PT84287B - Processo para a preparacao de acidos quinolinodioicos 2-substituidos - Google Patents

Processo para a preparacao de acidos quinolinodioicos 2-substituidos

Info

Publication number
PT84287B
PT84287B PT84287A PT8428787A PT84287B PT 84287 B PT84287 B PT 84287B PT 84287 A PT84287 A PT 84287A PT 8428787 A PT8428787 A PT 8428787A PT 84287 B PT84287 B PT 84287B
Authority
PT
Portugal
Prior art keywords
substd
opt
alkyl
benzyl
phenyl
Prior art date
Application number
PT84287A
Other languages
English (en)
Other versions
PT84287A (en
Inventor
Serge Leger
Robert N Young
Robert Zamboni
Original Assignee
Merck Frosst Canada Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Frosst Canada Inc filed Critical Merck Frosst Canada Inc
Publication of PT84287A publication Critical patent/PT84287A/pt
Publication of PT84287B publication Critical patent/PT84287B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/12Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/18Halogen atoms or nitro radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/36Sulfur atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
PT84287A 1986-02-14 1987-02-13 Processo para a preparacao de acidos quinolinodioicos 2-substituidos PT84287B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CA501932 1986-02-14

Publications (2)

Publication Number Publication Date
PT84287A PT84287A (en) 1987-03-01
PT84287B true PT84287B (pt) 1989-09-14

Family

ID=4132478

Family Applications (1)

Application Number Title Priority Date Filing Date
PT84287A PT84287B (pt) 1986-02-14 1987-02-13 Processo para a preparacao de acidos quinolinodioicos 2-substituidos

Country Status (14)

Country Link
EP (1) EP0233763B1 (pt)
JP (1) JPH0686432B2 (pt)
KR (1) KR870007920A (pt)
AT (1) ATE60584T1 (pt)
AU (1) AU595286B2 (pt)
DE (1) DE3767730D1 (pt)
DK (1) DK168534B1 (pt)
ES (1) ES2031498T3 (pt)
GR (1) GR3001474T3 (pt)
IE (1) IE59889B1 (pt)
IL (1) IL81569A (pt)
NZ (1) NZ219249A (pt)
PT (1) PT84287B (pt)
ZA (1) ZA871064B (pt)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0271287A3 (en) * 1986-12-11 1990-06-13 Merck Frosst Canada Inc. Quinoline dioic acids and amides
US4920130A (en) * 1987-11-02 1990-04-24 Rorer Pharamceutical Corp. Quinoline derivatives and use thereof as antagonists of leukotriene D4
US4920132A (en) * 1987-11-03 1990-04-24 Rorer Pharmaceutical Corp. Quinoline derivatives and use thereof as antagonists of leukotriene D4
US4920131A (en) * 1987-11-03 1990-04-24 Rorer Pharmaceutical Corp. Quinoline derivatives and use thereof as antagonists of leukotriene D4
US5004743A (en) * 1987-11-25 1991-04-02 Merck Frosst Canada, Inc. Pyridyl styrene dialkanoic acids as anti-leukotriene agents
EP0318093A3 (en) * 1987-11-25 1990-12-05 Merck Frosst Canada Inc. Diarylquinoline diacids and their use as medicaments
US5204358A (en) * 1987-11-25 1993-04-20 Merck Frosst Canada, Inc. Hetaryl styryl quinolines as leukotriene inhibitors
US5104882A (en) * 1987-11-25 1992-04-14 Merck Frosst Canada, Inc. Diarylstrylquinoline diacids and pharmaceutical compositions thereof
AU617386B2 (en) * 1987-12-01 1991-11-28 Leo Pharmaceutical Products Ltd. A/S (Lovens Kemiske Fabrik Produktionsaktieselskab) Substituted quinolines
GB8728051D0 (en) * 1987-12-01 1988-01-06 Leo Pharm Prod Ltd Chemical compounds
US4883878A (en) * 1988-02-08 1989-11-28 Merck & Co. Inc. Process for unsymmetrical dithioacetals and dithioketals
EP0349062A1 (en) * 1988-06-27 1990-01-03 Merck Frosst Canada Inc. Quinoline ether alkanoic acid
US5070022A (en) * 1988-12-22 1991-12-03 Merck & Co., Inc. Enzymic process for preparing leukotriene antagonists
NZ233752A (en) * 1989-05-24 1993-05-26 Merck Frosst Canada Inc Substituted quinoline derivatives, preparation and pharmaceutical compositions thereof
US4996214A (en) * 1990-06-28 1991-02-26 Smithkline Beecham Corporation Quinolinyl substituted phenyl/thioalkanoic acid substituted propionic acids and leucotriene antagonist use thereof
US5856322A (en) * 1990-10-12 1999-01-05 Merck Frosst Canada, Inc. Unsaturated hydroxyalkylquinoline acids as leukotriene antagonists
US5266568A (en) * 1990-10-12 1993-11-30 Merck Frosst Canada, Inc. Hydroxyalkylquinoline ether acids as leukotriene antagonists
ES2079586T3 (es) * 1990-10-12 1996-01-16 Merck Frosst Canada Inc Acidos de eter de hidroxialquilquinolina como antagonistas de leucotrienos.
DK0480717T3 (da) * 1990-10-12 1999-02-08 Merck Frosst Canada Inc Umættede hydroxyalkylquinolinsyrer som leukotrienantagonister
EP0480716A1 (en) * 1990-10-12 1992-04-15 Merck Frosst Canada Inc. Saturated hydroxyalkylquinoline acids as leukotriene antagonists
US5212180A (en) * 1991-02-21 1993-05-18 Merck Frosst Canada, Inc. Quinoline-containing ketoacids as leukotriene antagonists
IE920499A1 (en) * 1991-02-21 1992-08-26 Merck Frosst Canada Inc Quinoline-containing ketoacids as leukotriene antagonists
US5276044A (en) * 1991-08-14 1994-01-04 Allergan, Inc. Leukotriene receptor antagonist and antihistamine complex pharmaceutical compositions
US5270324A (en) * 1992-04-10 1993-12-14 Merck Frosst Canada, Inc. Fluorinated hydroxyalkylquinoline acids as leukotriene antagonists
CA2136241C (en) * 1992-06-22 2004-01-27 Richard Frenette Fluorinated quinoline indoles as inhibitors of the biosynthesis of leukotrienes
US5964261A (en) * 1996-05-29 1999-10-12 Baxter International Inc. Implantation assembly
US20030216571A1 (en) * 1999-12-28 2003-11-20 Yoshiaki Kuroki Tricyclic compounds

