OA11864A - Substituted benzolactam compounds. - Google Patents

Substituted benzolactam compounds. Download PDF

Info

Publication number: OA11864A
Authority: OA; OAPI
Prior art keywords: compound; disorder; disorders; oxo; formula
Prior art date: 1999-05-06

Application number

OA1200100264A

Other languages

English (en)

Inventor

Susan Beth Sobolov-Jaynes

Original Assignee

Pfizer Prod Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-05-06

Filing date

2000-04-13

Publication date

2006-03-03

2000-04-13 Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc

2006-03-03 Publication of OA11864A publication Critical patent/OA11864A/en

Links

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239000001257 hydrogen Substances 0.000 claims abstract description 31
150000002431 hydrogen Chemical class 0.000 claims abstract description 20
125000000217 alkyl group Chemical group 0.000 claims abstract description 19
125000005678 ethenylene group Chemical group [H]C([*:1])=C([H])[*:2] 0.000 claims abstract description 15
229910052799 carbon Inorganic materials 0.000 claims abstract description 14
125000001153 fluoro group Chemical group F* 0.000 claims abstract description 14
125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims abstract description 13
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QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical group [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 claims abstract description 9
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Classifications

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- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems

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OA1200100264A 1999-05-06 2000-04-13 Substituted benzolactam compounds. OA11864A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US13285899P	1999-05-06	1999-05-06

Publications (1)

Publication Number	Publication Date
OA11864A true OA11864A (en)	2006-03-03

Family

ID=22455915

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
OA1200100264A OA11864A (en)	1999-05-06	2000-04-13	Substituted benzolactam compounds.

Country Status (40)

Country	Link
EP (1)	EP1175417B1 (fr)
JP (1)	JP2002544128A (fr)
KR (1)	KR20020015319A (fr)
CN (1)	CN1349527A (fr)
AP (1)	AP2001002314A0 (fr)
AR (1)	AR036320A1 (fr)
AT (1)	ATE257478T1 (fr)
AU (1)	AU3572800A (fr)
BG (1)	BG106141A (fr)
BR (1)	BR0010673A (fr)
CA (1)	CA2373079A1 (fr)
CR (1)	CR6505A (fr)
CZ (1)	CZ20013977A3 (fr)
DE (1)	DE60007625T2 (fr)
DK (1)	DK1175417T3 (fr)
DZ (1)	DZ3040A1 (fr)
EA (1)	EA200101050A1 (fr)
EE (1)	EE200100586A (fr)
ES (1)	ES2211520T3 (fr)
GE (1)	GEP20043224B (fr)
GT (1)	GT200000063A (fr)
HK (1)	HK1046144A1 (fr)
HR (1)	HRP20010821A2 (fr)
HU (1)	HUP0201135A3 (fr)
IL (1)	IL145945A0 (fr)
IS (1)	IS6122A (fr)
MA (1)	MA26731A1 (fr)
MY (1)	MY133207A (fr)
NO (1)	NO20015395L (fr)
NZ (1)	NZ514697A (fr)
OA (1)	OA11864A (fr)
PA (1)	PA8494901A1 (fr)
PE (1)	PE20010119A1 (fr)
PL (1)	PL351919A1 (fr)
PT (1)	PT1175417E (fr)
TN (1)	TNSN00095A1 (fr)
TR (1)	TR200103222T2 (fr)
UY (1)	UY26135A1 (fr)
WO (1)	WO2000068224A1 (fr)
ZA (1)	ZA200109116B (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB0108982D0 (en)	2001-04-10	2001-05-30	Merck Sharp & Dohme	Therapeutic agents
EP1460061A4 (fr) *	2001-12-27	2006-05-31	Toray Finechemicals Co Ltd	Processus de production de derive heterocyclique sature azote 1-alcoxycarbonyle
DE602004027798D1 (de)	2003-03-12	2010-08-05	Univ Arizona State	Verfahren zur regulierung von angiogenese mit apelin-zusammensetzungen
US7790745B2 (en)	2005-10-21	2010-09-07	Bristol-Myers Squibb Company	Tetrahydroisoquinoline LXR Modulators
WO2009109001A1 (fr) *	2008-03-04	2009-09-11	Adelaide Research & Innovation Pty Ltd	Procédé de prévention et/ou de traitement d’une maladie, d’une condition ou d’un état associés à une fonction réduite des neurones dopaminergiques
JP6156074B2 (ja) *	2013-11-08	2017-07-05	住友化学株式会社	スクシンイミド化合物及びその用途

