|
US4820715A
(en)
*
|
1984-06-28 |
1989-04-11 |
Bristol-Myers Company |
Anti-emetic quinuclidinyl benzamides
|
|
US4816416A
(en)
*
|
1986-08-27 |
1989-03-28 |
Paul Averback |
Microspheric bodies for use in screening therapies for Azheimer's disease and related conditions
|
|
US5231170A
(en)
*
|
1986-08-27 |
1993-07-27 |
Paul Averback |
Antibodies to dense microspheres
|
|
DE3780276T2
(de)
*
|
1986-12-16 |
1993-02-25 |
Robins Co Inc A H |
Angstloesende n-(1-azabicyclo(2.2.2)oct-3-yl)benzamide und -thiobenzamide.
|
|
DE3751404T2
(de)
*
|
1986-12-17 |
1995-12-21 |
Glaxo Group Ltd |
Verwendung von heterocyclischen Verbindungen zur Behandlung von Bewusstseinsstörungen.
|
|
US5190954A
(en)
*
|
1986-12-17 |
1993-03-02 |
Glaxo Group Limited |
Methods for the treatment of cognitive disorders
|
|
US5246941A
(en)
*
|
1986-12-17 |
1993-09-21 |
Glaxo Group Limited |
Method for the treatment of depression
|
|
US5244909A
(en)
*
|
1986-12-17 |
1993-09-14 |
Glaxo Group Limited |
Methods for the treatment of cognitive disorders
|
|
US5200414A
(en)
*
|
1986-12-17 |
1993-04-06 |
Glaxo Group Limited |
Methods for the treatment of cognitive disorders
|
|
JP2608078B2
(ja)
*
|
1986-12-17 |
1997-05-07 |
グラクソ、グループ、リミテッド |
医 薬
|
|
GB8720805D0
(en)
*
|
1987-09-04 |
1987-10-14 |
Naylor R J |
2-alkoxy-n-(1-azabicyclo(2 2 2)oct-3-yl)benzamides & thiobenzamides
|
|
EP0311724A1
(fr)
*
|
1987-10-16 |
1989-04-19 |
Synthelabo |
R-N-(1-azabicyclo[2.2.2]oct-3-yl) benzamides et thiobenzamides anxiolytiques
|
|
US4863919A
(en)
*
|
1988-02-01 |
1989-09-05 |
A. H. Robins Company, Incorporated |
Method of enhancing memory or correcting memory deficiency with arylamido(and arylthiomido)-azabicycloalkanes
|
|
EP0353371A1
(fr)
*
|
1988-08-04 |
1990-02-07 |
Synthelabo |
R-N-(1-azabicyclo[2.2.2]oct-3-yl)benzamides et thiobenzamides améliorant la mémoire
|
|
US5229407A
(en)
*
|
1988-09-01 |
1993-07-20 |
Glaxo Group Limited |
Medicaments
|
|
GB8820651D0
(en)
*
|
1988-09-01 |
1988-10-05 |
Glaxo Group Ltd |
Medicaments
|
|
DE4009565A1
(de)
*
|
1990-03-24 |
1991-09-26 |
Merck Patent Gmbh |
Indolderivate
|
|
EP0492020A1
(fr)
*
|
1990-12-21 |
1992-07-01 |
Merrell Dow Pharmaceuticals Inc. |
Utilisation de certains esters de la hexahydro-8-hydroxy-2,6-méthano-2H-quinolizine-3(4H)-one et des composés apparentés pour le traitement des maladies cognitives
|
|
ZA92278B
(en)
*
|
1991-02-01 |
1992-10-28 |
Akzo Nv |
3-quinuclidine derivatives
|
|
AU654013B2
(en)
*
|
1991-03-13 |
1994-10-20 |
Regents Of The University Of Minnesota |
2-hydroxy-3(4-iodophenyl)-1-(4-phenylpiperidinyl) propane
|
|
IT1250629B
(it)
*
|
1991-07-04 |
1995-04-21 |
Boehringer Ingelheim Italia |
Uso dei derivati dell'acido benzimidazolin-2-oxo-1-carbossilico.
