PT92242A - Processo para a preparacao de um analogo de fluoxetina - Google Patents
Processo para a preparacao de um analogo de fluoxetinaInfo
- Publication number
- PT92242A PT92242A PT92242A PT9224289A PT92242A PT 92242 A PT92242 A PT 92242A PT 92242 A PT92242 A PT 92242A PT 9224289 A PT9224289 A PT 9224289A PT 92242 A PT92242 A PT 92242A
- Authority
- PT
- Portugal
- Prior art keywords
- fluoxetine
- analogue
- preparation
- fluoxetine analogue
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C217/00—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton
- C07C217/02—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C217/48—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated and containing rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US27017788A | 1988-11-14 | 1988-11-14 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PT92242A true PT92242A (pt) | 1990-05-31 |
| PT92242B PT92242B (pt) | 1995-07-06 |
Family
ID=23030229
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT92242A PT92242B (pt) | 1988-11-14 | 1989-11-09 | Processo para a preparacao de um analogo de fluoxetina |
Country Status (15)
| Country | Link |
|---|---|
| EP (1) | EP0369685B1 (pt) |
| JP (1) | JP2776919B2 (pt) |
| CN (1) | CN1042704A (pt) |
| AU (1) | AU622942B2 (pt) |
| CA (1) | CA2002483C (pt) |
| DE (1) | DE68922277T2 (pt) |
| DK (1) | DK560289A (pt) |
| ES (1) | ES2071663T3 (pt) |
| FI (1) | FI895328A7 (pt) |
| HU (1) | HUT58041A (pt) |
| IL (1) | IL92245A0 (pt) |
| NZ (1) | NZ231354A (pt) |
| PT (1) | PT92242B (pt) |
| SU (1) | SU1750417A3 (pt) |
| ZA (1) | ZA898513B (pt) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5250571A (en) * | 1988-11-14 | 1993-10-05 | Eli Lilly And Company | (S)-norfluoxetine in method of inhibiting serotonin uptake |
| FI910897A7 (fi) * | 1990-02-28 | 1991-08-29 | Lilly Co Eli | (S)-norfluoksetiiniin liittyviä parannuksia |
| CA2039103A1 (en) * | 1990-03-29 | 1991-09-30 | David Wayne Robertson | Improvements in and relating to the selective occupation of serotonin 1c receptors |
| US5589511A (en) * | 1990-08-13 | 1996-12-31 | Sepracor Inc. | Method for treating migraine headaches using optically pure S(+) fluoxetine |
| US5708035A (en) * | 1991-02-04 | 1998-01-13 | Sepracor Inc. | Methods of use and compositions of R(-) fluoxetine |
| US5136078A (en) * | 1991-02-26 | 1992-08-04 | Eli Lilly And Company | Synthesis of b-cyanohydrins |
| US5136079A (en) * | 1991-02-26 | 1992-08-04 | Eli Lilly And Company | Regioselective synthesis |
| EP0798285A3 (en) * | 1991-03-01 | 1997-10-08 | Monsanto Company | 3,4,4-Trifluoro-3-butenoic acid or its methyl ester |
| ES2101650B1 (es) * | 1995-06-29 | 1998-01-16 | Lilly Sa | Procedimiento de preparacion de n-metil-3-fenil-3-(p-trifluorometilfenoxi) propilamina. |
| ES2101654B1 (es) * | 1995-07-24 | 1998-01-16 | Lilly Sa | Procedimiento de preparacion de n-metil-3-fenil-3-(p-trifluorometilfe noxi) propilamina. |
| ES2101655B1 (es) * | 1995-07-28 | 1998-01-16 | Lilly Sa | Procedimiento de preparacion de n-metil-3-fenil-3-(p-trifluorometilfe noxi) propilamina. |
| ES2103682B1 (es) * | 1995-09-20 | 1998-04-01 | Lilly Sa | Composicion farmaceutica oral de fluoxetina, solida y con caracteristicas organolepticas mejoradas. |
| ES2120368B1 (es) * | 1996-06-14 | 1999-07-01 | Almirall Prodesfarma Sa | Procedimiento de obtencion de n-metil-3-(p-trifluorometilfenoxi)-3-fenilpropilamina y sus sales farmaceuticamente aceptables. |
