PL357713A1 - Inhibitory kaspaz i ich zastosowania - Google Patents
Inhibitory kaspaz i ich zastosowaniaInfo
- Publication number
- PL357713A1 PL357713A1 PL01357713A PL35771301A PL357713A1 PL 357713 A1 PL357713 A1 PL 357713A1 PL 01357713 A PL01357713 A PL 01357713A PL 35771301 A PL35771301 A PL 35771301A PL 357713 A1 PL357713 A1 PL 357713A1
- Authority
- PL
- Poland
- Prior art keywords
- caspase inhibitors
- caspase
- inhibitors
- Prior art date
Links
- 102000011727 Caspases Human genes 0.000 title 1
- 108010076667 Caspases Proteins 0.000 title 1
- 239000003112 inhibitor Substances 0.000 title 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
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- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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- C07D213/28—Radicals substituted by singly-bound oxygen or sulphur atoms
- C07D213/30—Oxygen atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
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- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
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- C07—ORGANIC CHEMISTRY
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- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Physical Education & Sports Medicine (AREA)
- Oncology (AREA)
- Neurology (AREA)
- Diabetes (AREA)
- Neurosurgery (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Communicable Diseases (AREA)
- Biomedical Technology (AREA)
- Hematology (AREA)
- Virology (AREA)
- Dermatology (AREA)
- Rheumatology (AREA)
- Immunology (AREA)
- Cardiology (AREA)
- Pulmonology (AREA)
- Heart & Thoracic Surgery (AREA)
- Endocrinology (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Addiction (AREA)
- Molecular Biology (AREA)
- Urology & Nephrology (AREA)
- Obesity (AREA)
- Emergency Medicine (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US20636200P | 2000-05-23 | 2000-05-23 | |
| US21700600P | 2000-07-10 | 2000-07-10 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PL357713A1 true PL357713A1 (pl) | 2004-07-26 |
Family
ID=26901274
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL01357713A PL357713A1 (pl) | 2000-05-23 | 2001-05-23 | Inhibitory kaspaz i ich zastosowania |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US7053057B2 (pl) |
| EP (1) | EP1283827A2 (pl) |
| JP (1) | JP2003534325A (pl) |
| KR (1) | KR20020025959A (pl) |
| AP (1) | AP2002002407A0 (pl) |
| AR (1) | AR028619A1 (pl) |
| AU (1) | AU2001265008A1 (pl) |
| CA (1) | CA2380935A1 (pl) |
| MX (1) | MXPA02000823A (pl) |
| NO (1) | NO20020343L (pl) |
| NZ (1) | NZ516918A (pl) |
| PE (1) | PE20020058A1 (pl) |
| PL (1) | PL357713A1 (pl) |
| SK (1) | SK1192002A3 (pl) |
| TR (1) | TR200200767T1 (pl) |
| WO (1) | WO2001090070A2 (pl) |
Families Citing this family (48)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2000061542A1 (en) | 1999-04-09 | 2000-10-19 | Cytovia, Inc. | Caspase inhibitors and the use thereof |
| AU6894800A (en) | 1999-08-06 | 2001-03-05 | Vertex Pharmaceuticals Incorporated | Caspase inhibitors and uses thereof |
| IL148426A0 (en) | 1999-08-27 | 2002-09-12 | Cytovia Inc | α-HYDROXY ACID DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME |
| PE20011350A1 (es) | 2000-05-19 | 2002-01-15 | Vertex Pharma | PROFARMACO DE UN INHIBIDOR DE ENZIMA CONVERTIDORA DE INTERLEUCINA-1ß (ICE) |
| US6878743B2 (en) | 2001-09-18 | 2005-04-12 | Sunesis Pharmaceuticals, Inc. | Small molecule inhibitors of caspases |
| US7410956B2 (en) | 2002-02-11 | 2008-08-12 | Vertex Pharmaceuticals Incorporated | Caspase inhibitor prodrugs |
| US7960398B2 (en) | 2002-04-19 | 2011-06-14 | Vertex Pharmaceuticals Incorporated | Regulation of TNF-alpha |
| JP2006502415A (ja) * | 2002-10-10 | 2006-01-19 | ベクトン・ディキンソン・アンド・カンパニー | カスパーゼ阻害剤を有するサンプル収集システム |
| EP1626732B1 (en) * | 2003-05-22 | 2013-04-03 | CHIESI FARMACEUTICI S.p.A. | Means for preventing and treating cellular death and their biological applications |
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| AU7775991A (en) | 1990-04-04 | 1991-10-30 | Immunex Corporation | Interleukin 1beta protease |
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| CN1297354A (zh) | 1998-03-16 | 2001-05-30 | 西托维亚公司 | 二肽卡斯帕酶抑制剂及其用途 |
| US6045990A (en) * | 1998-07-09 | 2000-04-04 | Baust; John M. | Inclusion of apoptotic regulators in solutions for cell storage at low temperature |
-
2001
- 2001-05-23 EP EP01939497A patent/EP1283827A2/en not_active Withdrawn
- 2001-05-23 US US09/863,649 patent/US7053057B2/en not_active Expired - Fee Related
- 2001-05-23 CA CA002380935A patent/CA2380935A1/en not_active Abandoned
- 2001-05-23 KR KR1020027000995A patent/KR20020025959A/ko not_active Ceased
- 2001-05-23 AP APAP/P/2002/002407A patent/AP2002002407A0/en unknown
- 2001-05-23 JP JP2001586259A patent/JP2003534325A/ja active Pending
- 2001-05-23 PE PE2001000468A patent/PE20020058A1/es not_active Application Discontinuation
- 2001-05-23 SK SK119-2002A patent/SK1192002A3/sk unknown
- 2001-05-23 AU AU2001265008A patent/AU2001265008A1/en not_active Abandoned
- 2001-05-23 WO PCT/US2001/017075 patent/WO2001090070A2/en not_active Ceased
- 2001-05-23 TR TR2002/00767T patent/TR200200767T1/xx unknown
- 2001-05-23 NZ NZ516918A patent/NZ516918A/en unknown
- 2001-05-23 AR ARP010102477A patent/AR028619A1/es unknown
- 2001-05-23 MX MXPA02000823A patent/MXPA02000823A/es not_active Application Discontinuation
- 2001-05-23 PL PL01357713A patent/PL357713A1/pl not_active Application Discontinuation
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2002
- 2002-01-22 NO NO20020343A patent/NO20020343L/no not_active Application Discontinuation
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| Publication number | Publication date |
|---|---|
| AR028619A1 (es) | 2003-05-14 |
| SK1192002A3 (en) | 2002-09-10 |
| PE20020058A1 (es) | 2002-01-31 |
| CA2380935A1 (en) | 2001-11-29 |
| NO20020343D0 (no) | 2002-01-22 |
| WO2001090070A3 (en) | 2002-04-11 |
| EP1283827A2 (en) | 2003-02-19 |
| MXPA02000823A (es) | 2002-07-30 |
| US20020061853A1 (en) | 2002-05-23 |
| NZ516918A (en) | 2004-06-25 |
| US7053057B2 (en) | 2006-05-30 |
| KR20020025959A (ko) | 2002-04-04 |
| JP2003534325A (ja) | 2003-11-18 |
| WO2001090070A2 (en) | 2001-11-29 |
| TR200200767T1 (tr) | 2002-09-23 |
| AU2001265008A1 (en) | 2001-12-03 |
| NO20020343L (no) | 2002-03-21 |
| AP2002002407A0 (en) | 2002-03-31 |
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