PL372288A1 - Sposób wytwarzania chlorku benzoizoksazolometanosulfonylu i jego amidowanie z wytworzeniem zonisamidu - Google Patents
Sposób wytwarzania chlorku benzoizoksazolometanosulfonylu i jego amidowanie z wytworzeniem zonisamiduInfo
- Publication number
- PL372288A1 PL372288A1 PL03372288A PL37228803A PL372288A1 PL 372288 A1 PL372288 A1 PL 372288A1 PL 03372288 A PL03372288 A PL 03372288A PL 37228803 A PL37228803 A PL 37228803A PL 372288 A1 PL372288 A1 PL 372288A1
- Authority
- PL
- Poland
- Prior art keywords
- amidation
- sulfonyl chloride
- methane sulfonyl
- benzisoxazole methane
- zonisamide
- Prior art date
Links
- IRNDEKGGGVTALN-UHFFFAOYSA-N 1,2-benzoxazole;methane;sulfuryl dichloride Chemical compound C.ClS(Cl)(=O)=O.C1=CC=C2C=NOC2=C1 IRNDEKGGGVTALN-UHFFFAOYSA-N 0.000 title 1
- 230000009435 amidation Effects 0.000 title 1
- 238000007112 amidation reaction Methods 0.000 title 1
- 238000000034 method Methods 0.000 title 1
- UBQNRHZMVUUOMG-UHFFFAOYSA-N zonisamide Chemical compound C1=CC=C2C(CS(=O)(=O)N)=NOC2=C1 UBQNRHZMVUUOMG-UHFFFAOYSA-N 0.000 title 1
- 229960002911 zonisamide Drugs 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/20—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Psychiatry (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US35891602P | 2002-02-22 | 2002-02-22 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PL372288A1 true PL372288A1 (pl) | 2005-07-11 |
Family
ID=27766019
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL03372288A PL372288A1 (pl) | 2002-02-22 | 2003-02-24 | Sposób wytwarzania chlorku benzoizoksazolometanosulfonylu i jego amidowanie z wytworzeniem zonisamidu |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US6936720B2 (pl) |
| EP (1) | EP1472236A4 (pl) |
| JP (1) | JP2005526049A (pl) |
| KR (1) | KR20040099279A (pl) |
| CN (1) | CN1636002A (pl) |
| AU (1) | AU2003219889A1 (pl) |
| CA (1) | CA2475598A1 (pl) |
| HR (1) | HRP20040766A2 (pl) |
| IL (1) | IL158238A0 (pl) |
| IS (1) | IS7406A (pl) |
| MX (1) | MXPA04008109A (pl) |
| NO (1) | NO20043972L (pl) |
| PL (1) | PL372288A1 (pl) |
| WO (1) | WO2003072552A1 (pl) |
| ZA (1) | ZA200407018B (pl) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2003298248A1 (en) * | 2003-01-10 | 2004-08-10 | Dipharma S.P.A. | A process for the preparation of benzo(d)isoxazol-3-yl-methanesulfonic acid and the intermediates thereof |
| DK1583748T3 (da) * | 2003-01-13 | 2010-04-19 | Dainippon Sumitomo Pharma Co | Fremgangsmåde til fremstilling af 1,2-dichlorethanfrie krystaller af zonisamid og særdeles rene krystaller af zonisamid |
| US7081539B2 (en) * | 2004-03-25 | 2006-07-25 | Dainippon Sumitomo Pharma Co., Ltd. | One-pot process for the preparation of 1,2-benzisoxazole-3-methanesulfonamide |
| US20060084814A1 (en) * | 2004-05-20 | 2006-04-20 | Siva Kumar Bobba V | Process for the preparation of zonisamide |
| US7745471B2 (en) | 2004-06-18 | 2010-06-29 | Chemagis Ltd. | Derivatives of 1,2-benzisoxazole-3-methane sulfonic acid as novel intermediates for the synthesis of zonisamide |
| AU2006243000B2 (en) | 2005-05-05 | 2011-05-26 | Macrophage Pharma Limited | Alpha aminoacid ester-drug conjugates hydrolysable by carboxylesterase |
| WO2007016209A2 (en) * | 2005-07-28 | 2007-02-08 | Teva Pharmaceutical Industries Ltd. | Pure 1,2-benzisoxazole-3-methane-sulfonic acid sodium salt and purification process |
