PL398491A1 - Diazabicykliczny związek (cis)-3-(5,6-dichloro-3-pirydynylo)-3,6-diazabicyklo[3,2,0]-heptan, środek do leczenia i ich zastosowanie - Google Patents

Diazabicykliczny związek (cis)-3-(5,6-dichloro-3-pirydynylo)-3,6-diazabicyklo[3,2,0]-heptan, środek do leczenia i ich zastosowanie

Info

Publication number: PL398491A1
Authority: PL; Poland
Prior art keywords: diazabicyclo; pyridinyl; dichloro; heptane; cis
Prior art date: 2000-04-27

Application number

PL398491A

Other languages

English (en)

Inventor

Michael R. Schrimpf

Karin R. Tietje

Richard B. Toupence

Jianguo Ji

Anwer Basha

William H. Bunnelle

Jerome F. Daanen

Jennifer M. Pace

Kevin B. Sippy

Original Assignee

Abbott Laboratories

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-04-27

Filing date

2001-04-27

Publication date

2012-06-04

2001-04-12 Priority claimed from US09/833,914 external-priority patent/US6809105B2/en

2001-04-27 Application filed by Abbott Laboratories filed Critical Abbott Laboratories

2012-06-04 Publication of PL398491A1 publication Critical patent/PL398491A1/pl

Links

MBQYQLWSBRANKQ-IMTBSYHQSA-N (1s,5s)-3-(5,6-dichloropyridin-3-yl)-3,6-diazabicyclo[3.2.0]heptane Chemical compound N1=C(Cl)C(Cl)=CC(N2C[C@H]3NC[C@H]3C2)=C1 MBQYQLWSBRANKQ-IMTBSYHQSA-N 0.000 title 1
150000001875 compounds Chemical class 0.000 title 1
239000003814 drug Substances 0.000 title 1
229940124597 therapeutic agent Drugs 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Psychiatry (AREA)
Pain & Pain Management (AREA)
Psychology (AREA)
Addiction (AREA)
Hospice & Palliative Care (AREA)
Anesthesiology (AREA)
Urology & Nephrology (AREA)
Gynecology & Obstetrics (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

PL398491A 2000-04-27 2001-04-27 Diazabicykliczny związek (cis)-3-(5,6-dichloro-3-pirydynylo)-3,6-diazabicyklo[3,2,0]-heptan, środek do leczenia i ich zastosowanie PL398491A1 (pl)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US55994300A	2000-04-27	2000-04-27
US09/833,914 US6809105B2 (en)	2000-04-27	2001-04-12	Diazabicyclic central nervous system active agents

Publications (1)

Publication Number	Publication Date
PL398491A1 true PL398491A1 (pl)	2012-06-04

Family

ID=27072208

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
PL01358340A PL358340A1 (pl)	2000-04-27	2001-04-27	Diazabicykliczne środki aktywne wobec centralnegoukładu nerwowego
PL398491A PL398491A1 (pl)	2000-04-27	2001-04-27	Diazabicykliczny związek (cis)-3-(5,6-dichloro-3-pirydynylo)-3,6-diazabicyklo[3,2,0]-heptan, środek do leczenia i ich zastosowanie

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
PL01358340A PL358340A1 (pl)	2000-04-27	2001-04-27	Diazabicykliczne środki aktywne wobec centralnegoukładu nerwowego

Country Status (22)

Country	Link
EP (3)	EP2295437A1 (pl)
JP (2)	JP4981232B2 (pl)
KR (4)	KR100947188B1 (pl)
CN (3)	CN100430398C (pl)
AR (1)	AR030421A1 (pl)
AU (2)	AU6655901A (pl)
BG (2)	BG66151B1 (pl)
BR (1)	BR0107246A (pl)
CA (2)	CA2683045A1 (pl)
CZ (4)	CZ301324B6 (pl)
HK (1)	HK1054375A1 (pl)
HU (1)	HUP0300602A3 (pl)
IL (3)	IL152231A0 (pl)
MX (1)	MXPA02010594A (pl)
MY (3)	MY145722A (pl)
NO (1)	NO324250B1 (pl)
NZ (1)	NZ521734A (pl)
PE (1)	PE20011305A1 (pl)
PL (2)	PL358340A1 (pl)
SK (2)	SK287273B6 (pl)
TW (4)	TWI357903B (pl)
WO (1)	WO2001081347A2 (pl)

