PT94805A - Processo para a preparacao de um macrolido antiparasitario relacionado com as milbemicinas - Google Patents

Processo para a preparacao de um macrolido antiparasitario relacionado com as milbemicinas

Info

Publication number: PT94805A
Authority: PT; Portugal
Prior art keywords: milbemicines; antiparasitary; preparation; macrolide; macrolide related
Prior art date: 1989-07-26

Application number

PT94805A

Other languages

English (en)

Other versions

PT94805B (pt

Inventor

Hiroshi Maeda

Satoshi Nishiyama

Yasuhiro Kojiima

David Austen Perry

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1989-07-26

Filing date

1990-07-24

Publication date

1991-03-20

1990-07-24 Application filed by Pfizer filed Critical Pfizer

1991-03-20 Publication of PT94805A publication Critical patent/PT94805A/pt

1997-05-28 Publication of PT94805B publication Critical patent/PT94805B/pt

Links

239000003120 macrolide antibiotic agent Substances 0.000 title 1
241000238876 Acari Species 0.000 abstract 1
241000238631 Hexapoda Species 0.000 abstract 1
241000244206 Nematoda Species 0.000 abstract 1
241000970979 Streptomyces griseochromogenes Species 0.000 abstract 1
241000607479 Yersinia pestis Species 0.000 abstract 1
239000003242 anti bacterial agent Substances 0.000 abstract 1
239000003096 antiparasitic agent Substances 0.000 abstract 1
229940125687 antiparasitic agent Drugs 0.000 abstract 1
230000003115 biocidal effect Effects 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
244000078703 ectoparasite Species 0.000 abstract 1
YYJNOYZRYGDPNH-MFKUBSTISA-N fenpyroximate Chemical compound C=1C=C(C(=O)OC(C)(C)C)C=CC=1CO/N=C/C=1C(C)=NN(C)C=1OC1=CC=CC=C1 YYJNOYZRYGDPNH-MFKUBSTISA-N 0.000 abstract 1
230000004151 fermentation Effects 0.000 abstract 1
238000000855 fermentation Methods 0.000 abstract 1
244000005700 microbiome Species 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
- C12P—FERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
- C12P19/00—Preparation of compounds containing saccharide radicals
- C12P19/44—Preparation of O-glycosides, e.g. glucosides
- C12P19/60—Preparation of O-glycosides, e.g. glucosides having an oxygen of the saccharide radical directly bound to a non-saccharide heterocyclic ring or a condensed ring system containing a non-saccharide heterocyclic ring, e.g. coumermycin, novobiocin
- C12P19/62—Preparation of O-glycosides, e.g. glucosides having an oxygen of the saccharide radical directly bound to a non-saccharide heterocyclic ring or a condensed ring system containing a non-saccharide heterocyclic ring, e.g. coumermycin, novobiocin the hetero ring having eight or more ring members and only oxygen as ring hetero atoms, e.g. erythromycin, spiramycin, nystatin
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/22—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains four or more hetero rings
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
- A—HUMAN NECESSITIES
- A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
- A23K—FODDER
- A23K20/00—Accessory food factors for animal feeding-stuffs
- A23K20/10—Organic substances
- A23K20/195—Antibiotics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics

Landscapes

Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Zoology (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Polymers & Plastics (AREA)
Wood Science & Technology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Animal Husbandry (AREA)
Dentistry (AREA)
Plant Pathology (AREA)
Tropical Medicine & Parasitology (AREA)
Environmental Sciences (AREA)
Pest Control & Pesticides (AREA)
Agronomy & Crop Science (AREA)
Food Science & Technology (AREA)
Bioinformatics & Cheminformatics (AREA)
Obesity (AREA)
Genetics & Genomics (AREA)
Diabetes (AREA)
Biotechnology (AREA)
Microbiology (AREA)
Biochemistry (AREA)
General Engineering & Computer Science (AREA)
Hematology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Micro-Organisms Or Cultivation Processes Thereof (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

PT94805A 1989-07-26 1990-07-24 Processo para a preparacao de um macrolido antiparasitario relacionado com as milbemicinas PT94805B (pt)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GB898917064A GB8917064D0 (en)	1989-07-26	1989-07-26	Antiparasitic agent

Publications (2)

Publication Number	Publication Date
PT94805A true PT94805A (pt)	1991-03-20
PT94805B PT94805B (pt)	1997-05-28

Family

ID=10660639

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PT94805A PT94805B (pt)	1989-07-26	1990-07-24	Processo para a preparacao de um macrolido antiparasitario relacionado com as milbemicinas

Country Status (19)

