PL429346A1 - (+)-rel-(1R,6R,1'R)-1-(1'-Bromoethyl)-9-oxabicyclo[4.3.0]nonan-8-one and method of obtaining (+)-rel-(1R,6R,1'R)-1-(1'-bromoethyl)-9-oxabicyclo[4.3.0]nonan-8-one - Google Patents
(+)-rel-(1R,6R,1'R)-1-(1'-Bromoethyl)-9-oxabicyclo[4.3.0]nonan-8-one and method of obtaining (+)-rel-(1R,6R,1'R)-1-(1'-bromoethyl)-9-oxabicyclo[4.3.0]nonan-8-oneInfo
- Publication number
- PL429346A1 PL429346A1 PL429346A PL42934619A PL429346A1 PL 429346 A1 PL429346 A1 PL 429346A1 PL 429346 A PL429346 A PL 429346A PL 42934619 A PL42934619 A PL 42934619A PL 429346 A1 PL429346 A1 PL 429346A1
- Authority
- PL
- Poland
- Prior art keywords
- nonan
- oxabicyclo
- bromoethyl
- rel
- obtaining
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 2
- CZLBIUWPNOXWTQ-UHFFFAOYSA-N CC=C1CCCCC1CC(O)=O Chemical compound CC=C1CCCCC1CC(O)=O CZLBIUWPNOXWTQ-UHFFFAOYSA-N 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- 238000010722 bromolactonization reaction Methods 0.000 abstract 1
- 238000004440 column chromatography Methods 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
Landscapes
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Abstract
Przedmiotem zgłoszenia jest związek o nazwie: (+)-rel-(1R,6R,1'R)-1-(1'-Bromoetylo)-9-oksabicyklo[4.3.0]nonan-8-on o wzorze 2, przedstawionym na rysunku. Zgłoszenie obejmuje też sposób otrzymywania(+)-rel-(1R,6R,1'R)-1-(1'-bromoetylo)-9-oksabicyklo[4.3.0]nonan-8-onu, polegający na tym, że kwas (+)-(2'-etylideno-cykloheksylo)octowy o wzorze 1 poddaje się reakcji bromolaktonizacji w której otrzymuje się (+)-rel-(1R,6R,1'R)-1-(1'-Bromoetylo)-9-oksabicyklo[4.3.0]nonan-8-on o wzorze 2, który oczyszcza się metodą chromatografii kolumnowej.The subject of the application is a compound named: (+) - rel- (1R, 6R, 1'R) -1- (1'-Bromoethyl) -9-oxabicyclo [4.3.0] nonan-8-one of the formula 2, shown in the drawing. The application also covers a method for the preparation of (+) - rel- (1R, 6R, 1'R) -1- (1'-bromoethyl) -9-oxabicyclo [4.3.0] nonan-8-one, which consists in the fact that the acid The (+) - (2'-ethylidene-cyclohexyl) acetic acid of formula 1 is subjected to a bromolactonization reaction to obtain (+) - rel- (1R, 6R, 1'R) -1- (1'-Bromoethyl) -9 -oxabicyclo [4.3.0] nonan-8-one of formula 2 which is purified by column chromatography.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PL429346(22)20190321A PL238102B1 (en) | 2019-03-21 | 2019-03-21 | (+)-rel-(1R,6R,1'R)-1-(1'-Bromoethyl)-9-oxabicyclo[4.3.0]nonan-8-one and method of obtaining (+)-rel-(1R,6R,1'R)-1-(1'-bromoethyl)-9-oxabicyclo[4.3.0]nonan-8-one |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PL429346(22)20190321A PL238102B1 (en) | 2019-03-21 | 2019-03-21 | (+)-rel-(1R,6R,1'R)-1-(1'-Bromoethyl)-9-oxabicyclo[4.3.0]nonan-8-one and method of obtaining (+)-rel-(1R,6R,1'R)-1-(1'-bromoethyl)-9-oxabicyclo[4.3.0]nonan-8-one |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PL429346A1 true PL429346A1 (en) | 2020-10-05 |
| PL238102B1 PL238102B1 (en) | 2021-07-05 |
Family
ID=72669270
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL429346(22)20190321A PL238102B1 (en) | 2019-03-21 | 2019-03-21 | (+)-rel-(1R,6R,1'R)-1-(1'-Bromoethyl)-9-oxabicyclo[4.3.0]nonan-8-one and method of obtaining (+)-rel-(1R,6R,1'R)-1-(1'-bromoethyl)-9-oxabicyclo[4.3.0]nonan-8-one |
Country Status (1)
| Country | Link |
|---|---|
| PL (1) | PL238102B1 (en) |
-
2019
- 2019-03-21 PL PL429346(22)20190321A patent/PL238102B1/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| PL238102B1 (en) | 2021-07-05 |
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