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE56702B1 (en) * 1982-12-01 1991-11-06 Usv Pharma Corp Antiinflammatory antiallergic compounds
US4625034A (en) * 1985-02-04 1986-11-25 Usv Pharmaceutical Corp. 1,2-Dihydro; 1,2,3,4-tetrahydro; 5,8 dihydro; and 5,6,7,8-tetrahydroquinoline derivatives
IE861607L (en) * 1985-06-18 1986-12-18 Bunce Roger A 2-substituted quinolines

Also Published As

Publication number Publication date
JPH0686432B2 (ja) 1994-11-02
ATE60584T1 (de) 1991-02-15
DK168534B1 (da) 1994-04-18
KR870007920A (ko) 1987-09-22
AU6871787A (en) 1987-08-20
DK72287D0 (da) 1987-02-13
AU595286B2 (en) 1990-03-29
EP0233763A2 (en) 1987-08-26
IL81569A (en) 1991-11-21
GR3001474T3 (en) 1992-10-08
JPS62258363A (ja) 1987-11-10
IL81569A0 (en) 1987-09-16
EP0233763A3 (en) 1988-10-19
DE3767730D1 (de) 1991-03-07
IE59889B1 (en) 1994-04-20
PT84287A (en) 1987-03-01
ZA871064B (en) 1987-10-28
EP0233763B1 (en) 1991-01-30
NZ219249A (en) 1990-07-26
DK72287A (da) 1987-08-15
ES2031498T3 (es) 1992-12-16
IE870334L (en) 1987-08-14

Similar Documents

Publication Publication Date Title
PT84287B (pt) Processo para a preparacao de acidos quinolinodioicos 2-substituidos
FR2342056A1 (fr) Solution de prise pour ciments ionomeres de verre dentaire
BE846610A (fr) Procede pour la preparation de nouveaux derives insolubles dans l'eau et a pouvoir d'absorption eleve
DK207175A (da) Fremgangsmade til fremstilling af cephalosporiner med alfa-acylaminoeddikesyresidekede
IT1039416B (it) Procedimento per la preparazione di acqua ossigenata
NL7902136A (nl) Ornithine- en argininezouten van keto-analogen van onontbeerlijke aminozuren met vertakte keten met farmacologische werking.
RO77320A (ro) Procedeu pentru purificarea sarurilor acidului clavulanic
IT8324409A0 (it) Sali di metallo alcalino di acidi procedimento per la preparazione di polietossicarbossilici.
MX4350E (es) Procedimiento para la preparacion de compuestos monoazoicos insolubles en agua
IT1042820B (it) Processo per la preparazione contemporanea di epsilon caprolattoni e acidi carbossilici
IT988272B (it) Procedimento per l eliminazione o per la lavorazione congiunta di residui di sali da tempra
IT1162868B (it) Procedimento per la preparazione dell'acido d 2 6 metossi 2 naftil propionico e suoi sali farmaceuticamente accettabili e nouvi intermedi per tale preparazione
BG27561A3 (bg) Метод за получаване на 7-в-/д-2-амино-2-/метил- сулфониламинофенил/ ацетиламино/ -3-r-3-цефем -4- карбонови киселини и техните соли
IT986994B (it) Procedimento per la preparazione di sali di addizione con acidi inorganici della urea
IT8049141A0 (it) Procedimento per preparare sali di acidi minerali di cisteammina
FR2320336A1 (fr) Procede pour ameliorer la solubilite de colorants acides dans l'eau
IT1040561B (it) Procedimento ed apparecchiatura per la depurazione spinta di soluzioni acquose di sali metallici
IT1141406B (it) Sali della cefapirina con aminoacidi
IT1047136B (it) Procedimento per la fabbricazione di dl 6 finel 2 3 5 6 tetraidro immidazo 2 1 8 tiazolo e relativi sali di addizione con acidi
DK141964C (da) Analogifremgangsmaade til fremstilling af isoquinolinderivatereller salte deraf med fysiologisk acceptable syrer
IT1080477B (it) Sali di amoxicillina con aminoacidi
FR2280475A1 (fr) Metal d'apport pour soudure
IT973235B (it) Procedimento per la preparazione di acidi monocarbossilici alifati ci superiori
IT1077985B (it) Procedimento per giuntare segmenti di aste o cilindri cavi ad esempio segmenti di guide d'onda
IT994096B (it) Procedimento per la produzione di sali di aurammina e soluzioni di sali di aurammina

Legal Events

Date Code Title Description
PC3A Transfer or assignment

Free format text: 19990427 MERCK FROSST CANADA & CO. CA

MM3A Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 20040806