PL376659A1 - Skondensowane związki heterocykliczne - Google Patents

Skondensowane związki heterocykliczne

Info

Publication number
PL376659A1
PL376659A1 PL376659A PL37665903A PL376659A1 PL 376659 A1 PL376659 A1 PL 376659A1 PL 376659 A PL376659 A PL 376659A PL 37665903 A PL37665903 A PL 37665903A PL 376659 A1 PL376659 A1 PL 376659A1
Authority
PL
Poland
Prior art keywords
heterocyclic compounds
fused heterocyclic
fused
compounds
heterocyclic
Prior art date
Application number
PL376659A
Other languages
English (en)
Inventor
Xi Chen
Xiaoqi Chen
Pingchen Fan
Juan Jaen
Leping Li
Jeffrey T. Mihalic
Original Assignee
Tularik Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Tularik Inc. filed Critical Tularik Inc.
Publication of PL376659A1 publication Critical patent/PL376659A1/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Psychiatry (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
PL376659A 2002-11-06 2003-11-06 Skondensowane związki heterocykliczne PL376659A1 (pl)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US42445602P 2002-11-06 2002-11-06

Publications (1)

Publication Number Publication Date
PL376659A1 true PL376659A1 (pl) 2006-01-09

Family

ID=32312811

Family Applications (1)

Application Number Title Priority Date Filing Date
PL376659A PL376659A1 (pl) 2002-11-06 2003-11-06 Skondensowane związki heterocykliczne

Country Status (16)

Country Link
US (2) US7253179B2 (pl)
EP (1) EP1562943A1 (pl)
JP (1) JP4547266B2 (pl)
KR (1) KR20050103184A (pl)
CN (2) CN101134757A (pl)
AU (1) AU2003285160B2 (pl)
BR (1) BR0316070A (pl)
CA (1) CA2505372A1 (pl)
EA (1) EA009421B1 (pl)
IS (1) IS7833A (pl)
MX (1) MXPA05004739A (pl)
NO (1) NO20052655L (pl)
NZ (1) NZ540328A (pl)
PL (1) PL376659A1 (pl)
WO (1) WO2004043958A1 (pl)
ZA (1) ZA200503654B (pl)

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US6809104B2 (en) 2001-05-04 2004-10-26 Tularik Inc. Fused heterocyclic compounds
US20070135425A1 (en) * 2001-05-04 2007-06-14 Amgen Inc. Fused heterocyclic compounds
EA009421B1 (ru) 2002-11-06 2007-12-28 Эмджен Инк. Конденсированные гетероциклические соединения
WO2004069798A1 (ja) 2003-02-10 2004-08-19 Banyu Pharmaceutical Co.,Ltd. ピペリジン誘導体を有効成分とするメラニン凝集ホルモン受容体拮抗剤
DE102010025663A1 (de) * 2010-06-30 2012-01-05 Karl-Heinz Glüsenkamp Neue beta-Aminoaldehyd-Derivate, Verfahren zu ihrer Herstellung und ihre chemische Verwendung als reaktive Intermediate
CA2807538A1 (en) * 2010-08-10 2012-02-16 Abbvie Inc. Novel trpv3 modulators
WO2012129491A1 (en) 2011-03-24 2012-09-27 Abbott Laboratories Trpv3 modulators
WO2013062964A2 (en) 2011-10-24 2013-05-02 Abbvie Inc. Novel trpv3 modulators
CN106588812B (zh) * 2016-12-07 2019-02-22 烟台大学 一种酰氯制备2，4-二取代噻唑啉类化合物的方法
JP7488267B2 (ja) * 2019-01-14 2024-05-21 ザイダス・ライフサイエンシーズ・リミテッド 新規な置換スルホニル尿素誘導体
HUP2200222A1 (hu) 2022-06-17 2023-12-28 Richter Gedeon Nyrt MCHR1 antagonisták a Prader-Willi szindróma kezelésére

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JPS63258474A (ja) 1986-08-15 1988-10-25 セドナ・ファ−マセウチカルズ・ビ−・ブイ カルバゾ−ル、ジベンゾフラン又はジベンゾチオフェン基を含む化合物の水酸基誘導体を調製するための方法
US5049655A (en) * 1989-03-22 1991-09-17 The Salk Institute For Biological Studies Melanin-concentrating hormones
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JP2002525054A (ja) 1998-09-17 2002-08-13 インサイト・ファーマスーティカルズ・インコーポレイテッド ヒトｇｐｃｒタンパク質
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Also Published As

Publication number Publication date
JP4547266B2 (ja) 2010-09-22
US7253179B2 (en) 2007-08-07
EP1562943A1 (en) 2005-08-17
NZ540328A (en) 2008-02-29
IS7833A (is) 2005-05-02
NO20052655D0 (no) 2005-06-02
JP2006508130A (ja) 2006-03-09
ZA200503654B (en) 2006-09-27
CN1735613A (zh) 2006-02-15
EA009421B1 (ru) 2007-12-28
US20080058365A1 (en) 2008-03-06
CA2505372A1 (en) 2004-05-27
AU2003285160A1 (en) 2004-06-03
CN1330651C (zh) 2007-08-08
MXPA05004739A (es) 2005-08-02
KR20050103184A (ko) 2005-10-27
AU2003285160B2 (en) 2009-06-04
CN101134757A (zh) 2008-03-05
NO20052655L (no) 2005-07-26
US20040147538A1 (en) 2004-07-29
EA200500770A1 (ru) 2005-12-29
WO2004043958A1 (en) 2004-05-27
BR0316070A (pt) 2005-09-27

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Legal Events

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REFS Decisions on refusal to grant patents (taken after the publication of the particulars of the applications)