| US5936124A (en) * | 1998-06-22 | 1999-08-10 | Sepacor Inc. | Fluoxetine process from benzoylpropionic acid |
| US6025517A (en) * | 1998-08-03 | 2000-02-15 | Sepracor Inc. | Fluoxetine process from benzoylacetonitrile |
| US7034059B2 (en) | 2001-07-02 | 2006-04-25 | Sepracor Inc. | Methods of using norfluoxetine |
| US7439399B2 (en) * | 2004-06-28 | 2008-10-21 | Teva Pharmaceutical Fine Chemicals | Processes for the preparation of atomoxetine hydrochloride |
| ITMI20061987A1 (it) * | 2006-10-16 | 2008-04-17 | Archimica Srl | Processo per la sintesi di arilossipropilammine ed eteroarilossipropilammine. |
| WO2023039408A1 (en) * | 2021-09-07 | 2023-03-16 | The Trustees Of Columbia University In The City Of New York | Methods of treating chronic obstructive pulmonary disease including compounds useful therein |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4626549A (en) | 1974-01-10 | 1986-12-02 | Eli Lilly And Company | Treatment of obesity with aryloxyphenylpropylamines |
| US4313896A (en) * | 1974-01-10 | 1982-02-02 | Eli Lilly And Company | Aryloxyphenylpropylamines |
| US4868344A (en) * | 1988-03-30 | 1989-09-19 | Aldrich-Boranes, Inc. | Novel process of producing phenyl or substituted phenylalkylamine pharmaceutical agents and novel chiral intermediates of high enantiomeric purity useful therein |
-
1989
- 1989-11-08 CA CA002002483A patent/CA2002483C/en not_active Expired - Fee Related
- 1989-11-08 IL IL92245A patent/IL92245A0/xx unknown
- 1989-11-08 ZA ZA898513A patent/ZA898513B/xx unknown
- 1989-11-09 HU HU895848A patent/HUT58041A/hu unknown
- 1989-11-09 PT PT92242A patent/PT92242B/pt not_active IP Right Cessation
- 1989-11-09 SU SU894742384A patent/SU1750417A3/ru active
- 1989-11-09 FI FI895328A patent/FI895328A7/fi not_active Application Discontinuation
- 1989-11-09 DK DK560289A patent/DK560289A/da not_active Application Discontinuation
- 1989-11-09 AU AU44516/89A patent/AU622942B2/en not_active Ceased
- 1989-11-10 DE DE68922277T patent/DE68922277T2/de not_active Expired - Fee Related
- 1989-11-10 NZ NZ231354A patent/NZ231354A/en unknown
- 1989-11-10 JP JP1293785A patent/JP2776919B2/ja not_active Expired - Lifetime
- 1989-11-10 EP EP89311634A patent/EP0369685B1/en not_active Expired - Lifetime
- 1989-11-10 CN CN89108468A patent/CN1042704A/zh active Pending
- 1989-11-10 ES ES89311634T patent/ES2071663T3/es not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| ZA898513B (en) | 1991-07-31 |
| FI895328A7 (fi) | 1990-05-15 |
| HUT58041A (en) | 1992-01-28 |
| JP2776919B2 (ja) | 1998-07-16 |
| EP0369685A3 (en) | 1991-03-27 |
| PT92242B (pt) | 1995-07-06 |
| DE68922277T2 (de) | 1995-09-21 |
| CN1042704A (zh) | 1990-06-06 |
| JPH02193951A (ja) | 1990-07-31 |
| CA2002483C (en) | 1999-08-17 |
| EP0369685B1 (en) | 1995-04-19 |
| NZ231354A (en) | 1991-05-28 |
| CA2002483A1 (en) | 1990-05-14 |
| AU622942B2 (en) | 1992-04-30 |
| EP0369685A2 (en) | 1990-05-23 |
| DK560289D0 (da) | 1989-11-09 |
| SU1750417A3 (ru) | 1992-07-23 |
| DK560289A (da) | 1990-05-15 |
| IL92245A0 (en) | 1990-07-26 |
| HU895848D0 (en) | 1990-01-28 |
| ES2071663T3 (es) | 1995-07-01 |
| DE68922277D1 (de) | 1995-05-24 |
| AU4451689A (en) | 1990-05-17 |
| FI895328A0 (fi) | 1989-11-09 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM3A | Annulment or lapse |
Free format text: LAPSE DUE TO NON-PAYMENT OF FEES Effective date: 19960831 |