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2001
- 2001-04-26 MY MYPI20055633A patent/MY145722A/en unknown
- 2001-04-26 MY MYPI20011984A patent/MY137020A/en unknown
- 2001-04-27 KR KR1020097021390A patent/KR100947188B1/ko not_active Expired - Fee Related
- 2001-04-27 AR ARP010101990A patent/AR030421A1/es active IP Right Grant
- 2001-04-27 KR KR1020027014385A patent/KR100899950B1/ko not_active Expired - Fee Related
- 2001-04-27 SK SK1681-2002A patent/SK287273B6/sk not_active IP Right Cessation
- 2001-04-27 CZ CZ20023765A patent/CZ301324B6/cs not_active IP Right Cessation
- 2001-04-27 HU HU0300602A patent/HUP0300602A3/hu unknown
- 2001-04-27 EP EP10177411A patent/EP2295437A1/en not_active Withdrawn
- 2001-04-27 MX MXPA02010594A patent/MXPA02010594A/es active IP Right Grant
- 2001-04-27 CZ CZ20080677A patent/CZ302072B6/cs not_active IP Right Cessation
- 2001-04-27 CN CNB018117112A patent/CN100430398C/zh not_active Expired - Fee Related
- 2001-04-27 PL PL01358340A patent/PL358340A1/pl unknown
- 2001-04-27 SK SK10-2010A patent/SK287658B6/sk not_active IP Right Cessation
- 2001-04-27 AU AU6655901A patent/AU6655901A/xx active Pending
- 2001-04-27 KR KR1020097010331A patent/KR100947187B1/ko not_active Expired - Fee Related
- 2001-04-27 CA CA002683045A patent/CA2683045A1/en not_active Abandoned
- 2001-04-27 JP JP2001578437A patent/JP4981232B2/ja not_active Expired - Fee Related
- 2001-04-27 CA CA002407094A patent/CA2407094C/en not_active Expired - Fee Related
- 2001-04-27 KR KR1020087031655A patent/KR100961406B1/ko not_active Expired - Fee Related
- 2001-04-27 PL PL398491A patent/PL398491A1/pl unknown
- 2001-04-27 PE PE2001000385A patent/PE20011305A1/es not_active Application Discontinuation
- 2001-04-27 CN CN2010102450796A patent/CN101935322A/zh active Pending
- 2001-04-27 EP EP01944118A patent/EP1284976A2/en not_active Withdrawn
- 2001-04-27 HK HK03104885.7A patent/HK1054375A1/zh unknown
- 2001-04-27 IL IL15223101A patent/IL152231A0/xx not_active IP Right Cessation
- 2001-04-27 BR BR0107246-3A patent/BR0107246A/pt not_active IP Right Cessation
- 2001-04-27 WO PCT/US2001/013798 patent/WO2001081347A2/en not_active Ceased
- 2001-04-27 CN CN2012103509141A patent/CN102863441A/zh active Pending
- 2001-04-27 AU AU2001266559A patent/AU2001266559C1/en not_active Ceased
- 2001-04-27 CZ CZ20090553A patent/CZ302038B6/cs not_active IP Right Cessation
- 2001-04-27 EP EP10177450A patent/EP2298775A1/en not_active Withdrawn
- 2001-04-27 NZ NZ521734A patent/NZ521734A/en not_active IP Right Cessation
- 2001-04-27 CZ CZ20100538A patent/CZ302795B6/cs not_active IP Right Cessation
- 2001-05-22 TW TW097145362A patent/TWI357903B/zh not_active IP Right Cessation
- 2001-05-22 TW TW095100404A patent/TWI323733B/zh not_active IP Right Cessation
- 2001-05-22 TW TW100130949A patent/TW201141871A/zh unknown
- 2001-05-22 TW TW090110172A patent/TWI311137B/zh not_active IP Right Cessation
2002
- 2002-10-24 NO NO20025107A patent/NO324250B1/no not_active IP Right Cessation
- 2002-11-21 BG BG107303A patent/BG66151B1/bg unknown
2005
- 2005-03-07 MY MYPI20094589A patent/MY168244A/en unknown
2006
- 2006-08-06 IL IL177316A patent/IL177316A/en not_active IP Right Cessation
2009
- 2009-12-29 IL IL203035A patent/IL203035A/en not_active IP Right Cessation
2010
- 2010-03-17 BG BG110620A patent/BG110620A/bg unknown
2011
- 2011-09-15 JP JP2011202172A patent/JP2012041349A/ja not_active Withdrawn

