OA13039A - 3-(1-[3-(1,3-benzothiazol-6-yl)propylcarbamoyl]cycloalkyl)propanoic acid derivatives as NEP inhibitors. - Google Patents

3-(1-[3-(1,3-benzothiazol-6-yl)propylcarbamoyl]cycloalkyl)propanoic acid derivatives as NEP inhibitors. Download PDF

Info

Publication number: OA13039A
Authority: OA; OAPI
Prior art keywords: disorder; methyl; compound; compounds; sexual
Prior art date: 2003-03-14

Application number

OA1200500261A

Other languages

English (en)

Inventor

David Hepworth

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-03-14

Filing date

2004-03-09

Publication date

2006-11-10

2003-03-14 Priority claimed from GB0305916A external-priority patent/GB0305916D0/en

2003-12-16 Priority claimed from GB0329143A external-priority patent/GB0329143D0/en

2004-03-09 Application filed by Pfizer filed Critical Pfizer

2006-11-10 Publication of OA13039A publication Critical patent/OA13039A/en

Links

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Rheumatology (AREA)
Gynecology & Obstetrics (AREA)
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Pregnancy & Childbirth (AREA)
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Gastroenterology & Hepatology (AREA)

OA1200500261A 2003-03-14 2004-03-09 3-(1-[3-(1,3-benzothiazol-6-yl)propylcarbamoyl]cycloalkyl)propanoic acid derivatives as NEP inhibitors. OA13039A (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB0305916A GB0305916D0 (en)	2003-03-14	2003-03-14	New N-phenpropylcyclopentyl-substituted glutaramide derivatives as NEP inhibitors
GB0329143A GB0329143D0 (en)	2003-12-16	2003-12-16	Novel pharmaceuticals

Publications (1)

Publication Number	Publication Date
OA13039A true OA13039A (en)	2006-11-10

Family

ID=32992599

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
OA1200500261A OA13039A (en)	2003-03-14	2004-03-09	3-(1-[3-(1,3-benzothiazol-6-yl)propylcarbamoyl]cycloalkyl)propanoic acid derivatives as NEP inhibitors.

Country Status (25)

Country	Link
US (1)	US20040180941A1 (fr)
EP (1)	EP1606272A1 (fr)
JP (1)	JP3923512B2 (fr)
KR (1)	KR20050110003A (fr)
AP (1)	AP2005003393A0 (fr)
AR (1)	AR043551A1 (fr)
AU (1)	AU2004220269A1 (fr)
BR (1)	BRPI0408377A (fr)
CA (1)	CA2519072A1 (fr)
CL (1)	CL2004000512A1 (fr)
EA (1)	EA200501204A1 (fr)
EC (1)	ECSP056017A (fr)
HR (1)	HRP20050797A2 (fr)
IS (1)	IS8003A (fr)
MA (1)	MA27720A1 (fr)
MX (1)	MXPA05009788A (fr)
NL (1)	NL1025709C2 (fr)
NO (1)	NO20054169L (fr)
OA (1)	OA13039A (fr)
PA (1)	PA8597401A1 (fr)
PE (1)	PE20050310A1 (fr)
TN (1)	TNSN05227A1 (fr)
TW (1)	TW200504038A (fr)
UY (1)	UY28226A1 (fr)
WO (1)	WO2004080985A1 (fr)

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WO2006027680A1 (fr) *	2004-09-10	2006-03-16	Pfizer Limited	Derives d'acide 3-(1-carbamoylcyclohexyl)propionique comme inhibiteurs de l'enzyme endopeptidase neutre
WO2006066361A1 (fr) *	2004-12-24	2006-06-29	The University Of Queensland	Procede de traitement ou prophylaxie
JP2009502961A (ja)	2005-07-29	2009-01-29	コンサートファーマシューティカルズインコーポレイテッド	新規な医薬組成物
US20070178141A1 (en) *	2005-09-07	2007-08-02	Bebaas, Inc.	Vitamin B12 compositions
US20130131007A1 (en)	2005-09-07	2013-05-23	Bebaas, Inc.	Vitamin b12 compositions
AU2007229322B2 (en) *	2006-03-20	2012-04-05	Novartis Ag	Method of treatment or prophylaxis inflammatory pain
WO2008021666A2 (fr) *	2006-08-18	2008-02-21	Morton Grove Pharmaceuticals, Inc.	Compositions stables de lévétiracétam et procédés
KR101177866B1 (ko)	2011-03-24	2012-08-28	주식회사 케이엠더블유	케이블 접속 장치
WO2019241588A1 (fr) *	2018-06-14	2019-12-19	Astrazeneca Uk Limited	Méthodes de traitement d'une dysfonction érectile avec une composition pharmaceutique d'inhibiteur de phosphodiestérase 5 spécifique de cgmp
WO2019241585A1 (fr) *	2018-06-14	2019-12-19	Astrazeneca Uk Limited	Méthodes de traitement d'une dysfonction érectile avec une composition pharmaceutique d'inhibiteur de phosphodiestérase 5 spécifique de cgmp
SG11202102791SA (en)	2018-09-25	2021-04-29	Antabio Sas	Indane derivatives for use in the treatment of bacterial infection
IL292775A (en) *	2019-11-08	2022-07-01	Vella Bioscience Inc	preparations containing cannabidiol (cbd) that act peripherally and their use to improve female sexual function or to treat female sexual disorders
GB202402524D0 (en) *	2024-02-22	2024-04-10	Futura Medical Developments Ltd	Topical composition

