PL361616A1 - Sposób wytwarzania 16,17-[(cykloheksylometyleno) bis (oksy)]-11,21-dihydroksypregna-1,4-dieno-3,20-dionu lub jego 21-izomaślanu przez transketalizację - Google Patents

Sposób wytwarzania 16,17-[(cykloheksylometyleno) bis (oksy)]-11,21-dihydroksypregna-1,4-dieno-3,20-dionu lub jego 21-izomaślanu przez transketalizację

Info

Publication number
PL361616A1
PL361616A1 PL01361616A PL36161601A PL361616A1 PL 361616 A1 PL361616 A1 PL 361616A1 PL 01361616 A PL01361616 A PL 01361616A PL 36161601 A PL36161601 A PL 36161601A PL 361616 A1 PL361616 A1 PL 361616A1
Authority
PL
Poland
Prior art keywords
oxy
bis
cyclohexylmethylen
isobutyrat
transketalisation
Prior art date
Application number
PL01361616A
Other languages
English (en)
Other versions
PL205674B1 (pl
Inventor
Beate Schmidt
Original Assignee
Altana Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Altana Pharma Ag filed Critical Altana Pharma Ag
Publication of PL361616A1 publication Critical patent/PL361616A1/pl
Publication of PL205674B1 publication Critical patent/PL205674B1/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005—Oxygen-containing hetero ring
    • C07J71/0026—Oxygen-containing hetero ring cyclic ketals
    • C07J71/0031—Oxygen-containing hetero ring cyclic ketals at positions 16, 17

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Liquid Crystal Substances (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
PL361616A 2000-11-10 2001-11-06 Sposób wytwarzania 16,17-[(cykloheksylometyleno) bis (oksy)]-11,21-dihydroksypregna-1,4-dieno-3,20-dionu PL205674B1 (pl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP00124626 2000-11-10
PCT/EP2001/012808 WO2002038584A1 (en) 2000-11-10 2001-11-06 Process for the production of 16,17-[(cyclohexylmethylen)bis(oxy)]-11,21-dihydroxy-pregna-1,4-dien-3,20-dion or its 21-isobutyrat by transketalisation

Publications (2)

Publication Number Publication Date
PL361616A1 true PL361616A1 (pl) 2004-10-04
PL205674B1 PL205674B1 (pl) 2010-05-31

Family

ID=8170345

Family Applications (1)

Application Number Title Priority Date Filing Date
PL361616A PL205674B1 (pl) 2000-11-10 2001-11-06 Sposób wytwarzania 16,17-[(cykloheksylometyleno) bis (oksy)]-11,21-dihydroksypregna-1,4-dieno-3,20-dionu

Country Status (22)

Country Link
US (1) US7468433B2 (pl)
EP (1) EP1335929B1 (pl)
JP (1) JP4456811B2 (pl)
KR (2) KR20070116185A (pl)
CN (1) CN1264855C (pl)
AT (1) ATE478888T1 (pl)
AU (1) AU2953602A (pl)
BR (1) BR0115220A (pl)
CA (1) CA2430196C (pl)
CZ (1) CZ303885B6 (pl)
DE (1) DE60142920D1 (pl)
EA (1) EA006231B1 (pl)
ES (1) ES2351184T3 (pl)
HU (1) HU228432B1 (pl)
IL (1) IL155274A0 (pl)
MX (1) MXPA03004123A (pl)
NO (1) NO325286B1 (pl)
NZ (1) NZ525707A (pl)
PL (1) PL205674B1 (pl)
SK (1) SK287545B6 (pl)
WO (1) WO2002038584A1 (pl)
ZA (1) ZA200303121B (pl)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY143936A (en) * 2003-03-27 2011-07-29 Nycomed Gmbh Process for preparing crystalline ciclesonide with defined particle size
CN100404545C (zh) * 2003-03-27 2008-07-23 尼科梅德有限责任公司 具有规定粒径的结晶环缩松的制备方法
CN100338089C (zh) * 2004-08-12 2007-09-19 重庆医药工业研究院有限责任公司 一种哮喘病治疗药物环索奈德的新的制备方法
CN100345864C (zh) * 2004-10-29 2007-10-31 天津药业研究院有限公司 一种治疗呼吸道疾病的甾体药物的制备方法及其中间体
WO2007054974A2 (en) * 2005-09-28 2007-05-18 Arch Pharmalab Limited A green chemistry process for the preparation of pregnadiene esters
WO2008015696A2 (en) * 2006-05-23 2008-02-07 Cadila Healthcare Limited Process for preparing ciclesonide
CA2663737A1 (en) 2006-09-19 2008-03-27 Cipla Limited Processes for the preparation of ciclesonide and its crystal form
US9109005B2 (en) 2012-02-23 2015-08-18 Boehringer Ingelheim International Gmbh Method for manufacturing of ciclesonide
EP3250211B1 (en) 2015-01-30 2021-12-22 Coral Drugs Pvt. Ltd. Novel process for preparation of glucocorticoid steroids
US20180126000A1 (en) 2016-06-02 2018-05-10 Abbvie Inc. Glucocorticoid receptor agonist and immunoconjugates thereof
BR112020010694A2 (pt) 2017-12-01 2020-11-10 Abbvie Inc. agonista de receptor de glicocorticoides e imunoconjugados do mesmo