Country	Link
US (1)	US5073567A (pt)
EP (1)	EP0410615B1 (pt)
JP (1)	JPH0692414B2 (pt)
KR (1)	KR930005872B1 (pt)
AT (1)	ATE100106T1 (pt)
AU (1)	AU615620B2 (pt)
CA (1)	CA2021894C (pt)
DE (1)	DE69005935T2 (pt)
DK (1)	DK0410615T3 (pt)
ES (1)	ES2062378T3 (pt)
FI (1)	FI94262C (pt)
GB (1)	GB8917064D0 (pt)
HU (1)	HUT57832A (pt)
IE (1)	IE63136B1 (pt)
IL (1)	IL95133A (pt)
NO (1)	NO903312L (pt)
NZ (1)	NZ234644A (pt)
PT (1)	PT94805B (pt)
ZA (1)	ZA905842B (pt)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB9125818D0 (en) *	1991-12-04	1992-02-05	Pfizer Ltd	Antiparasitic agents
GB9205007D0 (en) *	1992-03-07	1992-04-22	Pfizer Ltd	Antiparasitic agents
US5707817A (en) *	1993-02-05	1998-01-13	Colorado State University Research Foundation	Carbohydrate-based vaccine and diagnostic reagent for trichinosis
US5541075A (en) *	1993-02-05	1996-07-30	Heska Corporation	Carbohydrate-based vaccine and diagnostic reagent for trichinosis
EP0739344B1 (en) *	1994-01-14	1998-11-11	Pfizer Inc.	Antiparasitic pyrrolobenzoxazine compounds
GB9402916D0 (en) *	1994-02-16	1994-04-06	Pfizer Ltd	Antiparasitic agents
FR2754541B1 (fr) *	1996-10-15	1998-12-24	Air Liquide	Procede et installation pour la separation d'un melange d'hydrogene et/ou d'au moins un hydrocarbure et/ou d'azote et/ou d'oxyde de carbone
AU9785698A (en)	1997-10-02	1999-04-27	Microcide Pharmaceuticals, Inc.	Fungal efflux pump inhibitors
GB9825402D0 (en)	1998-11-19	1999-01-13	Pfizer Ltd	Antiparasitic formulations
CA2460692C (en)	2001-09-17	2012-12-18	Eli Lilly And Company	Pesticidal formulations
EP2327410A1 (en)	2009-10-28	2011-06-01	Consiglio Nazionale Delle Ricerche - Infm Istituto Nazionale Per La Fisica Della Materia	Avermectins and milbemycins for the treatment of flavivirus infections
EP2886640A1 (en)	2013-12-18	2015-06-24	Riga Technical University	Process for isolation of milbemycins A3 and A4

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS4914624A (pt) *	1972-06-08	1974-02-08
DK165119C (da) *	1984-06-05	1993-03-01	American Cyanamid Co	Antibiotiske forbindelser betegnet ll-f28249alfa, beta, gamma, delta, epsilon, zeta, eta, theta, iota, kappa, my og ny og pharmaceutisk or pharmakologisk acceptable salte deraf samt fremgangsmaade til deres fremstilling
US4587247A (en) *	1985-02-25	1986-05-06	Merck & Co., Inc.	Substituted and unsubstituted 13-(alkoxy)methoxy derivatives of the avermectin aglycones, compositions and use
NZ215917A (en) *	1985-05-02	1989-10-27	Merck & Co Inc	22-oh milbemycin derivatives and parasiticidal compositions
DE3750495T2 (de) *	1986-07-24	1995-02-23	Beecham Group Plc	Milbemycin-Derivate mit parasitenabtötender Aktivität, ein Verfahren zu ihrer Herstellung und die sie enthaltenden Zusammensetzungen.

1989
- 1989-07-26 GB GB898917064A patent/GB8917064D0/en active Pending
1990
- 1990-07-13 DE DE90307708T patent/DE69005935T2/de not_active Expired - Fee Related
- 1990-07-13 DK DK90307708.9T patent/DK0410615T3/da active
- 1990-07-13 AT AT90307708T patent/ATE100106T1/de not_active IP Right Cessation
- 1990-07-13 ES ES90307708T patent/ES2062378T3/es not_active Expired - Lifetime
- 1990-07-13 EP EP90307708A patent/EP0410615B1/en not_active Expired - Lifetime
- 1990-07-19 IL IL9513390A patent/IL95133A/en not_active IP Right Cessation
- 1990-07-24 PT PT94805A patent/PT94805B/pt not_active IP Right Cessation
- 1990-07-24 CA CA002021894A patent/CA2021894C/en not_active Expired - Fee Related
- 1990-07-25 US US07/557,885 patent/US5073567A/en not_active Expired - Fee Related
- 1990-07-25 FI FI903727A patent/FI94262C/fi not_active IP Right Cessation
- 1990-07-25 ZA ZA905842A patent/ZA905842B/xx unknown
- 1990-07-25 AU AU59849/90A patent/AU615620B2/en not_active Ceased
- 1990-07-25 IE IE269490A patent/IE63136B1/en not_active IP Right Cessation
- 1990-07-25 KR KR1019900011286A patent/KR930005872B1/ko not_active Expired - Fee Related
- 1990-07-25 NZ NZ234644A patent/NZ234644A/xx unknown
- 1990-07-25 NO NO90903312A patent/NO903312L/no unknown
- 1990-07-26 JP JP2198945A patent/JPH0692414B2/ja not_active Expired - Lifetime
- 1990-07-26 HU HU904642A patent/HUT57832A/hu unknown

