PL3827005T3 - Pirydopirymidyny jako inhibitory receptora histaminowego h4 - Google Patents

Pirydopirymidyny jako inhibitory receptora histaminowego h4

Info

Publication number
PL3827005T3
PL3827005T3 PL19742760.2T PL19742760T PL3827005T3 PL 3827005 T3 PL3827005 T3 PL 3827005T3 PL 19742760 T PL19742760 T PL 19742760T PL 3827005 T3 PL3827005 T3 PL 3827005T3
Authority
PL
Poland
Prior art keywords
pyridopyrimidines
histamine
receptor inhibitors
inhibitors
receptor
Prior art date
Application number
PL19742760.2T
Other languages
English (en)
Inventor
Gonzalo HERNÁNDEZ HERRERO
Neftalí GARCÍA DOMÍNGUEZ
Arturo ZAZPE ARCE
Roberto Olivera Tizne
Bárbara NOVERGES PEDRO
Reyes CORCÓSTEGUI VIVAR
Paloma Tato Cerdeiras
Original Assignee
Faes Farma, S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Faes Farma, S.A. filed Critical Faes Farma, S.A.
Publication of PL3827005T3 publication Critical patent/PL3827005T3/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
PL19742760.2T 2018-07-25 2019-07-24 Pirydopirymidyny jako inhibitory receptora histaminowego h4 PL3827005T3 (pl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP18382559 2018-07-25
PCT/EP2019/069905 WO2020020939A1 (en) 2018-07-25 2019-07-24 Pyridopyrimidines as histamine h4-receptor inhibitors

Publications (1)

Publication Number Publication Date
PL3827005T3 true PL3827005T3 (pl) 2022-11-28

Family

ID=63207688

Family Applications (1)

Application Number Title Priority Date Filing Date
PL19742760.2T PL3827005T3 (pl) 2018-07-25 2019-07-24 Pirydopirymidyny jako inhibitory receptora histaminowego h4

Country Status (29)

Country Link
US (1) US12492199B2 (pl)
EP (1) EP3827005B1 (pl)
JP (1) JP7093462B2 (pl)
KR (1) KR102603203B1 (pl)
CN (1) CN112739699B (pl)
AU (1) AU2019310889B2 (pl)
BR (1) BR112021001270A2 (pl)
CA (1) CA3107556C (pl)
CL (1) CL2021000184A1 (pl)
CO (1) CO2021001925A2 (pl)
DK (1) DK3827005T3 (pl)
EA (1) EA202190339A1 (pl)
EC (1) ECSP21010874A (pl)
ES (1) ES2929227T3 (pl)
HR (1) HRP20221250T1 (pl)
HU (1) HUE059824T2 (pl)
LT (1) LT3827005T (pl)
MA (1) MA53372B1 (pl)
MX (1) MX2021000966A (pl)
MY (1) MY206632A (pl)
PE (1) PE20211638A1 (pl)
PH (1) PH12021550143A1 (pl)
PL (1) PL3827005T3 (pl)
PT (1) PT3827005T (pl)
RS (1) RS63661B1 (pl)
SA (1) SA521421098B1 (pl)
SG (1) SG11202100575QA (pl)
WO (1) WO2020020939A1 (pl)
ZA (1) ZA202101092B (pl)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR102923602B1 (ko) * 2019-05-31 2026-02-06 키에시 파르마슈티시 엣스. 피. 에이. P2x3 억제제로서 피리도피리미딘 유도체
JP2023084709A (ja) * 2020-04-28 2023-06-20 Meiji Seikaファルマ株式会社 ヒスタミンh4受容体調節作用を有する新規二環化合物

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1789399A1 (en) 2004-08-31 2007-05-30 AstraZeneca AB Quinazolinone derivatives and their use as b-raf inhibitors
JP2008280341A (ja) 2007-04-12 2008-11-20 Sumitomo Chemical Co Ltd ヒドラジド化合物およびその防除用途
EP2077263A1 (en) 2008-01-02 2009-07-08 Vereniging voor christelijk hoger onderwijs, wetenschappelijk onderzoek en patiëntenzorg Quinazolines and related heterocyclic compounds and their therapeutic use
JP2012504157A (ja) * 2008-09-30 2012-02-16 アストラゼネカ アクチボラグ 複素環式jakキナーゼ阻害剤
US8481732B2 (en) 2009-03-20 2013-07-09 Incyte Corporation Substituted heterocyclic compounds
EP2270002A1 (en) 2009-06-18 2011-01-05 Vereniging voor Christelijk Hoger Onderwijs, Wetenschappelijk Onderzoek en Patiëntenzorg Quinazoline derivatives as histamine H4-receptor inhibitors for use in the treatment of inflammatory disorders
US20110319409A1 (en) 2010-06-23 2011-12-29 Cox Christopher D 7-aza-quinazoline pde10 inhibitors
WO2013060881A1 (en) 2011-10-27 2013-05-02 Vereniging Voor Christelijk Hoger Onderwijs, Wetenschappelijk Onderzoek En Patientenzorg Pyridopyrimidines and their therapeutic use
MX372736B (es) 2012-09-28 2020-06-19 Cancer Research Tech Ltd Inhibidores de azaquinazolina de la proteina quinasa c atipica.
EP3040334A1 (en) 2014-12-29 2016-07-06 Faes Farma, S.A. New benzimidazole derivatives as antihistamine agents
WO2018190778A1 (en) 2017-04-12 2018-10-18 Thammasat University Inspection procedure of the authenticity of brand-named leather bag

Also Published As

Publication number Publication date
KR20210038909A (ko) 2021-04-08
JP7093462B2 (ja) 2022-06-29
SA521421098B1 (ar) 2024-02-08
ES2929227T3 (es) 2022-11-25
CO2021001925A2 (es) 2021-03-08
AU2019310889B2 (en) 2022-03-31
EP3827005A1 (en) 2021-06-02
BR112021001270A2 (pt) 2021-04-20
PH12021550143A1 (en) 2021-09-13
MY206632A (en) 2024-12-27
PT3827005T (pt) 2022-11-04
JP2021531304A (ja) 2021-11-18
US12492199B2 (en) 2025-12-09
EA202190339A1 (ru) 2021-05-20
ECSP21010874A (es) 2021-03-31
LT3827005T (lt) 2022-11-10
US20210300922A1 (en) 2021-09-30
KR102603203B1 (ko) 2023-11-16
NZ773053A (en) 2023-10-27
RS63661B1 (sr) 2022-11-30
WO2020020939A1 (en) 2020-01-30
HRP20221250T1 (hr) 2022-12-09
CA3107556A1 (en) 2020-01-30
CN112739699B (zh) 2023-11-28
MX2021000966A (es) 2021-07-06
MA53372A (fr) 2021-06-02
AU2019310889A1 (en) 2021-03-11
HUE059824T2 (hu) 2023-01-28
ZA202101092B (en) 2022-09-28
SG11202100575QA (en) 2021-02-25
CN112739699A (zh) 2021-04-30
PE20211638A1 (es) 2021-08-24
EP3827005B1 (en) 2022-08-17
CA3107556C (en) 2022-10-25
CL2021000184A1 (es) 2021-07-09
DK3827005T3 (da) 2022-09-19
MA53372B1 (fr) 2022-10-31

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