PT100329A - Composicoes a base de di-hidro-4-(3,5-di-terc-butil-4-hidroxi-benzilideno)-metil-2h-1,2-oxazin-3(4h)-ona sob forma micronizada - Google Patents
Composicoes a base de di-hidro-4-(3,5-di-terc-butil-4-hidroxi-benzilideno)-metil-2h-1,2-oxazin-3(4h)-ona sob forma micronizadaInfo
- Publication number
- PT100329A PT100329A PT100329A PT10032992A PT100329A PT 100329 A PT100329 A PT 100329A PT 100329 A PT100329 A PT 100329A PT 10032992 A PT10032992 A PT 10032992A PT 100329 A PT100329 A PT 100329A
- Authority
- PT
- Portugal
- Prior art keywords
- micronized
- terc
- oxazin
- benzylidene
- hydro
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title abstract 2
- 239000004480 active ingredient Substances 0.000 abstract 1
- 230000003110 anti-inflammatory effect Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
- A61K9/145—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
Landscapes
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
- Cosmetics (AREA)
- Lubricants (AREA)
- Compositions Of Macromolecular Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US07/680,997 US5271944A (en) | 1991-04-05 | 1991-04-05 | Pharmacologically enhanced formulations |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PT100329A true PT100329A (pt) | 1993-07-30 |
| PT100329B PT100329B (pt) | 1999-06-30 |
Family
ID=24733350
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT100329A PT100329B (pt) | 1991-04-05 | 1992-04-01 | Composicoes a base de di-hidro-4-(3,5-di-terc-butil-4-hidroxi-benzilideno)-metil-2h-1,2-oxazin-3(4h)-ona sob forma micronizada |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US5271944A (pt) |
| EP (1) | EP0599914B1 (pt) |
| AT (1) | ATE155687T1 (pt) |
| AU (1) | AU1876792A (pt) |
| CA (1) | CA2052901C (pt) |
| CH (1) | CH683824A5 (pt) |
| DE (1) | DE69221150T2 (pt) |
| DK (1) | DK0599914T3 (pt) |
| ES (1) | ES2108130T3 (pt) |
| FR (1) | FR2674754B1 (pt) |
| IE (1) | IE74211B1 (pt) |
| IT (1) | ITTO920303A1 (pt) |
| NZ (1) | NZ242233A (pt) |
| PT (1) | PT100329B (pt) |
| WO (1) | WO1992017163A1 (pt) |
| ZA (1) | ZA922482B (pt) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2684298B1 (fr) * | 1991-12-03 | 1994-03-11 | Rhone Poulenc Rorer Sa | Nouvelles compositions pharmaceutiques solides a base de derives de lapiperidine substitues en 1,4. |
| AU701042B2 (en) * | 1995-02-28 | 1999-01-21 | Aventisub Llc | Pharmaceutical composition for piperidinoalkanol compounds |
| KR100514264B1 (ko) * | 1997-08-26 | 2005-09-15 | 아벤티스 파마슈티칼스 인크. | 피페리디노알칸올-충혈완화제 조합용 제약 조성물 |
| AU5721301A (en) * | 2000-04-24 | 2001-11-07 | Teva Pharma | Zolpidem hemitartrate |
| EP1604663A1 (en) | 2000-04-24 | 2005-12-14 | Teva Pharmaceutical Industries Ltd | Zolpidem Hemitartrate Form H Solvate |
| AU2002244247B2 (en) | 2001-03-01 | 2007-12-13 | Harbor Biosciences, Inc. | Use of certain steroids for treatment of blood cell deficiencies |
| US20060280761A1 (en) * | 2002-03-11 | 2006-12-14 | Health Plus International, Inc. | Nanofluidized B-12 composition and process for treating pernicious anemia |
| US6861066B2 (en) | 2002-03-11 | 2005-03-01 | Health Plus International Inc. | Method for the delivery of a biologically active agent |
| BE1015641A4 (fr) * | 2003-05-26 | 2005-07-05 | Mariani Jean Paul | Micronisation 70. |
| CA2542499A1 (en) * | 2003-10-16 | 2005-04-28 | Teva Pharmaceutical Industries Ltd. | Preparation of candesartan cilexetil |
| CA2552003A1 (en) * | 2004-01-05 | 2005-07-28 | Teva Pharmaceutical Industries Ltd. | Methods for the production of sildenafil base and citrate salt |
| EP1713795A2 (en) * | 2004-02-11 | 2006-10-25 | Teva Pharmaceutical Industries Ltd. | Candesartan cilexetil polymorphs |
| AU2005330504B2 (en) | 2004-09-29 | 2010-10-28 | Harbor Biosciences, Inc. | Steroid analogs and characterization and treatment methods |
