PL369449A1 - Solwaty chlorowodorku lerkanidypiny i nowe krystaliczne postacie chlorowodorku lerkanidypiny - Google Patents

Solwaty chlorowodorku lerkanidypiny i nowe krystaliczne postacie chlorowodorku lerkanidypiny

Info

Publication number: PL369449A1
Authority: PL; Poland
Prior art keywords: lercanidipine hydrochloride; solvates; crystalline forms; new crystalline; lercanidipine
Prior art date: 2001-08-06

Application number

PL02369449A

Other languages

English (en)

Inventor

Amedeo Leonardi

Iasi Gianluca De

Fausto Bonifacio

Original Assignee

Recordati Ireland Limited

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-08-06

Filing date

2002-08-05

Publication date

2005-04-18

2002-08-05 Application filed by Recordati Ireland Limited filed Critical Recordati Ireland Limited

2005-04-18 Publication of PL369449A1 publication Critical patent/PL369449A1/pl

Links

WMFYOYKPJLRMJI-UHFFFAOYSA-N Lercanidipine hydrochloride Chemical compound Cl.COC(=O)C1=C(C)NC(C)=C(C(=O)OC(C)(C)CN(C)CCC(C=2C=CC=CC=2)C=2C=CC=CC=2)C1C1=CC=CC([N+]([O-])=O)=C1 WMFYOYKPJLRMJI-UHFFFAOYSA-N 0.000 title abstract 5
229960002162 lercanidipine hydrochloride Drugs 0.000 title abstract 5
239000012453 solvate Substances 0.000 title abstract 3
239000013543 active substance Substances 0.000 abstract 1
239000003960 organic solvent Substances 0.000 abstract 1
239000008194 pharmaceutical composition Substances 0.000 abstract 1
238000007614 solvation Methods 0.000 abstract 1
239000002904 solvent Substances 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/80—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D211/84—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen directly attached to ring carbon atoms
- C07D211/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/12—Drugs for disorders of the metabolism for electrolyte homeostasis
- A61P3/14—Drugs for disorders of the metabolism for electrolyte homeostasis for calcium homeostasis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Life Sciences & Earth Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Rheumatology (AREA)
Obesity (AREA)
Hematology (AREA)
Endocrinology (AREA)
Diabetes (AREA)
Hydrogenated Pyridines (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

PL02369449A 2001-08-06 2002-08-05 Solwaty chlorowodorku lerkanidypiny i nowe krystaliczne postacie chlorowodorku lerkanidypiny PL369449A1 (pl)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
IT2001MI001727A ITMI20011727A1 (it)	2001-08-06	2001-08-06	Solvati della lercanidipina cloridrato e nuove forme cristalline della lercanidipina cloridrato ottenute da essi

Publications (1)

Publication Number	Publication Date
PL369449A1 true PL369449A1 (pl)	2005-04-18

Family

ID=11448246

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PL02369449A PL369449A1 (pl)	2001-08-06	2002-08-05	Solwaty chlorowodorku lerkanidypiny i nowe krystaliczne postacie chlorowodorku lerkanidypiny

Country Status (21)

Country	Link
EP (1)	EP1423367B1 (pl)
JP (1)	JP2005502648A (pl)
KR (1)	KR100912664B1 (pl)
CN (1)	CN100494175C (pl)
AR (1)	AR037230A1 (pl)
AT (1)	ATE294162T1 (pl)
AU (1)	AU2002331390B2 (pl)
BR (1)	BR0211738A (pl)
DE (1)	DE60203919D1 (pl)
EA (1)	EA200400279A1 (pl)
ES (1)	ES2209684T1 (pl)
HR (1)	HRP20040157A2 (pl)
HU (1)	HUP0401161A3 (pl)
IL (2)	IL153916A0 (pl)
IT (1)	ITMI20011727A1 (pl)
MX (1)	MXPA04001073A (pl)
NO (1)	NO20040479L (pl)
PE (1)	PE20030350A1 (pl)
PL (1)	PL369449A1 (pl)
UY (1)	UY27409A1 (pl)
WO (1)	WO2003014085A1 (pl)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
KR100651212B1 (ko)	2004-10-27	2006-12-01	제일약품주식회사	무정형 레르카니디핀의 제조방법
AR052918A1 (es)	2005-02-25	2007-04-11	Recordati Ireland Ltd	Clorhidrato de lercanidipina amorfo
WO2007031865A2 (en)	2005-09-16	2007-03-22	Glenmark Pharmaceuticals Limited	Polymorphic form of lercanidipine hydrochloride and process for the preparation thereof
CN101868442A (zh) *	2007-03-05	2010-10-20	阿克塔维什集团Ptc公司	盐酸乐卡地平多晶型物和1,1,n-三甲基-n-(3,3-二苯基丙基)-2-氨基乙酰醋酸乙酯的改进制法
WO2008136393A1 (ja) *	2007-04-27	2008-11-13	Ajinomoto Co., Inc.	ラクタム化合物の結晶形およびその製造方法
EP2585051B2 (en)	2010-06-23	2020-04-08	KRKA, tovarna zdravil, d.d., Novo mesto	Pharmaceutical oral dosage forms comprising lercanidipine and enalapril and their pharmaceutically acceptable salts
WO2012085249A2 (en)	2010-12-24	2012-06-28	Krka, D.D., Novo Mesto	Homogenous pharmaceutical oral dosage forms comprising lercanidipine and enalapril or their pharmaceutically acceptable salts

