PT83323A - Processo para a preparacao de novos tripeptideos n-alquilados e de composicoes farmaceuticas que os contem - Google Patents
Processo para a preparacao de novos tripeptideos n-alquilados e de composicoes farmaceuticas que os contemInfo
- Publication number
- PT83323A PT83323A PT83323A PT8332386A PT83323A PT 83323 A PT83323 A PT 83323A PT 83323 A PT83323 A PT 83323A PT 8332386 A PT8332386 A PT 8332386A PT 83323 A PT83323 A PT 83323A
- Authority
- PT
- Portugal
- Prior art keywords
- tripeptidees
- alkylated
- pharmaceutical compositions
- compositions containing
- preparing new
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
- C07K5/022—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
- C07K5/0222—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Molecular Biology (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19853532035 DE3532035A1 (de) | 1985-09-09 | 1985-09-09 | Neue n-alkylierte tripeptide, verfahren zu ihrer herstellung, sie enthaltende medikamente und deren verwendung |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PT83323A true PT83323A (pt) | 1986-10-01 |
| PT83323B PT83323B (pt) | 1989-05-12 |
Family
ID=6280419
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT83323A PT83323B (pt) | 1985-09-09 | 1986-09-08 | Processo para a preparacao de novos tripeptideos n-alquilados e de composicoes farmaceuticas que os contem |
Country Status (13)
| Country | Link |
|---|---|
| EP (1) | EP0214570A3 (pt) |
| JP (1) | JPS6261995A (pt) |
| KR (1) | KR870003134A (pt) |
| AU (1) | AU6243286A (pt) |
| DE (1) | DE3532035A1 (pt) |
| DK (1) | DK427786A (pt) |
| ES (1) | ES2001665A6 (pt) |
| FI (1) | FI863593L (pt) |
| GR (1) | GR862287B (pt) |
| HU (1) | HUT42507A (pt) |
| IL (1) | IL79966A0 (pt) |
| PT (1) | PT83323B (pt) |
| ZA (1) | ZA866807B (pt) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3538749A1 (de) * | 1985-10-31 | 1987-05-07 | Merck Patent Gmbh | Peptide |
| US8669281B1 (en) | 2013-03-14 | 2014-03-11 | Alkermes Pharma Ireland Limited | Prodrugs of fumarates and their use in treating various diseases |
| KR102085557B1 (ko) | 2013-03-14 | 2020-03-06 | 엘커메스 파마 아일랜드 리미티드 | 푸마레이트의 프로드럭 및 다양한 질환을 치료하는데 있어서의 이들의 용도 |
| JP6337135B2 (ja) | 2014-02-24 | 2018-06-06 | アルカーメス ファーマ アイルランド リミテッド | フマル酸エステルのスルホンアミドプロドラッグ及びスルフィンアミドプロドラッグ並びに種々の疾患の治療におけるその使用 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4483850A (en) * | 1982-05-10 | 1984-11-20 | Merck & Co., Inc. | N-Terminal substituted oligopeptide converting enzyme inhibitors |
| DE3413710A1 (de) * | 1984-04-12 | 1985-10-24 | Hoechst Ag, 6230 Frankfurt | Verfahren zur behandlung der herzinsuffizienz |
-
1985
- 1985-09-09 DE DE19853532035 patent/DE3532035A1/de not_active Withdrawn
-
1986
- 1986-08-29 EP EP86111972A patent/EP0214570A3/de not_active Withdrawn
- 1986-09-05 ES ES8601664A patent/ES2001665A6/es not_active Expired
- 1986-09-05 FI FI863593A patent/FI863593L/fi not_active Application Discontinuation
- 1986-09-08 KR KR1019860007497A patent/KR870003134A/ko not_active Withdrawn
- 1986-09-08 DK DK427786A patent/DK427786A/da not_active Application Discontinuation
- 1986-09-08 AU AU62432/86A patent/AU6243286A/en not_active Abandoned
- 1986-09-08 ZA ZA866807A patent/ZA866807B/xx unknown
- 1986-09-08 IL IL79966A patent/IL79966A0/xx unknown
- 1986-09-08 GR GR862287A patent/GR862287B/el unknown
- 1986-09-08 JP JP61209771A patent/JPS6261995A/ja active Pending
- 1986-09-08 PT PT83323A patent/PT83323B/pt not_active IP Right Cessation
- 1986-09-08 HU HU863881A patent/HUT42507A/hu unknown
Also Published As
| Publication number | Publication date |
|---|---|
| KR870003134A (ko) | 1987-04-15 |
| DE3532035A1 (de) | 1987-03-26 |
| PT83323B (pt) | 1989-05-12 |
| ZA866807B (en) | 1987-04-29 |
| FI863593A7 (fi) | 1987-03-10 |
| FI863593L (fi) | 1987-03-10 |
| AU6243286A (en) | 1987-03-12 |
| IL79966A0 (en) | 1986-12-31 |
| HUT42507A (en) | 1987-07-28 |
| ES2001665A6 (es) | 1988-06-01 |
| GR862287B (en) | 1987-01-12 |
| EP0214570A3 (de) | 1989-11-15 |
| JPS6261995A (ja) | 1987-03-18 |
| DK427786D0 (da) | 1986-09-08 |
| FI863593A0 (fi) | 1986-09-05 |
| DK427786A (da) | 1987-03-10 |
| EP0214570A2 (de) | 1987-03-18 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM3A | Annulment or lapse |
Free format text: LAPSE DUE TO NON-PAYMENT OF FEES Effective date: 19940430 |