PL2253619T3 - Sól aminowa pochodnej karbostyrylowej - Google Patents

Sól aminowa pochodnej karbostyrylowej

Info

Publication number: PL2253619T3
Authority: PL; Poland
Prior art keywords: amine salt; carbostyril derivative; carbostyril; derivative; amine
Prior art date: 2004-01-21

Application number

PL10174397T

Other languages

English (en)

Inventor

Yoshihiro Nishioka

Shinji Aki

Shigekazu Fujita

Yoshinao Onishi

Shun-Ichiro Sumida

Original Assignee

Otsuka Pharma Co Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2004-01-21

Filing date

2005-01-20

Publication date

2012-08-31

2005-01-20 Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd

2012-08-31 Publication of PL2253619T3 publication Critical patent/PL2253619T3/pl

Links

-1 Amine salt Chemical class 0.000 title 1
LISFMEBWQUVKPJ-UHFFFAOYSA-N quinolin-2-ol Chemical class C1=CC=C2NC(=O)C=CC2=C1 LISFMEBWQUVKPJ-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
- C07D215/22—Oxygen atoms attached in position 2 or 4
- C07D215/227—Oxygen atoms attached in position 2 or 4 only one oxygen atom which is attached in position 2
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/08—Solutions
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P39/00—General protective or antinoxious agents
- A61P39/06—Free radical scavengers or antioxidants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Diabetes (AREA)
Immunology (AREA)
Epidemiology (AREA)
Biochemistry (AREA)
Emergency Medicine (AREA)
Endocrinology (AREA)
Hematology (AREA)
Obesity (AREA)
Ophthalmology & Optometry (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Dermatology (AREA)
Urology & Nephrology (AREA)
Gastroenterology & Hepatology (AREA)
Pulmonology (AREA)
Toxicology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)
Quinoline Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

PL10174397T 2004-01-21 2005-01-20 Sól aminowa pochodnej karbostyrylowej PL2253619T3 (pl)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
JP2004013402		2004-01-21
EP05704144.4A EP1706383B1 (en)	2004-01-21	2005-01-20	Amine salt of carbostyril derivative useful for the treatment of, inter alia, gastric ulcer
EP10174397A EP2253619B1 (en)	2004-01-21	2005-01-20	Amine salt of carbostyril derivative

Publications (1)

Publication Number	Publication Date
PL2253619T3 true PL2253619T3 (pl)	2012-08-31

Family

ID=34805383

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
PL05704144T PL1706383T3 (pl)	2004-01-21	2005-01-20	Sól aminowa pochodnej karbostyrylowej użyteczna do leczenia między innymi wrzodu żołądka
PL10174397T PL2253619T3 (pl)	2004-01-21	2005-01-20	Sól aminowa pochodnej karbostyrylowej

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
PL05704144T PL1706383T3 (pl)	2004-01-21	2005-01-20	Sól aminowa pochodnej karbostyrylowej użyteczna do leczenia między innymi wrzodu żołądka

Country Status (22)

Country	Link
US (2)	US7732611B2 (pl)
EP (2)	EP1706383B1 (pl)
JP (1)	JP4516962B2 (pl)
KR (1)	KR100844762B1 (pl)
CN (1)	CN1934086B (pl)
AR (1)	AR047438A1 (pl)
AT (1)	ATE549318T1 (pl)
AU (1)	AU2005206430B2 (pl)
BR (1)	BRPI0506982A (pl)
CA (1)	CA2553231C (pl)
CY (2)	CY1112723T1 (pl)
DK (2)	DK1706383T3 (pl)
ES (2)	ES2382133T3 (pl)
HU (1)	HUE027990T2 (pl)
MY (1)	MY148416A (pl)
PL (2)	PL1706383T3 (pl)
PT (2)	PT1706383E (pl)
RU (1)	RU2372336C2 (pl)
SG (1)	SG149854A1 (pl)
SI (2)	SI2253619T1 (pl)
TW (1)	TWI340650B (pl)
WO (1)	WO2005070892A1 (pl)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US6187197B1 (en) *	1998-10-28	2001-02-13	Marvin Haddock	Multi-stage engine coolant recycling process
TWI340650B (en) *	2004-01-21	2011-04-21	Otsuka Pharma Co Ltd	Amine saly of carbostyril derivative
WO2009022674A1 (en) *	2007-08-10	2009-02-19	Otsuka Pharmaceutical Co., Ltd.	Medical composition containing rebamipide
WO2009126695A2 (en) *	2008-04-08	2009-10-15	Dynamis Therapeutics, Inc.	Method for treating or preventing dry eye disorders using alkylamino-polyhydroxyalkanes
US20110124682A1 (en) *	2008-06-19	2011-05-26	Sumida Shun-Ichiro	Pharmaceutical composition comprising rebamipide
CN103476753B (zh) *	2011-02-25	2015-12-09	诺弗米克斯有限公司	新的瑞巴派特复合物和共晶体

