PL365950A1 - Heterocykliczne sulfonamidowe inhibitory procesu wytwarzania beta amyloidu - Google Patents

Heterocykliczne sulfonamidowe inhibitory procesu wytwarzania beta amyloidu

Info

Publication number
PL365950A1
PL365950A1 PL01365950A PL36595001A PL365950A1 PL 365950 A1 PL365950 A1 PL 365950A1 PL 01365950 A PL01365950 A PL 01365950A PL 36595001 A PL36595001 A PL 36595001A PL 365950 A1 PL365950 A1 PL 365950A1
Authority
PL
Poland
Prior art keywords
beta amyloid
amyloid production
heterocyclic sulfonamide
sulfonamide inhibitors
inhibitors
Prior art date
Application number
PL01365950A
Other languages
English (en)
Inventor
Anthony Frank Kreft
Derek Cecil Cole
Kevin Roger Woller
Joseph Raymond Stock
George Diamanitis
Dennis Michael Kurbrak
Kristina Martha Kutterer
William Jay Moore
David Scott Casebier
Original Assignee
Wyeth
Arqule, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22966854&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL365950(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Wyeth, Arqule, Inc. filed Critical Wyeth
Publication of PL365950A1 publication Critical patent/PL365950A1/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D307/64—Sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/30—Hetero atoms other than halogen
    • C07D333/34—Sulfur atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
PL01365950A 2000-12-13 2001-12-11 Heterocykliczne sulfonamidowe inhibitory procesu wytwarzania beta amyloidu PL365950A1 (pl)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US25510500P 2000-12-13 2000-12-13

Publications (1)

Publication Number Publication Date
PL365950A1 true PL365950A1 (pl) 2005-01-24

Family

ID=22966854

Family Applications (1)

Application Number Title Priority Date Filing Date
PL01365950A PL365950A1 (pl) 2000-12-13 2001-12-11 Heterocykliczne sulfonamidowe inhibitory procesu wytwarzania beta amyloidu

Country Status (27)

Country Link
US (5) US6610734B2 (pl)
EP (1) EP1341779B1 (pl)
JP (2) JP2004517892A (pl)
KR (1) KR100869061B1 (pl)
CN (2) CN1800176A (pl)
AR (1) AR035516A1 (pl)
AT (1) ATE330950T1 (pl)
AU (1) AU2002245123B2 (pl)
BR (1) BR0116063A (pl)
CA (1) CA2436526C (pl)
CY (1) CY1105441T1 (pl)
DE (1) DE60121032T2 (pl)
DK (1) DK1341779T3 (pl)
EA (1) EA009035B1 (pl)
ES (1) ES2267853T3 (pl)
HU (1) HUP0303857A3 (pl)
IL (3) IL156268A0 (pl)
MX (1) MXPA03005255A (pl)
NO (1) NO328885B1 (pl)
NZ (2) NZ526213A (pl)
PL (1) PL365950A1 (pl)
PT (1) PT1341779E (pl)
SG (1) SG128491A1 (pl)
SI (1) SI1341779T1 (pl)
TW (1) TWI235155B (pl)
WO (1) WO2002057252A2 (pl)
ZA (1) ZA200304135B (pl)

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EP3586839A1 (en) 2008-07-28 2020-01-01 Blanchette Rockefeller Neurosciences, Institute Pkc-activating compounds for the treatment of neurodegenerative diseases
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US9802954B2 (en) 2011-08-24 2017-10-31 Boehringer Ingelheim International Gmbh Piperidino-dihydrothienopyrimidine sulfoxides and their use for treating COPD and asthma
BR112015017251B1 (pt) 2013-01-18 2021-10-26 Cardioxyl Pharmaceuticals, Inc. Composições farmacêuticas compreendendo doadores de nitroxil, misturas e usos das referidas composições farmacêuticas
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Also Published As

Publication number Publication date
US20020183361A1 (en) 2002-12-05
IL188853A0 (en) 2011-08-01
DE60121032D1 (de) 2006-08-03
IL156268A (en) 2008-04-13
JP2004517892A (ja) 2004-06-17
EP1341779A2 (en) 2003-09-10
AU2002245123B2 (en) 2007-05-24
CA2436526A1 (en) 2002-07-25
WO2002057252A3 (en) 2002-12-12
WO2002057252A2 (en) 2002-07-25
EA009035B1 (ru) 2007-10-26
DE60121032T2 (de) 2007-01-11
SG128491A1 (en) 2007-01-30
CN1263750C (zh) 2006-07-12
CN1800176A (zh) 2006-07-12
US6610734B2 (en) 2003-08-26
US20050196813A1 (en) 2005-09-08
NZ538100A (en) 2006-07-28
US7691884B2 (en) 2010-04-06
KR20040018318A (ko) 2004-03-03
TWI235155B (en) 2005-07-01
PT1341779E (pt) 2006-10-31
NO20032645L (no) 2003-08-05
US20100022594A1 (en) 2010-01-28
EP1341779B1 (en) 2006-06-21
IL156268A0 (en) 2004-01-04
NO20032645D0 (no) 2003-06-11
JP2010265280A (ja) 2010-11-25
DK1341779T3 (da) 2006-10-30
HUP0303857A2 (hu) 2004-03-29
US20110034513A1 (en) 2011-02-10
CN1503790A (zh) 2004-06-09
CY1105441T1 (el) 2010-07-28
US6878742B2 (en) 2005-04-12
CA2436526C (en) 2010-10-19
KR100869061B1 (ko) 2008-11-17
MXPA03005255A (es) 2004-10-14
BR0116063A (pt) 2004-08-03
EA200300674A1 (ru) 2004-06-24
ATE330950T1 (de) 2006-07-15
ZA200304135B (en) 2004-09-03
NO328885B1 (no) 2010-06-07
SI1341779T1 (sl) 2006-12-31
US7842718B2 (en) 2010-11-30
ES2267853T3 (es) 2007-03-16
US20030229127A1 (en) 2003-12-11
NZ526213A (en) 2005-05-27
AR035516A1 (es) 2004-06-02
HUP0303857A3 (en) 2007-07-30
HK1059619A1 (en) 2004-07-09

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