|
|
US5723103A
(en)
*
|
1994-12-09 |
1998-03-03 |
Vanderbilt University |
Substituted benzamides and radioligand analogs and methods of use
|
|
SE0000540D0
(sv)
|
2000-02-18 |
2000-02-18 |
Astrazeneca Ab |
New compounds
|
|
US6492385B2
(en)
|
2000-08-18 |
2002-12-10 |
Pharmacia & Upjohn Company |
Quinuclidine-substituted heteroaryl moieties for treatment of disease
|
|
US6479510B2
(en)
|
2000-08-18 |
2002-11-12 |
Pharmacia & Upjohn Company |
Quinuclidine-substituted aryl compounds for treatment of disease
|
|
WO2002016357A2
(fr)
|
2000-08-18 |
2002-02-28 |
Pharmacia & Upjohn Company |
Composes aryle substitues par quinuclidine destines au traitement de maladies
|
|
AU2001282875A1
(en)
|
2000-08-21 |
2002-03-04 |
Pharmacia And Upjohn Company |
Quinuclidine-substituted heteroaryl moieties for treatment of disease
|
|
US6599916B2
(en)
|
2000-08-21 |
2003-07-29 |
Pharmacia & Upjohn Company |
Quinuclidine-substituted heteroaryl moieties for treatment of disease
|
|
PE20021019A1
(es)
|
2001-04-19 |
2002-11-13 |
Upjohn Co |
Grupos azabiciclicos sustituidos
|
|
AR036041A1
(es)
*
|
2001-06-12 |
2004-08-04 |
Upjohn Co |
Compuestos aromaticos heterociclicos sustituidos con quinuclidina y composiciones farmaceuticas que los contienen
|
|
JP2005504059A
(ja)
*
|
2001-08-24 |
2005-02-10 |
ファルマシア アンド アップジョン カンパニー リミティド ライアビリティー カンパニー |
疾患を処置するための置換アリール7−アザ[2.2.1]ビシクロヘプタン
|
|
CA2458375A1
(fr)
|
2001-08-24 |
2003-03-06 |
Pharmacia & Upjohn Company |
Heteroaryl-7-aza¬2.2.1|bicycloheptanes substitues destines au traitement de maladies
|
|
DE60218493D1
(de)
*
|
2001-09-12 |
2007-04-12 |
Pharmacia & Upjohn Co Llc |
Substituierte 7-aza-ä2.2.1übicycloheptane für die behandlung von krankheiten
|
|
CA2462453C
(fr)
|
2001-10-02 |
2009-07-28 |
Pharmacia & Upjohn Company |
Composes d'heteoraryle fusionne substitues par azabicyclo utiles pour le traitement de maladies
|
|
JP2005510482A
(ja)
*
|
2001-10-16 |
2005-04-21 |
アストラゼネカ・アクチエボラーグ |
線維筋痛症候群の治療方法
|
|
US6849620B2
(en)
|
2001-10-26 |
2005-02-01 |
Pfizer Inc |
N-(azabicyclo moieties)-substituted hetero-bicyclic aromatic compounds for the treatment of disease
|
|
JP2005511574A
(ja)
*
|
2001-10-26 |
2005-04-28 |
ファルマシア アンド アップジョン カンパニー リミティド ライアビリティー カンパニー |
Nachrアゴニストとしてのn−アザビシクロ−置換ヘテロ二環式カルボキサミド
|
|
CA2466375A1
(fr)
*
|
2001-11-08 |
2003-05-15 |
Pharmacia & Upjohn Company |
Composes heteroaryles substitues azabicycliques pour le traitement de maladies
|
|
MXPA04004373A
(es)
|
2001-11-09 |
2004-08-11 |
Upjohn Co |
Compuestos heterociclicos condensados con fenilo azabiciclo para el tratamiento de enfermedades.
|
|
DE10162375A1
(de)
*
|
2001-12-19 |
2003-07-10 |
Bayer Ag |
Bicyclische N-Aryl-amide
|
|
DE10164139A1
(de)
*
|
2001-12-27 |
2003-07-10 |
Bayer Ag |
2-Heteroarylcarbonsäureamide
|
|
EP1480977A2
(fr)
*
|
2002-02-15 |
2004-12-01 |
PHARMACIA & UPJOHN COMPANY |
Composes aryle substitues permettant de traiter une maladie
|
|
CA2476624A1
(fr)
*
|
2002-02-19 |
2003-08-28 |
Pharmacia & Upjohn Company |
Composes azabicycliques servant a traiter des maladies
|
|
CA2476681A1
(fr)
*
|
2002-02-19 |
2003-08-28 |
Bruce N. Rogers |
Carboxamides hetero-aromatiques n-pontes bicycliques condenses destines au traitement de maladies
|
|
WO2003072578A1
(fr)
*
|
2002-02-20 |
2003-09-04 |
Pharmacia & Upjohn Company |
Composes azabicycliques presentant une activite de recepteurs d'alfa 7 nicotinique acetylcholine
|
|
DE10234424A1
(de)
|
2002-07-29 |
2004-02-12 |
Bayer Ag |
Benzothiophen-, Benzofuran- und Indolharnstoffe
|
|
US7176198B2
(en)
|
2002-08-01 |
2007-02-13 |
Pfizer Inc. |
1H-pyrazole and 1H-pyrrole-azabicyclic compounds for the treatment of disease
|
|
GB0220581D0
(en)
|
2002-09-04 |
2002-10-09 |
Novartis Ag |
Organic Compound
|
|
MXPA05003317A
(es)
*
|
2002-09-25 |
2005-07-05 |
Memory Pharm Corp |
Indazoles, benzotiazoles y benzoisotiazoles asi como preparacion y usos de los mismos.
