PL371127A1 - Pochodne 6-amino-morfinianu, metody ich otrzymywania oraz ich zastosowania - Google Patents

Pochodne 6-amino-morfinianu, metody ich otrzymywania oraz ich zastosowania

Info

Publication number: PL371127A1
Authority: PL; Poland
Prior art keywords: aminomorphinane; derivatives; production; compounds; formula
Prior art date: 2001-12-17

Application number

PL02371127A

Other languages

English (en)

Inventor

Johannes Schütz

Helmut Schmidhammer

Original Assignee

Alcasynn Pharmaceuticals Gmbh

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-12-17

Filing date

2002-12-16

Publication date

2005-06-13

2002-12-16 Application filed by Alcasynn Pharmaceuticals Gmbh filed Critical Alcasynn Pharmaceuticals Gmbh

2005-06-13 Publication of PL371127A1 publication Critical patent/PL371127A1/pl

Links

ITJUMAAPIQSIHR-YPTPCZDSSA-N (1S,9R,10R)-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2,4,6-trien-13-amine Chemical class C1C(N)CC[C@H]2[C@]3([H])NCC[C@@]21C1=CC=CC=C1C3 ITJUMAAPIQSIHR-YPTPCZDSSA-N 0.000 title 1
150000001875 compounds Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D489/00—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:
- C07D489/06—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: with a hetero atom directly attached in position 14
- C07D489/08—Oxygen atom
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
- A—HUMAN NECESSITIES
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- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P29/02—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P37/02—Immunomodulators
- A—HUMAN NECESSITIES
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- A61P37/02—Immunomodulators
- A61P37/04—Immunostimulants
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- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
- A61P5/40—Mineralocorticosteroids, e.g. aldosterone; Drugs increasing or potentiating the activity of mineralocorticosteroids
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- A—HUMAN NECESSITIES
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- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Veterinary Medicine (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Immunology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Addiction (AREA)
Pain & Pain Management (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Anesthesiology (AREA)
Diabetes (AREA)
Rheumatology (AREA)
Psychiatry (AREA)
Physical Education & Sports Medicine (AREA)
Epidemiology (AREA)
Hematology (AREA)
Emergency Medicine (AREA)
Urology & Nephrology (AREA)
Endocrinology (AREA)
Orthopedic Medicine & Surgery (AREA)
Gastroenterology & Hepatology (AREA)
Pulmonology (AREA)
Transplantation (AREA)
Vascular Medicine (AREA)
Obesity (AREA)
Child & Adolescent Psychology (AREA)

PL02371127A 2001-12-17 2002-12-16 Pochodne 6-amino-morfinianu, metody ich otrzymywania oraz ich zastosowania PL371127A1 (pl)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE10161963A DE10161963A1 (de)	2001-12-17	2001-12-17	6-Aminomorphinanderivate, Herstellungsverfahren dafür und deren Verwendung

Publications (1)

Publication Number	Publication Date
PL371127A1 true PL371127A1 (pl)	2005-06-13

Family

ID=7709535

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PL02371127A PL371127A1 (pl)	2001-12-17	2002-12-16	Pochodne 6-amino-morfinianu, metody ich otrzymywania oraz ich zastosowania

Country Status (18)

