PL197005A1 - Sposob wytwarzania nowych pochodnych prostaglandyn - Google Patents
Sposob wytwarzania nowych pochodnych prostaglandynInfo
- Publication number
- PL197005A1 PL197005A1 PL19700577A PL19700577A PL197005A1 PL 197005 A1 PL197005 A1 PL 197005A1 PL 19700577 A PL19700577 A PL 19700577A PL 19700577 A PL19700577 A PL 19700577A PL 197005 A1 PL197005 A1 PL 197005A1
- Authority
- PL
- Poland
- Prior art keywords
- making new
- prostaglandin derivatives
- new prostaglandin
- derivatives
- making
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/24—Oxygen or sulfur atoms
- C07D207/26—2-Pyrrolidones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C53/00—Saturated compounds having only one carboxyl group bound to an acyclic carbon atom or hydrogen
- C07C53/126—Acids containing more than four carbon atoms
- C07C53/128—Acids containing more than four carbon atoms the carboxylic group being bound to a carbon atom bound to at least two other carbon atoms, e.g. neo-acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
- C07F9/40—Esters thereof
- C07F9/4003—Esters thereof the acid moiety containing a substituent or a structure which is considered as characteristic
- C07F9/4006—Esters of acyclic acids which can have further substituents on alkyl
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyrrole Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IL49325A IL49325A (en) | 1976-03-31 | 1976-03-31 | 8-aza-11-deoxy-pge1 derivatives,their preparation and pharmaceutical compositions containing them |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PL197005A1 true PL197005A1 (pl) | 1978-10-09 |
| PL107643B1 PL107643B1 (pl) | 1980-02-29 |
Family
ID=11048789
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL1977197005A PL107643B1 (pl) | 1976-03-31 | 1977-03-29 | Sposob wytwarzania nowych pochodnych prostaglandyn |
| PL1977210101A PL107544B1 (pl) | 1976-03-31 | 1977-03-29 | Sposob wytwarzania nowych pochodnych prostaglandyn |
| PL1977210102A PL108289B1 (pl) | 1976-03-31 | 1977-03-29 | Sposob wytwarzania nowych pochodnych prostaglandynmethod of producing new derivatives of prostaglandins |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL1977210101A PL107544B1 (pl) | 1976-03-31 | 1977-03-29 | Sposob wytwarzania nowych pochodnych prostaglandyn |
| PL1977210102A PL108289B1 (pl) | 1976-03-31 | 1977-03-29 | Sposob wytwarzania nowych pochodnych prostaglandynmethod of producing new derivatives of prostaglandins |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US4115401A (pl) |
| JP (1) | JPS52142060A (pl) |
| BE (1) | BE852941A (pl) |
| CA (1) | CA1074804A (pl) |
| CH (2) | CH624101A5 (pl) |
| DD (1) | DD130352A5 (pl) |
| DE (1) | DE2714129A1 (pl) |
| ES (1) | ES457385A1 (pl) |
| FR (1) | FR2346332A1 (pl) |
| GB (1) | GB1574246A (pl) |
| HU (1) | HU178040B (pl) |
| IL (1) | IL49325A (pl) |
| IT (1) | IT1075373B (pl) |
| NL (1) | NL7703503A (pl) |
| NO (1) | NO149428C (pl) |
| PL (3) | PL107643B1 (pl) |
| SE (1) | SE417603B (pl) |
| SU (3) | SU676162A3 (pl) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE7906017L (sv) * | 1978-07-11 | 1980-02-13 | Glaxo Group Ltd | Prostanoida foreningar |
| US4320136A (en) * | 1980-08-11 | 1982-03-16 | E. I. Du Pont De Nemours And Company | 8-Aza-16,16-difluoroprostanoids |
| US4456613A (en) * | 1982-12-27 | 1984-06-26 | E. I. Du Pont De Nemours And Company | 6-Keto- and 6-hydroxy-8-azaprostanoids and anti-ulcer use thereof |
| US4530933A (en) * | 1982-12-27 | 1985-07-23 | E. I. Du Pont De Nemours And Company | 8-Aza-13-thiaprostanoids and a method of use thereof as anti-ulcer agents |
| EA005293B1 (ru) | 1999-12-22 | 2004-12-30 | Пфайзер Продактс Инк. | Производные пирролидин-2-она и их применение при лечении остеопороза |
| EA200300379A1 (ru) * | 2000-11-27 | 2003-08-28 | Пфайзер Продактс Инк. | Селективные агонисты рецептора ep4 в лечении остеопороза |
