PH24886A - Pyridonecarboxylic acid derivatives - Google Patents

Pyridonecarboxylic acid derivatives

Info

Publication number: PH24886A
Authority: PH; Philippines
Prior art keywords: sup; sub; acid derivatives; pyridonecarboxylic acid; hydrogen
Prior art date: 1985-06-26

Application number

PH33956A

Other languages

English (en)

Inventor

Isao Nayakawa

Shohgo Atarashi

Original Assignee

Daiichi Seiyaku Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1985-06-26

Filing date

1986-06-26

Publication date

1990-12-26

1986-06-26 Application filed by Daiichi Seiyaku Co filed Critical Daiichi Seiyaku Co

1990-12-26 Publication of PH24886A publication Critical patent/PH24886A/en

Links

YSLIPUSJNFIFAB-UHFFFAOYSA-N 2-oxopyridine-1-carboxylic acid Chemical class OC(=O)N1C=CC=CC1=O YSLIPUSJNFIFAB-UHFFFAOYSA-N 0.000 title 1
UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 2
229910052739 hydrogen Inorganic materials 0.000 abstract 2
239000001257 hydrogen Substances 0.000 abstract 2
125000004777 2-fluoroethyl group Chemical group [H]C([H])(F)C([H])([H])* 0.000 abstract 1
125000006414 CCl Chemical group ClC* 0.000 abstract 1
239000002253 acid Substances 0.000 abstract 1
125000000217 alkyl group Chemical group 0.000 abstract 1
230000000845 anti-microbial effect Effects 0.000 abstract 1
125000001559 cyclopropyl group Chemical group [H]C1([H])C([H])([H])C1([H])* 0.000 abstract 1
125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 abstract 1
125000000555 isopropenyl group Chemical group [H]\C([H])=C(\*)C([H])([H])[H] 0.000 abstract 1
125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 abstract 1
125000000391 vinyl group Chemical group [H]C([*])=C([H])[H] 0.000 abstract 1
229920002554 vinyl polymer Polymers 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Communicable Diseases (AREA)
Public Health (AREA)
Oncology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Pyridine Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Pyrrole Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Table Devices Or Equipment (AREA)
Stringed Musical Instruments (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

PH33956A 1985-06-26 1986-06-26 Pyridonecarboxylic acid derivatives PH24886A (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
JP13983085		1985-06-26
JP27999185		1985-12-12

Publications (1)

Publication Number	Publication Date
PH24886A true PH24886A (en)	1990-12-26

Family

ID=26472527

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PH33956A PH24886A (en)	1985-06-26	1986-06-26	Pyridonecarboxylic acid derivatives

Country Status (18)

