PT1002792E - Compostos de 2-aminopropano-1,3-diol, sua utilizacao medicinal e intermediariosda sintese dos mesmos - Google Patents

Compostos de 2-aminopropano-1,3-diol, sua utilizacao medicinal e intermediariosda sintese dos mesmos

Info

Publication number
PT1002792E
PT1002792E PT98911211T PT98911211T PT1002792E PT 1002792 E PT1002792 E PT 1002792E PT 98911211 T PT98911211 T PT 98911211T PT 98911211 T PT98911211 T PT 98911211T PT 1002792 E PT1002792 E PT 1002792E
Authority
PT
Portugal
Prior art keywords
compound
same
diole
aminopropane
medicinal
Prior art date
Application number
PT98911211T
Other languages
English (en)
Inventor
Tetsuro Fujita
Kunitomo Adachi
Koji Teshima
Yoshiyuki Aoki
Tokushi Hanano
Yukio Hoshino
Original Assignee
Mitsubishi Pharma Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mitsubishi Pharma Corp filed Critical Mitsubishi Pharma Corp
Publication of PT1002792E publication Critical patent/PT1002792E/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/01—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms
    • C07C255/16—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms containing cyano groups and singly-bound oxygen atoms bound to the same carbon atom of an acyclic carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C225/00—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones
    • C07C225/02—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C225/14—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being unsaturated
    • C07C225/16—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being unsaturated and containing six-membered aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C215/00—Compounds containing amino and hydroxy groups bound to the same carbon skeleton
    • C07C215/02—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C215/22—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated
    • C07C215/28—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated and containing six-membered aromatic rings
    • C07C215/34—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated and containing six-membered aromatic rings containing hydroxy groups and carbon atoms of six-membered aromatic rings bound to the same carbon atom of the carbon skeleton and at least one hydroxy group bound to another carbon atom of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C223/00—Compounds containing amino and —CHO groups bound to the same carbon skeleton
    • C07C223/02—Compounds containing amino and —CHO groups bound to the same carbon skeleton having amino groups bound to acyclic carbon atoms of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804—Compounds having Si-O-C linkages

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pulmonology (AREA)
  • Transplantation (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
PT98911211T 1997-04-04 1998-04-03 Compostos de 2-aminopropano-1,3-diol, sua utilizacao medicinal e intermediariosda sintese dos mesmos PT1002792E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP8625597 1997-04-04

Publications (1)

Publication Number Publication Date
PT1002792E true PT1002792E (pt) 2004-12-31

Family

ID=13881722

Family Applications (2)

Application Number Title Priority Date Filing Date
PT98911211T PT1002792E (pt) 1997-04-04 1998-04-03 Compostos de 2-aminopropano-1,3-diol, sua utilizacao medicinal e intermediariosda sintese dos mesmos
PT03003623T PT1319651E (pt) 1997-04-04 1998-04-03 Composto 2-aminopropano-1,3-diol, sua utilizacao farmaceutica e seus intermediarios sinteticos

Family Applications After (1)

Application Number Title Priority Date Filing Date
PT03003623T PT1319651E (pt) 1997-04-04 1998-04-03 Composto 2-aminopropano-1,3-diol, sua utilizacao farmaceutica e seus intermediarios sinteticos

Country Status (18)

Country Link
US (2) USRE39072E1 (pt)
EP (2) EP1002792B1 (pt)
JP (1) JP4045364B2 (pt)
KR (1) KR100551931B1 (pt)
CN (2) CN1290819C (pt)
AT (2) ATE271028T1 (pt)
AU (1) AU735853B2 (pt)
BR (1) BR9808481A (pt)
CA (1) CA2286315C (pt)
DE (2) DE69830756T2 (pt)
DK (2) DK1319651T3 (pt)
ES (2) ES2226110T3 (pt)
IL (3) IL155065A (pt)
NZ (1) NZ500713A (pt)
PT (2) PT1002792E (pt)
RU (1) RU2198162C2 (pt)
SI (2) SI1002792T1 (pt)
WO (1) WO1998045249A1 (pt)

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CA2483594C (en) 2002-05-16 2011-02-15 Novartis Ag Use of edg receptor binding agents in cancer
GB0217152D0 (en) 2002-07-24 2002-09-04 Novartis Ag Organic compounds
AU2003273865A1 (en) * 2002-09-13 2004-04-30 Novartis Ag Amino-propanol derivatives
MXPA05003254A (es) * 2002-09-24 2005-06-08 Novartis Ag Agonistas del receptor de esfingosina-1-fosfato en el tratamiento de trastornos de desmielinacion.
RU2229290C1 (ru) * 2003-02-19 2004-05-27 Государственное образовательное учреждение высшего профессионального образования Московская медицинская академия им. И.М. Сеченова Применение бисопролола в качестве антицитокинового средства
DE202004021680U1 (de) * 2003-04-08 2010-04-22 Novartis Ag Feste pharmazeutische Zusammensetzung
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US7524887B2 (en) 2003-06-06 2009-04-28 Sanofi-Aventis Deutschland Gmbh 2-amino-1,3-propanediol compounds for the treatment of acute pain
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TWI355934B (en) 2004-02-24 2012-01-11 Sankyo Co Pharmaceutical composition for treatment or prophy
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JP4919374B2 (ja) * 2004-07-29 2012-04-18 第一三共株式会社 免疫抑制剤としての医薬組成物
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Also Published As

Publication number Publication date
CA2286315C (en) 2007-03-06
RU2198162C2 (ru) 2003-02-10
DE69830756D1 (de) 2005-08-04
KR100551931B1 (ko) 2006-02-16
IL155065A (en) 2004-01-04
AU735853B2 (en) 2001-07-19
DK1319651T3 (da) 2005-08-01
US6214873B1 (en) 2001-04-10
IL155065A0 (en) 2003-10-31
ES2226110T3 (es) 2005-03-16
DE69830756T2 (de) 2006-05-04
ATE298740T1 (de) 2005-07-15
SI1002792T1 (en) 2004-12-31
CN1259117A (zh) 2000-07-05
EP1002792A1 (en) 2000-05-24
IL155066A (en) 2004-06-20
DK1002792T3 (da) 2004-11-22
EP1319651A3 (en) 2004-01-02
CN1480450A (zh) 2004-03-10
EP1002792A4 (en) 2002-03-20
AU6523098A (en) 1998-10-30
BR9808481A (pt) 2000-05-23
DE69825056T2 (de) 2005-08-25
USRE39072E1 (en) 2006-04-18
WO1998045249A1 (en) 1998-10-15
ATE271028T1 (de) 2004-07-15
CN1290819C (zh) 2006-12-20
EP1319651A2 (en) 2003-06-18
CA2286315A1 (en) 1998-10-15
SI1319651T1 (en) 2005-10-31
EP1319651B1 (en) 2005-06-29
ES2240868T3 (es) 2005-10-16
IL155066A0 (en) 2003-10-31
IL132208A0 (en) 2001-03-19
JP4045364B2 (ja) 2008-02-13
CN1137086C (zh) 2004-02-04
IL132208A (en) 2003-07-31
KR20010006004A (ko) 2001-01-15
DE69825056D1 (de) 2004-08-19
EP1002792B1 (en) 2004-07-14
NZ500713A (en) 2000-07-28
PT1319651E (pt) 2005-09-30

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