PT91716A - Processo para a preparacao de antibioticos beta-lactamicos - Google Patents

Processo para a preparacao de antibioticos beta-lactamicos

Info

Publication number
PT91716A
PT91716A PT91716A PT9171689A PT91716A PT 91716 A PT91716 A PT 91716A PT 91716 A PT91716 A PT 91716A PT 9171689 A PT9171689 A PT 9171689A PT 91716 A PT91716 A PT 91716A
Authority
PT
Portugal
Prior art keywords
beta
preparation
lactamic antibiotics
lactamic
antibiotics
Prior art date
Application number
PT91716A
Other languages
English (en)
Other versions
PT91716B (pt
Inventor
George Burton
John Hargreaves Bateson
Stephen Cristopher Martin Fell
Original Assignee
Beecham Group Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Beecham Group Plc filed Critical Beecham Group Plc
Publication of PT91716A publication Critical patent/PT91716A/pt
Publication of PT91716B publication Critical patent/PT91716B/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/22—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with radicals containing only hydrogen and carbon atoms, attached in position 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D505/00—Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
PT91716A 1988-09-16 1989-09-14 Processo para a preparacao de antibioticos beta-lactamicos PT91716B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB888821797A GB8821797D0 (en) 1988-09-16 1988-09-16 Novel compounds

Publications (2)

Publication Number Publication Date
PT91716A true PT91716A (pt) 1990-03-30
PT91716B PT91716B (pt) 1995-05-31

Family

ID=10643729

Family Applications (1)

Application Number Title Priority Date Filing Date
PT91716A PT91716B (pt) 1988-09-16 1989-09-14 Processo para a preparacao de antibioticos beta-lactamicos

Country Status (8)

Country Link
US (1) US5064649A (pt)
EP (1) EP0359536A3 (pt)
JP (1) JPH02121995A (pt)
KR (1) KR900004746A (pt)
AU (1) AU4140489A (pt)
DK (1) DK453489A (pt)
GB (1) GB8821797D0 (pt)
PT (1) PT91716B (pt)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0395219B1 (en) * 1989-03-30 1998-09-30 Pfizer Inc. Cephalosporins and their homologues, process for their preparation and pharmaceutical compositions
GB8920793D0 (en) * 1989-09-14 1989-11-01 Beecham Group Plc Novel compounds
MY106399A (en) * 1990-07-24 1995-05-30 Pfizer Cephalosporins and homologeus, preparation and pharmaceutical composition
GB9019743D0 (en) * 1990-09-10 1990-10-24 Beecham Group Plc Novel compounds
US5169843A (en) * 1990-10-22 1992-12-08 Bristol-Myers Squibb Company Antibiotic C-3 cyclobutenedione substituted (1-carba) cephalosporin compounds, cmpositions, and methods of use thereof
PT620225E (pt) * 1993-04-16 2003-03-31 Basilea Pharmaceutica Ag Derivados de cefalosporina
US5523400A (en) * 1993-04-16 1996-06-04 Hoffmann-La Roche Inc. Cephalosporin antibiotics
US5856474A (en) * 1994-04-25 1999-01-05 Biochemie Gesellschaft, M.B.H. Cephalosporin synthesis
EP0761673A1 (en) * 1995-09-12 1997-03-12 F. Hoffmann-La Roche Ag Cephalosporin derivatives
US5804577A (en) * 1995-09-12 1998-09-08 Hoffmann-La Roche Inc. Cephalosporin derivatives
CN114728008A (zh) * 2019-08-29 2022-07-08 加利福尼亚大学董事会 鉴定β-内酰胺酶的化合物及其使用方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4870168A (en) * 1987-02-26 1989-09-26 Bristol-Myers Company 3-Unsaturated alkyl cephems from 3-triflyl cephems

Also Published As

Publication number Publication date
DK453489D0 (da) 1989-09-14
DK453489A (da) 1990-03-17
JPH02121995A (ja) 1990-05-09
AU4140489A (en) 1990-03-22
US5064649A (en) 1991-11-12
PT91716B (pt) 1995-05-31
GB8821797D0 (en) 1988-10-19
KR900004746A (ko) 1990-04-12
EP0359536A3 (en) 1991-11-13
EP0359536A2 (en) 1990-03-21

Similar Documents

Publication Publication Date Title
PT82989B (pt) Processo para a preparacao de antibioticos beta-lactamicos
PT90523A (pt) Processo para a preparacao de adsorvatos de ranitidina
PT90119A (pt) Processo para a preparacao de um adocante
PT93785A (pt) Processo para a preparacao de derivados de 3-substituido-2-oxindole
BR8802484A (pt) Processo para a preparacao de isocianatos
PT90293A (pt) Processo para a preparacao de macrolidos
PT92534A (pt) Processo para a preparacao de compostos azabiciclicos
PT91068A (pt) Processo para a preparacao de compostos biarilo
PT91895A (pt) Processo para a preparacao de 9h-purinas substituidas
BR8906327A (pt) Processo para a preparacao de organoclorossilanos
PT91872A (pt) Processo para a preparacao de compostos azabiciclicos
PT90854A (pt) Processo para a preparacao de 1-aril-2-naftoilaminas
PT92638A (pt) Processo para a preparacao de poliazamacrociclos mono-n-alquilados
PT90266A (pt) Processo para a preparacao de compostos azabiciclicos
PT92365A (pt) Processo para a preparacao de (s)-alfa-etil-2-oxo-1-pirrolidinoacetamida
PT90435A (pt) Processo aperfeicoado para a preparacao de uma cetimina
BR9001503A (pt) Processo para a preparacao de alquil-halogenossilanos
PT93629A (pt) Processo para a preparacao de derivados de tieno-triazolo-diazepina
PT91027A (pt) Processo para a preparacao de derivados peptidicos
PT89775A (pt) Processo para a preparacao de derivados de isoquinolina
PT92539A (pt) Processo para a preparacao de derivados de anfotericina b
BR8803678A (pt) Processo para a preparacao de polieteramidas
BR8903367A (pt) Processo para a preparacao de organoclorossilanos
PT92507A (pt) Processo para a preparacao de alfa-ciano-beta-oxopropionamidas
PT93631A (pt) Processo para a preparacao de derivados de tieno-triazolo-diazepina

Legal Events

Date Code Title Description
FG3A Patent granted, date of granting

Effective date: 19941124

MM3A Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 19960531