PL380663A1 - Amorficzne postaci rizedronianu monosodowego - Google Patents
Amorficzne postaci rizedronianu monosodowegoInfo
- Publication number
- PL380663A1 PL380663A1 PL380663A PL38066305A PL380663A1 PL 380663 A1 PL380663 A1 PL 380663A1 PL 380663 A PL380663 A PL 380663A PL 38066305 A PL38066305 A PL 38066305A PL 380663 A1 PL380663 A1 PL 380663A1
- Authority
- PL
- Poland
- Prior art keywords
- amorphous forms
- risedronate monosodium
- risedronate
- monosodium
- amorphous
- Prior art date
Links
- DRFDPXKCEWYIAW-UHFFFAOYSA-M Risedronate sodium Chemical compound [Na+].OP(=O)(O)C(P(O)([O-])=O)(O)CC1=CC=CN=C1 DRFDPXKCEWYIAW-UHFFFAOYSA-M 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
- C07F9/576—Six-membered rings
- C07F9/58—Pyridine rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Physical Education & Sports Medicine (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CZ20040292A CZ298383B6 (cs) | 2004-02-26 | 2004-02-26 | Amorfní forma risedronátu monosodného |
| CZ20040798A CZ298328B6 (cs) | 2004-07-08 | 2004-07-08 | Semikrystalická forma risedronátu monosodného, zpusob jeho prípravy a léková forma ho obsahující |
| CZ20040880A CZ298491B6 (cs) | 2004-08-12 | 2004-08-12 | Zpusob prípravy amorfní formy risedronátu monosodného |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PL380663A1 true PL380663A1 (pl) | 2007-02-19 |
| PL213481B1 PL213481B1 (pl) | 2013-03-29 |
Family
ID=34915827
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL05706666T PL1723157T5 (pl) | 2004-02-26 | 2005-02-28 | Amorficzne postaci rizedronianu monosodowego |
| PL380663A PL213481B1 (pl) | 2004-02-26 | 2005-02-28 | Amorficzne postaci rizedronianu monosodowego, sposób wytwarzania i preparat farmaceutyczny |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL05706666T PL1723157T5 (pl) | 2004-02-26 | 2005-02-28 | Amorficzne postaci rizedronianu monosodowego |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US7618953B2 (pl) |
| EP (1) | EP1723157B2 (pl) |
| DE (1) | DE602005003557D1 (pl) |
| EA (1) | EA009737B1 (pl) |
| PL (2) | PL1723157T5 (pl) |
| SK (1) | SK50782006A3 (pl) |
| UA (1) | UA83900C2 (pl) |
| WO (1) | WO2005082915A1 (pl) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE602005001873T2 (de) | 2004-03-03 | 2008-04-24 | Chemi S.P.A., Cinisello Balsamo | Amorphe 3-Pyridyl-1-Hydroxyethyliden-1,1-Bisphosphonsäure Mononatriumsalz und Verfahren zu deren Herstellung |
| JP2008514722A (ja) * | 2004-09-30 | 2008-05-08 | ドクター レディズ ラボラトリーズ リミテッド | 非結晶性アトルバスタチンカルシウム |
| US7872144B2 (en) * | 2005-06-13 | 2011-01-18 | Jubilant Organosys Limited | Process for producing biphosphonic acids and forms thereof |
| GB0519891D0 (en) * | 2005-09-30 | 2005-11-09 | Pliva Hrvatska D O O | Pharmaceutically acceptable salts and hydrates |
| JP5354858B2 (ja) * | 2006-05-09 | 2013-11-27 | 株式会社Adeka | スルホンアミド化合物の金属塩を含有するポリエステル樹脂組成物 |
| JP2009536639A (ja) | 2006-05-11 | 2009-10-15 | アイエヌディー−スイフト ラボラトリーズ リミテッド | 純リセドロン酸または塩を調製するための方法 |
