PL2632927T3 - Boroniany jako inhibitory arginazy - Google Patents

Boroniany jako inhibitory arginazy

Info

Publication number
PL2632927T3
PL2632927T3 PL11779904.9T PL11779904T PL2632927T3 PL 2632927 T3 PL2632927 T3 PL 2632927T3 PL 11779904 T PL11779904 T PL 11779904T PL 2632927 T3 PL2632927 T3 PL 2632927T3
Authority
PL
Poland
Prior art keywords
boronates
arginase inhibitors
arginase
inhibitors
Prior art date
Application number
PL11779904.9T
Other languages
English (en)
Inventor
Zandt Michael Van
Jr. Gunnar Erik Jagdmann
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of PL2632927T3 publication Critical patent/PL2632927T3/pl

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/69—Boron compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/08—Plasma substitutes; Perfusion solutions; Dialytics or haemodialytics; Drugs for electrolytic or acid-base disorders, e.g. hypovolemic shock
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Pulmonology (AREA)
  • Cardiology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Hospice & Palliative Care (AREA)
  • Vascular Medicine (AREA)
  • Psychiatry (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
PL11779904.9T 2010-10-26 2011-10-19 Boroniany jako inhibitory arginazy PL2632927T3 (pl)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US40676010P 2010-10-26 2010-10-26

Publications (1)

Publication Number Publication Date
PL2632927T3 true PL2632927T3 (pl) 2016-09-30

Family

ID=44913403

Family Applications (1)

Application Number Title Priority Date Filing Date
PL11779904.9T PL2632927T3 (pl) 2010-10-26 2011-10-19 Boroniany jako inhibitory arginazy

Country Status (19)

Country Link
US (5) US9233985B2 (pl)
EP (3) EP2632927B1 (pl)
JP (1) JP5909239B2 (pl)
CN (2) CN106008569B9 (pl)
AU (1) AU2011320732B2 (pl)
BR (1) BR112013010099B1 (pl)
CA (1) CA2815536C (pl)
DK (1) DK2632927T3 (pl)
ES (2) ES2568680T3 (pl)
HK (1) HK1223104A1 (pl)
HR (1) HRP20160305T1 (pl)
HU (1) HUE027317T2 (pl)
IL (1) IL225926A (pl)
MX (1) MX336381B (pl)
PL (1) PL2632927T3 (pl)
RS (1) RS54750B1 (pl)
SI (1) SI2632927T1 (pl)
SM (1) SMT201600141B (pl)
WO (1) WO2012058065A1 (pl)

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Publication number Publication date
CA2815536A1 (en) 2012-05-03
DK2632927T3 (en) 2016-04-11
US20190054101A1 (en) 2019-02-21
CN106008569B (zh) 2020-04-03
BR112013010099A2 (pt) 2016-09-06
EP3034509A1 (en) 2016-06-22
HRP20160305T1 (hr) 2016-07-01
EP3034509B1 (en) 2020-04-22
US20150191492A1 (en) 2015-07-09
CN103249737B (zh) 2016-06-08
US10603330B2 (en) 2020-03-31
CN103249737A (zh) 2013-08-14
AU2011320732B2 (en) 2018-07-05
ES2794006T3 (es) 2020-11-17
IL225926A (en) 2016-09-29
JP2013542223A (ja) 2013-11-21
CN106008569B9 (zh) 2020-05-22
MX336381B (es) 2016-01-18
US20170000808A1 (en) 2017-01-05
WO2012058065A1 (en) 2012-05-03
EP2632927B1 (en) 2016-02-10
SI2632927T1 (sl) 2016-08-31
HK1223104A1 (en) 2017-07-21
IL225926A0 (en) 2013-06-27
CN106008569A (zh) 2016-10-12
CA2815536C (en) 2019-10-01
JP5909239B2 (ja) 2016-04-26
US9233985B2 (en) 2016-01-12
EP3719024A1 (en) 2020-10-07
BR112013010099B1 (pt) 2021-08-10
US9440995B2 (en) 2016-09-13
MX2013004491A (es) 2013-11-04
HUE027317T2 (en) 2016-10-28
US10098902B2 (en) 2018-10-16
US11389464B2 (en) 2022-07-19
EP2632927A1 (en) 2013-09-04
SMT201600141B (it) 2016-07-01
RS54750B1 (sr) 2016-10-31
US20120129806A1 (en) 2012-05-24
ES2568680T3 (es) 2016-05-03
AU2011320732A1 (en) 2013-11-21
HK1225390A1 (zh) 2017-09-08
US20200246362A1 (en) 2020-08-06

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