Country	Link
US (4)	US5098912A (ja)
EP (1)	EP0207420B1 (ja)
JP (2)	JPH0745491B2 (ja)
KR (1)	KR930005001B1 (ja)
AT (1)	ATE75740T1 (ja)
AU (1)	AU589978B2 (ja)
CA (1)	CA1301760C (ja)
DE (1)	DE3685157D1 (ja)
DK (1)	DK170641B1 (ja)
ES (1)	ES8707520A1 (ja)
FI (1)	FI87071C (ja)
GR (1)	GR861649B (ja)
IE (1)	IE59188B1 (ja)
IL (1)	IL79189A (ja)
NO (1)	NO167090C (ja)
PH (1)	PH24886A (ja)
PT (1)	PT82839B (ja)
YU (1)	YU46526B (ja)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE3508816A1 (de) *	1985-01-10	1986-07-10	Bayer Ag, 5090 Leverkusen	6,7-disubstituierte 1-cyclopropyl-1,4-dihydro-4-oxo-1,8-naphtyridin-3-carbonsaeuren
US4920120A (en) *	1988-01-25	1990-04-24	Warner-Lambert Company	Antibacterial agents
US5585491A (en) *	1988-01-25	1996-12-17	Otsuka Pharmaceutical Co., Ltd.	Antibacterial agents
CA1332605C (en) *	1988-10-03	1994-10-18	Yasuhiro Nishitani	Pyridonecarboxylic acids
ES2137942T3 (es) *	1990-11-30	2000-01-01	Warner Lambert Co	Estereoisomeros individuales de 7-(3-(aminoalquil)-1-pirrolidinil)-quinolonas y de naftiridonas utilizados como agentes antibacterianos.
US5364861A (en) *	1990-11-30	1994-11-15	Warner-Lambert Company	Optical isomers of 7-[3-(1,1-dialkylmethyl-1-amino-1-pyrrolidinyl]-quinolones and naphthyridones as antibacterial agents
US5157128A (en) *	1990-11-30	1992-10-20	Warner-Lambert Company	Certain optically active substituted α,α-dialkyl-pyrrolidine-3-methamines useful as intermediates
US5258528A (en) *	1990-11-30	1993-11-02	Warner-Lambert Company	Individual stereoisomers of pyrrolidine methanamines substituted on the ring nitrogen by a 1-phenylethyl group
EP0550016A1 (en) *	1991-12-31	1993-07-07	Korea Research Institute Of Chemical Technology	Novel quinolone carboxylic acid derivatives and processes for preparing same
DK0807630T3 (da) *	1995-02-02	2003-09-01	Daiichi Seiyaku Co	Heterocykliske forbindelser
DE69635812T2 (de) *	1995-11-22	2006-10-19	Daiichi Pharmaceutical Co., Ltd.	Substituierte aminocycloalkylpyrrolidinderivate
US6121285A (en)	1995-11-22	2000-09-19	Daiichi Pharmaceutical Co., Ltd.	Substituted aminocycloalkylpyrrolidine derivatives and cis-substituted aminocycloalkylpyrrolidine derivatives
DE69732635T2 (de)	1996-07-12	2005-12-29	Daiichi Pharmaceutical Co., Ltd.	Cis-substituierte aminocyclopropanderivate
KR20010012740A (ko) *	1997-05-21	2001-02-26	스즈키 다다시	시스-이치환된 아미노사이클로알킬 피롤리딘 유도체
ZA984527B (en) *	1997-05-30	1998-12-03	Daiichi Seiyaku Co	Substituted cyclobutylamine derivative
ES2321042T3 (es) *	1997-09-15	2009-06-01	THE PROCTER & GAMBLE COMPANY	Quinolonas antimicrobianas, composiciones y usos de las mismas.
US6387928B1 (en)	1997-09-15	2002-05-14	The Procter & Gamble Co.	Antimicrobial quinolones, their compositions and uses
PT1082300E (pt) *	1998-05-29	2004-02-27	Upjohn Co	Monometanossulfonato de 3-¬(1'-n-metilamino)etil-n-benzil\|pirrolidina
DE60011264T2 (de) *	1999-03-10	2005-07-14	Daiichi Pharmaceutical Co., Ltd.	Aminomethylpyrrolidin-derivate mit aromatischen substituenten
EP1250587A1 (en) *	2000-01-28	2002-10-23	Pion, Inc.	MEASUREMENT OF SOLUBILITY-pH PROFILES
EP1336611B1 (en) *	2000-11-20	2007-09-05	Daiichi Pharmaceutical Co., Ltd.	Dehalogeno compounds
SG144936A1 (en)	2003-09-10	2008-08-28	Kyorin Seiyaku Kk	7-(4-substituted-3-cyclopropylaminomethyl-1- pyrrolidinyl)quinolonecarboxylic acid derivative
JP4619952B2 (ja) *	2003-09-29	2011-01-26	第一三共株式会社	８−シアノキノロンカルボン酸誘導体
PL2001862T3 (pl) *	2006-03-28	2011-09-30	Warner Chilcott Co Llc	Jabłczany oraz odmiany polimorficzne kwasu (3S,5S)-7-[3-amino-5-metylo-piperydynylo]-1-cyklopropylo-1,4-dihydro-8-metoksy-4-okso-3-chinolinokarboksylowego
EP1999106B1 (en) *	2006-03-28	2012-06-27	TaiGen Biotechnology Co., Ltd.	A hydride reduction process for preparing quinolone intermediates
WO2007110835A2 (en) *	2006-03-28	2007-10-04	The Procter & Gamble Company	A coupling process for preparing quinolone intermediates
CA2688008A1 (en) *	2007-05-24	2008-11-27	Kyorin Pharmaceutical Co., Ltd.	Mutilin derivative having heterocyclic aromatic ring carboxylic acid structure in substituent at 14-position
CN116606280A (zh) *	2023-03-13	2023-08-18	广东工业大学	一种氟喹诺酮类化合物及其在制备抗菌药物中的应用

