OA12735A - Salts forms of E-2-methoxy-N-(3-(4-(3-methyl-pyridin-3-yloxy)-phenylamino)-quinazolin-6-YL)-allyl)-acetamide, its preparation ant its use against cancer. - Google Patents
Salts forms of E-2-methoxy-N-(3-(4-(3-methyl-pyridin-3-yloxy)-phenylamino)-quinazolin-6-YL)-allyl)-acetamide, its preparation ant its use against cancer. Download PDFInfo
- Publication number
- OA12735A OA12735A OA1200400161A OA1200400161A OA12735A OA 12735 A OA12735 A OA 12735A OA 1200400161 A OA1200400161 A OA 1200400161A OA 1200400161 A OA1200400161 A OA 1200400161A OA 12735 A OA12735 A OA 12735A
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- OA
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- Prior art keywords
- cancer
- methyl
- acetamide
- pyridin
- methoxy
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Classifications
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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Landscapes
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- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US34088501P | 2001-12-12 | 2001-12-12 |
Publications (1)
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|---|---|
| OA12735A true OA12735A (en) | 2006-06-29 |
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| OA1200400161A OA12735A (en) | 2001-12-12 | 2002-11-11 | Salts forms of E-2-methoxy-N-(3-(4-(3-methyl-pyridin-3-yloxy)-phenylamino)-quinazolin-6-YL)-allyl)-acetamide, its preparation ant its use against cancer. |
Country Status (34)
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| US (1) | US6844349B2 (sr) |
| EP (1) | EP1456199A1 (sr) |
| JP (1) | JP4202926B2 (sr) |
| KR (1) | KR20040065259A (sr) |
| CN (1) | CN1608062A (sr) |
| AP (1) | AP2004003059A0 (sr) |
| AR (1) | AR037772A1 (sr) |
| AU (1) | AU2002366581A1 (sr) |
| BR (1) | BR0214876A (sr) |
| CA (1) | CA2469889A1 (sr) |
| DO (1) | DOP2002000544A (sr) |
| EA (1) | EA007412B1 (sr) |
| EC (1) | ECSP045148A (sr) |
| GE (1) | GEP20063872B (sr) |
| GT (1) | GT200200272A (sr) |
| HR (1) | HRP20040530A2 (sr) |
| HU (1) | HUP0402662A2 (sr) |
| IL (1) | IL161915A0 (sr) |
| IS (1) | IS7227A (sr) |
| MA (1) | MA27095A1 (sr) |
| MX (1) | MXPA04005678A (sr) |
| NO (1) | NO20042925L (sr) |
| NZ (1) | NZ532436A (sr) |
| OA (1) | OA12735A (sr) |
| PA (1) | PA8561401A1 (sr) |
| PE (1) | PE20030716A1 (sr) |
| PL (1) | PL370858A1 (sr) |
| RS (1) | RS46404A (sr) |
| TN (1) | TNSN04112A1 (sr) |
| TW (1) | TW200301103A (sr) |
| UA (1) | UA75482C2 (sr) |
| UY (1) | UY27572A1 (sr) |
| WO (1) | WO2003050108A1 (sr) |
| ZA (1) | ZA200402995B (sr) |
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| WO2005044264A1 (en) * | 2003-10-27 | 2005-05-19 | Merck & Co., Inc. | Ccr-2 antagonist salt |
| US20050192298A1 (en) * | 2004-02-27 | 2005-09-01 | Pfizer Inc | Crystal forms of E-2-Methoxy-N-(3-{4-[3-methyl-4-(6-methyl-pyridin-3-yloxy)-phenylamino]-quinazolin-6-yl}-allyl)-acetamide |
| WO2005121124A1 (en) * | 2004-06-07 | 2005-12-22 | Pfizer Products Inc. | Complexes of e-2-methoxy-n-(3-{4-[3-methyl-pyridin-3-yloxy)-phenylamino]-quinazolin-6-yl}-allyl)-acetamide and methods of preparing same |
| PL216369B1 (pl) | 2004-07-27 | 2014-03-31 | Gilead Sciences | Pochodne fosfonianowe, kompozycje farmaceutyczne zawierające te pochodne oraz zastosowanie tych pochodnych do wytwarzania leku do hamowania wirusa HIV |
| JP2008542354A (ja) * | 2005-06-03 | 2008-11-27 | ファイザー・プロダクツ・インク | 癌治療におけるerbB2阻害剤と他の治療薬の併用 |
| CA2610491A1 (en) * | 2005-06-03 | 2006-12-07 | Pfizer Products Inc. | Bicyclic derivatives for the treatment of abnormal cell growth |
| DK2020996T3 (da) * | 2006-05-16 | 2012-02-27 | Gilead Sciences Inc | Fremgangsmåder og sammensætninger til behandling af hæmatologiske sygdomme |
| RU2009126576A (ru) | 2006-12-12 | 2011-01-20 | Такеда Фармасьютикал Компани Лимитед (Jp) | Конденсированное гетероциклическое соединение |
| PT2125786E (pt) * | 2006-12-21 | 2011-04-21 | Pfizer Prod Inc | Sal succinato de 2-((4-(1-metil-4-(piridin-4-il)-1hpirazol- 3-il)fenoxi)metil)quinolina |
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| UA108618C2 (uk) | 2009-08-07 | 2015-05-25 | Застосування c-met-модуляторів в комбінації з темозоломідом та/або променевою терапією для лікування раку | |
| US9265739B2 (en) | 2010-06-02 | 2016-02-23 | The Trustees Of The University Of Pennsylvania | Methods and use of compounds that bind to HER2/neu receptor complex |
| US8993634B2 (en) | 2010-06-02 | 2015-03-31 | The Trustees Of The University Of Pennsylvania | Methods and use of compounds that bind to Her2/neu receptor complex |
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| EP3806887A4 (en) | 2018-06-13 | 2022-04-06 | California Institute of Technology | Nanoparticles for crossing the blood brain barrier and methods of treatment using the same |
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| US6884418B1 (en) | 1989-08-04 | 2005-04-26 | Berlex Laboratories, Inc. | Use of ligand-mimicking agents and anti-neoplastic drugs in cancer therapy |
| GB9510757D0 (en) * | 1994-09-19 | 1995-07-19 | Wellcome Found | Therapeuticaly active compounds |
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| MXPA02012870A (es) * | 2000-06-22 | 2003-05-14 | Pfizer Prod Inc | Derivados biciclicos sustituidos para el tratamiento del crecimiento celular anormal. |
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- 2002-11-11 BR BR0214876-5A patent/BR0214876A/pt not_active IP Right Cessation
- 2002-11-11 EP EP02804543A patent/EP1456199A1/en not_active Withdrawn
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- 2002-11-11 CN CNA028248554A patent/CN1608062A/zh active Pending
- 2002-11-11 CA CA002469889A patent/CA2469889A1/en not_active Abandoned
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- 2002-11-11 MX MXPA04005678A patent/MXPA04005678A/es active IP Right Grant
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- 2002-11-11 OA OA1200400161A patent/OA12735A/en unknown
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- 2002-11-11 WO PCT/IB2002/004708 patent/WO2003050108A1/en not_active Ceased
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- 2002-12-09 UY UY27572A patent/UY27572A1/es not_active Application Discontinuation
- 2002-12-10 US US10/315,862 patent/US6844349B2/en not_active Expired - Fee Related
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