| WO2007016208A2 (en) * | 2005-07-28 | 2007-02-08 | Teva Pharmaceutical Industries Ltd. | 1,2-benzisoxazole-3-methane-sulfonic acid ammonium salt |
| US7268234B2 (en) * | 2005-09-16 | 2007-09-11 | Dainippon Sumitomo Pharma Co., Ltd. | Method for sulfonation of 1,2-benzisoxazole-3-acetic acid |
| US7375233B2 (en) | 2005-12-16 | 2008-05-20 | Apotex Pharmachem Inc. | Process for the preparation of zonisamide and the intermediates thereof |
| CN102329278A (zh) * | 2010-07-13 | 2012-01-25 | 深圳市资福药业有限公司 | 一种唑尼沙胺晶体、其制备方法和包含其的药物组合物 |
| KR102704441B1 (ko) * | 2016-11-25 | 2024-09-09 | 삼성디스플레이 주식회사 | 증착용 마스크, 이의 제조 방법, 표시 장치의 제조장치 및 표시 장치의 제조 방법 |
| CN106810507B (zh) * | 2017-01-23 | 2019-06-21 | 珠海市海瑞德生物科技有限公司 | 一种唑尼沙胺的绿色环保合成方法 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS6033114B2 (ja) | 1976-12-16 | 1985-08-01 | 大日本製薬株式会社 | １，２−ベンズイソキサゾ−ル誘導体 |
| US4172896A (en) * | 1978-06-05 | 1979-10-30 | Dainippon Pharmaceutical Co., Ltd. | Methane-sulfonamide derivatives, the preparation thereof and composition comprising the same |
| DE3884966T2 (de) * | 1987-12-29 | 1994-02-03 | Dainippon Pharmaceutical Co | Mittel zur behandlung der ischämischen gehirnkrankheit. |
| CA2440030A1 (en) * | 2001-03-02 | 2002-09-12 | Teva Pharmaceutical Industries Ltd. | Process for the preparation of 1,2-benzisoxazole-3-acetic acid |
| IL158239A0 (en) * | 2001-08-30 | 2004-05-12 | Teva Pharma | Zonisamide intermediate and synthesis |
-
2003
- 2003-02-24 PL PL03372288A patent/PL372288A1/pl not_active Application Discontinuation
- 2003-02-24 CA CA002475598A patent/CA2475598A1/en not_active Abandoned
- 2003-02-24 HR HR20040766A patent/HRP20040766A2/hr not_active Application Discontinuation
- 2003-02-24 WO PCT/US2003/005690 patent/WO2003072552A1/en not_active Ceased
- 2003-02-24 EP EP03716172A patent/EP1472236A4/en not_active Withdrawn
- 2003-02-24 MX MXPA04008109A patent/MXPA04008109A/es unknown
- 2003-02-24 JP JP2003571258A patent/JP2005526049A/ja active Pending
- 2003-02-24 KR KR10-2004-7013020A patent/KR20040099279A/ko not_active Ceased
- 2003-02-24 CN CNA038043289A patent/CN1636002A/zh active Pending
- 2003-02-24 US US10/373,554 patent/US6936720B2/en not_active Expired - Fee Related
- 2003-02-24 AU AU2003219889A patent/AU2003219889A1/en not_active Abandoned
- 2003-02-24 IL IL15823803A patent/IL158238A0/xx unknown
-
2004
- 2004-08-17 IS IS7406A patent/IS7406A/is unknown
- 2004-09-02 ZA ZA200407018A patent/ZA200407018B/en unknown
- 2004-09-22 NO NO20043972A patent/NO20043972L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| WO2003072552A1 (en) | 2003-09-04 |
| WO2003072552A8 (en) | 2004-09-23 |
| US20040014983A1 (en) | 2004-01-22 |
| IL158238A0 (en) | 2004-05-12 |
| CN1636002A (zh) | 2005-07-06 |
| EP1472236A4 (en) | 2006-04-19 |
| IS7406A (is) | 2004-08-17 |
| HRP20040766A2 (en) | 2005-02-28 |
| EP1472236A1 (en) | 2004-11-03 |
| AU2003219889A1 (en) | 2003-09-09 |
| CA2475598A1 (en) | 2003-09-04 |
| MXPA04008109A (es) | 2004-11-26 |
| JP2005526049A (ja) | 2005-09-02 |
| NO20043972L (no) | 2004-09-22 |
| ZA200407018B (en) | 2006-06-28 |
| KR20040099279A (ko) | 2004-11-26 |
| US6936720B2 (en) | 2005-08-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| REFS | Decisions on refusal to grant patents (taken after the publication of the particulars of the applications) |