OA11245A - Sertraline salts and sustained-release dosage forms of sertraline - Google Patents

Info

Publication number

OA11245A

OA11245A OA9900305A OA9900305A OA11245A OA 11245 A OA11245 A OA 11245A OA 9900305 A OA9900305 A OA 9900305A OA 9900305 A OA9900305 A OA 9900305A OA 11245 A OA11245 A OA 11245A

Authority

OA

OAPI

Prior art keywords

sertraline

dosage form

sertraiine

daim

release

Prior art date

1997-07-01

Links

• Espacenet
• Global Dossier
• Discuss

• VGKDLMBJGBXTGI-SJCJKPOMSA-N sertraline Chemical class C1([C@@H]2CC[C@@H](C3=CC=CC=C32)NC)=CC=C(Cl)C(Cl)=C1 VGKDLMBJGBXTGI-SJCJKPOMSA-N 0.000 title claims abstract description 747
• 229960002073 sertraline Drugs 0.000 title claims abstract description 741
• 239000002552 dosage form Substances 0.000 title claims abstract description 290
• 238000013268 sustained release Methods 0.000 title claims abstract description 158
• 239000012730 sustained-release form Substances 0.000 title claims abstract description 158
• 238000000034 method Methods 0.000 claims abstract description 170
• QTBSBXVTEAMEQO-UHFFFAOYSA-M Acetate Chemical compound CC([O-])=O QTBSBXVTEAMEQO-UHFFFAOYSA-M 0.000 claims abstract description 117
• CKLJMWTZIZZHCS-REOHCLBHSA-N L-aspartic acid Chemical class OC(=O)[C@@H](N)CC(O)=O CKLJMWTZIZZHCS-REOHCLBHSA-N 0.000 claims abstract description 91
• JVTAAEKCZFNVCJ-REOHCLBHSA-N L-lactic acid Chemical compound C[C@H](O)C(O)=O JVTAAEKCZFNVCJ-REOHCLBHSA-N 0.000 claims abstract description 86
• 230000008569 process Effects 0.000 claims abstract description 74
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