PT2968351T - Formulações de dosagem de modulador de recetores de opioides - Google Patents

Formulações de dosagem de modulador de recetores de opioides

Info

Publication number
PT2968351T
PT2968351T PT14774006T PT14774006T PT2968351T PT 2968351 T PT2968351 T PT 2968351T PT 14774006 T PT14774006 T PT 14774006T PT 14774006 T PT14774006 T PT 14774006T PT 2968351 T PT2968351 T PT 2968351T
Authority
PT
Portugal
Prior art keywords
opioid receptor
receptor modulator
dosage formulations
modulator dosage
formulations
Prior art date
Application number
PT14774006T
Other languages
English (en)
Inventor
Jozef Ceulemans Jens
Costello Tim
Maria Jozef Jans Eugeen
Erna H Heyns Philip
Original Assignee
Allergan Holdings Unlimited Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=51528071&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PT2968351(T) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Allergan Holdings Unlimited Company filed Critical Allergan Holdings Unlimited Company
Publication of PT2968351T publication Critical patent/PT2968351T/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/4174Arylalkylimidazoles, e.g. oxymetazolin, naphazoline, miconazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/286Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/501Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Organic Chemistry (AREA)
  • Inorganic Chemistry (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Biochemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
PT14774006T 2013-03-14 2014-03-10 Formulações de dosagem de modulador de recetores de opioides PT2968351T (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US13/829,984 US9675587B2 (en) 2013-03-14 2013-03-14 Opioid receptor modulator dosage formulations

Publications (1)

Publication Number Publication Date
PT2968351T true PT2968351T (pt) 2018-11-19

Family

ID=51528071

Family Applications (1)

Application Number Title Priority Date Filing Date
PT14774006T PT2968351T (pt) 2013-03-14 2014-03-10 Formulações de dosagem de modulador de recetores de opioides

Country Status (20)

Country Link
US (9) US9675587B2 (pt)
EP (3) EP2968351B1 (pt)
JP (2) JP6449225B2 (pt)
KR (1) KR102435440B1 (pt)
CN (2) CN110917159A (pt)
AU (1) AU2014241076B2 (pt)
BR (1) BR112015022753A8 (pt)
CA (2) CA3254178A1 (pt)
CY (1) CY1120892T1 (pt)
DK (1) DK2968351T3 (pt)
EA (1) EA031559B1 (pt)
ES (1) ES2693374T3 (pt)
HU (1) HUE042748T2 (pt)
IL (2) IL241561B (pt)
PL (1) PL2968351T3 (pt)
PT (1) PT2968351T (pt)
SI (1) SI2968351T1 (pt)
TR (1) TR201815953T4 (pt)
TW (1) TWI648071B (pt)
WO (1) WO2014159245A1 (pt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
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US9675587B2 (en) 2013-03-14 2017-06-13 Allergan Holdings Unlimited Company Opioid receptor modulator dosage formulations
EP3297609A1 (en) * 2015-05-22 2018-03-28 Novartis AG Pharmaceutical compositions
CN105250232B (zh) * 2015-09-29 2018-08-14 江苏汇智知识产权服务有限公司 一种伊卢多啉肠溶片及其制备方法
EP3515434A4 (en) 2016-09-20 2020-02-26 Sun Pharmaceutical Industries Limited PROCESSES FOR THE PREPARATION OF ELUXADOLINE
WO2018069770A1 (en) * 2016-10-14 2018-04-19 Allergan Holdings Unlimited Company Methods of treatment using eluxadoline
US12285411B2 (en) * 2019-09-10 2025-04-29 Aurobindo Pharma Ltd Pharmaceutical composition comprising eluxadoline, process of preparation and use thereof
CA3166250A1 (en) 2020-02-05 2021-08-12 Gregory G. Plucinski Drug products for intranasal administration and uses thereof