| RU2288913C2 (ru) | 2001-07-16 | 2006-12-10 | Ф.Хоффманн-Ля Рош Аг | Аналоги простагландинов, способ их получения и фармацевтическая композиция, обладающая селективной агонистической активностью в отношении рецептора ep4 |
| RU2296122C2 (ru) * | 2001-07-16 | 2007-03-27 | Ф.Хоффманн-Ля Рош Аг | Производные 2-пирролидона в качестве простаноидных агонистов и фармацевтическая композиция |
| IL159996A0 (en) | 2001-07-23 | 2004-06-20 | Ono Pharmaceutical Co | Remedies for diseases with bone mass loss having ep4 agonist as the active ingredient |
| JP4547912B2 (ja) | 2002-03-05 | 2010-09-22 | 小野薬品工業株式会社 | 8−アザプロスタグランジン誘導体化合物およびその化合物を有効成分として含有する薬剤 |
| CA2479222A1 (en) * | 2002-03-18 | 2003-09-25 | Pfizer Products Inc. | Use of selective ep4 receptor agonists for the treatment of liver failure, loss of patency of the ductus arteriosus, glaucoma or ocular hypertension |
| CN1735597A (zh) * | 2003-01-10 | 2006-02-15 | 霍夫曼-拉罗奇有限公司 | 作为前列腺素激动剂的2-哌啶酮衍生物 |
| US7179820B2 (en) | 2003-06-06 | 2007-02-20 | Allergan, Inc. | Piperidinyl prostaglandin E analogs |
| US20080058375A1 (en) * | 2004-01-08 | 2008-03-06 | Elworthy Todd R | 2-Piperidone derivatives as prostaglandin antagonists |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3975399A (en) * | 1974-08-06 | 1976-08-17 | E. I. Du Pont De Nemours And Company | 1,5-Disubstituted-2-pyrrolidinones, -3-pyrrolin-2-ones, and -4-pyrrolin-2-ones |
-
1976
- 1976-03-31 IL IL49325A patent/IL49325A/xx unknown
-
1977
- 1977-03-28 BE BE176164A patent/BE852941A/xx not_active IP Right Cessation
- 1977-03-28 GB GB12991/77A patent/GB1574246A/en not_active Expired
- 1977-03-29 PL PL1977197005A patent/PL107643B1/pl unknown
- 1977-03-29 DD DD7700198124A patent/DD130352A5/xx unknown
- 1977-03-29 PL PL1977210101A patent/PL107544B1/pl unknown
- 1977-03-29 PL PL1977210102A patent/PL108289B1/pl unknown
- 1977-03-30 DE DE19772714129 patent/DE2714129A1/de not_active Withdrawn
- 1977-03-30 CA CA275,134A patent/CA1074804A/en not_active Expired
- 1977-03-30 SE SE7703698A patent/SE417603B/xx unknown
- 1977-03-30 HU HU77LA913A patent/HU178040B/hu unknown
- 1977-03-30 CH CH400377A patent/CH624101A5/fr not_active IP Right Cessation
- 1977-03-30 NO NO771134A patent/NO149428C/no unknown
- 1977-03-31 IT IT21906/77A patent/IT1075373B/it active
- 1977-03-31 FR FR7709650A patent/FR2346332A1/fr active Granted
- 1977-03-31 JP JP3742877A patent/JPS52142060A/ja active Pending
- 1977-03-31 ES ES457385A patent/ES457385A1/es not_active Expired
- 1977-03-31 SU SU772465855A patent/SU676162A3/ru active
- 1977-03-31 NL NL7703503A patent/NL7703503A/xx not_active Application Discontinuation
- 1977-03-31 US US05/783,284 patent/US4115401A/en not_active Expired - Lifetime
-
1978
- 1978-03-30 SU SU782594353A patent/SU837321A3/ru active
- 1978-03-30 SU SU782595450A patent/SU715019A3/ru active
-
1980
- 1980-09-17 CH CH697780A patent/CH628032A5/fr not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| SU676162A3 (ru) | 1979-07-25 |
| IL49325A0 (en) | 1976-05-31 |
| DE2714129A1 (de) | 1977-10-13 |
| NO149428B (no) | 1984-01-09 |
| SU837321A3 (ru) | 1981-06-07 |
| SE417603B (sv) | 1981-03-30 |
| CA1074804A (en) | 1980-04-01 |
| IL49325A (en) | 1979-11-30 |
| NO771134L (no) | 1977-10-03 |
| PL108289B1 (pl) | 1980-03-31 |
| PL107544B1 (pl) | 1980-02-29 |
| NL7703503A (nl) | 1977-10-04 |
| IT1075373B (it) | 1985-04-22 |
| CH628032A5 (fr) | 1982-02-15 |
| CH624101A5 (pl) | 1981-07-15 |
| BE852941A (fr) | 1977-09-28 |
| HU178040B (en) | 1982-02-28 |
| NO149428C (no) | 1984-04-18 |
| JPS52142060A (en) | 1977-11-26 |
| SE7703698L (sv) | 1977-10-01 |
| ES457385A1 (es) | 1978-02-01 |
| US4115401A (en) | 1978-09-19 |
| FR2346332A1 (fr) | 1977-10-28 |
| DD130352A5 (de) | 1978-03-22 |
| SU715019A3 (ru) | 1980-02-05 |
| GB1574246A (en) | 1980-09-03 |
| FR2346332B1 (pl) | 1980-05-09 |
| PL107643B1 (pl) | 1980-02-29 |
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