OA12413A - Combination of GABA agonists and aldose reductase inhibitors. - Google Patents

Combination of GABA agonists and aldose reductase inhibitors. Download PDF

Info

Publication number: OA12413A
Authority: OA; OAPI
Prior art keywords: prodrug; gaba; pharmaceutically acceptable; pharmaceutical composition; diabetic
Prior art date: 2000-11-30

Application number

OA1200300138A

Other languages

English (en)

Inventor

Banavara Lakshman Mylari

Original Assignee

Pfizer Prod Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-11-30

Filing date

2001-11-19

Publication date

2004-09-30

2001-11-19 Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc

2004-09-30 Publication of OA12413A publication Critical patent/OA12413A/en

Links

239000003477 4 aminobutyric acid receptor stimulating agent Substances 0.000 title claims abstract description 56
239000003288 aldose reductase inhibitor Substances 0.000 title description 32
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239000000651 prodrug Substances 0.000 claims abstract description 81
239000008194 pharmaceutical composition Substances 0.000 claims abstract description 36
208000002249 Diabetes Complications Diseases 0.000 claims abstract description 9
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208000032131 Diabetic Neuropathies Diseases 0.000 claims abstract description 6
206010012689 Diabetic retinopathy Diseases 0.000 claims abstract description 6
208000033679 diabetic kidney disease Diseases 0.000 claims abstract description 6
208000032781 Diabetic cardiomyopathy Diseases 0.000 claims abstract description 5
206010063547 Diabetic macroangiopathy Diseases 0.000 claims abstract description 5
206010054044 Diabetic microangiopathy Diseases 0.000 claims abstract description 5
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BTCSSZJGUNDROE-UHFFFAOYSA-N gamma-aminobutyric acid Chemical compound NCCCC(O)=O BTCSSZJGUNDROE-UHFFFAOYSA-N 0.000 claims description 21
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Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

OA1200300138A 2000-11-30 2001-11-19 Combination of GABA agonists and aldose reductase inhibitors. OA12413A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US25044800P	2000-11-30	2000-11-30

Publications (1)

Publication Number	Publication Date
OA12413A true OA12413A (en)	2004-09-30

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OA1200300138A OA12413A (en)	2000-11-30	2001-11-19	Combination of GABA agonists and aldose reductase inhibitors.

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US (1)	US6720348B2 (fr)
EP (1)	EP1337272A2 (fr)
JP (1)	JP2004514700A (fr)
KR (1)	KR20030059287A (fr)
CN (1)	CN1477976A (fr)
AP (1)	AP2001002359A0 (fr)
AR (1)	AR031432A1 (fr)
AU (1)	AU2002215160A1 (fr)
BG (1)	BG107812A (fr)
BR (1)	BR0115776A (fr)
CA (1)	CA2430309A1 (fr)
CR (1)	CR6962A (fr)
CZ (1)	CZ20031387A3 (fr)
DO (1)	DOP2001000294A (fr)
EA (1)	EA200300433A1 (fr)
EC (1)	ECSP034629A (fr)
EE (1)	EE200300249A (fr)
HR (1)	HRP20030419A2 (fr)
HU (1)	HUP0302555A3 (fr)
IL (1)	IL155710A0 (fr)
IS (1)	IS6787A (fr)
MA (1)	MA26965A1 (fr)
MX (1)	MXPA03004871A (fr)
NO (1)	NO20032387L (fr)
OA (1)	OA12413A (fr)
PA (1)	PA8534201A1 (fr)
PE (1)	PE20020598A1 (fr)
PL (1)	PL365378A1 (fr)
SK (1)	SK6092003A3 (fr)
SV (1)	SV2003000752A (fr)
TN (1)	TNSN01170A1 (fr)
UY (1)	UY27044A1 (fr)
WO (1)	WO2002043763A2 (fr)
ZA (1)	ZA200303340B (fr)

