PT92032A - Processo para a preparacao de esteres de alquilo de cadeia ramificada do acido 2-{4-(2-piperidino-etoxi)-benzoil}-benzoico e de composicoes farmaceuticas que os contem - Google Patents

Processo para a preparacao de esteres de alquilo de cadeia ramificada do acido 2-{4-(2-piperidino-etoxi)-benzoil}-benzoico e de composicoes farmaceuticas que os contem

Info

Publication number
PT92032A
PT92032A PT92032A PT9203289A PT92032A PT 92032 A PT92032 A PT 92032A PT 92032 A PT92032 A PT 92032A PT 9203289 A PT9203289 A PT 9203289A PT 92032 A PT92032 A PT 92032A
Authority
PT
Portugal
Prior art keywords
etoxy
piperidine
benzoyl
contain
preparation
Prior art date
Application number
PT92032A
Other languages
English (en)
Other versions
PT92032B (pt
Inventor
Martin Bickel
Jurgen Blumbach
Bansi Lal
Ramanujam Rajagopalan
Alihussein Nomanbhaidohadwalla
Richard Helmut Rupp
Swati Bal-Tembe
Narayan Sudhindra Punekar
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of PT92032A publication Critical patent/PT92032A/pt
Publication of PT92032B publication Critical patent/PT92032B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/08Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
    • C07D295/084Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/088Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
PT92032A 1988-10-21 1989-10-19 Processo para a preparacao de esteres de alquilo de cadeia ramificada do acido 2-{4-(2-piperidino-etoxi)-benzoil}-benzoico e de composicoes farmaceuticas que os contem PT92032B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP88117521 1988-10-21

Publications (2)

Publication Number Publication Date
PT92032A true PT92032A (pt) 1990-04-30
PT92032B PT92032B (pt) 1995-06-30

Family

ID=8199477

Family Applications (1)

Application Number Title Priority Date Filing Date
PT92032A PT92032B (pt) 1988-10-21 1989-10-19 Processo para a preparacao de esteres de alquilo de cadeia ramificada do acido 2-{4-(2-piperidino-etoxi)-benzoil}-benzoico e de composicoes farmaceuticas que os contem

Country Status (25)

Country Link
EP (1) EP0364941B1 (pt)
JP (1) JP2851077B2 (pt)
KR (1) KR0163567B1 (pt)
CN (1) CN1025615C (pt)
AT (1) ATE118489T1 (pt)
AU (1) AU628404B2 (pt)
CA (1) CA1333905C (pt)
CZ (1) CZ280193B6 (pt)
DE (1) DE68921132T2 (pt)
DK (1) DK168012B1 (pt)
EG (1) EG19053A (pt)
ES (1) ES2068869T3 (pt)
FI (1) FI93355C (pt)
GR (1) GR3015493T3 (pt)
HU (1) HU207306B (pt)
IE (1) IE66246B1 (pt)
IL (1) IL92049A0 (pt)
NO (1) NO175255C (pt)
NZ (1) NZ231087A (pt)
PH (1) PH30769A (pt)
PT (1) PT92032B (pt)
RU (1) RU1782232C (pt)
SK (1) SK596189A3 (pt)
SU (1) SU1766253A3 (pt)
ZA (1) ZA897953B (pt)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5821252A (en) * 1988-10-21 1998-10-13 Hoechst Aktiengesellschaft Method of blocking nerve conduction by treatment with branched-chain esters of 2- 4-(2-piperidine-ethoxy)-benzoyl!-benzoic acid and pharmaceutically acceptable salts thereof
US5998401A (en) * 1995-02-28 1999-12-07 Eli Lilly And Company Naphthyl compounds, intermediates, compositions, and methods
US5811421A (en) * 1995-07-31 1998-09-22 Eli Lilly And Company Naphthyl and dihydronaphthyl intermediates, compounds, compositions, and methods

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1057372A (fr) * 1951-05-26 1954-03-08 Hoechst Ag éthers basiques et leur préparation
US2681340A (en) 1951-05-26 1954-06-15 Hoechst Ag Amino esters
DE3508398A1 (de) * 1985-03-08 1986-11-06 Hoechst Ag, 6230 Frankfurt Fungizide mittel auf der basis von 3-(hetero)-arylpropylaminen sowie neue (hetero)-aryl-propylamine und verfahren zu ihrer herstellung

Also Published As

Publication number Publication date
NO894184L (no) 1990-04-23
NZ231087A (en) 1991-09-25
FI894973A0 (fi) 1989-10-19
KR0163567B1 (ko) 1998-12-01
IL92049A0 (en) 1990-07-12
EG19053A (en) 1994-07-30
CN1025615C (zh) 1994-08-10
JPH02169585A (ja) 1990-06-29
FI93355B (fi) 1994-12-15
DE68921132D1 (de) 1995-03-23
HUT52081A (en) 1990-06-28
PT92032B (pt) 1995-06-30
NO175255B (no) 1994-06-13
RU1782232C (ru) 1992-12-15
NO894184D0 (no) 1989-10-20
CN1042146A (zh) 1990-05-16
GR3015493T3 (en) 1995-06-30
IE66246B1 (en) 1995-12-27
NO175255C (no) 1994-09-21
DK168012B1 (da) 1994-01-17
AU628404B2 (en) 1992-09-17
EP0364941B1 (en) 1995-02-15
FI93355C (fi) 1995-03-27
DK522789A (da) 1990-04-22
AU4356489A (en) 1990-04-26
PH30769A (en) 1997-10-17
HU895383D0 (en) 1990-01-28
ZA897953B (en) 1990-07-25
KR900006287A (ko) 1990-05-07
CZ596189A3 (en) 1995-06-14
CA1333905C (en) 1995-01-10
SU1766253A3 (ru) 1992-09-30
HU207306B (en) 1993-03-29
DE68921132T2 (de) 1995-07-13
IE893400L (en) 1990-04-21
SK279536B6 (sk) 1998-12-02
ATE118489T1 (de) 1995-03-15
DK522789D0 (da) 1989-10-20
SK596189A3 (en) 1998-12-02
JP2851077B2 (ja) 1999-01-27
EP0364941A1 (en) 1990-04-25
ES2068869T3 (es) 1995-05-01
CZ280193B6 (cs) 1995-11-15

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