PL363960A1 - Pochodne oksazolidynonów jako środki przeciwbakteryjne - Google Patents

Pochodne oksazolidynonów jako środki przeciwbakteryjne

Info

Publication number: PL363960A1
Authority: PL; Poland
Prior art keywords: antimicrobials; oxazolidinone derivatives; oxazolidinone; derivatives
Prior art date: 2000-07-17

Application number

PL01363960A

Other languages

English (en)

Inventor

Anita Mehta

Sudershan K. Arora

Biswajit Das

Abhijit Ray

Sonali Rudra

Ashok Rattan

Original Assignee

Ranbaxy Laboratories Limited

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-07-17

Filing date

2001-07-16

Publication date

2004-11-29

2001-07-16 Application filed by Ranbaxy Laboratories Limited filed Critical Ranbaxy Laboratories Limited

2004-11-29 Publication of PL363960A1 publication Critical patent/PL363960A1/pl

Links

IZXIZTKNFFYFOF-UHFFFAOYSA-N 2-Oxazolidone Chemical class O=C1NCCO1 IZXIZTKNFFYFOF-UHFFFAOYSA-N 0.000 title 1
239000004599 antimicrobial Substances 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

PL01363960A 2000-07-17 2001-07-16 Pochodne oksazolidynonów jako środki przeciwbakteryjne PL363960A1 (pl)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
IN654DE2000		2000-07-17
PCT/IB2001/001262 WO2002006278A1 (en)	2000-07-17	2001-07-16	Oxazolidinone derivatives as antimicrobials

Publications (1)

Publication Number	Publication Date
PL363960A1 true PL363960A1 (pl)	2004-11-29

Family

ID=11097070

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PL01363960A PL363960A1 (pl)	2000-07-17	2001-07-16	Pochodne oksazolidynonów jako środki przeciwbakteryjne

Country Status (16)

Country	Link
US (2)	US6734307B2 (pl)
EP (1)	EP1303511A1 (pl)
JP (1)	JP2004504321A (pl)
CN (1)	CN1447808A (pl)
AU (2)	AU2001269370B2 (pl)
BR (1)	BR0112826A (pl)
CA (1)	CA2415965A1 (pl)
CZ (1)	CZ2003228A3 (pl)
HU (1)	HUP0302918A2 (pl)
MX (1)	MXPA03000503A (pl)
NZ (1)	NZ523700A (pl)
PL (1)	PL363960A1 (pl)
RU (1)	RU2292345C9 (pl)
SK (1)	SK1402003A3 (pl)
WO (1)	WO2002006278A1 (pl)
ZA (1)	ZA200300471B (pl)

