PH27000A - Heteroaryl derivatives and pharmaceutical compositions containing them - Google Patents

Heteroaryl derivatives and pharmaceutical compositions containing them Download PDF

Info

Publication number
PH27000A
PH27000A PH36319A PH36319A PH27000A PH 27000 A PH27000 A PH 27000A PH 36319 A PH36319 A PH 36319A PH 36319 A PH36319 A PH 36319A PH 27000 A PH27000 A PH 27000A
Authority
PH
Philippines
Prior art keywords
phenyl
dihydro
oxo
propanamide
pyrazol
Prior art date
Application number
PH36319A
Other languages
English (en)
Inventor
Gianfederico Doria
Anna Maria Isetta
Mario Ferrari
Domenico Trizio
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB878700477A external-priority patent/GB8700477D0/en
Priority claimed from GB878717282A external-priority patent/GB8717282D0/en
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of PH27000A publication Critical patent/PH27000A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • C07D491/044—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
    • C07D491/052—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring the oxygen-containing ring being six-membered
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/04—Immunostimulants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Immunology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pyridine Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
PH36319A 1987-01-09 1988-01-04 Heteroaryl derivatives and pharmaceutical compositions containing them PH27000A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB878700477A GB8700477D0 (en) 1987-01-09 1987-01-09 Heteroaryl 2-cyano-3-oxo-propanamide derivatives
GB878717282A GB8717282D0 (en) 1987-07-22 1987-07-22 Heteroaryl 3-oxo-propanenitrile derivatives

Publications (1)

Publication Number Publication Date
PH27000A true PH27000A (en) 1993-02-01

Family

ID=26291768

Family Applications (1)

Application Number Title Priority Date Filing Date
PH36319A PH27000A (en) 1987-01-09 1988-01-04 Heteroaryl derivatives and pharmaceutical compositions containing them

Country Status (23)

Country Link
US (1) US4816467A (da)
EP (1) EP0274443B1 (da)
JP (1) JP2672312B2 (da)
KR (1) KR960002852B1 (da)
CN (1) CN1025500C (da)
AU (1) AU598893B2 (da)
CA (1) CA1310647C (da)
CZ (1) CZ277972B6 (da)
DE (1) DE3862937D1 (da)
DK (1) DK8088A (da)
ES (1) ES2029003T3 (da)
FI (1) FI89489C (da)
GR (1) GR3002032T3 (da)
HU (1) HU198722B (da)
IE (1) IE60620B1 (da)
IL (1) IL85004A (da)
MY (1) MY103348A (da)
NO (1) NO165841C (da)
NZ (1) NZ223113A (da)
PH (1) PH27000A (da)
PT (1) PT86516B (da)
SU (1) SU1695826A3 (da)
YU (2) YU46787B (da)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2061644T3 (es) * 1987-04-09 1994-12-16 Du Pont Indazoles sustituidos insecticidas.
GB8814586D0 (en) * 1988-06-20 1988-07-27 Erba Carlo Spa Tricyclic 3-oxo-propanenitrile derivatives & process for their preparation
GB8814587D0 (en) * 1988-06-20 1988-07-27 Erba Carlo Spa Condensed pyrazole 3-oxo-propanenitrile derivatives & process for their preparation
GB2227741B (en) * 1989-02-06 1992-08-05 Erba Carlo Spa Condensed 3-oxo-propanenitrile derivatives and process for their preparation
GB8907799D0 (en) * 1989-04-06 1989-05-17 Erba Carlo Spa Heteroaryl-3-oxo-propanenitrile derivatives useful in the treatment of rheumatoid arthritis and other autoimmune diseases
US5260328A (en) * 1989-04-06 1993-11-09 Farmitalia Carlo Erba Srl Phenyl-indenopurazol 3-oxo-propanamide derivatives useful in the treatment of rheumatoid arthritis
GB8916290D0 (en) * 1989-07-17 1989-08-31 Erba Carlo Spa Heteroaryl-3-oxo-propanenitrile derivatives useful in stimulating myelopoiesis
WO1991017748A1 (de) * 1990-05-18 1991-11-28 Hoechst Aktiengesellschaft Isoxazol-4-carbonsäureamide und hydroxyalkyliden-cyanessigsäureamide, diese verbindungen enthaltende arzneimittel und deren verwendung
US5547975A (en) * 1994-09-20 1996-08-20 Talley; John J. Benzopyranopyrazolyl derivatives for the treatment of inflammation
US5886016A (en) * 1995-09-15 1999-03-23 G.D. Searle & Co. Benzopyranopyrazolyl derivatives for the treatment of inflammation
UA48989C2 (uk) * 1995-11-06 2002-09-16 Орто-Макнейл Фармасьютікел, Інк. Похідні 1-арилсульфоніл, арил(тіо)карбонілпіридазину, спосіб їх одержання, фармацевтична композиція та спосіб лікування
GB9720899D0 (en) * 1997-10-01 1997-12-03 Pharmacia & Upjohn Spa Condensed heterocyclic compounds
ES2637801T3 (es) * 2000-04-11 2017-10-17 Genentech, Inc. Anticuerpos multivalentes y usos de los mismos
ES2286275T3 (es) * 2001-09-19 2007-12-01 Pharmacia Corporation Compuestos de pirazolo sustituidos para el tratamiento de la inflamacion.
EP1651276A4 (en) * 2003-08-08 2009-05-06 Barnes Jewish Hospital EMULSION PARTICLES FOR IMAGING AND THERAPY AND USE METHOD THEREFOR
US20060035242A1 (en) 2004-08-13 2006-02-16 Michelitsch Melissa D Prion-specific peptide reagents
CA2650574A1 (en) * 2006-04-27 2007-11-08 Barnes-Jewish Hospital Detection and imaging of target tissue
MX2012005518A (es) 2009-11-13 2012-06-19 Merck Serono Sa Derivados de pirazol amina triciclica.
CN102086212B (zh) * 2009-12-03 2013-06-12 沈阳药科大学 抗真菌剂-2，3，4，5-四氢-4H-苯并[b]噻喃并[4，3-c]吡唑-2-甲酰胺衍生物
WO2018075564A1 (en) 2016-10-17 2018-04-26 University Of Maryland, College Park Multispecific antibodies targeting human immunodeficiency virus and methods of using the same