|
|
WO2004039815A2
(fr)
*
|
2002-11-01 |
2004-05-13 |
Pharmacia & Upjohn Company Llc |
Composes possedant une activite d'agoniste du recepteur nicotinique $g(a)7 et d'antagoniste du recepteur 5ht3 pour traiter des maladies du systeme nerveux central
|
|
RU2389729C2
(ru)
*
|
2003-12-22 |
2010-05-20 |
Мемори Фармасьютиклз Корпорейшн |
1н-индазолы, 1, 2-бензизоксазолы и 1, 2-бензизотиазолы, их получение и применение
|
|
EP1735306A2
(fr)
|
2004-03-25 |
2006-12-27 |
Memory Pharmaceuticals Corporation |
Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, et leur preparation et leurs utilisations
|
|
CA2567977A1
(fr)
*
|
2004-04-22 |
2006-01-05 |
Memory Pharmaceutical Corporation |
Indoles, 1h-indazoles, 1,2-benzisoxazoles, 1,2-benzoisothiazoles, leur preparation et leurs utilisations
|
|
NZ551712A
(en)
*
|
2004-05-07 |
2010-07-30 |
Memory Pharm Corp |
1H-indazoles, benzothiazoles, 1,2-benzoisoxazoles, 1,2-benzoisothiazoles, and chromones and preparations and uses thereof
|
|
AR049401A1
(es)
|
2004-06-18 |
2006-07-26 |
Novartis Ag |
Aza-biciclononanos
|
|
GB0415746D0
(en)
|
2004-07-14 |
2004-08-18 |
Novartis Ag |
Organic compounds
|
|
CA2591817A1
(fr)
|
2004-12-22 |
2006-06-29 |
Memory Pharmaceuticals Corporation |
Ligands du recepteur alpha-7 nicotinique ainsi que preparation et utilisations de ceux-ci
|
|
US8106066B2
(en)
*
|
2005-09-23 |
2012-01-31 |
Memory Pharmaceuticals Corporation |
Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, pyrazolopyridines, isothiazolopyridines, and preparation and uses thereof
|
|
GB0521508D0
(en)
|
2005-10-21 |
2005-11-30 |
Novartis Ag |
Organic compounds
|
|
GB0525673D0
(en)
|
2005-12-16 |
2006-01-25 |
Novartis Ag |
Organic compounds
|
|
GB0525672D0
(en)
*
|
2005-12-16 |
2006-01-25 |
Novartis Ag |
Organic compounds
|
|
US20080242688A1
(en)
*
|
2007-03-19 |
2008-10-02 |
Astrazeneca Ab |
Method 741
|
|
EP2344636B1
(fr)
*
|
2008-10-09 |
2017-12-06 |
Howard Hughes Medical Institute |
Canaux ioniques chimériques inédits activés par la fixation d'un ligand et leurs procédés d'utilisation
|
|
LT2889033T
(lt)
|
2008-11-19 |
2018-07-10 |
Forum Pharmaceuticals Inc. |
Šizofrenijos negatyvių simptomų gydymas (r)-7-chlor-n-(chinuklidin-3-il)benzo[b]tiofen-2-karboksamidu ir jo farmaciniu požiūriu priimtinomis druskomis
|
|
JP5808319B2
(ja)
*
|
2009-05-11 |
2015-11-10 |
フォルム ファーマシューティカルズ、インコーポレイテッド |
アセチルコリンエステラーゼ阻害剤と組み合わせた特定のα7ニコチン酸受容体を用いた認知障害の治療
|
|
PE20170923A1
(es)
|
2010-05-17 |
2017-07-12 |
Forum Pharmaceuticals Inc |
Una forma cristalina de clorhidrato de (r)-7-cloro-n-(quinuclidin-3-il)benzo[b]tiofeno-2-carboxamida monohidratado
|
|
JP6263469B2
(ja)
|
2011-07-15 |
2018-01-17 |
ノバルティス アーゲー |
アザ二環式ジ−アリールエーテルの塩およびその製造方法またはその前駆体の製造方法
|
|
EP3461481A1
(fr)
|
2012-05-08 |
2019-04-03 |
Forum Pharmaceuticals Inc. |
Procédés de maintien, de traitement ou d'amélioration de la fonction cognitive
|
|
WO2017060287A1
(fr)
*
|
2015-10-05 |
2017-04-13 |
Sandoz Ag |
Procédé pour la préparation d'encenicline à partir de chlorure d'acide 7-chloro-benzo[b]thiophène-2-carboxylique et de (r)-quinuclidin-3-amine en présence d'imidazole
|