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IE55898B1 (en) *	1982-09-09	1991-02-14	Warner Lambert Co	Antibacterial agents
US4665079A (en) *	1984-02-17	1987-05-12	Warner-Lambert Company	Antibacterial agents
DE3318145A1 (de) *	1983-05-18	1984-11-22	Bayer Ag, 5090 Leverkusen	7-amino-1-cyclopropyl-6,8-difluor-1,4-dihydro-4-oxo-3-chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel
JPS60228479A (ja) *	1984-04-26	1985-11-13	Toyama Chem Co Ltd	１，４−ジヒドロ−４−オキソナフチリジン誘導体およびその塩
IE58742B1 (en) *	1984-07-20	1993-11-05	Warner Lambert Co	Substituted-9-fluoro-3-methyl-7-oxo-2,3-dihydro-7h-pyrido[1,2,3-de] [1,4]benzoxauine-6-carboxylic acids; sibstituted-5-amino-6-6fluoro-4-oxo.1,4-dihydroquinoline-3 carboxylic acids; substituted-5-amino-6-fluoro-1,4-dihydro-4-oxo-1.8-naphthyridine-3-carboxylic acids; derivatives thereof; pharmaceutical compositions comprising the compounds; and processes for producing the compounds
DE3509546A1 (de) *	1985-03-16	1986-09-25	Bayer Ag, 5090 Leverkusen	7-amino-1-(subst.cyclopropyl)-1,4-dihydro-4-oxo-3-chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel
US4657913A (en) *	1985-04-18	1987-04-14	Warner-Lambert Company	Trifluoro- quinoline -3- carboxylic acids and their use as anti-bacterial agents
EP0242789A3 (en) *	1986-04-25	1990-09-05	Dainippon Pharmaceutical Co., Ltd.	Novel quinoline derivates and processes for preparation thereof
US4851418A (en) *	1987-08-21	1989-07-25	Warner-Lambert Company	Naphthyridine antibacterial agents containing an α-amino acid in the side chain of the 7-substituent
US4920120A (en) *	1988-01-25	1990-04-24	Warner-Lambert Company	Antibacterial agents

1986
- 1986-06-23 EP EP86108547A patent/EP0207420B1/en not_active Expired - Lifetime
- 1986-06-23 AT AT86108547T patent/ATE75740T1/de not_active IP Right Cessation
- 1986-06-23 IL IL79189A patent/IL79189A/xx not_active IP Right Cessation
- 1986-06-23 DE DE8686108547T patent/DE3685157D1/de not_active Expired - Lifetime
- 1986-06-24 FI FI862688A patent/FI87071C/fi not_active IP Right Cessation
- 1986-06-25 ES ES556754A patent/ES8707520A1/es not_active Expired
- 1986-06-25 GR GR861649A patent/GR861649B/el unknown
- 1986-06-25 AU AU59245/86A patent/AU589978B2/en not_active Expired
- 1986-06-25 CA CA000512446A patent/CA1301760C/en not_active Expired - Lifetime
- 1986-06-25 NO NO862559A patent/NO167090C/no not_active IP Right Cessation
- 1986-06-25 IE IE169686A patent/IE59188B1/en not_active IP Right Cessation
- 1986-06-25 PT PT82839A patent/PT82839B/pt unknown
- 1986-06-26 DK DK304686A patent/DK170641B1/da not_active IP Right Cessation
- 1986-06-26 JP JP61150581A patent/JPH0745491B2/ja not_active Expired - Lifetime
- 1986-06-26 PH PH33956A patent/PH24886A/en unknown
- 1986-06-26 YU YU112086A patent/YU46526B/sh unknown
- 1986-06-26 KR KR1019860005150A patent/KR930005001B1/ko not_active Expired - Lifetime
1989
- 1989-12-12 US US07/449,160 patent/US5098912A/en not_active Expired - Lifetime
1991
- 1991-12-24 US US07/812,830 patent/US5416222A/en not_active Expired - Lifetime
1993
- 1993-06-21 JP JP5148887A patent/JP2686705B2/ja not_active Expired - Lifetime
1994
- 1994-03-04 US US08/205,638 patent/US5380874A/en not_active Expired - Lifetime
1995
- 1995-03-20 US US08/406,594 patent/US5476950A/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
IL79189A (en)	1990-07-12
ATE75740T1 (de)	1992-05-15
IE59188B1 (en)	1994-01-26
AU589978B2 (en)	1989-10-26
DK304686D0 (da)	1986-06-26
CA1301760C (en)	1992-05-26
JPS62234082A (ja)	1987-10-14
GR861649B (en)	1986-10-30
YU112086A (en)	1991-04-30
IL79189A0 (en)	1986-09-30
FI87071B (fi)	1992-08-14
EP0207420B1 (en)	1992-05-06
DE3685157D1 (de)	1992-06-11
KR930005001B1 (ko)	1993-06-11
ES556754A0 (es)	1987-08-01
US5416222A (en)	1995-05-16
AU5924586A (en)	1987-01-08
NO167090C (no)	1991-10-02
JPH0745491B2 (ja)	1995-05-17
YU46526B (sh)	1993-11-16
JPH09143157A (ja)	1997-06-03
FI87071C (fi)	1992-11-25
DK304686A (da)	1987-02-23
FI862688A0 (fi)	1986-06-24
NO862559D0 (no)	1986-06-25
NO862559L (no)	1986-12-29
US5380874A (en)	1995-01-10
IE861696L (en)	1986-12-26
ES8707520A1 (es)	1987-08-01
EP0207420A2 (en)	1987-01-07
DK170641B1 (da)	1995-11-20
US5476950A (en)	1995-12-19
JP2686705B2 (ja)	1997-12-08
PT82839A (en)	1986-07-01
FI862688L (fi)	1986-12-27
EP0207420A3 (en)	1988-04-20
US5098912A (en)	1992-03-24
PT82839B (pt)	1988-04-21
NO167090B (no)	1991-06-24
KR870000321A (ko)	1987-02-17