Country	Link
US (2)	US7538118B2 (pl)
EP (1)	EP1456212B1 (pl)
JP (1)	JP5017629B2 (pl)
CN (1)	CN1604900A (pl)
AT (1)	ATE347555T1 (pl)
AU (1)	AU2002356660B2 (pl)
BR (1)	BR0215027A (pl)
CA (1)	CA2470809C (pl)
DE (2)	DE10161963A1 (pl)
DK (1)	DK1456212T3 (pl)
ES (1)	ES2278083T3 (pl)
HU (1)	HUP0500024A3 (pl)
NO (1)	NO20043016L (pl)
NZ (1)	NZ533966A (pl)
PL (1)	PL371127A1 (pl)
RU (1)	RU2306314C2 (pl)
WO (1)	WO2003051888A1 (pl)
ZA (1)	ZA200404752B (pl)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE10161963A1 (de) *	2001-12-17	2003-07-03	Johannes Schuetz	6-Aminomorphinanderivate, Herstellungsverfahren dafür und deren Verwendung
TW200619206A (en) *	2004-09-29	2006-06-16	Anormed Inc	Chemokine-binding heterocyclic compound salts, and methods of use thereof
WO2006126529A1 (ja) *	2005-05-25	2006-11-30	Shionogi & Co., Ltd.	６，７－不飽和－７－カルバモイル置換モルヒナン誘導体
EP1762569A1 (en) *	2005-09-12	2007-03-14	Alcasynn Pharmaceuticals Gmbh	Novel 6-amino-morphinan derivatives, method of manufacturing them and their application as analgesics
KR20080065664A (ko) *	2005-11-09	2008-07-14	도레이 가부시끼가이샤	기능성 장장해의 치료 또는 예방제
WO2007140272A2 (en) *	2006-05-26	2007-12-06	Pharmacofore, Inc.	Controlled release of phenolic opioids
RU2363468C1 (ru) *	2008-04-03	2009-08-10	Сергей Константинович Судаков	Применение производных налоксона и налтрексона для приготовления обезболивающих лекарственных средств
FR2939796B1 (fr) *	2008-12-11	2010-12-17	Sanofi Aventis	Derives bicycliques de morphine-6-glucuronide, leur preparation et leur application en therapeutique
US8946419B2 (en)	2009-02-23	2015-02-03	Mallinckrodt Llc	(+)-6-hydroxy-morphinan or (+)-6-amino-morphinan derivatives
EP2440562B1 (en) *	2009-06-11	2016-08-10	Mallinckrodt LLC	Preparation of 6-alpha-amino n-substituted morphinans by catalytic hydrogen transfer
ES2465066T3 (es) *	2009-06-11	2014-06-05	Mallinckrodt Llc	Aminación reductora de 6-ceto-normorfinanos por transferencia de hidrógeno catalítica
JP5867081B2 (ja) *	2010-01-29	2016-02-24	東レ株式会社	胆道疾患の治療又は予防剤
EP2420503A1 (en)	2010-07-27	2012-02-22	Universität Innsbruck	Process for the synthesis of 14-oxygenated morphinan-6-ones
BR112013011593B1 (pt)	2010-11-12	2022-02-22	Shionogi & Co., Ltd	Sal de ácido p-toluenossulfônico
CN103717601A (zh)	2011-06-09	2014-04-09	马林克罗特有限公司	通过催化氢转移对6-酮基吗啡喃的还原胺化
DE102012112839A1 (de)	2012-12-21	2014-06-26	L'Air Liquide, Société Anonyme pour l'Etude et l'Exploitation des Procédés Georges Claude	Verfahren zur Inbetriebnahme einer Anlage für die Herstellung von Propylen
WO2015139847A1 (en) *	2014-03-21	2015-09-24	Chironwells Gmbh	6-(amino acid)-morphinan derivatives in combination with permeation enhancers for use as an orally, rectally, transdermally or nasally administered medicament
TWI775723B (zh)	2015-03-17	2022-09-01	日商日本化美化股份有限公司	嗎啡喃衍生物
JP6840155B6 (ja)	2016-09-16	2025-06-17	日本ケミファ株式会社	モルヒナン誘導体のオピオイドδ受容体アゴニスト関連疾患の治療のための使用
WO2020012248A1 (en)	2018-07-13	2020-01-16	Alkermes Pharma Ireland Limited	Novel naphthylenyl compounds for long-acting injectable compositions and related methods
WO2020012245A1 (en)	2018-07-13	2020-01-16	Alkermes Pharma Ireland Limited	Thienothiophene-naltrexone prodrugs for long-acting injectable compositions
WO2020094634A1 (en)	2018-11-05	2020-05-14	Alkermes Pharma Ireland Limited	Thiophene prodrugs of naltroxene for long-acting injectable compositions and related methods

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US136951A (en) *		1873-03-18		Improvement in truss bridges
JPS4118823B1 (pl) *	1964-02-03	1966-10-31
US4730048A (en) *	1985-12-12	1988-03-08	Regents Of The University Of Minnesota	Gut-selective opiates
US4806556A (en) *	1985-12-12	1989-02-21	Regents Of The University Of Minnesota	Gut-selective opiates
US4912114A (en) *	1988-03-18	1990-03-27	Sandoz Ltd.	Morphinan derivatives
ES2121988T3 (es) *	1992-01-23	1998-12-16	Toray Industries	Derivado de morfinano y uso medicinal.
KR100341950B1 (ko) *	1993-07-19	2002-11-29	도레이 가부시끼가이샤	뇌세포보호제
AU686203B2 (en) *	1993-07-23	1998-02-05	Toray Industries, Inc.	Morphinan derivative and medicinal use
US5869669A (en) *	1996-07-26	1999-02-09	Penick Corporation	Preparation of 14-hydroxynormorphinones from normorphinone dienol acylates
WO1999038869A1 (en) *	1998-01-29	1999-08-05	Monash University	Therapeutic compounds
US6469030B2 (en) *	1999-11-29	2002-10-22	Adolor Corporation	Methods for the treatment and prevention of ileus
CA2403252A1 (en) *	2000-03-15	2001-09-20	Wolfgang Sadee	Neutral antagonists and use thereof in treating drug abuse
DE10161963A1 (de) *	2001-12-17	2003-07-03	Johannes Schuetz	6-Aminomorphinanderivate, Herstellungsverfahren dafür und deren Verwendung

