PL374884A1 - Wytwarzanie 1H-imidazo[4,5-c]chinolino-4-amin z zastosowaniem jako związków pośrednich 1H-imidazo[4,5-c]chinolino-4-ftalimidów - Google Patents

Wytwarzanie 1H-imidazo[4,5-c]chinolino-4-amin z zastosowaniem jako związków pośrednich 1H-imidazo[4,5-c]chinolino-4-ftalimidów

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Publication number
PL374884A1
PL374884A1 PL03374884A PL37488403A PL374884A1 PL 374884 A1 PL374884 A1 PL 374884A1 PL 03374884 A PL03374884 A PL 03374884A PL 37488403 A PL37488403 A PL 37488403A PL 374884 A1 PL374884 A1 PL 374884A1
Authority
PL
Poland
Prior art keywords
imidazo
quinolin
preparation
intermediates
amines via
Prior art date
Application number
PL03374884A
Other languages
English (en)
Inventor
Merli Valeriano
Paola Daverio
Stefano Bianchi
Original Assignee
Teva Gyogyszergyar Zartköruen Mukodo Reszvenytarsasag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teva Gyogyszergyar Zartköruen Mukodo Reszvenytarsasag filed Critical Teva Gyogyszergyar Zartköruen Mukodo Reszvenytarsasag
Publication of PL374884A1 publication Critical patent/PL374884A1/pl

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
PL03374884A 2002-07-23 2003-07-23 Wytwarzanie 1H-imidazo[4,5-c]chinolino-4-amin z zastosowaniem jako związków pośrednich 1H-imidazo[4,5-c]chinolino-4-ftalimidów PL374884A1 (pl)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US39760702P 2002-07-23 2002-07-23

Publications (1)

Publication Number Publication Date
PL374884A1 true PL374884A1 (pl) 2005-11-14

Family

ID=30771087

Family Applications (1)

Application Number Title Priority Date Filing Date
PL03374884A PL374884A1 (pl) 2002-07-23 2003-07-23 Wytwarzanie 1H-imidazo[4,5-c]chinolino-4-amin z zastosowaniem jako związków pośrednich 1H-imidazo[4,5-c]chinolino-4-ftalimidów

Country Status (17)

Country Link
US (3) US6852861B2 (pl)
EP (1) EP1543002B1 (pl)
JP (1) JP2006502121A (pl)
KR (1) KR20050028047A (pl)
CN (1) CN1315828C (pl)
AT (1) ATE338044T1 (pl)
AU (1) AU2003259226A1 (pl)
CA (1) CA2493227A1 (pl)
DE (1) DE60308040T2 (pl)
DK (1) DK1543002T3 (pl)
ES (1) ES2271650T3 (pl)
HR (1) HRP20050159A2 (pl)
IL (1) IL166309A (pl)
MX (1) MXPA05000893A (pl)
PL (1) PL374884A1 (pl)
PT (1) PT1543002E (pl)
WO (1) WO2004009593A1 (pl)

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US20090075980A1 (en) * 2003-10-03 2009-03-19 Coley Pharmaceutical Group, Inc. Pyrazolopyridines and Analogs Thereof
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WO2005123080A2 (en) 2004-06-15 2005-12-29 3M Innovative Properties Company Nitrogen-containing heterocyclyl substituted imidazoquinolines and imidazonaphthyridines
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EP1831214A1 (en) * 2004-12-27 2007-09-12 Usv Limited A process for preparation of 4-amino-1-isobutyl-1h-imidazo[4,5-c]-quinoline (imiquimod)
EP1831226B1 (en) 2004-12-30 2012-08-08 3M Innovative Properties Company Chiral tetracyclic compounds inducing interferon biosynthesis
US8436176B2 (en) * 2004-12-30 2013-05-07 Medicis Pharmaceutical Corporation Process for preparing 2-methyl-1-(2-methylpropyl)-1H-imidazo[4,5-c][1,5]naphthyridin-4-amine
KR20070107685A (ko) * 2004-12-30 2007-11-07 다케다 야쿠힌 고교 가부시키가이샤 1-(2-메틸프로필)-1H-이미다조[4,5-c][1,5]나프티리딘-4-아민 에탄술포네이트 및1-(2-메틸프로필)-1H-이미다조[4,5-c][1,5]나프티리딘-4-아민 메탄술포네이트
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Also Published As

Publication number Publication date
US20050113404A1 (en) 2005-05-26
CA2493227A1 (en) 2004-01-29
IL166309A0 (en) 2006-01-15
DE60308040D1 (de) 2006-10-12
ES2271650T3 (es) 2007-04-16
IL166309A (en) 2010-04-15
JP2006502121A (ja) 2006-01-19
US6852861B2 (en) 2005-02-08
KR20050028047A (ko) 2005-03-21
US20070060755A1 (en) 2007-03-15
EP1543002B1 (en) 2006-08-30
HRP20050159A2 (en) 2005-08-31
DK1543002T3 (da) 2006-12-27
US7153967B2 (en) 2006-12-26
ATE338044T1 (de) 2006-09-15
DE60308040T2 (de) 2007-04-19
PT1543002E (pt) 2006-11-30
CN1681814A (zh) 2005-10-12
WO2004009593A1 (en) 2004-01-29
EP1543002A1 (en) 2005-06-22
US20040138459A1 (en) 2004-07-15
CN1315828C (zh) 2007-05-16
AU2003259226A1 (en) 2004-02-09
MXPA05000893A (es) 2005-09-30

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