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4880368A (en) * 1983-10-24 1989-11-14 Siegfried C. Hasl In-mold label transfer apparatus
ES8506753A1 (es) 1983-11-24 1985-08-01 Frumtost Zyma S A Procedimiento para la obtencion de un corticoide de accion antipsoriatica
IT1196142B (it) * 1984-06-11 1988-11-10 Sicor Spa Procedimento per la preparazione di 16,17-acetali di derivati pregnanici e nuovi composti ottenuti
SE8604059D0 (sv) * 1986-09-25 1986-09-25 Astra Pharma Prod A method of controlling the epimeric distribution in the preparation of 16,17-acetals of pregnane derivatives
GR1001529B (el) * 1990-09-07 1994-03-31 Elmuquimica Farm Sl Μέ?οδος για την λήψη νέων 21-εστέρων της 16-17-ακετάλης της πρ να-1,4-διενο-3,20-διόνης.
FR2675146A1 (fr) 1991-04-10 1992-10-16 Roussel Uclaf Nouveaux derives sterouides de la pregna-1,4-diene-3,20-dione, leur preparation, leur application a la preparation de derives 16,17-methylene dioxy substitues et nouveaux intermediaires.
DK0701565T3 (da) 1993-04-02 1999-07-12 Byk Gulden Lomberg Chem Fab Nye prednisolonderivater
DE19635498A1 (de) 1996-09-03 1998-03-26 Byk Gulden Lomberg Chem Fab Verfahren zur Epimerenanreicherung

Also Published As

Publication number Publication date
CN1473164A (zh) 2004-02-04
NO325286B1 (no) 2008-03-17
IL155274A0 (en) 2003-11-23
HUP0302220A3 (en) 2007-11-28
BR0115220A (pt) 2003-10-07
PL205674B1 (pl) 2010-05-31
JP4456811B2 (ja) 2010-04-28
KR20070116185A (ko) 2007-12-06
NO20031964L (no) 2003-04-30
WO2002038584A1 (en) 2002-05-16
SK5552003A3 (en) 2003-08-05
SK287545B6 (sk) 2011-01-04
JP2004513181A (ja) 2004-04-30
EA200300504A1 (ru) 2003-12-25
KR100809510B1 (ko) 2008-03-04
NO20031964D0 (no) 2003-04-30
CA2430196A1 (en) 2002-05-16
EA006231B1 (ru) 2005-10-27
ZA200303121B (en) 2004-04-23
US20050080063A1 (en) 2005-04-14
CZ303885B6 (cs) 2013-06-12
MXPA03004123A (es) 2004-09-10
ATE478888T1 (de) 2010-09-15
AU2953602A (en) 2002-05-21
US7468433B2 (en) 2008-12-23
EP1335929B1 (en) 2010-08-25
EP1335929A1 (en) 2003-08-20
DE60142920D1 (de) 2010-10-07
HK1058043A1 (en) 2004-04-30
ES2351184T3 (es) 2011-02-01
HU228432B1 (hu) 2013-03-28
CA2430196C (en) 2010-01-26
NZ525707A (en) 2004-11-26
HUP0302220A2 (hu) 2003-10-28
CN1264855C (zh) 2006-07-19
KR20030081329A (ko) 2003-10-17

Similar Documents

Publication Publication Date Title
EP0164636A3 (en) A process for the preparation of 16,17 acetals of pregnane derivatives and compounds obtained therefrom
PL361616A1 (pl) Sposób wytwarzania 16,17-[(cykloheksylometyleno) bis (oksy)]-11,21-dihydroksypregna-1,4-dieno-3,20-dionu lub jego 21-izomaślanu przez transketalizację
AU6530990A (en) Process for the manufacture of budesonide
EE03927B1 (et) Meetod R-epimeeri suhtelise sisalduse suurendamiseks [11B,16a(R/S)]-16,17-[(tsükloheksüülmetüleen)bis(oksü)]-11-hüdroksü-21-(2-metüül-1-oksopropoksü)pregna-1,4-dieen-3,20-diooni R/S-epimeerses segus ja selle segu valmistamismeetod
UA6044A1 (uk) Спосіб одержання метіленових похідних андроста-1,4 -діен-3,17-діона
WO2001051451A3 (en) Methods for manufacturing betulinic acid
HUT61570A (en) Process for producing pregna-1,4-diene-3,20-dione derivatives
WO2002026759A3 (de) 17α-FLUORALKYLSTEROIDE, VERFAHREN ZU DEREN HERSTELLUNG UND DIESE VERBINDUNGEN ENTHALTENDE PHARMAZEUTISCHE ZUSAMMENSETZUNGEN
AU2003224308A1 (en) Stereospecific reduction of sapogen-3-ones
AU2713584A (en) Preparation 21-hydroxy-20-keto-delta 16 steroids and intermediates
YU63004A (sh) Postupak za izradu 7alfa-metilsteroida
PL372217A1 (pl) Sposób wytwarzania kwasu 6alfa,9alfa-difluoro-17alfa-(1-oksopropoksy)-11beta-hydroksy-16alfa-metylo-3-oksoandrosta-1,4-dieno-17beta-karbotiowego
PL358032A1 (pl) Nowe zastosowanie 22R-(11, 16 )-16,17-[butylideno-bis(oksy)]-11,21-dihydroksypregna-1,4-dieno-3,20-dionu
WO2004033478A3 (en) Fatty acid modified forms of glucocorticoids and their use as anti-inflammatory
MXPA03005372A (es) Androgenos 14 (15) -insaturados, 15- y/o 16-sustituidos, con perfil de actividad mixto androgenico-progestacional.
MXPA03011751A (es) Proceso para preparar 21-acetato de 11b,17a, 21-trihidroxi-6a-metilpregna-1, 4-dieno-3, 20- diona.
WO2004074305A3 (en) Process for the production of 2-oxa-3-one androstane derivatives
MXPA03005224A (es) Esteroides de metileno como androgenos novedosos.
JPS5762300A (en) 17alpha-cyanosteroid

Legal Events

Date Code Title Description
RECP Rectifications of patent specification