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US3238215A (en) *	1963-10-17	1966-03-01	Sterling Drug Inc	1-[(3-, 2-, and 1-indolyl)-lower-alkyl-, lower-alkenyl-, and lower-alkynyl]piperidines
IT1066857B (it) *	1965-12-15	1985-03-12	Acraf	Derivati della s ipiazolo 4.3 a piridina e processi per la loro preparazione
US3511836A (en) *	1967-12-13	1970-05-12	Pfizer & Co C	2,4,6,7-tetra substituted quinazolines
NL175059C (nl) *	1974-02-23		Boehringer Mannheim Gmbh	Bereiding van bloeddrukverlagende stoffen en van preparaten die ze bevatten.
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FR2421888A1 (fr) *	1978-02-06	1979-11-02	Synthelabo	Amides d'alkylene-diamines et leur application en therapeutique
IT1094076B (it) *	1978-04-18	1985-07-26	Acraf	Cicloalchiltriazoli
JPS56110665A (en) *	1980-02-08	1981-09-01	Yamanouchi Pharmaceut Co Ltd	Sulfamoyl-substituted phenetylamine derivative and its preparation
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2004
- 2004-03-08 PA PA20048597401A patent/PA8597401A1/es unknown
- 2004-03-09 BR BRPI0408377-6A patent/BRPI0408377A/pt not_active IP Right Cessation
- 2004-03-09 WO PCT/IB2004/000822 patent/WO2004080985A1/fr not_active Ceased
- 2004-03-09 EA EA200501204A patent/EA200501204A1/ru unknown
- 2004-03-09 CA CA002519072A patent/CA2519072A1/fr not_active Abandoned
- 2004-03-09 OA OA1200500261A patent/OA13039A/en unknown
- 2004-03-09 AU AU2004220269A patent/AU2004220269A1/en not_active Abandoned
- 2004-03-09 HR HR20050797A patent/HRP20050797A2/hr not_active Application Discontinuation
- 2004-03-09 MX MXPA05009788A patent/MXPA05009788A/es unknown
- 2004-03-09 JP JP2006500337A patent/JP3923512B2/ja not_active Expired - Fee Related
- 2004-03-09 EP EP04718706A patent/EP1606272A1/fr not_active Withdrawn
- 2004-03-09 KR KR1020057017229A patent/KR20050110003A/ko not_active Ceased
- 2004-03-09 AP AP2005003393A patent/AP2005003393A0/xx unknown
- 2004-03-10 PE PE2004000259A patent/PE20050310A1/es not_active Application Discontinuation
- 2004-03-11 UY UY28226A patent/UY28226A1/es not_active Application Discontinuation
- 2004-03-11 AR ARP040100785A patent/AR043551A1/es unknown
- 2004-03-12 US US10/800,065 patent/US20040180941A1/en not_active Abandoned
- 2004-03-12 NL NL1025709A patent/NL1025709C2/nl not_active IP Right Cessation
- 2004-03-12 CL CL200400512A patent/CL2004000512A1/es unknown
- 2004-03-12 TW TW093106666A patent/TW200504038A/zh unknown
2005
- 2005-08-29 IS IS8003A patent/IS8003A/is unknown
- 2005-09-07 NO NO20054169A patent/NO20054169L/no not_active Application Discontinuation
- 2005-09-14 EC EC2005006017A patent/ECSP056017A/es unknown
- 2005-09-14 TN TNP2005000227A patent/TNSN05227A1/fr unknown
- 2005-09-14 MA MA28498A patent/MA27720A1/fr unknown