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AU2003243603A1 (en) *	2002-06-13	2003-12-31	Board Of Regents, The University Of Texas System	Methods and compositions involving aldose reductase inhibitors
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2001
- 2001-11-19 CA CA002430309A patent/CA2430309A1/fr not_active Abandoned
- 2001-11-19 MX MXPA03004871A patent/MXPA03004871A/es unknown
- 2001-11-19 IL IL15571001A patent/IL155710A0/xx unknown
- 2001-11-19 JP JP2002545733A patent/JP2004514700A/ja not_active Withdrawn
- 2001-11-19 OA OA1200300138A patent/OA12413A/en unknown
- 2001-11-19 KR KR10-2003-7007221A patent/KR20030059287A/ko not_active Ceased
- 2001-11-19 WO PCT/IB2001/002214 patent/WO2002043763A2/fr not_active Ceased
- 2001-11-19 EP EP01983740A patent/EP1337272A2/fr not_active Withdrawn
- 2001-11-19 EA EA200300433A patent/EA200300433A1/ru unknown
- 2001-11-19 CN CNA018195954A patent/CN1477976A/zh active Pending
- 2001-11-19 PL PL01365378A patent/PL365378A1/xx not_active Application Discontinuation
- 2001-11-19 HU HU0302555A patent/HUP0302555A3/hu unknown
- 2001-11-19 AU AU2002215160A patent/AU2002215160A1/en not_active Abandoned
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- 2001-11-19 HR HR20030419A patent/HRP20030419A2/hr not_active Application Discontinuation
- 2001-11-19 SK SK609-2003A patent/SK6092003A3/sk not_active Application Discontinuation
- 2001-11-19 AP APAP/P/2001/002359A patent/AP2001002359A0/en unknown
- 2001-11-19 BR BR0115776-0A patent/BR0115776A/pt not_active IP Right Cessation
- 2001-11-19 EE EEP200300249A patent/EE200300249A/xx unknown
- 2001-11-26 DO DO2001000294A patent/DOP2001000294A/es unknown
- 2001-11-27 PE PE2001001187A patent/PE20020598A1/es not_active Application Discontinuation
- 2001-11-28 AR ARP010105542A patent/AR031432A1/es not_active Application Discontinuation
- 2001-11-28 UY UY27044A patent/UY27044A1/es not_active Application Discontinuation
- 2001-11-29 TN TNTNSN01170A patent/TNSN01170A1/fr unknown
- 2001-11-29 US US09/997,039 patent/US6720348B2/en not_active Expired - Fee Related
- 2001-11-30 SV SV2001000752A patent/SV2003000752A/es unknown
- 2001-11-30 PA PA20018534201A patent/PA8534201A1/es unknown
2003
- 2003-04-14 IS IS6787A patent/IS6787A/is unknown
- 2003-04-24 CR CR6962A patent/CR6962A/es not_active Application Discontinuation
- 2003-04-30 ZA ZA200303340A patent/ZA200303340B/en unknown
- 2003-05-13 BG BG107812A patent/BG107812A/bg unknown
- 2003-05-20 MA MA27166A patent/MA26965A1/fr unknown
- 2003-05-27 NO NO20032387A patent/NO20032387L/no not_active Application Discontinuation
- 2003-05-28 EC EC2003004629A patent/ECSP034629A/es unknown

Also Published As

Publication number	Publication date
MA26965A1 (fr)	2004-12-20
JP2004514700A (ja)	2004-05-20
US6720348B2 (en)	2004-04-13
PE20020598A1 (es)	2002-07-08
CZ20031387A3 (cs)	2004-04-14
PL365378A1 (en)	2005-01-10
EE200300249A (et)	2003-10-15
BR0115776A (pt)	2004-01-13
NO20032387D0 (no)	2003-05-27
EA200300433A1 (ru)	2003-10-30
KR20030059287A (ko)	2003-07-07
HUP0302555A3 (en)	2005-06-28
HUP0302555A2 (hu)	2003-11-28
TNSN01170A1 (fr)	2005-11-10
UY27044A1 (es)	2002-07-31
EP1337272A2 (fr)	2003-08-27
AU2002215160A1 (en)	2002-06-11
MXPA03004871A (es)	2003-08-19
BG107812A (bg)	2004-02-27
DOP2001000294A (es)	2002-08-30
HRP20030419A2 (en)	2004-08-31
SK6092003A3 (en)	2004-07-07
ECSP034629A (es)	2003-07-25
IL155710A0 (en)	2003-11-23
WO2002043763A3 (fr)	2003-03-13
WO2002043763A2 (fr)	2002-06-06
IS6787A (is)	2003-04-14
SV2003000752A (es)	2003-01-13
US20020077319A1 (en)	2002-06-20
AR031432A1 (es)	2003-09-24
AP2001002359A0 (en)	2001-12-31
PA8534201A1 (es)	2002-10-24
NO20032387L (no)	2003-05-27
CR6962A (es)	2004-02-02
CN1477976A (zh)	2004-02-25
ZA200303340B (en)	2004-04-30
CA2430309A1 (fr)	2002-06-06

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