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS517614Y2 (pl) *	1971-02-12	1976-03-01
FI80022C (fi) *	1982-07-05	1990-04-10	Otsuka Pharma Co Ltd	Foerfarande foer framstaellning av ett nytt, terapeutiskt anvaendbart karbostyrilderivat.
JPS597168A (ja)	1982-07-05	1984-01-14	Otsuka Pharmaceut Co Ltd	カルボスチリル誘導体
DE69207560T2 (de) *	1991-06-07	1996-06-27	Otsuka Pharma Co Ltd	Antidiabetikum
TW227558B (pl) *	1992-05-14	1994-08-01	Otsuka Pharma Co Ltd
US5415872A (en) *	1992-06-22	1995-05-16	Digestive Care Inc.	Compositions of gastric acid-resistant microspheres containing salts of bile acids
JP2872546B2 (ja) *	1992-11-26	1999-03-17	大塚製薬株式会社	腸粘膜障害保護剤
CA2150546C (en) *	1993-10-21	2004-11-09	Takahide Matsuda	Agent for inhibiting production of interleukin-8
AU8003194A (en)	1993-11-05	1995-05-23	Otsuka Pharmaceutical Co., Ltd.	Bismuth salt of carbostyril derivatives for the treatment of peptic ulcers
JP3621463B2 (ja) *	1995-04-26	2005-02-16	大塚製薬株式会社	カルボスチリル誘導体ビスマス塩
AR004214A1 (es)	1995-10-12	1998-11-04	Otsuka Pharma Co Ltd	Una preparación de gotas oftálmicas para la cura de enfermedades oftálmicas
GB9613455D0 (en) *	1996-06-27	1996-08-28	Aston Molecules Ltd	Analogues or derivatives of quercetin
JP2005519949A (ja) *	2002-03-11	2005-07-07	ノバルティスアクチエンゲゼルシャフト	ナテグリニドの塩
KR20040104020A (ko)	2003-06-02	2004-12-10	진양제약주식회사	신규 레바미피드 리지네이트와 레바미피드 아르기니네이트및 이 신규 레바미피드 리지네이트와 레바미피드아르기니네이트를 유효성분으로 함유하는 약학적 제제
TWI340650B (en) *	2004-01-21	2011-04-21	Otsuka Pharma Co Ltd	Amine saly of carbostyril derivative
JP4719917B2 (ja)	2007-03-30	2011-07-06	国立大学法人岡山大学	アズキ加工食品のアズキ原料品種判定方法