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US5574159A (en) 1992-02-03 1996-11-12 Delta Pharmaceuticals, Inc. Opioid compounds and methods for making therefor
US5240929A (en) 1992-08-03 1993-08-31 Warner-Lambert Company 2-heterocyclic-5-hydroxy-1,3-pyrimidines useful as antiinflammatory agents
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WO1996022997A1 (en) 1995-01-27 1996-08-01 Novo Nordisk A/S Compounds with growth hormone releasing properties
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US6518292B1 (en) 1999-03-12 2003-02-11 Bristol-Myers Squibb Co. Heterocyclic aromatic compounds usefuls as growth hormone secretagogues
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WO2002024657A2 (en) 2000-09-20 2002-03-28 Schering Corporation Substituted imidazoles as dual histamine h1 and h3 agonists or antagonists
CN100400040C (zh) 2000-10-30 2008-07-09 詹森药业有限公司 三肽酶抑制剂
EP1387673B1 (en) * 2001-05-11 2010-12-29 Endo Pharmaceuticals Inc. Abuse-resistant controlled-release opioid dosage form
BR0213327A (pt) 2001-10-15 2004-10-13 Janssen Pharmaceutica Nv Derivados de 4-fenil-4-[1h-imidazol-2-il]-piperidina substituìdos e sua aplicação como agonistas de delta opióides não-peptìdicos seletivos
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WO2007043061A1 (en) * 2005-10-11 2007-04-19 Ipca Laboratories Ltd. Anti-malarial combination and methods of formulation
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KR101590596B1 (ko) 2007-07-09 2016-02-01 퓨리엑스 파마슈티컬스, 인코포레이티드 신규한 결정 및 5-({[2-아미노-3-(4-카르바모일-2,6-다이메틸-페닐)-프로피오닐]-[1-(4-페닐-1h-이미다졸-2-일)-에틸]-아미노}-메틸)-2-메톡시-벤조산의 제조 방법
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Also Published As

Publication number Publication date
US11090291B2 (en) 2021-08-17
US10188632B2 (en) 2019-01-29
JP2019014744A (ja) 2019-01-31
US12097187B2 (en) 2024-09-24
US11229627B1 (en) 2022-01-25
CA2906472A1 (en) 2014-10-02
US20170304268A1 (en) 2017-10-26
SI2968351T1 (sl) 2019-01-31
IL241561B (en) 2019-09-26
CN110917159A (zh) 2020-03-27
ES2693374T3 (es) 2018-12-11
AU2014241076B2 (en) 2018-07-19
US11311516B2 (en) 2022-04-26
HK1218514A1 (en) 2017-02-24
EP2968351A4 (en) 2016-08-24
CA3254178A1 (en) 2025-05-13
US20220040151A1 (en) 2022-02-10
IL268718B (en) 2021-04-29
EP2968351A1 (en) 2016-01-20
KR102435440B1 (ko) 2022-08-22
US20220008394A1 (en) 2022-01-13
US20210030720A1 (en) 2021-02-04
EA201591768A1 (ru) 2016-03-31
EA031559B1 (ru) 2019-01-31
BR112015022753A2 (pt) 2017-07-18
EP3865131A1 (en) 2021-08-18
US20230293493A1 (en) 2023-09-21
EP2968351B1 (en) 2018-08-29
IL268718A (en) 2019-10-31
PL2968351T3 (pl) 2019-03-29
TR201815953T4 (tr) 2018-11-21
CN105228629A (zh) 2016-01-06
KR20150140681A (ko) 2015-12-16
US20210205269A1 (en) 2021-07-08
DK2968351T3 (en) 2018-11-26
JP6449225B2 (ja) 2019-01-09
EP3456321A1 (en) 2019-03-20
BR112015022753A8 (pt) 2019-11-26
JP6666975B2 (ja) 2020-03-18
US9675587B2 (en) 2017-06-13
HUE042748T2 (hu) 2019-07-29
WO2014159245A1 (en) 2014-10-02
US20140271854A1 (en) 2014-09-18
CY1120892T1 (el) 2019-12-11
US11484527B2 (en) 2022-11-01
US11160792B2 (en) 2021-11-02
AU2014241076A1 (en) 2015-10-01
JP2016516694A (ja) 2016-06-09
US20210205268A1 (en) 2021-07-08
US20220096440A1 (en) 2022-03-31
US11007179B2 (en) 2021-05-18
TW201444590A (zh) 2014-12-01
TWI648071B (zh) 2019-01-21

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