PT92375A - Processo para a preparacao de nucleosidos pirimidina substituida em 5 por propinilo esteroficados e de formulacoes farmaceuticos anti-virais que os contem - Google Patents

Processo para a preparacao de nucleosidos pirimidina substituida em 5 por propinilo esteroficados e de formulacoes farmaceuticos anti-virais que os contem

Info

Publication number
PT92375A
PT92375A PT92375A PT9237589A PT92375A PT 92375 A PT92375 A PT 92375A PT 92375 A PT92375 A PT 92375A PT 9237589 A PT9237589 A PT 9237589A PT 92375 A PT92375 A PT 92375A
Authority
PT
Portugal
Prior art keywords
preparation
pharmaceutical formulations
steroficated
propinyl
contain
Prior art date
Application number
PT92375A
Other languages
English (en)
Other versions
PT92375B (pt
Inventor
Saad George Rahim
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wellcome Found filed Critical Wellcome Found
Publication of PT92375A publication Critical patent/PT92375A/pt
Publication of PT92375B publication Critical patent/PT92375B/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06—Pyrimidine radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/20—Antivirals for DNA viruses
    • A61P31/22—Antivirals for DNA viruses for herpes viruses

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Virology (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
PT92375A 1988-11-23 1989-11-22 Processo para a preparacao de nucleosidos pirimidina substituida em 5 por propinilo esteroficados e de formulacoes farmaceuticos anti-virais que os contem PT92375B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB888827339A GB8827339D0 (en) 1988-11-23 1988-11-23 Antiviral compounds

Publications (2)

Publication Number Publication Date
PT92375A true PT92375A (pt) 1990-05-31
PT92375B PT92375B (pt) 1995-07-18

Family

ID=10647307

Family Applications (1)

Application Number Title Priority Date Filing Date
PT92375A PT92375B (pt) 1988-11-23 1989-11-22 Processo para a preparacao de nucleosidos pirimidina substituida em 5 por propinilo esteroficados e de formulacoes farmaceuticos anti-virais que os contem

Country Status (25)

Country Link
EP (1) EP0375164B1 (pt)
JP (1) JPH0753748B2 (pt)
CN (1) CN1022570C (pt)
AT (1) ATE104676T1 (pt)
AU (1) AU620471B2 (pt)
CA (1) CA2003607A1 (pt)
DD (1) DD289534A5 (pt)
DE (1) DE68914809T2 (pt)
DK (1) DK586489A (pt)
ES (1) ES2063147T3 (pt)
FI (1) FI895572A7 (pt)
GB (1) GB8827339D0 (pt)
HU (1) HU204842B (pt)
IE (1) IE893731L (pt)
IL (1) IL92402A0 (pt)
MC (1) MC2071A1 (pt)
MY (1) MY104976A (pt)
NO (1) NO171168C (pt)
NZ (1) NZ231478A (pt)
PH (1) PH26745A (pt)
PL (1) PL162956B1 (pt)
PT (1) PT92375B (pt)
RU (1) RU1831486C (pt)
YU (1) YU47096B (pt)
ZA (1) ZA898926B (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK0465297T3 (da) * 1990-07-04 1996-02-19 Merrell Pharma Inc 9-Purinylphosphonsyre-derivater
US5494912A (en) * 1991-06-26 1996-02-27 Merrell Pharmaceuticals Inc. 9-purinyl phosphonic acid derivitives for treating gout
GB9125271D0 (en) * 1991-11-27 1992-01-29 Wellcome Found Anti-hbv pyrimidine nucleoside
WO2022008025A1 (en) * 2020-07-05 2022-01-13 Since & Technology Development Fund Authority 2-hydroxyiminopyrimidine nucleosides and derivitives and antiviral uses thereto

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4211773A (en) * 1978-10-02 1980-07-08 Sloan Kettering Institute For Cancer Research 5-Substituted 1-(2'-Deoxy-2'-substituted-β-D-arabinofuranosyl)pyrimidine nucleosides
GB8629892D0 (en) * 1986-12-15 1987-01-28 Wellcome Found Antiviral compounds
EP0346108A3 (en) * 1988-06-09 1991-04-24 The Wellcome Foundation Limited Anti-infective nucleosides