Also Published As

Publication number	Publication date
PE20050310A1 (es)	2005-05-04
AR043551A1 (es)	2005-08-03
HRP20050797A2 (en)	2006-02-28
IS8003A (is)	2005-08-29
AU2004220269A1 (en)	2004-09-23
PA8597401A1 (es)	2005-05-24
NL1025709A1 (nl)	2004-09-16
CL2004000512A1 (es)	2005-01-21
WO2004080985A1 (fr)	2004-09-23
MA27720A1 (fr)	2006-01-02
NO20054169L (no)	2005-12-07
EA200501204A1 (ru)	2006-06-30
NL1025709C2 (nl)	2005-03-14
US20040180941A1 (en)	2004-09-16
TNSN05227A1 (fr)	2007-06-11
JP2006526572A (ja)	2006-11-24
EP1606272A1 (fr)	2005-12-21
MXPA05009788A (es)	2005-10-26
TW200504038A (en)	2005-02-01
JP3923512B2 (ja)	2007-06-06
BRPI0408377A (pt)	2006-03-21
NO20054169D0 (no)	2005-09-07
ECSP056017A (es)	2006-01-27
UY28226A1 (es)	2004-11-08
AP2005003393A0 (en)	2005-09-30
CA2519072A1 (fr)	2004-09-23
KR20050110003A (ko)	2005-11-22

Publication	Publication Date	Title
WO2006027680A1 (fr)	2006-03-16	Derives d'acide 3-(1-carbamoylcyclohexyl)propionique comme inhibiteurs de l'enzyme endopeptidase neutre
SK18182002A3 (sk)	2004-04-06	Deriváty glutaramidu substituované cyklopentylskupinou ako inhibítory neutrálnej endopeptidázy
US11485727B2 (en)	2022-11-01	N-methyl, n-(6-(methoxy)pyridazin-3-yl) amine derivatives as autotaxin (ATX) modulators
RS75303A (sr)	2006-12-15	Derivati n-fenilpropilciklopentil-supstituisanog glutaramida kao nep inhibitori za fsad
US20040180941A1 (en)	2004-09-16	3-(1-[3-(1,3-Benzothiazol-6-yl)propylcarbamoyl]cycloalkyl)propanoic acid derivatives as NEP inhibitors
US20080167371A1 (en)	2008-07-10	Diaryl, Dipyridinyl and Aryl-Pyridinyl Derivatives and Uses Thereof
MXPA02009697A (es)	2003-03-27	Compuestos de eter difenilico utiles en terapia.
US12391667B2 (en)	2025-08-19	N-methyl, n-(6-(methoxy)pyridazin-3-yl) amine derivatives as Autotaxin (ATX) modulators for the treatment of inflammatory airway or fibrotic diseases
US11465982B2 (en)	2022-10-11	Pyridazines
US20090005354A1 (en)	2009-01-01	New Amino Derivatives and Their Use as Pharmaceuticals
US20040063643A1 (en)	2004-04-01	Bombesin antagonists
US20070185078A1 (en)	2007-08-09	Substituted triazole derivatives as oxytocin antagonists
JPH07500604A (ja)	1995-01-19	高血圧治療用エチルアラニンアミノジオール化合物
AU2005247699A1 (en)	2005-12-08	Aminopyridine derivatives as selective dopamine D3 agonists
US20030105097A1 (en)	2003-06-05	Alkylamide compounds
US20050267096A1 (en)	2005-12-01	New indazole and indolone derivatives and their use pharmaceuticals
US20100222365A1 (en)	2010-09-02	Substituted triazole deriviatives as oxytocin antagonists
US7618972B2 (en)	2009-11-17	Substituted triazole derivatives as oxytocin antagonists
JP2003012626A (ja)	2003-01-15	アルキルアミド化合物
ZA200506500B (en)	2006-11-29	3-(1-[3-(1,3-benzothiazol-6-YL)propylcarbamoyl]cycloalykl)propanoic acid derivatives as nep inhibitors
KR20070022795A (ko)	2007-02-27	선택적 도파민 ｄ3 효능제로서의 아미노피리딘 유도체
CA2751866A1 (fr)	2010-08-19	Derives de n-[(6-aza-bicyclo[3.2.1]oct-1-yl)-aryl-methyl]-benzamide, leur preparation et leur application en therapeutique
HK1055109A (en)	2003-12-24	Cyclopentyl-substituted glutaramide derivatives as inhibitors of neutral endopeptidase