PE20120689A1 - Derivados de 5-fluoro-2-oxopirimidina-1(2h)-carboxilato - Google Patents

Derivados de 5-fluoro-2-oxopirimidina-1(2h)-carboxilato

Info

Publication number: PE20120689A1
Authority: PE; Peru
Prior art keywords: fluoro; oxopyrimidine; optionally substituted; carboxylate; compounds
Prior art date: 2009-08-07

Application number

PE2012000170A

Other languages

English (en)

Spanish (es)

Inventor

Timothy Boebel

Kristy Bryan

Beth Lorsbach

Timothy Martin

W Owen

Mark Pobanz

Scott Thornburgh

Jeffery Webster

Chenglin Yao

Original Assignee

Dow Agrosciences Llc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2009-08-07

Filing date

2010-08-05

Publication date

2012-06-06

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535293&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PE20120689(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2010-08-05 Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc

2012-06-06 Publication of PE20120689A1 publication Critical patent/PE20120689A1/es

Links

HRHMGDXHJNYKSR-UHFFFAOYSA-N OC(=O)N1C=C(F)C=NC1=O Chemical class OC(=O)N1C=C(F)C=NC1=O HRHMGDXHJNYKSR-UHFFFAOYSA-N 0.000 title abstract 2
150000001875 compounds Chemical class 0.000 abstract 3
-1 2,2-DIMETHYL-PROPYL Chemical class 0.000 abstract 1
101000977048 Streptomyces cinnamonensis Uncharacterized protein in mutB 3'region Proteins 0.000 abstract 1
239000002253 acid Substances 0.000 abstract 1
MMNNNCCLKAWPPZ-UHFFFAOYSA-N ethyl 4-amino-5-fluoro-2-oxopyrimidine-1-carboxylate Chemical compound CCOC(=O)N1C=C(F)C(N)=NC1=O MMNNNCCLKAWPPZ-UHFFFAOYSA-N 0.000 abstract 1
239000000417 fungicide Substances 0.000 abstract 1
229910052736 halogen Inorganic materials 0.000 abstract 1
150000002367 halogens Chemical group 0.000 abstract 1
CJEOHCPDDTWSQV-UHFFFAOYSA-N o-phenyl 4-amino-5-fluoro-2-oxopyrimidine-1-carbothioate Chemical compound C1=C(F)C(N)=NC(=O)N1C(=S)OC1=CC=CC=C1 CJEOHCPDDTWSQV-UHFFFAOYSA-N 0.000 abstract 1
230000002265 prevention Effects 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
- A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
- A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
- A01N47/16—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof the nitrogen atom being part of a heterocyclic ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/20—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D239/22—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to ring carbon atoms

Landscapes

Life Sciences & Earth Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Environmental Sciences (AREA)
Engineering & Computer Science (AREA)
Dentistry (AREA)
General Health & Medical Sciences (AREA)
Wood Science & Technology (AREA)
Zoology (AREA)
Plant Pathology (AREA)
Pest Control & Pesticides (AREA)
Agronomy & Crop Science (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Plural Heterocyclic Compounds (AREA)

PE2012000170A 2009-08-07 2010-08-05 Derivados de 5-fluoro-2-oxopirimidina-1(2h)-carboxilato PE20120689A1 (es)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US23223209P	2009-08-07	2009-08-07

Publications (1)

Publication Number	Publication Date
PE20120689A1 true PE20120689A1 (es)	2012-06-06

Family

ID=43535293

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PE2012000170A PE20120689A1 (es)	2009-08-07	2010-08-05	Derivados de 5-fluoro-2-oxopirimidina-1(2h)-carboxilato

Country Status (28)