2005
- 2005-01-18 TW TW094101386A patent/TWI340650B/zh not_active IP Right Cessation
- 2005-01-19 MY MYPI20050200A patent/MY148416A/en unknown
- 2005-01-20 ES ES10174397T patent/ES2382133T3/es not_active Expired - Lifetime
- 2005-01-20 JP JP2006520510A patent/JP4516962B2/ja not_active Expired - Lifetime
- 2005-01-20 BR BRPI0506982-3A patent/BRPI0506982A/pt not_active IP Right Cessation
- 2005-01-20 ES ES05704144.4T patent/ES2544327T3/es not_active Expired - Lifetime
- 2005-01-20 HU HUE05704144A patent/HUE027990T2/en unknown
- 2005-01-20 PT PT57041444T patent/PT1706383E/pt unknown
- 2005-01-20 AU AU2005206430A patent/AU2005206430B2/en not_active Ceased
- 2005-01-20 RU RU2006129945/04A patent/RU2372336C2/ru not_active IP Right Cessation
- 2005-01-20 WO PCT/JP2005/001034 patent/WO2005070892A1/en not_active Ceased
- 2005-01-20 SI SI200531494T patent/SI2253619T1/sl unknown
- 2005-01-20 AT AT10174397T patent/ATE549318T1/de active
- 2005-01-20 PL PL05704144T patent/PL1706383T3/pl unknown
- 2005-01-20 EP EP05704144.4A patent/EP1706383B1/en not_active Expired - Lifetime
- 2005-01-20 KR KR1020067016600A patent/KR100844762B1/ko not_active Expired - Fee Related
- 2005-01-20 DK DK05704144.4T patent/DK1706383T3/en active
- 2005-01-20 US US10/586,453 patent/US7732611B2/en not_active Expired - Fee Related
- 2005-01-20 CA CA2553231A patent/CA2553231C/en not_active Expired - Fee Related
- 2005-01-20 PL PL10174397T patent/PL2253619T3/pl unknown
- 2005-01-20 DK DK10174397.9T patent/DK2253619T3/da active
- 2005-01-20 EP EP10174397A patent/EP2253619B1/en not_active Expired - Lifetime
- 2005-01-20 SG SG200900369-0A patent/SG149854A1/en unknown
- 2005-01-20 PT PT10174397T patent/PT2253619E/pt unknown
- 2005-01-20 SI SI200531992T patent/SI1706383T1/sl unknown
- 2005-01-20 AR ARP050100199A patent/AR047438A1/es not_active Application Discontinuation
- 2005-01-20 CN CN2005800086478A patent/CN1934086B/zh not_active Expired - Fee Related
2010
- 2010-04-26 US US12/662,610 patent/US8222276B2/en not_active Expired - Fee Related
2012
- 2012-05-11 CY CY20121100442T patent/CY1112723T1/el unknown
2015
- 2015-10-06 CY CY20151100891T patent/CY1116773T1/el unknown

Also Published As

Publication number	Publication date
SI1706383T1 (sl)	2015-09-30
US7732611B2 (en)	2010-06-08
WO2005070892A1 (en)	2005-08-04
MY148416A (en)	2013-04-30
KR20060123566A (ko)	2006-12-01
EP1706383A1 (en)	2006-10-04
DK1706383T3 (en)	2015-08-03
CA2553231C (en)	2012-03-13
CA2553231A1 (en)	2005-08-04
ES2544327T3 (es)	2015-08-28
US20100210684A1 (en)	2010-08-19
AR047438A1 (es)	2006-01-18
CY1112723T1 (el)	2016-02-10
US20070155787A1 (en)	2007-07-05
DK2253619T3 (da)	2012-04-16
PT2253619E (pt)	2012-03-29
SI2253619T1 (sl)	2012-04-30
AU2005206430B2 (en)	2008-12-11
RU2006129945A (ru)	2008-02-27
ATE549318T1 (de)	2012-03-15
TW200529873A (en)	2005-09-16
PT1706383E (pt)	2015-10-15
ES2382133T3 (es)	2012-06-05
AU2005206430A1 (en)	2005-08-04
CN1934086B (zh)	2013-01-02
RU2372336C2 (ru)	2009-11-10
EP1706383B1 (en)	2015-07-22
KR100844762B1 (ko)	2008-07-07
CY1116773T1 (el)	2017-03-15
EP2253619A1 (en)	2010-11-24
HUE027990T2 (en)	2016-11-28
BRPI0506982A (pt)	2007-07-03
US8222276B2 (en)	2012-07-17
SG149854A1 (en)	2009-02-27
PL1706383T3 (pl)	2015-12-31
HK1148527A1 (en)	2011-09-09
JP2007514641A (ja)	2007-06-07
HK1101327A1 (en)	2007-10-12
JP4516962B2 (ja)	2010-08-04
TWI340650B (en)	2011-04-21
EP2253619B1 (en)	2012-03-14
CN1934086A (zh)	2007-03-21

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