PL358412A1 - Kompozycje zawierające związki chinazolinowe i sposoby ich wykorzystania - Google Patents

Kompozycje zawierające związki chinazolinowe i sposoby ich wykorzystania

Info

Publication number
PL358412A1
PL358412A1 PL01358412A PL35841201A PL358412A1 PL 358412 A1 PL358412 A1 PL 358412A1 PL 01358412 A PL01358412 A PL 01358412A PL 35841201 A PL35841201 A PL 35841201A PL 358412 A1 PL358412 A1 PL 358412A1
Authority
PL
Poland
Prior art keywords
methods
compositions utilizing
quinazolinones
utilizing quinazolinones
compositions
Prior art date
Application number
PL01358412A
Other languages
English (en)
Other versions
PL204525B1 (pl
Inventor
Jeffrey T. Finer
Gustav Bergnes
Bainian Feng
Whitney W. Smith
John C. Chabala
David J.Jr. Morgans
Original Assignee
Cytokinetics, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cytokinetics, Inc. filed Critical Cytokinetics, Inc.
Publication of PL358412A1 publication Critical patent/PL358412A1/pl
Publication of PL204525B1 publication Critical patent/PL204525B1/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88—Oxygen atoms
    • C07D239/90—Oxygen atoms with acyclic radicals attached in position 2 or 3
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88—Oxygen atoms
    • C07D239/91—Oxygen atoms with aryl or aralkyl radicals attached in position 2 or 3

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Immunology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Transplantation (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
  • Paints Or Removers (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Investigating Or Analysing Biological Materials (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
  • Medicinal Preparation (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Fats And Perfumes (AREA)
PL358412A 2000-06-21 2001-04-27 Związki chinazolinowe , ich zastosowanie oraz kompozycje farmaceutyczne zawierające te związki PL204525B1 (pl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US21310400P 2000-06-21 2000-06-21
US09/699,047 US6545004B1 (en) 1999-10-27 2000-10-24 Methods and compositions utilizing quinazolinones

Publications (2)

Publication Number Publication Date
PL358412A1 true PL358412A1 (pl) 2004-08-09
PL204525B1 PL204525B1 (pl) 2010-01-29

Family

ID=26907773

Family Applications (1)

Application Number Title Priority Date Filing Date
PL358412A PL204525B1 (pl) 2000-06-21 2001-04-27 Związki chinazolinowe , ich zastosowanie oraz kompozycje farmaceutyczne zawierające te związki

Country Status (23)

Country Link
US (7) US6545004B1 (pl)
EP (2) EP1296959B1 (pl)
JP (1) JP4854906B2 (pl)
KR (1) KR100847788B1 (pl)
CN (1) CN1229353C (pl)
AT (1) ATE323684T1 (pl)
AU (3) AU5927001A (pl)
BR (1) BR0111898A (pl)
CA (1) CA2413426C (pl)
CY (1) CY1105070T1 (pl)
CZ (1) CZ303007B6 (pl)
DE (1) DE60118921T2 (pl)
DK (1) DK1296959T3 (pl)
ES (1) ES2262649T3 (pl)
HU (1) HU229078B1 (pl)
IL (1) IL153554A (pl)
MX (1) MXPA02012627A (pl)
NO (1) NO324440B1 (pl)
NZ (1) NZ523233A (pl)
PL (1) PL204525B1 (pl)
PT (1) PT1296959E (pl)
SI (1) SI1296959T1 (pl)
WO (1) WO2001098278A1 (pl)

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HUP0301201A3 (en) 2004-03-29
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CA2413426C (en) 2011-01-04
US7294634B2 (en) 2007-11-13
CN1437585A (zh) 2003-08-20
AU5927001A (en) 2002-01-02
BR0111898A (pt) 2003-05-13
US6831085B1 (en) 2004-12-14
US6545004B1 (en) 2003-04-08
IL153554A0 (en) 2003-07-06
HUP0301201A2 (hu) 2003-12-29
KR100847788B1 (ko) 2008-07-23
HK1053837A1 (en) 2003-11-07
CZ20024178A3 (cs) 2003-05-14
ES2262649T3 (es) 2006-12-01
PL204525B1 (pl) 2010-01-29
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NZ523233A (en) 2004-10-29
PT1296959E (pt) 2006-07-31
US20040023996A1 (en) 2004-02-05
NO324440B1 (no) 2007-10-15
US7105668B1 (en) 2006-09-12
US6630479B1 (en) 2003-10-07
IL153554A (en) 2009-09-01
DK1296959T3 (da) 2006-07-31
AU2006236024A1 (en) 2006-12-07
CN1229353C (zh) 2005-11-30
DE60118921D1 (de) 2006-05-24
ATE323684T1 (de) 2006-05-15
HU229078B1 (en) 2013-07-29
EP1707563A3 (en) 2007-06-06
JP4854906B2 (ja) 2012-01-18
AU2001259270B2 (en) 2006-08-24
NO20026172L (no) 2003-02-20
KR20030047903A (ko) 2003-06-18
CA2413426A1 (en) 2001-12-27
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JP2004501140A (ja) 2004-01-15
US6562831B1 (en) 2003-05-13
EP1707563A2 (en) 2006-10-04
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EP1296959A1 (en) 2003-04-02
CY1105070T1 (el) 2009-11-04

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