Country	Link
US (1)	US8318758B2 (2)
EP (1)	EP2462133B1 (2)
JP (1)	JP5818791B2 (2)
KR (1)	KR101792286B1 (2)
CN (1)	CN102548979B (2)
AU (1)	AU2010279408B2 (2)
BR (1)	BR112012002807B1 (2)
CA (1)	CA2769251C (2)
CL (1)	CL2012000314A1 (2)
CO (1)	CO6491089A2 (2)
CR (1)	CR20120033A (2)
DK (1)	DK2462133T3 (2)
EA (1)	EA022930B1 (2)
EC (1)	ECSP12011651A (2)
ES (1)	ES2506169T3 (2)
HN (1)	HN2012000261A (2)
IL (1)	IL217954A (2)
IN (1)	IN2012DN00695A (2)
MX (1)	MX2012001623A (2)
NI (1)	NI201200019A (2)
NZ (1)	NZ597638A (2)
PE (1)	PE20120689A1 (2)
PL (1)	PL2462133T3 (2)
PT (1)	PT2462133E (2)
RS (1)	RS53658B1 (2)
UA (1)	UA106086C2 (2)
WO (1)	WO2011017544A1 (2)
ZA (1)	ZA201305992B (2)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ES2471371T3 (es) *	2009-08-07	2014-06-26	Dow Agrosciences Llc	Derivados de N1-sulfonil-5-fluoropirimidinona
CA2894510A1 (en)	2012-12-28	2014-07-03	Dow Agrosciences Llc	N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2h)-carboxamide derivatives
MX2015008443A (es) *	2012-12-28	2015-09-23	Dow Agrosciences Llc	Derivados de 1-(benzoilo-sustituido) -5-fluoro-4-imino-3-metil-3, 4-dihidropirimidin-2 (1h)-ona.
RU2638556C2 (ru)	2012-12-28	2017-12-14	Адама Мактешим Лтд.	Производные n-(замещенного)-5-фтор-4-имино-3-метил-2-оксо-3,4-дигидропиримидин-1(2н)-карбоксилата
AU2013370494B2 (en)	2012-12-31	2017-08-17	Adama Makhteshim Ltd.	3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1H)-one derivatives as fungicides
NZ722419A (en)	2013-12-31	2018-01-26	Adama Makhteshim Ltd	Synergistic fungicidal mixtures and compositions for fungal control
CA2935594C (en)	2013-12-31	2022-05-03	Nakyen Choy	5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
WO2016040193A1 (en)	2014-09-08	2016-03-17	Samumed, Llc	3-(1h-imidazo[4,5-c]pyridin-2-yl)-1h-pyrazolo[3,4-b]pyridine and therapeutic uses thereof
BR112018009252A2 (pt)	2015-11-06	2018-11-06	Samumed Llc	tratamento da osteoartrite
LT3464285T (lt)	2016-06-01	2022-12-27	Biosplice Therapeutics, Inc.	N-(5-(3-(7-(3-fluorfenil)-3h-imidazo[4,5-c]piridin-2-il)-1h-indazol-5-il)piridin-3-il)- 3-metilbutanamido gamybos būdas
EP3655396A1 (en)	2017-07-17	2020-05-27	Adama Makhteshim Ltd.	Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
EP3876717A1 (en)	2018-11-05	2021-09-15	Adama Makhteshim Ltd.	Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof
PY2057637A (es)	2019-09-23	2021-10-05	Adama Makhteshim Ltd	Proceso para preparar 5-(fluoro-4-imino-3-metil)-1-tosil-3,4-dihidropirimidin-(1h)-ona y derivados del compuesto

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3368938A (en) *	1966-01-13	1968-02-13	Hoffmann La Roche	Controlling fungi with 5-fluorocytosine
ATE216999T1 (de) *	1996-03-11	2002-05-15	Syngenta Participations Ag	Pyrimidin-4-on derivate als pestizidesmittel
WO2004037159A2 (en) *	2002-10-23	2004-05-06	Obetherapy Biotechnology	Compounds, compositions and methods for modulating fat metabolism
BRPI0810821A8 (pt) *	2007-04-27	2015-09-15	Asubio Pharma Co Ltd	Derivados de anéis aromáticos de seis membros contendo nitrogênio e produtos farmacêuticos contendo os mesmos
CN102215691B (zh) *	2008-08-01	2015-02-04	陶氏益农公司	5-氟胞嘧啶作为杀真菌剂的用途