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB8403866D0 (en) *	1984-02-14	1984-03-21	Recordati Chem Pharm	Diphenylalkylaminoalkyl esters
US5912351A (en) *	1995-05-12	1999-06-15	Recordati, S.A. Chemical And Pharmaceutical Company	Anhydrous 1,4-Dihydropyridines and salts thereof

2001
- 2001-08-06 IT IT2001MI001727A patent/ITMI20011727A1/it unknown
2002
- 2002-08-02 AR ARP020102957A patent/AR037230A1/es not_active Application Discontinuation
- 2002-08-05 EP EP02767318A patent/EP1423367B1/en not_active Expired - Lifetime
- 2002-08-05 PL PL02369449A patent/PL369449A1/pl unknown
- 2002-08-05 HU HU0401161A patent/HUP0401161A3/hu unknown
- 2002-08-05 WO PCT/EP2002/008700 patent/WO2003014085A1/en not_active Ceased
- 2002-08-05 MX MXPA04001073A patent/MXPA04001073A/es not_active Application Discontinuation
- 2002-08-05 JP JP2003519035A patent/JP2005502648A/ja active Pending
- 2002-08-05 ES ES02767318T patent/ES2209684T1/es active Pending
- 2002-08-05 EA EA200400279A patent/EA200400279A1/ru unknown
- 2002-08-05 KR KR1020047001791A patent/KR100912664B1/ko not_active Expired - Fee Related
- 2002-08-05 CN CNB028155114A patent/CN100494175C/zh not_active Expired - Fee Related
- 2002-08-05 DE DE60203919T patent/DE60203919D1/de not_active Expired - Lifetime
- 2002-08-05 AT AT02767318T patent/ATE294162T1/de not_active IP Right Cessation
- 2002-08-05 HR HR20040157A patent/HRP20040157A2/hr not_active Application Discontinuation
- 2002-08-05 IL IL15391602A patent/IL153916A0/xx unknown
- 2002-08-05 BR BR0211738-0A patent/BR0211738A/pt not_active IP Right Cessation
- 2002-08-05 AU AU2002331390A patent/AU2002331390B2/en not_active Ceased
- 2002-08-06 UY UY27409A patent/UY27409A1/es not_active Application Discontinuation
- 2002-08-06 PE PE2002000716A patent/PE20030350A1/es not_active Application Discontinuation
2003
- 2003-01-13 IL IL153916A patent/IL153916A/en unknown
2004
- 2004-02-03 NO NO20040479A patent/NO20040479L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
HUP0401161A3 (en)	2009-04-28
ATE294162T1 (de)	2005-05-15
CN1538958A (zh)	2004-10-20
WO2003014085A1 (en)	2003-02-20
KR20040030932A (ko)	2004-04-09
IL153916A0 (en)	2003-07-31
EP1423367A1 (en)	2004-06-02
DE60203919D1 (de)	2005-06-02
NO20040479L (no)	2004-02-03
EA200400279A1 (ru)	2004-06-24
MXPA04001073A (es)	2005-02-17
HUP0401161A2 (hu)	2004-09-28
EP1423367B1 (en)	2005-04-27
HRP20040157A2 (en)	2004-08-31
IL153916A (en)	2008-07-08
CN100494175C (zh)	2009-06-03
AR037230A1 (es)	2004-11-03
BR0211738A (pt)	2004-09-28
AU2002331390B2 (en)	2008-06-05
KR100912664B1 (ko)	2009-08-17
UY27409A1 (es)	2003-03-31
ITMI20011727A0 (it)	2001-08-06
ES2209684T1 (es)	2004-07-01
ITMI20011727A1 (it)	2003-02-06
JP2005502648A (ja)	2005-01-27
PE20030350A1 (es)	2003-06-06

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AU2002352986A1 (en)	2003-06-23	Compositions containing 1,3-dicarbonyl chelating agents for stripping residues from semiconductors
IL161857A0 (en)	2005-11-20	Pharmaceutical compositions of 5,7,14-triazatetracycloÄ10.3.1.0(2,11).0(4,9)Ü-hexadeca-2(11)3,5,7,9-pentaene
EA200401169A1 (ru)	2005-04-28	Аминометилзамещенные тетрациклиновые соединения
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NO20033732L (no)	2003-10-22	N-substituerte ikke-aryl-heterosykliske NMDA/NR2B-antagonister, og farmasoytiske preparater som omfatter slike forbindelser.
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WO2005087700A3 (en)	2006-10-19	Bisphenyl compounds useful as vitamin d3 receptor agonists
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WO2001004116A3 (en)	2001-08-23	Neurotrophic pyrrolidines and piperidines, and related compositions containing them
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