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4268516A (en) * 1978-10-11 1981-05-19 Pfizer Inc. [1]Benzothiopyrano[4,3-c]pyrazoles as immunoregulatory agents
EP0022446A1 (de) * 1979-04-06 1981-01-21 F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft Verfahren zur Herstellung von Biotinestern und von Biotin
EP0057932A1 (en) * 1981-02-11 1982-08-18 E.I. Du Pont De Nemours And Company Antiinflammatory and/or analgesic 3,4-dihydro(or 1,4-dihydro)-2-((substituted)thiol)-(1)-benzopyrano(3,4-d)imidazoles and their corresponding sulfoxides and sulfones
PH21213A (en) * 1984-10-26 1987-08-21 Fujisawa Pharmaceutical Co Benzene- and pyrazole- fused heterocyclic compound and pharmaceutical composition comprising the same

Also Published As

Publication number Publication date
KR960002852B1 (ko) 1996-02-27
PT86516B (pt) 1991-12-31
DK8088A (da) 1988-07-10
ES2029003T3 (es) 1992-07-16
CZ277972B6 (en) 1993-07-14
YU1088A (en) 1989-08-31
DK8088D0 (da) 1988-01-08
MY103348A (en) 1993-06-30
AU1003788A (en) 1988-07-14
CZ17988A3 (en) 1993-02-17
EP0274443B1 (en) 1991-05-29
IE60620B1 (en) 1994-07-27
CN1025500C (zh) 1994-07-20
JPS63174988A (ja) 1988-07-19
KR880008987A (ko) 1988-09-13
HUT47113A (en) 1989-01-30
AU598893B2 (en) 1990-07-05
CA1310647C (en) 1992-11-24
GR3002032T3 (en) 1992-12-30
NO880068L (no) 1988-07-11
FI89489B (fi) 1993-06-30
IE880002L (en) 1988-07-09
IL85004A (en) 1991-11-21
FI880078A0 (fi) 1988-01-08
FI880078A7 (fi) 1988-07-10
NO880068D0 (no) 1988-01-08
NO165841B (no) 1991-01-07
JP2672312B2 (ja) 1997-11-05
NO165841C (no) 1991-04-17
FI89489C (fi) 1993-10-11
YU46787B (sh) 1994-06-10
IL85004A0 (en) 1988-06-30
HU198722B (en) 1989-11-28
DE3862937D1 (de) 1991-07-04
PT86516A (en) 1988-02-01
EP0274443A1 (en) 1988-07-13
SU1695826A3 (ru) 1991-11-30
US4816467A (en) 1989-03-28
CN88100153A (zh) 1988-07-27
NZ223113A (en) 1989-07-27
YU79489A (en) 1989-10-31

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