2010
- 2010-08-05 BR BR112012002807-3A patent/BR112012002807B1/pt active IP Right Grant
- 2010-08-05 DK DK10807174.7T patent/DK2462133T3/en active
- 2010-08-05 EA EA201270255A patent/EA022930B1/ru not_active IP Right Cessation
- 2010-08-05 US US12/851,304 patent/US8318758B2/en active Active
- 2010-08-05 EP EP10807174.7A patent/EP2462133B1/en active Active
- 2010-08-05 PL PL10807174T patent/PL2462133T3/pl unknown
- 2010-08-05 IN IN695DEN2012 patent/IN2012DN00695A/en unknown
- 2010-08-05 AU AU2010279408A patent/AU2010279408B2/en not_active Ceased
- 2010-08-05 MX MX2012001623A patent/MX2012001623A/es active IP Right Grant
- 2010-08-05 CA CA2769251A patent/CA2769251C/en not_active Expired - Fee Related
- 2010-08-05 PT PT108071747T patent/PT2462133E/pt unknown
- 2010-08-05 UA UAA201202680A patent/UA106086C2/uk unknown
- 2010-08-05 KR KR1020127005932A patent/KR101792286B1/ko not_active Expired - Fee Related
- 2010-08-05 NZ NZ597638A patent/NZ597638A/en unknown
- 2010-08-05 CN CN201080045339.3A patent/CN102548979B/zh active Active
- 2010-08-05 PE PE2012000170A patent/PE20120689A1/es not_active Application Discontinuation
- 2010-08-05 WO PCT/US2010/044585 patent/WO2011017544A1/en not_active Ceased
- 2010-08-05 RS RS20140630A patent/RS53658B1/sr unknown
- 2010-08-05 ES ES10807174.7T patent/ES2506169T3/es active Active
- 2010-08-05 JP JP2012523954A patent/JP5818791B2/ja active Active
2012
- 2012-01-18 CR CR20120033A patent/CR20120033A/es unknown
- 2012-01-27 CO CO12012413A patent/CO6491089A2/es active IP Right Grant
- 2012-02-02 HN HN2012000261A patent/HN2012000261A/es unknown
- 2012-02-03 NI NI201200019A patent/NI201200019A/es unknown
- 2012-02-05 IL IL217954A patent/IL217954A/en active IP Right Grant
- 2012-02-06 CL CL2012000314A patent/CL2012000314A1/es unknown
- 2012-02-07 EC ECSP12011651 patent/ECSP12011651A/es unknown
2013
- 2013-08-14 ZA ZA2013/05992A patent/ZA201305992B/en unknown

Also Published As

Publication number	Publication date
CL2012000314A1 (es)	2012-10-05
IN2012DN00695A (2)	2015-06-19
CO6491089A2 (es)	2012-07-31
EP2462133B1 (en)	2014-09-24
KR20120043069A (ko)	2012-05-03
US8318758B2 (en)	2012-11-27
DK2462133T3 (en)	2015-01-05
ECSP12011651A (es)	2012-03-30
ES2506169T3 (es)	2014-10-13
IL217954A0 (en)	2012-03-29
AU2010279408B2 (en)	2015-09-10
NZ597638A (en)	2014-06-27
HK1172892A1 (en)	2013-05-03
US20110034491A1 (en)	2011-02-10
BR112012002807A2 (pt)	2015-10-13
BR112012002807B1 (pt)	2018-07-10
WO2011017544A1 (en)	2011-02-10
CA2769251A1 (en)	2011-02-10
HN2012000261A (es)	2015-01-05
RS53658B1 (sr)	2015-04-30
AU2010279408A1 (en)	2012-02-09
EP2462133A1 (en)	2012-06-13
EP2462133A4 (en)	2013-01-16
IL217954A (en)	2016-02-29
ZA201305992B (en)	2014-10-29
UA106086C2 (uk)	2014-07-25
EA201270255A1 (ru)	2012-07-30
CR20120033A (es)	2012-03-22
EA022930B1 (ru)	2016-03-31
PT2462133E (pt)	2014-12-26
PL2462133T3 (pl)	2015-03-31
MX2012001623A (es)	2012-04-11
NI201200019A (es)	2012-05-22
CA2769251C (en)	2018-05-15
KR101792286B1 (ko)	2017-10-31
CN102548979A (zh)	2012-07-04
BR112012002807A8 (pt)	2017-07-11
JP2013501726A (ja)	2013-01-17
JP5818791B2 (ja)	2015-11-18
CN102548979B (zh)	2015-05-13

