PT88468A - Process for the preparation of macrolide compounds - Google Patents

Process for the preparation of macrolide compounds

Info

Publication number: PT88468A
Authority: PT; Portugal
Prior art keywords: preparation; group; macrolide compounds; chem; compound
Prior art date: 1987-09-11

Application number

PT88468A

Other languages

English (en)

Other versions

PT88468B (pt

Inventor

Michael V J Ramsay

Anthony H Shingler

Simon C Dolan

Stephen Freeman

Oswy Z Pereira

Original Assignee

American Cyanamid Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1987-09-11

Filing date

1988-09-09

Publication date

1988-10-01

1988-09-09 Application filed by American Cyanamid Co filed Critical American Cyanamid Co

1988-10-01 Publication of PT88468A publication Critical patent/PT88468A/pt

1992-11-30 Publication of PT88468B publication Critical patent/PT88468B/pt

Links

150000001875 compounds Chemical class 0.000 title abstract 4
239000003120 macrolide antibiotic agent Substances 0.000 title 1
239000000543 intermediate Substances 0.000 abstract 3
125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 2
125000003668 acetyloxy group Chemical group [H]C([H])([H])C(=O)O[*] 0.000 abstract 1
125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 abstract 1
125000005843 halogen group Chemical group 0.000 abstract 1
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
-1 hydroxy, methoxy Chemical group 0.000 abstract 1
125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 abstract 1
125000006239 protecting group Chemical group 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/22—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains four or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Engineering & Computer Science (AREA)
Biochemistry (AREA)
Biotechnology (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Tropical Medicine & Parasitology (AREA)
Saccharide Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Steroid Compounds (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Cephalosporin Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Physical Or Chemical Processes And Apparatus (AREA)

PT88468A 1987-09-11 1988-09-09 Processo para a preparacao de um composto macrolido PT88468B (pt)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GB878721373A GB8721373D0 (en)	1987-09-11	1987-09-11	Chemical process

Publications (2)

Publication Number	Publication Date
PT88468A true PT88468A (pt)	1988-10-01
PT88468B PT88468B (pt)	1992-11-30

Family

ID=10623610

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PT88468A PT88468B (pt)	1987-09-11	1988-09-09	Processo para a preparacao de um composto macrolido

Country Status (17)

Country	Link
EP (1)	EP0307221B1 (pt)
JP (1)	JPH01163182A (pt)
KR (1)	KR890005116A (pt)
AT (1)	ATE90101T1 (pt)
AU (1)	AU621063B2 (pt)
BR (1)	BR8804664A (pt)
CA (1)	CA1333600C (pt)
DD (1)	DD274421A5 (pt)
DE (1)	DE3881458T2 (pt)
DK (1)	DK168524B1 (pt)
ES (1)	ES2040863T3 (pt)
GB (1)	GB8721373D0 (pt)
HU (2)	HU203353B (pt)
IE (1)	IE62759B1 (pt)
NZ (1)	NZ226118A (pt)
PT (1)	PT88468B (pt)
ZA (1)	ZA886739B (pt)

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4429209A (en) *	1981-10-19	1984-01-31	Duro Dyne Corporation	Resistance welding pin
ES8802229A1 (es) *	1985-04-30	1988-04-16	Glaxo Group Ltd	Un procedimiento para preparar nuevos derivados lactonicos macrociclicos.
DE3782481T2 (de) *	1986-09-12	1993-05-19	American Cyanamid Co	23-deoxy-derivate von ll-f28249-verbindungen.
US4806527A (en) *	1987-03-16	1989-02-21	Merck & Co., Inc.	Avermectin derivatives

1987
- 1987-09-11 GB GB878721373A patent/GB8721373D0/en active Pending
1988
- 1988-09-09 IE IE274588A patent/IE62759B1/en not_active IP Right Cessation
- 1988-09-09 PT PT88468A patent/PT88468B/pt not_active IP Right Cessation
- 1988-09-09 AU AU22089/88A patent/AU621063B2/en not_active Ceased
- 1988-09-09 HU HU884659A patent/HU203353B/hu not_active IP Right Cessation
- 1988-09-09 BR BR8804664A patent/BR8804664A/pt active Search and Examination
- 1988-09-09 CA CA000576930A patent/CA1333600C/en not_active Expired - Fee Related
- 1988-09-09 HU HU903199A patent/HU207085B/hu not_active IP Right Cessation
- 1988-09-09 KR KR1019880011658A patent/KR890005116A/ko not_active Ceased
- 1988-09-09 EP EP88308345A patent/EP0307221B1/en not_active Expired - Lifetime
- 1988-09-09 DD DD88319668A patent/DD274421A5/de not_active IP Right Cessation
- 1988-09-09 NZ NZ226118A patent/NZ226118A/en unknown
- 1988-09-09 DK DK504788A patent/DK168524B1/da not_active IP Right Cessation
- 1988-09-09 ES ES198888308345T patent/ES2040863T3/es not_active Expired - Lifetime
- 1988-09-09 JP JP63224828A patent/JPH01163182A/ja active Pending
- 1988-09-09 ZA ZA886739A patent/ZA886739B/xx unknown
- 1988-09-09 DE DE88308345T patent/DE3881458T2/de not_active Expired - Fee Related
- 1988-09-09 AT AT88308345T patent/ATE90101T1/de not_active IP Right Cessation