Also Published As

Publication number	Publication date
IE902694A1 (en)	1991-02-27
AU5984990A (en)	1991-01-31
JPH0368581A (ja)	1991-03-25
DE69005935T2 (de)	1994-04-28
NO903312D0 (no)	1990-07-25
AU615620B2 (en)	1991-10-03
IL95133A (en)	1994-11-11
FI903727A0 (fi)	1990-07-25
EP0410615B1 (en)	1994-01-12
US5073567A (en)	1991-12-17
HU904642D0 (en)	1991-01-28
KR930005872B1 (ko)	1993-06-25
JPH0692414B2 (ja)	1994-11-16
ES2062378T3 (es)	1994-12-16
GB8917064D0 (en)	1989-09-13
ATE100106T1 (de)	1994-01-15
PT94805B (pt)	1997-05-28
DE69005935D1 (de)	1994-02-24
NO903312L (no)	1991-01-28
KR910003111A (ko)	1991-02-26
CA2021894A1 (en)	1991-01-27
EP0410615A1 (en)	1991-01-30
NZ234644A (en)	1991-11-26
FI94262C (fi)	1995-08-10
FI94262B (fi)	1995-04-28
IE63136B1 (en)	1995-03-22
HUT57832A (en)	1991-12-30
DK0410615T3 (da)	1994-02-14
CA2021894C (en)	1996-09-17
ZA905842B (en)	1992-03-25

Legal Events

Date

Code

Title

Description

1991-03-20

BB1A

Laying open of patent application

Effective date: 19901019

1997-05-30

FG3A

Patent granted, date of granting

Effective date: 19970214

2000-12-29

MM3A

Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 20000831

Publication	Publication Date	Title
OA09249A (fr)	1992-06-30	Composés de macrolides.
PT89806A (pt)	1989-10-04	Processo de preparacao de antibioticos macrolidos antiparasiticos
HU904642D0 (en)	1991-01-28	Process for producing active agent against parasites
KR940011630A (ko)	1994-06-21	구충제 화합물 제조용의 스트렙토마이세스 균주 및 이의 사용방법
BR8803390A (pt)	1989-01-24	Antibioticos ab-006,processo para preparacao dos antibioticos ab-006,microorganismo,cultura biologicamente pura do microorganismo,composto selecionado e composicao fungicidas e ou como inseticida
ES2068178T3 (es)	1995-04-16	Nuevos derivados 23-imino de compuesto 23-ceto.
AU584946B2 (en)	1989-06-08	Organic chemical compound, microbiological processes for its preparation, and its use
CA2024825A1 (en)	1991-03-12	13-halo-23-imino derivatives of ll-f28249 compounds and their use as endo- and ectoparasiticidal insecticidal, acaricidal and nematocidal agents
PT90621A (pt)	1989-11-30	Processo para a preparacao de novas avermectinas com um anel furano clivado e um grupo hidroxi 8a
BR9403200A (pt)	1995-04-11	Derivado de amido-tiofosfato, composição para controlar insetos, nematódeos ou ácaros, processo para controlar insetos, namatódeos ou ácaros, uso de derivados de amido-tiofosfato, e, processo para produzir um derivado de amido-tiofosfato
ES506478A0 (es)	1983-02-16	Un procedimiento para la preparacion de nuevas lactonas macrociclicas.
CA2024824A1 (en)	1991-06-23	13-alkyl-23-imino derivatives of ll-f28249 compounds and their use as endo- and ectoparasiticidal insecticidal, acaricidal and nematocidal agents
AU3836593A (en)	1993-11-11	Active principle based on avermectins, related strain and process for the preparation thereof, as well as veterinary composition containing it
PT93258A (pt)	1990-08-31	Processo para a preparacao de um antibiotico de eter policiclico acidico
DK0412464T3 (da)	1992-12-07	Butalactin, en fremgangsmåde til dets fremstilling og dets anvendelse som lægemiddel
BR8802952A (pt)	1989-01-10	Composto,processo para a preparacao de um composto,composicao inseticida ou acaricida e processo para combater pestes de insetos ou acarinos