PT100672A - Processo para a preparacao de intermediarios de sertralina e compostos assim obtidos - Google Patents

Processo para a preparacao de intermediarios de sertralina e compostos assim obtidos

Info

Publication number: PT100672A
Authority: PT; Portugal
Prior art keywords: preparation; pct; sertraline; compounds; intermediaries
Prior art date: 1991-07-11

Application number

PT100672A

Other languages

English (en)

Other versions

PT100672B (pt

Inventor

Michael Trevelyan Williams

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1991-07-11

Filing date

1992-07-09

Publication date

1993-09-30

1992-07-09 Application filed by Pfizer filed Critical Pfizer

1993-09-30 Publication of PT100672A publication Critical patent/PT100672A/pt

1999-06-30 Publication of PT100672B publication Critical patent/PT100672B/pt

Links

150000001875 compounds Chemical class 0.000 title abstract 4
238000000034 method Methods 0.000 title abstract 2
229960002073 sertraline Drugs 0.000 title abstract 2
VGKDLMBJGBXTGI-SJCJKPOMSA-N sertraline Chemical compound C1([C@@H]2CC[C@@H](C3=CC=CC=C32)NC)=CC=C(Cl)C(Cl)=C1 VGKDLMBJGBXTGI-SJCJKPOMSA-N 0.000 title abstract 2
125000004178 (C1-C4) alkyl group Chemical group 0.000 abstract 1
239000000935 antidepressant agent Substances 0.000 abstract 1
239000000543 intermediate Substances 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C233/00—Carboxylic acid amides
- C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C233/12—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by halogen atoms or by nitro or nitroso groups
- C07C233/14—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by halogen atoms or by nitro or nitroso groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by a carbon atom of a ring other than a six-membered aromatic ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2602/00—Systems containing two condensed rings
- C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
- C07C2602/04—One of the condensed rings being a six-membered aromatic ring
- C07C2602/10—One of the condensed rings being a six-membered aromatic ring the other ring being six-membered, e.g. tetraline

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Epoxy Compounds (AREA)

PT100672A 1991-07-11 1992-07-09 Processo para a preparacao de intermediarios de sertralina e compostos assim obtidos PT100672B (pt)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GB919114947A GB9114947D0 (en)	1991-07-11	1991-07-11	Process for preparing sertraline

Publications (2)

Publication Number	Publication Date
PT100672A true PT100672A (pt)	1993-09-30
PT100672B PT100672B (pt)	1999-06-30

Family

ID=10698170

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PT100672A PT100672B (pt)	1991-07-11	1992-07-09	Processo para a preparacao de intermediarios de sertralina e compostos assim obtidos

Country Status (14)

Country	Link
US (1)	US5463126A (pt)
EP (1)	EP0594666B1 (pt)
JP (1)	JP2566374B2 (pt)
AT (1)	ATE127779T1 (pt)
CA (1)	CA2109817C (pt)
DE (1)	DE69204840T2 (pt)
DK (1)	DK0594666T3 (pt)
ES (1)	ES2078749T3 (pt)
FI (1)	FI112210B (pt)
GB (1)	GB9114947D0 (pt)
GR (1)	GR3017766T3 (pt)
IE (1)	IE67822B1 (pt)
PT (1)	PT100672B (pt)
WO (1)	WO1993001162A1 (pt)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2777000B1 (fr) *	1998-04-01	2002-09-27	Catalys	Procede de preparation de la sertraline racemique
IL132500A0 (en)	1998-10-29	2001-03-19	Pfizer Prod Inc	Stereoselective microbial reduction of a racemic tetralone
JP2002531427A (ja) *	1998-11-27	2002-09-24	テバファーマシューティカルインダストリーズリミティド	セルトラリン塩酸塩多形体
US6500987B1 (en)	1998-11-27	2002-12-31	Teva Pharmaceutical Industries Ltd.	Sertraline hydrochloride polymorphs
RU2161851C1 (ru) *	1999-05-24	2001-01-10	Научно-производственное внедренческое предприятие "Феррогидродинамика"	Электрическая машина
US6495721B1 (en) *	1999-08-09	2002-12-17	Teva Pharmaceutical Industries Ltd.	Sertraline hydrochloride Form II and methods for the preparation thereof
TWI260315B (en) *	1999-10-29	2006-08-21	Ciba Sc Holding Ag	Polymorphic forms of sertraline hydrochloride
US7442838B2 (en) *	1999-10-29	2008-10-28	Ciba Specialty Chemicals Corp.	Polymorphic forms of sertraline hydrochloride
US20050119351A1 (en) *	1999-10-29	2005-06-02	Van Der Schaaf Paul A.	Polymorphic forms of sertraline hydrochloride
PL356452A1 (en) *	1999-12-21	2004-06-28	Teva Pharmaceutical Industries Ltd.	Novel sertraline hydrochloride polymorphs, processes for preparing them, compositions containing them and methods of using them
IL151691A0 (en)	2000-03-14	2003-04-10	Teva Pharma	Novel process for preparing (+)-cis-sertraline
US6720003B2 (en) *	2001-02-16	2004-04-13	Andrx Corporation	Serotonin reuptake inhibitor formulations
WO2003093217A1 (en) *	2002-04-29	2003-11-13	Teva Pharmaceutical Industries Ltd.	Process for preparation of polymorphic form ii of sertraline hydrochloride, pharmaceutical formulations and methods of administration thereof
US20060014838A1 (en) *	2004-07-14	2006-01-19	Sudhakar Valluri	Process for converting trans-sertraline to cis-sertraline
WO2025046526A1 (ko) *	2023-09-01	2025-03-06	환인제약 주식회사	설트랄린 또는 이의 염을 포함하는 약학적 조성물