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WO2003008389A1 (en) *	2001-07-16	2003-01-30	Ranbaxy Laboratories Limited	Oxazolidinone derivatives as potential antimicrobials
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US6956040B2 (en)	2001-07-16	2005-10-18	Ranbaxy Laboratories Limited	Oxazolidinone piperazinyl derivatives as potential antimicrobials
FR2828488B1 (fr) *	2001-08-08	2005-06-10	Oreal	Composition pour la teinture de fibres keratiniques contenant une paraphenylenediamine substituee par un radical diazacycloheptane
CA2478502A1 (en) *	2002-04-01	2003-10-09	Cadila Healthcare Limited	Novel antiinfective compounds, process for their preparation and pharmaceutical compositions containing them
AU2003224345A1 (en) *	2002-04-30	2003-11-17	Orchid Chemicals & Pharmaceuticals	Antibacterial agents
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US6875784B2 (en)	2002-10-09	2005-04-05	Pharmacia & Upjohn Company	Antimibicrobial [3.1.0.] bicyclic oxazolidinone derivatives
GB0302094D0 (en)	2003-01-29	2003-02-26	Pharmagene Lab Ltd	EP4 receptor antagonists
EP1594852A1 (en) *	2003-02-07	2005-11-16	Ranbaxy Laboratories, Ltd.	Oxazolidinone derivatives as antimicrobials
US7223788B2 (en)	2003-02-14	2007-05-29	Sanofi-Aventis Deutschland Gmbh	Substituted N-aryl heterocycles, process for their preparation and their use as medicaments
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AU2003215861A1 (en) *	2003-04-07	2004-11-01	Ranbaxy Laboratories Limited	Oxazolidinone derivatives as antimicrobials
JP2006522791A (ja)	2003-04-09	2006-10-05	ファルマシア・アンド・アップジョン・カンパニー・エルエルシー	抗微生物性［３．１．０］ビシクロヘキシルフェニルオキサゾリジノン誘導体および類似体
WO2005003087A2 (en) *	2003-07-01	2005-01-13	Orchid Chemicals And Pharmaceuticals Ltd.	Oxazole derivatives as antibacterial agents
ATE471937T1 (de)	2003-07-02	2010-07-15	Merck Sharp & Dohme	Cyclopropylgruppensubstituierte oxazolidinonantibiotika und derivate davon
AU2004256086B2 (en) *	2003-07-02	2007-12-06	Kyorin Pharmaceutical Co., Ltd.	Oxazolidinone antibiotics and derivatives thereof
US20070185132A1 (en) *	2003-07-02	2007-08-09	Yasumichi Fukuda	Cyclopropyl group substituted oxazolidinone antibiotics and derivatives thereo
CA2529292A1 (en) *	2003-07-02	2005-01-20	Merck & Co., Inc.	Oxazolidinone antibiotics and derivatives thereof
GB0324269D0 (en)	2003-10-16	2003-11-19	Pharmagene Lab Ltd	EP4 receptor antagonists
WO2005051933A1 (en) *	2003-11-28	2005-06-09	Ranbaxy Laboratories Limited	An improved process for the synthesis of 4-(4-benzyloxy-carbonylamino-2-fluorophenyl)-piperazine-1-carboxylic acid tert-butyl ester, a key intermediate for oxazolidinone antimicrobials and compounds prepared thereby
WO2005082899A1 (en) *	2004-01-28	2005-09-09	Ranbaxy Laboratories Limited	Oxazolidinone derivatives as antimicrobials
US20090247545A1 (en) *	2004-10-11	2009-10-01	Mukund Keshao Gurjar	Substituted oxazolidinone derivatives
DE602006010702D1 (de)	2005-06-29	2010-01-07	Pharmacia & Upjohn Co Llc	Homomorpholinoxazolidinone als antibakterielle mittel
FR2895735B1 (fr)	2005-12-30	2008-04-18	Ecopack France	Valve a poche amelioree
US7728031B2 (en)	2006-02-24	2010-06-01	Abbott Laboratories	Octahydro-pyrrolo[3,4-b]pyrrole derivatives
KR20080110877A (ko)	2006-03-31	2008-12-19	재단법인 이쯔우 연구소	헤테로환을 갖는 신규 화합물
CN101809021B (zh)	2007-09-11	2013-04-24	雅培制药有限公司	八氢-吡咯并[3,4-b]吡咯n-氧化物
CN101883768A (zh) *	2007-10-02	2010-11-10	财团法人乙卯研究所	具有7元杂环的噁唑烷酮衍生物
WO2009132310A1 (en) *	2008-04-25	2009-10-29	Wisconsin Alumni Research Foundation	Inhibitors of udp-galactopyranose mutase thwart mycobacterial growth
EP2635589A1 (en)	2010-11-03	2013-09-11	Wockhardt Limited	Process for the preparation of phosphoric acid mono- (l-{4- [(s) -5- (acetylaminomethyl) - 2 - oxo - oxazolidin- 3 - yl]- 2, 6 - difluorophenyl} - 4 -methoxymethylpiperidin- 4 - yl) ester
UA112876C2 (uk)	2011-09-29	2016-11-10	Сюаньчжу Фарма Ко., Лтд.	Біарилгетероциклзаміщені оксазолідинонові антибактеріальні засоби
WO2015173664A1 (en)	2014-05-14	2015-11-19	Wockhardt Limited	Process for the preparation of (5s)-n-{3-[3,5-difluoro-4-(4-hydroxy-4-methoxymethyl-piperidin-1-yl)-phenyl]-2-oxo-oxazolidin-5-ylmethyl}-acetamide
US10080757B2 (en)	2016-03-11	2018-09-25	Wisconsin Alumni Research Foundation	Inhibitors of UDP-galactopyranose mutase
CN109020873B (zh) *	2018-07-16	2020-04-28	青岛农业大学	以靶标蛋白甾醇14α-脱甲基酶三维结构筛选的化合物及其在在制备杀菌剂中的应用
CA3121202A1 (en)	2018-11-30	2020-06-04	Nuvation Bio Inc.	Pyrrole and pyrazole compounds and methods of use thereof
MX2021012105A (es)	2019-04-03	2021-11-03	Aligos Therapeutics Inc	Compuestos de pirrol.
CA3183397A1 (en)	2020-06-18	2021-12-23	Daryl C. Drummond	Oxazolidinone compounds, liposome compositions comprising oxazolidinone compounds and methods of use thereof

