PT964855E - Processo para a fabricacao de derivados substituidos de pirimidina - Google Patents

Processo para a fabricacao de derivados substituidos de pirimidina

Info

Publication number
PT964855E
PT964855E PT98901950T PT98901950T PT964855E PT 964855 E PT964855 E PT 964855E PT 98901950 T PT98901950 T PT 98901950T PT 98901950 T PT98901950 T PT 98901950T PT 964855 E PT964855 E PT 964855E
Authority
PT
Portugal
Prior art keywords
pct
pyrimidine derivatives
substituted pyrimidine
manufacture
sec
Prior art date
Application number
PT98901950T
Other languages
English (en)
Inventor
Stucky Dr Gerhard
Beat Schmidt
Original Assignee
Lonza Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lonza Ag filed Critical Lonza Ag
Publication of PT964855E publication Critical patent/PT964855E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32One oxygen, sulfur or nitrogen atom
    • C07D239/34One oxygen atom
    • C07D239/36One oxygen atom as doubly bound oxygen atom or as unsubstituted hydroxy radical
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32One oxygen, sulfur or nitrogen atom
    • C07D239/38One sulfur atom
    • C07D239/40One sulfur atom as doubly bound sulfur atom or as unsubstituted mercapto radical

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
PT98901950T 1997-01-13 1998-01-08 Processo para a fabricacao de derivados substituidos de pirimidina PT964855E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH5597 1997-01-13

Publications (1)

Publication Number Publication Date
PT964855E true PT964855E (pt) 2002-04-29

Family

ID=4178290

Family Applications (1)

Application Number Title Priority Date Filing Date
PT98901950T PT964855E (pt) 1997-01-13 1998-01-08 Processo para a fabricacao de derivados substituidos de pirimidina

Country Status (11)

Country Link
US (1) US6114527A (pt)
EP (1) EP0964855B1 (pt)
JP (1) JP4143740B2 (pt)
AT (1) ATE207062T1 (pt)
AU (1) AU5862398A (pt)
CA (1) CA2275400C (pt)
DE (1) DE59801768D1 (pt)
DK (1) DK0964855T3 (pt)
ES (1) ES2165668T3 (pt)
PT (1) PT964855E (pt)
WO (1) WO1998030549A1 (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2240093T3 (es) * 1999-04-15 2005-10-16 Basf Aktiengesellschaft Procedimiento para la preparacion de pirimidinas substituidas.
US6281358B1 (en) 1999-04-15 2001-08-28 American Cyanamid Company Process for the preparation of substituted pyrimidines
US8299035B2 (en) 2008-05-15 2012-10-30 Taisho Pharmaceutucal Co., Ltd. 10a-azalide compound having 4-membered ring structure
EP3530645B1 (en) * 2016-10-19 2023-12-06 Agc Inc. Method for producing nitrogen-containing compound

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1806867C3 (de) * 1968-11-04 1974-07-18 Byk-Gulden Lomberg Chemische Fabrik Gmbh, 7750 Konstanz Verfahren zur Herstellung substituierter 4-Hydroxy pyrimidine
DE3811621A1 (de) * 1988-04-07 1989-10-26 Merck Patent Gmbh Verfahren zur herstellung von 1h-imidazol-5-carbon-saeureestern oder -nitrilen und von pyrrol-3,4-carbonsaeureestern oder -nitrilen sowie verwendung der hergestellten verbindungen zur synthese von pilocarpin

Also Published As

Publication number Publication date
JP4143740B2 (ja) 2008-09-03
US6114527A (en) 2000-09-05
ATE207062T1 (de) 2001-11-15
CA2275400A1 (en) 1998-07-16
EP0964855A1 (de) 1999-12-22
JP2001508058A (ja) 2001-06-19
WO1998030549A1 (de) 1998-07-16
EP0964855B1 (de) 2001-10-17
DE59801768D1 (de) 2001-11-22
ES2165668T3 (es) 2002-03-16
CA2275400C (en) 2008-07-15
AU5862398A (en) 1998-08-03
DK0964855T3 (da) 2001-11-19

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