2000513026A (ja)	2000-10-03
AU7226798A (en)	1998-12-30
PA8451801A1 (es)	2000-05-24
CA2293335A1 (en)	1998-12-17
HN1998000073A (es)	1999-01-08
KR20010013660A (ko)	2001-02-26
BR9810021A (pt)	2000-09-19
EP0988308A1 (en)	2000-03-29
AP9801253A0 (en)	1999-12-04
NO996108D0 (no)	1999-12-10
PE79899A1 (es)	1999-08-25
PL337606A1 (en)	2000-08-28
EA199901016A1 (ru)	2000-06-26
HUP0002252A2 (hu)	2000-12-28
GT199800074A (es)	1999-11-27
AR012244A1 (es)	2000-09-27
TR199902995T2 (xx)	2000-02-21
CO4940506A1 (es)	2000-07-24
HUP0002252A3 (en)	2002-01-28
ID24529A (id)	2000-07-20
TW448174B (en)	2001-08-01
CZ9904388A3 (cs)	2002-10-16
ZA985018B (en)	1999-12-10
HRP980316A2 (en)	1999-04-30
CN1259135A (zh)	2000-07-05
BG103947A (en)	2000-07-31
WO1998056800A1 (en)	1998-12-17
NO996108L (no)	2000-02-10
IL132767A0 (en)	2001-03-19
IS5251A (is)	1999-11-16
MA26505A1 (fr)	2004-12-20

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US6162794A (en)	2000-12-19	Erythromycin derivatives
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US20020025937A1 (en)	2002-02-28	9-oxime erythromycin derivatives
US6498146B1 (en)	2002-12-24	Erythromycin derivatives
US20020077302A1 (en)	2002-06-20	Tricyclic erythromycin derivatives
US6258785B1 (en)	2001-07-10	Crystalline 9-E-(O-methyl)oxime of 11, 12-dideoxy-3-de(2,6-dideoxy-3-C-methyl-3-O-methyl-α-L-ribohexopyranosyloxy)-6-O-methyl-12,11-(iminocarbonyl-(2-(3-(4-(3-pyridinyl)1H-imadazol-1-yl)propyl)hydrazono))-3-oxoerythromycin
EP0952157B1 (en)	2003-06-18	9A, 11B-Dehydro derivatives of 9-oxime-3-keto-6-0-methylerythromycin
NZ526120A (en)	2005-02-25	13-membered azalides and their use as antibiotic agents
MXPA99011494A (en)	2000-07-01	9-oxime erythromycin derivatives
MXPA01005055A (en)	2001-12-04	13-membered azalides and their use as antibiotic agents