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CA1320730C (en)	1987-10-16	1993-07-27	The Du Pont Merck Pharmaceutical Company	Aminomethyl oxooxazolidinyl aroylbenzene derivatives useful as antibacterial agents
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2001
- 2001-07-16 HU HU0302918A patent/HUP0302918A2/hu unknown
- 2001-07-16 PL PL01363960A patent/PL363960A1/pl not_active Application Discontinuation
- 2001-07-16 EP EP01947730A patent/EP1303511A1/en not_active Withdrawn
- 2001-07-16 RU RU2003103767/04A patent/RU2292345C9/ru not_active IP Right Cessation
- 2001-07-16 WO PCT/IB2001/001262 patent/WO2002006278A1/en not_active Ceased
- 2001-07-16 CZ CZ2003228A patent/CZ2003228A3/cs unknown
- 2001-07-16 CA CA002415965A patent/CA2415965A1/en not_active Abandoned
- 2001-07-16 JP JP2002512181A patent/JP2004504321A/ja active Pending
- 2001-07-16 US US09/906,215 patent/US6734307B2/en not_active Expired - Fee Related
- 2001-07-16 BR BR0112826-4A patent/BR0112826A/pt not_active IP Right Cessation
- 2001-07-16 AU AU2001269370A patent/AU2001269370B2/en not_active Ceased
- 2001-07-16 MX MXPA03000503A patent/MXPA03000503A/es unknown
- 2001-07-16 SK SK140-2003A patent/SK1402003A3/sk not_active Application Discontinuation
- 2001-07-16 NZ NZ523700A patent/NZ523700A/en unknown
- 2001-07-16 CN CN01814422A patent/CN1447808A/zh active Pending
- 2001-07-16 AU AU6937001A patent/AU6937001A/xx active Pending
2002
- 2002-01-21 US US10/483,905 patent/US20040242591A1/en not_active Abandoned
2003
- 2003-01-17 ZA ZA200300471A patent/ZA200300471B/en unknown

Also Published As

Publication number	Publication date
ZA200300471B (en)	2003-10-29
SK1402003A3 (en)	2003-08-05
US6734307B2 (en)	2004-05-11
RU2292345C2 (ru)	2007-01-27
HUP0302918A2 (hu)	2003-12-29
JP2004504321A (ja)	2004-02-12
MXPA03000503A (es)	2003-10-14
WO2002006278A1 (en)	2002-01-24
AU2001269370B2 (en)	2005-10-27
US20020103186A1 (en)	2002-08-01
RU2292345C9 (ru)	2007-05-10
US20040242591A1 (en)	2004-12-02
CA2415965A1 (en)	2002-01-24
NZ523700A (en)	2004-11-26
AU6937001A (en)	2002-01-30
CN1447808A (zh)	2003-10-08
EP1303511A1 (en)	2003-04-23
CZ2003228A3 (cs)	2003-06-18
BR0112826A (pt)	2003-06-24

Legal Events

Date	Code	Title	Description
2008-10-31	REFS	Decisions on refusal to grant patents (taken after the publication of the particulars of the applications)

Publication	Publication Date	Title
AU6937001A (en)	2002-01-30	Oxazolidinone derivatives as antimicrobials
EG22695A (en)	2003-06-30	Novel phenyl-propargylether derivatives
AU6053701A (en)	2001-12-17	2-aminocarbonyl-9h-purine derivatives
HRP20030055A2 (en)	2005-02-28	4-phenyl-pyridine derivatives
IL150841A0 (en)	2003-02-12	1h-imidazopyridine derivatives
GB0029531D0 (en)	2001-01-17	Speed govenor
GB0017508D0 (en)	2000-08-30	Antimicrobials
GB0017031D0 (en)	2000-08-30	Antimicrobials
EP1542696A4 (en)	2006-08-02	OXAZOLIDINONE DERIVATIVES AS ANTIMICROBIAL AGENTS
AU2002258054A1 (en)	2003-03-03	Oxazolidinone derivatives as antimicrobials
IL155103A0 (en)	2003-10-31	Substituted c-cyclohexylmethylamine derivatives
PL356565A1 (pl)	2004-06-28	Pochodne aminosulfonylobifenylu
IL150557A0 (en)	2003-02-12	Substituted aminomethyl-phenyl-cyclohexane derivatives
AU8993701A (en)	2002-04-15	Substituted 1-aminobutan-3-ol derivatives
GB0118407D0 (en)	2001-09-19	Oxazolidinone derivatives as antibacterial agents
IL150558A0 (en)	2003-02-12	Aminomethyl-phenyl-cyclohexanone derivatives
AU4754001A (en)	2001-10-15	Novel benzosultam oxazolidinone antibacterial agents
AU2163202A (en)	2002-04-22	5-amino-1-pentene-3-ol substituted derivatives
IL151598A0 (en)	2003-04-10	2-phenylpyran-4-one derivatives
AU2002216086A1 (en)	2002-07-08	Isothiazolecarboxamides as microbicides
HK1055427A (en)	2004-01-09	Oxazolidinone derivatives as antimicrobials
GB0017275D0 (en)	2000-08-30	Antimicrobials
AU2002219458A1 (en)	2003-03-03	Oxazolidinone derivatives as potential antimicrobials
GB0021639D0 (en)	2000-10-18	Maurotoxin derivatives
GB0021079D0 (en)	2000-10-11	Novel s-nitrosothiols