PT89370A - Processo para a preparacao de compostos derivados de mercapto-imidazolinas, dos seus intermedarios e de composicoes farmaceuticas contendo aqueles derivados - Google Patents

Processo para a preparacao de compostos derivados de mercapto-imidazolinas, dos seus intermedarios e de composicoes farmaceuticas contendo aqueles derivados

Info

Publication number
PT89370A
PT89370A PT89370A PT8937088A PT89370A PT 89370 A PT89370 A PT 89370A PT 89370 A PT89370 A PT 89370A PT 8937088 A PT8937088 A PT 8937088A PT 89370 A PT89370 A PT 89370A
Authority
PT
Portugal
Prior art keywords
imidazolines
mercapto
preparation
pharmaceutical compositions
compositions containing
Prior art date
Application number
PT89370A
Other languages
English (en)
Inventor
Lawrence Ivan Kruse
Stephen Torey Ross
Thomas Brent Leonard
Original Assignee
Smithkline Beckman Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beckman Corp filed Critical Smithkline Beckman Corp
Publication of PT89370A publication Critical patent/PT89370A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/30—Oxygen or sulfur atoms
    • C07D233/42—Sulfur atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C333/00—Derivatives of thiocarbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C333/14—Dithiocarbamic acids; Derivatives thereof
    • C07C333/16—Salts of dithiocarbamic acids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PT89370A 1987-12-31 1988-12-30 Processo para a preparacao de compostos derivados de mercapto-imidazolinas, dos seus intermedarios e de composicoes farmaceuticas contendo aqueles derivados PT89370A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/140,053 US4876266A (en) 1987-12-31 1987-12-31 1-aralkyl-2-mercaptoimidazolines as DBH inhibitors

Publications (1)

Publication Number Publication Date
PT89370A true PT89370A (pt) 1989-12-29

Family

ID=22489533

Family Applications (1)

Application Number Title Priority Date Filing Date
PT89370A PT89370A (pt) 1987-12-31 1988-12-30 Processo para a preparacao de compostos derivados de mercapto-imidazolinas, dos seus intermedarios e de composicoes farmaceuticas contendo aqueles derivados

Country Status (7)

Country Link
US (1) US4876266A (pt)
EP (1) EP0329900A1 (pt)
JP (1) JPH03501728A (pt)
AU (1) AU2911389A (pt)
PT (1) PT89370A (pt)
WO (1) WO1989006126A1 (pt)
ZA (1) ZA889708B (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3821464A1 (de) * 1988-06-25 1989-12-28 Degussa Verfahren zur herstellung substituierter organyloxysilylfunktioneller, cyclischer thioharnstoffe und diese verbindungen
WO2004083700A1 (de) * 2003-03-19 2004-09-30 Maschinenfabrik Reinhausen Gmbh Druckentlastungsventil
DE10312177B3 (de) * 2003-03-19 2004-06-17 Maschinenfabrik Reinhausen Gmbh Druckentlastungsventil
US9567316B2 (en) 2012-03-07 2017-02-14 The Mclean Hospital Corporation Aminoquinoline derivatives and uses thereof
EP3138863A1 (de) * 2015-09-01 2017-03-08 Sika Technology AG Emissionsarme epoxidharz-zusammensetzung

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2839561A (en) * 1955-02-10 1958-06-17 Bayer Ag Dithiocarbonic acid esters and production
GB1155580A (en) * 1965-10-21 1969-06-18 Geigy Ag J R New Imidazole Derivatives their Production and Use
GB1261345A (en) * 1968-03-07 1972-01-26 Ici Ltd Sulphur-containing benzyl derivatives and pesticidal compositions containing them
BE787477A (fr) * 1971-08-12 1973-02-12 Bayer Ag 1-phenyl-2-imino-imidazolidines, leur procede de preparation etleur application comme repulsifs a l'egard des oiseaux
DE2259627A1 (de) * 1972-12-06 1974-06-12 Hoechst Ag Imidazolyl-(2)-thio-alkansaeureester und verfahren zu ihrer herstellung
US4284641A (en) * 1977-08-26 1981-08-18 Burroughs Wellcome Co. Pharmaceutically active imidazole derivatives
GB2096987B (en) * 1981-04-22 1984-04-04 Farmos Oy Substituted imidazole and imidazole derivatives and their preparation and use
PT78388B (en) * 1983-04-12 1986-09-15 Smithkline Beckman Corp Dopamine-beta-hydroxylase inhibitors
US4532331A (en) * 1983-04-12 1985-07-30 Smithkline Beckman Corporation 1-Benzyl-2-aminomethyl imidazole derivatives
JPS614038A (ja) * 1984-06-18 1986-01-09 Asahi Chem Ind Co Ltd 新規な感光性組成物

Also Published As

Publication number Publication date
ZA889708B (en) 1989-12-27
WO1989006126A1 (en) 1989-07-13
AU2911389A (en) 1989-08-01
EP0329900A1 (en) 1989-08-30
US4876266A (en) 1989-10-24
JPH03501728A (ja) 1991-04-18

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Legal Events

Date Code Title Description
FC3A Refusal

Effective date: 19940721