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4269870A (en) *	1974-05-13	1981-05-26	Cooper Industries, Inc.	Solder flux and method
US4071489A (en) *	1976-03-08	1978-01-31	Rohm And Haas Company	Coating compositions from dicyclopentenyl acrylate and/or methacrylate
JPS5592293A (en) *	1978-12-28	1980-07-12	Sanwa Kagaku Kogyo Kk	Solid flux for soldering
US4536518A (en) *	1979-11-01	1985-08-20	Pfizer Inc.	Antidepressant derivatives of cis-4-phenyl-1,2,3,4-tetrahydro-1-naphthalenamine
JPS5910497A (ja) *	1982-07-12	1984-01-19	Hitachi Ltd	フラックス
JPH0773795B2 (ja) *	1985-07-02	1995-08-09	太陽インキ製造株式会社	はんだ付用水洗性フラツクス組成物
US4882339A (en) *	1987-07-10	1989-11-21	Ciba-Geigy Corporation	4-Amino-substituted 1,2-dihydroxynaphthalene derivatives useful in inhibiting 5-lipoxygenase activity in mammals
US5071875A (en) *	1989-09-25	1991-12-10	Northwestern University	Substituted 2-amidotetralins as melatonin agonists and antagonists

1991
- 1991-07-11 GB GB919114947A patent/GB9114947D0/en active Pending
1992
- 1992-07-03 AT AT92914143T patent/ATE127779T1/de not_active IP Right Cessation
- 1992-07-03 WO PCT/EP1992/001497 patent/WO1993001162A1/en not_active Ceased
- 1992-07-03 EP EP92914143A patent/EP0594666B1/en not_active Expired - Lifetime
- 1992-07-03 US US08/178,272 patent/US5463126A/en not_active Expired - Fee Related
- 1992-07-03 CA CA002109817A patent/CA2109817C/en not_active Expired - Fee Related
- 1992-07-03 ES ES92914143T patent/ES2078749T3/es not_active Expired - Lifetime
- 1992-07-03 DE DE69204840T patent/DE69204840T2/de not_active Expired - Fee Related
- 1992-07-03 JP JP5501953A patent/JP2566374B2/ja not_active Expired - Fee Related
- 1992-07-03 DK DK92914143.0T patent/DK0594666T3/da active
- 1992-07-09 PT PT100672A patent/PT100672B/pt not_active IP Right Cessation
- 1992-07-10 IE IE922248A patent/IE67822B1/en not_active IP Right Cessation
1994
- 1994-01-10 FI FI940106A patent/FI112210B/fi not_active IP Right Cessation
1995
- 1995-10-18 GR GR950402868T patent/GR3017766T3/el unknown

Also Published As

Publication number	Publication date
EP0594666B1 (en)	1995-09-13
EP0594666A1 (en)	1994-05-04
JP2566374B2 (ja)	1996-12-25
US5463126A (en)	1995-10-31
PT100672B (pt)	1999-06-30
GB9114947D0 (en)	1991-08-28
ATE127779T1 (de)	1995-09-15
WO1993001162A1 (en)	1993-01-21
GR3017766T3 (en)	1996-01-31
ES2078749T3 (es)	1995-12-16
CA2109817C (en)	1999-08-31
JPH06509080A (ja)	1994-10-13
IE922248A1 (en)	1993-01-13
FI940106L (fi)	1994-01-10
DK0594666T3 (da)	1995-11-13
IE67822B1 (en)	1996-05-01
DE69204840D1 (de)	1995-10-19
FI112210B (fi)	2003-11-14
FI940106A0 (fi)	1994-01-10
DE69204840T2 (de)	1996-02-22

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Legal Events

Date

Code

Title

Description

1993-09-30

BB1A

Laying open of patent application

Effective date: 19930507

1999-06-30

FG3A

Patent granted, date of granting

Effective date: 19990316

2007-10-03

MM4A

Annulment/lapse due to non-payment of fees, searched and examined patent

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 20070917