Also Published As

Publication number Publication date
YU221289A (en) 1991-02-28
MY104976A (en) 1994-07-30
RU1831486C (ru) 1993-07-30
DK586489A (da) 1990-05-24
NZ231478A (en) 1992-09-25
PL162956B1 (pl) 1994-01-31
CN1022570C (zh) 1993-10-27
CA2003607A1 (en) 1990-05-23
CN1042916A (zh) 1990-06-13
HU204842B (en) 1992-02-28
DK586489D0 (da) 1989-11-22
NO894658L (no) 1990-05-25
IE893731L (en) 1990-05-23
GB8827339D0 (en) 1988-12-29
IL92402A0 (en) 1990-07-26
ES2063147T3 (es) 1995-01-01
JPH0327394A (ja) 1991-02-05
AU620471B2 (en) 1992-02-20
EP0375164B1 (en) 1994-04-20
MC2071A1 (fr) 1990-10-03
PH26745A (en) 1992-09-28
DD289534A5 (de) 1991-05-02
NO171168C (no) 1993-02-03
JPH0753748B2 (ja) 1995-06-07
HUT52110A (en) 1990-06-28
NO171168B (no) 1992-10-26
ZA898926B (en) 1991-07-31
DE68914809D1 (de) 1994-05-26
AU4544289A (en) 1990-06-14
HU896136D0 (en) 1990-02-28
EP0375164A1 (en) 1990-06-27
FI895572A7 (fi) 1990-05-24
NO894658D0 (no) 1989-11-22
DE68914809T2 (de) 1994-08-11
FI895572A0 (fi) 1989-11-22
PT92375B (pt) 1995-07-18
YU47096B (sh) 1994-12-28
ATE104676T1 (de) 1994-05-15

Similar Documents

Publication Publication Date Title
PT100199A (pt) Combinacao antiviral de nucleosidos e processo para a sua preparacao
FI20001231A7 (fi) 2-Deoksi-2,3-didehydro-N-asetyylineuramiinihapon johdannaisia ja niiden analogeja ja niiden käyttö antiviraalisina aineina
DK224286D0 (da) 2',3'-dideoxy-nucleosider
NO2007016I2 (no) Nelarabin eller et farmasoytisk akseptabelt salt derav ( nelarabin=9-(beta-D-arabinofuranosyl-2-amino-6-metoksy-9H-purin)
DK0513917T4 (da) Antivirale kombinationer indeholdende nukleosidanaloger
PT94645A (pt) Processo para a preparacao de derivados de aminopirimidina com actividade fungicida e de composicoes fungicidas que os contem
PT97478A (pt) Processo de producao de derivados n-(3-fluoro-2-fosfonilmetoxipropilo) de bases puricas e pirimidicas heterociclicas e de composicoes farmaceuticas que os contem
PT84478B (pt) Processo para a preparacao de derivados de pirazolo-{3,4-d}-pirimidina e de composicoes farmaceuticas que os contem
PT90972A (pt) Processo para a preparacao de inibidores de ribonucleotido-redutase, nomeadamente, de tiocarbono-hidrazonas e/ou hidrazinas substituidas e seus derivados e de composicoes farmaceuticas que os contem em associacao com outros compostos antivirais
PT98121A (pt) Processo para a preparacao de novos 3,3'-ditio-bis (acidos propionicos) e seus esteres e de composicoes farmaceuticas que os contem
DE68900760D1 (de) Virushemmende nukleosidmischung.
PT99835A (pt) Processo para a preparacao de esteres da castanospermina com accao antiviral
PT91153A (pt) Processo para a preparacao de um ester de 9-(2-hidroxi-etoxi-metil)guanina e de composicoes que contem
DK291390A (da) Terapeutiske anvendelser af 2',5'-oligoadenylatderivater
PT87004A (pt) Process for the preparation of compositions for the treatment of viral infections and composites 3'-azide-2',3'-didesoxy-in osine and 3'-fluoro-2',3'-didesoxyguanosine
FI895572A0 (fi) Antivirala foereningar.
PT98186A (pt) Processo para a preparacao de purinil- e de pirimidinil-tetra-hidrofuranos e de composicoes farmaceuticas que os contem
BR9205877A (pt) Processo e composiçao para o tratamento de infecçoes por herpes.
DK0459176T3 (da) Oligophosphater med antiviral virkning
PT82258B (pt) Processo de preparacao de composicoes compreendendo interferao humano e nonilfenoxipolietanol para o tratamento de infeccoes virais por herpes simplex em humanos

Legal Events

Date Code Title Description
MM3A Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 19960930