Also Published As

Publication number	Publication date
BR0107246A (pt)	2002-10-01
KR20090121385A (ko)	2009-11-25
MY145722A (en)	2012-03-30
NO20025107D0 (no)	2002-10-24
CA2683045A1 (en)	2001-11-01
NO20025107L (no)	2002-12-19
TWI311137B (en)	2009-06-21
HUP0300602A2 (hu)	2003-06-28
AR030421A1 (es)	2003-08-20
BG107303A (bg)	2003-07-31
MY137020A (en)	2008-12-31
IL152231A0 (en)	2003-05-29
CZ20023765A3 (cs)	2003-02-12
EP1284976A2 (en)	2003-02-26
CN101935322A (zh)	2011-01-05
KR20090071654A (ko)	2009-07-01
AU2001266559B2 (en)	2005-03-03
KR20020093955A (ko)	2002-12-16
BG66151B1 (bg)	2011-08-31
HK1054375A1 (zh)	2003-11-28
TW200617013A (en)	2006-06-01
NZ521734A (en)	2004-10-29
MY168244A (en)	2018-10-15
BG110620A (bg)	2010-07-30
AU2001266559C1 (en)	2005-11-17
IL177316A0 (en)	2006-12-10
TWI357903B (en)	2012-02-11
JP2012041349A (ja)	2012-03-01
TWI323733B (en)	2010-04-21
NO324250B1 (no)	2007-09-17
JP4981232B2 (ja)	2012-07-18
IL203035A (en)	2010-12-30
IL177316A (en)	2010-06-30
KR100899950B1 (ko)	2009-05-28
EP2295437A1 (en)	2011-03-16
KR100947187B1 (ko)	2010-03-12
TW200909432A (en)	2009-03-01
CN1440410A (zh)	2003-09-03
KR20090013833A (ko)	2009-02-05
SK16812002A3 (sk)	2003-04-01
CN100430398C (zh)	2008-11-05
SK287658B6 (sk)	2011-05-06
KR100961406B1 (ko)	2010-06-09
CZ302072B6 (cs)	2010-09-29
TW201141871A (en)	2011-12-01
CZ302795B6 (cs)	2011-11-16
MXPA02010594A (es)	2003-05-14
EP2298775A1 (en)	2011-03-23
KR100947188B1 (ko)	2010-03-12
WO2001081347A3 (en)	2002-01-31
AU6655901A (en)	2001-11-07
WO2001081347A2 (en)	2001-11-01
CN102863441A (zh)	2013-01-09
JP2003531210A (ja)	2003-10-21
CA2407094A1 (en)	2001-11-01
SK287273B6 (sk)	2010-05-07
CZ301324B6 (cs)	2010-01-13
PE20011305A1 (es)	2001-12-31
HUP0300602A3 (en)	2005-12-28
PL358340A1 (pl)	2004-08-09
CZ302038B6 (cs)	2010-09-15
CA2407094C (en)	2009-11-17

Legal Events

Date	Code	Title	Description
2014-06-30	DISC	Decisions on discontinuance of the proceedings (taken after the publication of the particulars of the applications)

Publication	Publication Date	Title
MXPA02002898A (es)	2003-10-14	Pirazolopirimidinas como agentes terapeuticos.
ZA200306886B (en)	2004-07-16	Pyrazolopyrimidines as therapeutic agents.
IL150022A0 (en)	2002-12-01	Imidazo [1,3,5] triazinones and the use thereof
AU1393000A (en)	2000-06-26	1,4-diazabicyclo(3.2.2)nonane derivatives, their preparation and therapeutic application
IL157640A0 (en)	2004-03-28	Pyrazolopyrimidines as therapeutic agents
IL152231A0 (en)	2003-05-29	Diazabicyclic central nervous system active agents
ZA200202519B (en)	2004-01-28	Certain alkylene diamine-substituted pyrazolo[1,5,-a]-1,5-pyrimidines and pyrazolo[1,5-a]-1,3,5-triazines.
GB0027561D0 (en)	2000-12-27	Therapeutic agents
AU2001235595A1 (en)	2001-08-07	4-heteroaryl-1,4-diazabicyclo(3.2.2)nonane, preparation and therapeutic use thereof
PL349341A1 (en)	2002-07-15	Imidazo[4,5-c]-pyridine-4-on-derivatives
PL349364A1 (en)	2002-07-15	Use of pyridazino[4,5-b
MXPA03008894A (es)	2003-12-08	Uso de compuestos de imidazo[1,2-a]-piridin-3-il-amidas e imidazo [1,2-a]-piridin-3-il-aminas sustituidas como medicamentos.
ZA200110046B (en)	2003-03-06	Therapeutic agents.
ZA200109120B (en)	2003-11-13	Use of Arylalkanoylpyridazines.
GB2334672B (en)	2000-07-19	The Allenderry chair
SI1212327T1 (en)	2004-02-29	Pyrazolopyrimidines as therapeutic agents
ZA99132B (en)	2000-07-10	Therapeutic agents.
ZA200204584B (en)	2004-06-30	Therapeutic agents.
PL352760A1 (pl)	2003-09-08	Oksatiepino [6,5-b] dihydropirydyny, zawierające je kompozycje oraz sposoby wytwarzania
GB9920599D0 (en)	1999-11-03	The body seat
TW398311U (en)	2000-07-11	Illuminant inter-hit balls
TW386454U (en)	2000-04-01	The fitness equipment for sit/lie dual use
TW407477U (en)	2000-10-01	Multi-purpose chair structure
TW343509U (en)	1998-10-21	Multi-purpose cup
GB9910914D0 (en)	1999-07-07	The chair