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ES2147759T3 (es) *	1992-12-10	2000-10-01	Pfizer	Heterociclos no aromaticos sustituidos con aminometileno y uso como antagonistas de la sustancia p.
JP3042894B2 (ja) *	1995-07-07	2000-05-22	ファイザー製薬株式会社	サブスタンスｐアンタゴニストとしての置換ベンゾラクタム化合物
TW340842B (en) *	1995-08-24	1998-09-21	Pfizer	Substituted benzylaminopiperidine compounds
PT780375E (pt) *	1995-12-21	2002-12-31	Pfizer	3-¬(benzilo substituido em 5)amino\|-2-phenilpiperidinas como antagonistas da substancia p
TW426667B (en) *	1997-11-19	2001-03-21	Pfizer	Piperidinylaminomethyl trifluoromethyl cyclic ether compounds as substance P antagonists

2000
- 2000-04-13 IL IL14594500A patent/IL145945A0/xx unknown
- 2000-04-13 WO PCT/IB2000/000461 patent/WO2000068224A1/fr not_active Ceased
- 2000-04-13 PL PL00351919A patent/PL351919A1/xx not_active Application Discontinuation
- 2000-04-13 HR HR20010821A patent/HRP20010821A2/hr not_active Application Discontinuation
- 2000-04-13 AT AT00914335T patent/ATE257478T1/de not_active IP Right Cessation
- 2000-04-13 CA CA002373079A patent/CA2373079A1/fr not_active Abandoned
- 2000-04-13 GE GEAP20006190A patent/GEP20043224B/en unknown
- 2000-04-13 KR KR1020017014110A patent/KR20020015319A/ko not_active Ceased
- 2000-04-13 CZ CZ20013977A patent/CZ20013977A3/cs unknown
- 2000-04-13 PT PT00914335T patent/PT1175417E/pt unknown
- 2000-04-13 AU AU35728/00A patent/AU3572800A/en not_active Abandoned
- 2000-04-13 NZ NZ514697A patent/NZ514697A/en unknown
- 2000-04-13 EA EA200101050A patent/EA200101050A1/ru unknown
- 2000-04-13 OA OA1200100264A patent/OA11864A/en unknown
- 2000-04-13 HU HU0201135A patent/HUP0201135A3/hu unknown
- 2000-04-13 ES ES00914335T patent/ES2211520T3/es not_active Expired - Lifetime
- 2000-04-13 HK HK02107807.6A patent/HK1046144A1/zh unknown
- 2000-04-13 DK DK00914335T patent/DK1175417T3/da active
- 2000-04-13 EP EP00914335A patent/EP1175417B1/fr not_active Expired - Lifetime
- 2000-04-13 AP APAP/P/2001/002314A patent/AP2001002314A0/en unknown
- 2000-04-13 DE DE2000607625 patent/DE60007625T2/de not_active Expired - Fee Related
- 2000-04-13 JP JP2000616198A patent/JP2002544128A/ja active Pending
- 2000-04-13 CN CN00807267A patent/CN1349527A/zh active Pending
- 2000-04-13 EE EEP200100586A patent/EE200100586A/xx unknown
- 2000-04-13 TR TR2001/03222T patent/TR200103222T2/xx unknown
- 2000-04-13 BR BR0010673-9A patent/BR0010673A/pt not_active IP Right Cessation
- 2000-05-03 UY UY26135A patent/UY26135A1/es not_active Application Discontinuation
- 2000-05-03 MA MA25966A patent/MA26731A1/fr unknown
- 2000-05-03 TN TNTNSN00095A patent/TNSN00095A1/fr unknown
- 2000-05-03 PA PA20008494901A patent/PA8494901A1/es unknown
- 2000-05-03 DZ DZ000082A patent/DZ3040A1/fr active
- 2000-05-04 MY MYPI20001922A patent/MY133207A/en unknown
- 2000-05-04 AR ARP000102150A patent/AR036320A1/es unknown
- 2000-05-05 PE PE2000000418A patent/PE20010119A1/es not_active Application Discontinuation
- 2000-05-05 GT GT200000063A patent/GT200000063A/es unknown
2001
- 2001-10-23 IS IS6122A patent/IS6122A/is unknown
- 2001-11-05 ZA ZA200109116A patent/ZA200109116B/en unknown
- 2001-11-05 NO NO20015395A patent/NO20015395L/no not_active Application Discontinuation
- 2001-11-19 CR CR6505A patent/CR6505A/es not_active Application Discontinuation
- 2001-11-23 BG BG106141A patent/BG106141A/bg unknown