Also Published As

Publication number	Publication date
GB8721373D0 (en)	1987-10-21
HU203353B (en)	1991-07-29
ES2040863T3 (es)	1993-11-01
DE3881458D1 (de)	1993-07-08
DE3881458T2 (de)	1993-10-14
DK504788A (da)	1989-03-12
DK504788D0 (da)	1988-09-09
EP0307221A3 (en)	1989-10-25
PT88468B (pt)	1992-11-30
KR890005116A (ko)	1989-05-11
BR8804664A (pt)	1989-04-18
IE882745L (en)	1989-03-11
EP0307221B1 (en)	1993-06-02
AU621063B2 (en)	1992-03-05
DK168524B1 (da)	1994-04-11
ZA886739B (en)	1989-08-30
IE62759B1 (en)	1995-02-22
JPH01163182A (ja)	1989-06-27
HU207085B (en)	1993-03-01
AU2208988A (en)	1989-03-16
CA1333600C (en)	1994-12-20
HUT48258A (en)	1989-05-29
HU903199D0 (en)	1990-10-28
DD274421A5 (de)	1989-12-20
NZ226118A (en)	1989-12-21
EP0307221A2 (en)	1989-03-15
ATE90101T1 (de)	1993-06-15

Legal Events

Date

Code

Title

Description

1992-11-30

FG3A

Patent granted, date of granting

Effective date: 19920525

1997-03-31

MM3A

Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 19961130

Publication	Publication Date	Title
TW262474B (pt)	1995-11-11
EP0272110A3 (en)	1989-10-25	Erythromycin a derivatives and method for the preparation of the same
HUT57043A (en)	1991-11-28	Process for producing pharmaceutical solutions comprising macrolide
NO823836L (no)	1983-05-18	Fremgangsmaate ved fremstilling av antifibrinolytisk aktive forbindelser.
ES2005746A6 (es)	1989-03-16	Un procedimiento para la preparacion de un haluro de piridinio.
DK0781764T3 (da)	2000-07-10	Fremgangsmåde til fremstilling af alkoxyiminoacetamid-derivater
EP0298752A3 (en)	1989-11-08	Mercapto-substituted pyridine compounds and process for preparing the same
FI873443A7 (fi)	1987-08-07	Norfloxacinmellanprodukt.
ZA886739B (en)	1989-08-30	Process for the preparation of macrolide compounds
DE69007203D1 (de)	1994-04-14	Imidazolderivate, Verfahren zu deren Herstellung und diese enthaltende Antiulkusmittel.
BR8603787A (pt)	1987-03-17	Compostos heterociclicos,e,processo de sua preparacao e aplicacao
HU913900D0 (en)	1992-02-28	Method for producing 2-halogen-pyrrhole-3-carbonitrile derivatives
DK82583D0 (da)	1983-02-23	Furyloxazolyleddikesyrederivater og fremgangsmader til fremstilling deraf
HU910108D0 (en)	1991-08-28	Process for the production of macrolide compounds
NZ333414A (en)	2000-05-26	Preparation of substituted 3-aryl-5-haloalkyl-pyrazoles having herbicidal activity
PT91036A (pt)	1990-02-08	Processo para a preparacao de derivados de sulfonil-indolizina, uteis como intermediarios de sintese
DK162188A (da)	1988-09-27	Fremgangsmaade til fremstilling af pentandionderivater
AU8292787A (en)	1988-06-23	Fluorine-containing macrolide compounds and their use
ES2164258T3 (es)	2002-02-16	Procedimiento de preparacion de derivados de carbamoilmetilurea.
FI943596A7 (fi)	1994-08-02	Menetelmä terapeuttisesti käytt¦kelpoisten makrolidiyhdisteiden valmistamiseksi
SE9002445L (sv)	1990-07-16	Nytt cyklobutanderivat och foerfarande foer framstaellning av detsamma
FR2446818A1 (fr)	1980-08-14	Tetrahydro-2h-benzo(c)pyrroles utiles comme intermediaires