| EP2273994B1 (en) | 2008-04-03 | 2015-12-02 | NeurMedix, Inc. | Solid state forms of a pharmaceutical |
| TW201613888A (en) * | 2014-09-26 | 2016-04-16 | Helsinn Healthcare Sa | Crystalline forms of an NK-1 antagonist |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3033919A1 (de) * | 1980-09-09 | 1982-04-22 | Bayer Ag, 5090 Leverkusen | Feste arzneizubereitungen enthaltend nifedipin und verfahren zu ihrer herstellung |
| DE3204126A1 (de) * | 1982-02-06 | 1983-08-11 | Bayer Ag, 5090 Leverkusen | Pyrazoloxazine, -thiazine, -chinoline, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel |
| IT1187751B (it) * | 1985-10-15 | 1987-12-23 | Eurand Spa | Procedimento per la preparazione di formulazioni solidi di nifedipina ad elevata biodisponibilita' e ad effetto prolungato e formulazioni cosi' ottenute |
| US4912093A (en) * | 1986-10-01 | 1990-03-27 | Marion Laboratories, Inc. | Use of synthetic sulfated saccharides to enhance wound healing |
| DE3723327A1 (de) * | 1987-07-15 | 1989-02-02 | Hoechst Ag | Substituierte thienoimidazol-derivate, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische zubereitungen und ihre verwendung als magensaeuresekretionshemmer, magenschutzmittel sowie als medikament gegen intestinale entzuendungen |
| US4892870A (en) * | 1988-08-01 | 1990-01-09 | Biofor, Ltd. | Oxaza heterocycles and pharmaceutical compositions containing same |
-
1991
- 1991-04-05 US US07/680,997 patent/US5271944A/en not_active Expired - Fee Related
- 1991-10-07 CA CA002052901A patent/CA2052901C/en not_active Expired - Fee Related
-
1992
- 1992-03-31 DK DK92917294.8T patent/DK0599914T3/da active
- 1992-03-31 AU AU18767/92A patent/AU1876792A/en not_active Abandoned
- 1992-03-31 AT AT92917294T patent/ATE155687T1/de not_active IP Right Cessation
- 1992-03-31 ES ES92917294T patent/ES2108130T3/es not_active Expired - Lifetime
- 1992-03-31 EP EP92917294A patent/EP0599914B1/en not_active Expired - Lifetime
- 1992-03-31 WO PCT/US1992/002436 patent/WO1992017163A1/en not_active Ceased
- 1992-03-31 DE DE69221150T patent/DE69221150T2/de not_active Expired - Fee Related
- 1992-04-01 PT PT100329A patent/PT100329B/pt not_active IP Right Cessation
- 1992-04-02 IE IE921040A patent/IE74211B1/en not_active IP Right Cessation
- 1992-04-02 IT IT92TO000303A patent/ITTO920303A1/it not_active Application Discontinuation
- 1992-04-03 NZ NZ242233A patent/NZ242233A/xx unknown
- 1992-04-03 ZA ZA922482A patent/ZA922482B/xx unknown
- 1992-04-03 FR FR9204122A patent/FR2674754B1/fr not_active Expired - Fee Related
- 1992-04-06 CH CH1108/92A patent/CH683824A5/de not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| FR2674754A1 (fr) | 1992-10-09 |
| DK0599914T3 (da) | 1998-03-02 |
| ZA922482B (en) | 1992-12-30 |
| PT100329B (pt) | 1999-06-30 |
| EP0599914A4 (en) | 1994-08-24 |
| ITTO920303A0 (it) | 1992-04-02 |
| ATE155687T1 (de) | 1997-08-15 |
| CA2052901C (en) | 1997-12-23 |
| WO1992017163A1 (en) | 1992-10-15 |
| US5271944A (en) | 1993-12-21 |
| EP0599914A1 (en) | 1994-06-08 |
| DE69221150T2 (de) | 1998-02-26 |
| NZ242233A (en) | 1993-07-27 |
| IE74211B1 (en) | 1997-07-16 |
| ES2108130T3 (es) | 1997-12-16 |
| DE69221150D1 (de) | 1997-09-04 |
| CH683824A5 (de) | 1994-05-31 |
| IE921040A1 (en) | 1992-10-07 |
| ITTO920303A1 (it) | 1993-10-02 |
| AU1876792A (en) | 1992-11-02 |
| EP0599914B1 (en) | 1997-07-23 |
| CA2052901A1 (en) | 1992-10-06 |
| FR2674754B1 (fr) | 1994-01-14 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| BB1A | Laying open of patent application |
Effective date: 19930303 |
|
| FG3A | Patent granted, date of granting |
Effective date: 19990329 |
|
| MM3A | Annulment or lapse |
Free format text: LAPSE DUE TO NON-PAYMENT OF FEES Effective date: 20010930 |