2001
- 2001-12-17 DE DE10161963A patent/DE10161963A1/de not_active Ceased
2002
- 2002-12-16 CN CNA028251288A patent/CN1604900A/zh active Pending
- 2002-12-16 WO PCT/EP2002/014343 patent/WO2003051888A1/de not_active Ceased
- 2002-12-16 RU RU2004121952/04A patent/RU2306314C2/ru not_active IP Right Cessation
- 2002-12-16 JP JP2003552770A patent/JP5017629B2/ja not_active Expired - Fee Related
- 2002-12-16 HU HU0500024A patent/HUP0500024A3/hu unknown
- 2002-12-16 DK DK02804904T patent/DK1456212T3/da active
- 2002-12-16 AT AT02804904T patent/ATE347555T1/de active
- 2002-12-16 NZ NZ533966A patent/NZ533966A/en not_active IP Right Cessation
- 2002-12-16 BR BR0215027-1A patent/BR0215027A/pt not_active IP Right Cessation
- 2002-12-16 PL PL02371127A patent/PL371127A1/pl not_active Application Discontinuation
- 2002-12-16 AU AU2002356660A patent/AU2002356660B2/en not_active Ceased
- 2002-12-16 EP EP02804904A patent/EP1456212B1/de not_active Expired - Lifetime
- 2002-12-16 CA CA002470809A patent/CA2470809C/en not_active Expired - Fee Related
- 2002-12-16 DE DE50208918T patent/DE50208918D1/de not_active Expired - Lifetime
- 2002-12-16 US US10/499,133 patent/US7538118B2/en not_active Expired - Fee Related
- 2002-12-16 ES ES02804904T patent/ES2278083T3/es not_active Expired - Lifetime
2004
- 2004-06-15 ZA ZA2004/04752A patent/ZA200404752B/en unknown
- 2004-07-15 NO NO20043016A patent/NO20043016L/no not_active Application Discontinuation
2009
- 2009-04-27 US US12/430,495 patent/US20090209570A1/en not_active Abandoned

Also Published As

Publication number	Publication date
EP1456212A1 (de)	2004-09-15
BR0215027A (pt)	2004-11-09
EP1456212B1 (de)	2006-12-06
HUP0500024A3 (en)	2009-01-28
DE10161963A1 (de)	2003-07-03
ATE347555T1 (de)	2006-12-15
NZ533966A (en)	2006-05-26
HUP0500024A2 (hu)	2005-04-28
US20090209570A1 (en)	2009-08-20
CA2470809A1 (en)	2003-06-26
RU2306314C2 (ru)	2007-09-20
JP5017629B2 (ja)	2012-09-05
WO2003051888A1 (de)	2003-06-26
AU2002356660A1 (en)	2003-06-30
AU2002356660B2 (en)	2006-03-16
ES2278083T3 (es)	2007-08-01
US7538118B2 (en)	2009-05-26
DE50208918D1 (de)	2007-01-18
RU2004121952A (ru)	2006-01-20
US20050038061A1 (en)	2005-02-17
JP2005516937A (ja)	2005-06-09
CN1604900A (zh)	2005-04-06
ZA200404752B (en)	2005-04-26
NO20043016L (no)	2004-07-15
DK1456212T3 (da)	2007-04-02
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Publication	Publication Date	Title
PL371127A1 (pl)	2005-06-13	Pochodne 6-amino-morfinianu, metody ich otrzymywania oraz ich zastosowania
MXPA03010201A (es)	2006-02-09	Derivados de 2-piridin-ciclohexan-1,4-diamina sustituidos.
TW200510325A (en)	2005-03-16	2-acylamino-4-phenylthiazole derivatives, preparation thereof and therapeutic application thereof
MY134892A (en)	2007-12-31	Substituted 2-thio-3,5-dicyano-4-phenyl-6-aminopyridines and their use
PL369530A1 (pl)	2005-05-02	Związki chemiczne
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MXPA03006093A (es)	2005-02-14	Derivados de n(fenilsulfonil)glicina y su uso terapeutico.
MXPA03008754A (es)	2004-02-18	Derivados de piridina fundidos para utilizarse como agonistas receptores vaniloide para tratar dolor.
DE602004021472D1 (en)	2009-07-23	Pyrimiidinverbindungen
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DE50202504D1 (de)	2005-04-21	Neue 4-aminofuropyrimidine und ihre verwendung
HRP20080057T3 (en)	2008-02-29	9,10-alpha,alpha-oh-taxane analogs and methods for production thereof
AU2003290592A1 (en)	2004-06-18	Antitumor benzoylsulfonamides
PT1419163E (pt)	2005-10-31	Imidazopiridinas triciclicas
WO2002030870A3 (de)	2003-10-02	Substituierte c-cyclohexylmethylamin-derivate
WO2002010152A3 (de)	2002-08-01	Neue indolderivate und deren verwendung als arzneimittel
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WO2003037863A3 (de)	2004-08-12	Substituierte indole, verfahren zu deren herstellung und deren verwendung zur schmerzbekämpfung
UA74430C2 (uk)	2005-12-15	Похідні фенілгетероциклічних етерів як інгібітори зворотного захоплення серотоніну
GB0229081D0 (en)	2003-01-15	Multifunctional cationic photoinitiators, their preparation and use
AU2002357740A1 (en)	2003-06-23	Pyrazolo-pyridine derivatives as antiherpes agents
MXPA04004090A (es)	2004-07-08	Compuestos substituidos de 1h-quinolin-2-ona.
DE60201074D1 (en)	2004-09-30	Pyrazolopyridinderivate
TW200510323A (en)	2005-03-16	Process for the preparation of nonpeptide substituted spirobenzoazepine derivatives