Publication	Publication Date	Title
AU589978B2 (en)	1989-10-26	Pyridonecarboxylic acid derivatives
EP0193317A3 (en)	1987-11-11	Silane-crosslinkable copolymer compositions
IL81002A0 (en)	1987-03-31	Pyrazoline derivatives,processes for their preparation and pesticidal compositions containing the same
DE3670647D1 (de)	1990-05-31	Schaeumbare organopolysiloxanzusammensetzungen.
IT8521213A0 (it)	1985-06-19	Composizioni covulcanizzabili di fluoroelastomeri a migliorata stabilita' chimica.
IT8521867A0 (it)	1985-08-05	Composizioni covulcanizzabili di fluoroelastomeri a migliorata stabilita' chimica.
EP0247177A4 (en)	1988-04-06	BENZODIAZINONE-PYRIDAZINONE AND HYDROXY-PYRAZOLYL COMPOUNDS, CARDIOTONIC COMPOSITIONS CONTAINING THEM, AND USES THEREOF.
IL79287A0 (en)	1986-09-30	Herbicidal compositions containing diflufenican
FI873554A0 (fi)	1987-08-17	Stabiloitu antimikrobinen vetyperoksidikoostumus
DE3672446D1 (en)	1990-08-09	Pantothenolderivate.
AU5003085A (en)	1986-05-22	Imidazo-pyrrolo(3,4-b) pyridines
PL261454A1 (en)	1988-03-03	Herbicide containing novel 2-aryl-4,5,6,7-tetrahydroisoindolinones
GB2177916B (en)	1989-07-26	Coametic compositions.
GB2182328B (en)	1989-09-20	Diphenyl ether derivatives
Clair-Tisdall	1980	The Sources of Islam
AU2167588A (en)	1989-03-02	Diphenyl ether herbicides
NZ181038A (en)	1978-07-28	Anticonvulsive or antiar-rhythmic compositions comprising 1-(2,6-dimethyl phenoxy)-2-methylamino-propane
IE842800L (en)	1985-05-01	1,4-dihydropyridine heterocyclics.
GB2184352B (en)	1990-05-09	Compositions containing fructose.
AU572332B2 (en)	1988-05-05	1,2,5 - oxadiazole-urea herbicidal compositions
IT8541560A0 (it)	1985-05-31	L'invio di messaggi fonici. apparecchiatura elettronica, per
UA19097A (uk)	1997-12-25	D-1-ФЕHІЛ-2-МЕТИЛАМІHОПРОПАHОЛА 1-5,6,7-ТРИОКСИФЛАВОH-7-0-beta-D-ГЛЮКУРОHИДАТ, ЩО МАЄ ОКИСЛЮВАЛЬHУ ДІЮ ТА РОЗШИРЮЄ СУДИHИ
GR871254B (en)	1987-08-14	Writing table for the office home next to the telephone etc.
IE871382L (en)	1987-11-28	Antiviral compositions.
CS57284A1 (en)	1984-10-15	Zpusob vyroby 4,4 bis (4,6 difenyl 5 kyan 2 pyridyl)bifenylu