Also Published As

Publication number	Publication date
TR200103222T2 (tr)	2002-03-21
ZA200109116B (en)	2002-11-05
CN1349527A (zh)	2002-05-15
MA26731A1 (fr)	2004-12-20
ATE257478T1 (de)	2004-01-15
EA200101050A1 (ru)	2002-04-25
DZ3040A1 (fr)	2004-03-27
DE60007625D1 (de)	2004-02-12
GEP20043224B (en)	2004-04-26
PL351919A1 (en)	2003-06-30
CR6505A (es)	2004-03-24
NZ514697A (en)	2004-04-30
HUP0201135A3 (en)	2003-05-28
IS6122A (is)	2001-10-23
PA8494901A1 (es)	2003-12-10
PT1175417E (pt)	2004-04-30
HUP0201135A2 (en)	2002-09-28
HK1046144A1 (zh)	2002-12-27
NO20015395L (no)	2001-12-11
KR20020015319A (ko)	2002-02-27
BR0010673A (pt)	2002-02-19
PE20010119A1 (es)	2001-02-06
DE60007625T2 (de)	2004-11-18
AR036320A1 (es)	2004-09-01
TNSN00095A1 (fr)	2005-11-10
UY26135A1 (es)	2000-12-29
DK1175417T3 (da)	2004-04-05
CZ20013977A3 (cs)	2003-10-15
EP1175417B1 (fr)	2004-01-07
BG106141A (bg)	2002-07-31
JP2002544128A (ja)	2002-12-24
AP2001002314A0 (en)	2001-12-31
EP1175417A1 (fr)	2002-01-30
AU3572800A (en)	2000-11-21
NO20015395D0 (no)	2001-11-05
CA2373079A1 (fr)	2000-11-16
EE200100586A (et)	2003-02-17
IL145945A0 (en)	2002-07-25
MY133207A (en)	2007-10-31
GT200000063A (es)	2001-10-27
ES2211520T3 (es)	2004-07-16
HRP20010821A2 (en)	2002-12-31
WO2000068224A1 (fr)	2000-11-16

Publication	Publication Date	Title
US6180647B1 (en)	2001-01-30	Substituted benzolactam compounds as substance P antagonists
US5869672A (en)	1999-02-09	Huperzine A and analogs thereof
US4929731A (en)	1990-05-29	Method for the synthesis of huperzine A and analogs thereof and compounds useful therein
FR2563521A1 (fr)	1985-10-31	Derives de la 1,4-dihydro-4-oxonaphtyridine et leurs sels, procede pour leur production et agents antibacteriens les contenant
CN1662541A (zh)	2005-08-31	呋喃基化合物
US20030105124A1 (en)	2003-06-05	Substituted benzolactam compounds
CZ284789B6 (cs)	1999-03-17	Benzoxazinové deriváty, způsob jejich přípravy a farmaceutická kompozice tyto deriváty obsahující
CA2727669C (fr)	2016-08-23	Nouveaux derives de (piperazinyl ponte)-1-alcanone et leur utilisation comme inhibiteurs de p75
EP1175417B1 (fr)	2004-01-07	Composes de benzolactame substitues
US5604241A (en)	1997-02-18	Substituted benzylaminoquinuclidines as substance P antagonists
US6288225B1 (en)	2001-09-11	Substituted benzolactam compounds as substance P antagonists
OA11944A (en)	2006-04-12	1-Trifluoromethyl-4-hydroxy-7-piperidinyl-aminomethylchroman derivatives.
US5641785A (en)	1997-06-24	Oxazoloquinolinone derivatives, their preparation and their therapeutic application as inhibitors of monoamine oxidase
EP0385664B1 (fr)	1994-01-12	Benzoxazolones anti-inflammatoires
MXPA01011367A (en)	2002-06-05	Substituted benzolactam compounds
US20020052503A1 (en)	2002-05-02	Substituted benzolactam compounds as substance p antagonists
JPH0656806A (ja)	1994-03-01	モルホリン誘導体およびその製造方法
HK1035189A (en)	2001-11-16	2-aminopyridines containing fused ring substituents as nitric oxide synthase inhibitors
EP1100799A1 (fr)	2001-05-23	Preparation de derives de la camptothecine et de la nothapodytine
JPWO1996033992A1 (ja)	1998-06-30	光学活性キノリンカルボン酸誘導体およびその塩