Legal Events

Date	Code	Title	Description
2016-12-27	FG	Grant, registration
2019-03-27	FD	Application declared void or lapsed

Publication	Publication Date	Title
PE20120689A1 (es)	2012-06-06	Derivados de 5-fluoro-2-oxopirimidina-1(2h)-carboxilato
PE20120692A1 (es)	2012-06-08	Derivados de 5-fluoro-2-oxopirimidinona-1(2h)-carboxamida substituida-n1
PE20120690A1 (es)	2012-06-08	Derivados de 5-fluoropirimidinona
PE20120688A1 (es)	2012-06-06	Derivados de n1-acil-5-fluoropirimidinona
TN2011000346A1 (en)	2013-03-27	Benzoic acid (1-phenyl-2-pyridin-4-yl)ethyl esters as phosphodiesterase inhibitors
MX2015007883A (es)	2016-03-04	Compuestos para protección de células.
CO6341581A2 (es)	2011-11-21	Derivados de heteroarilo como inhibidores de dgat1
PE20091828A1 (es)	2009-12-21	Derivados de acido ciclopentanocarboxilico condensados sustituidos con acilamino como inhibidores de edg-2
PE20141726A1 (es)	2014-11-26	Heterociclilaminas como inhibidores de pi 3k
PE20050864A1 (es)	2005-10-31	Compuestos de heterociclilamino como inhibidores de 11-beta-hidroxiesteroide deshidrogenasa tipo 1
PE20121047A1 (es)	2012-08-02	Derivados de tiazolilpiperidina como fungicidas
CL2012000309A1 (es)	2012-10-05	Compuestos derivados de n1-sulfonil-5-fluoropirimidinona; composicion que los comprende; y metodo para el control y prevencion de un ataque fungico en una planta.
AR085960A1 (es)	2013-11-06	1,3-oxazinas como inhibidores de la bace1 y/o de la bace2
ES2590504T3 (es)	2016-11-22	N-ciclilamidas como nematicidas
PE20110420A1 (es)	2011-07-01	Nuevos derivados de 2-amidotiadiazol
UY32630A (es)	2010-12-31	Derivados de 7-aza-espiro[3.5]nonano-7-carboxilatos, su preparación y su aplicación en terapéutica.
PY0700623A (es)	2015-08-03	Acidos pirimidincarboxilicos 2-(arilo poli- sustituido)-6-amino-5-halo-4 y sus usos como herbicidas
PE20081487A1 (es)	2009-01-11	DERIVADOS DE NICOTINAMIDA COMO INHIBIDORES DE 11ßHSD1
PE20142164A1 (es)	2014-12-27	Inhibidores de diacilglicerol aciltransferasa 2
AR067915A1 (es)	2009-10-28	2-(2- fluor- fenil substituido )-6- amino-5- cloro-4- piridimidina carboxilatos y su uso como herbicidas
MX2014015501A (es)	2015-03-06	Carboxamidas heterociclicas fungicidas.
PE20141409A1 (es)	2014-10-01	Derivados de piridin-2(1h)-ona como inhibidores de jak
AR068115A1 (es)	2009-11-04	Derivado del acido pirazolcarboxilico metodo de produccion del mismo y fungicida
BR112016007427A2 (pt)	2017-05-02	compostos de pirazol-amida e usos dos mesmos
PE20090362A1 (es)	2009-04-04	Derivados de piperidina/piperazina como moduladores de dgat