| KR100775440B1 (ko) * | 2006-12-20 | 2007-11-12 | 동우신테크 주식회사 | 리세드로네이트 나트륨 헤미펜타히드레이트의 제조방법 |
| DE102007030370A1 (de) | 2007-06-29 | 2009-01-02 | Ratiopharm Gmbh | Essigsäure-Solvate von Risedronat, Polymorph hiervon, deren Herstellung und Verwendung sowie pharmazeutische Zusammensetzung, enthaltend diese |
| KR101010062B1 (ko) | 2008-04-11 | 2011-01-21 | 주식회사 대희화학 | 증발 결정화를 이용한 결정상 리세드로네이트 모노소듐모노하이드레이트의 제조방법 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1378234A1 (en) † | 1996-05-17 | 2004-01-07 | MERCK & CO. INC. | Effervescent bisphosphonate formulation |
| KR19990001564A (ko) † | 1997-06-16 | 1999-01-15 | 유충식 | 용해도를 개선한 아졸계 항진균제 및 이를 함유하는 제제 |
| CN1202828C (zh) † | 1999-05-21 | 2005-05-25 | 诺瓦提斯公司 | 二膦酸在制备抑制或逆转血管发生的药物中的用途 |
| PE20011061A1 (es) * | 2000-02-01 | 2001-11-20 | Procter & Gamble | Cristalizacion selectiva del acido 3-piridil-1-hidroxi-etiliden-1,1-bisfosfonico sodio como el hemipentahidrato o el monohidrato |
| GB2383042A (en) † | 2001-10-18 | 2003-06-18 | Cipla Ltd | Amorphous alendronate sodium |
| HRP20041051A2 (en) † | 2002-04-11 | 2005-02-28 | Teva Pharmaceutical Industries Ltd. | Novel polymorphs and pseudopolymorphs of risedronate sodium |
| CZ293349B6 (cs) | 2002-10-25 | 2004-04-14 | Léčiva, A.S. | Nová krystalická forma sodné soli kyseliny 3-pyridyl-1-hydroxyethyliden-1,1-bisfosfonové |
| CZ298639B6 (cs) † | 2004-02-05 | 2007-12-05 | Zentiva, A. S. | Krystalická forma risedronátu monosodného |
| DE602005001873T2 (de) † | 2004-03-03 | 2008-04-24 | Chemi S.P.A., Cinisello Balsamo | Amorphe 3-Pyridyl-1-Hydroxyethyliden-1,1-Bisphosphonsäure Mononatriumsalz und Verfahren zu deren Herstellung |
| US7872144B2 (en) † | 2005-06-13 | 2011-01-18 | Jubilant Organosys Limited | Process for producing biphosphonic acids and forms thereof |
-
2005
- 2005-02-28 US US10/590,694 patent/US7618953B2/en not_active Expired - Lifetime
- 2005-02-28 PL PL05706666T patent/PL1723157T5/pl unknown
- 2005-02-28 PL PL380663A patent/PL213481B1/pl unknown
- 2005-02-28 SK SK5078-2006A patent/SK50782006A3/sk not_active Application Discontinuation
- 2005-02-28 EA EA200601438A patent/EA009737B1/ru not_active IP Right Cessation
- 2005-02-28 UA UAA200610284A patent/UA83900C2/ru unknown
- 2005-02-28 EP EP05706666.4A patent/EP1723157B2/en not_active Expired - Lifetime
- 2005-02-28 DE DE602005003557T patent/DE602005003557D1/de not_active Expired - Lifetime
- 2005-02-28 WO PCT/CZ2005/000024 patent/WO2005082915A1/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| PL1723157T5 (pl) | 2018-01-31 |
| US20070142332A1 (en) | 2007-06-21 |
| EA009737B1 (ru) | 2008-02-28 |
| EP1723157A1 (en) | 2006-11-22 |
| UA83900C2 (en) | 2008-08-26 |
| EP1723157B1 (en) | 2007-11-28 |
| EP1723157B2 (en) | 2017-02-08 |
| EA200601438A1 (ru) | 2006-12-29 |
| WO2005082915A1 (en) | 2005-09-09 |
| PL1723157T3 (pl) | 2008-04-30 |
| US7618953B2 (en) | 2009-11-17 |
| PL213481B1 (pl) | 2013-03-29 |
| DE602005003557D1 (de) | 2008-01-10 |
| SK50782006A3 (sk) | 2007-03-01 |
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