PT97800A - Processo para a preparacao duma composicao repelente de insectos e acaros contendo derivados de morfolino-ureia - Google Patents

Processo para a preparacao duma composicao repelente de insectos e acaros contendo derivados de morfolino-ureia

Info

Publication number
PT97800A
PT97800A PT97800A PT9780091A PT97800A PT 97800 A PT97800 A PT 97800A PT 97800 A PT97800 A PT 97800A PT 9780091 A PT9780091 A PT 9780091A PT 97800 A PT97800 A PT 97800A
Authority
PT
Portugal
Prior art keywords
ureia
acars
insects
derivatives
preparation
Prior art date
Application number
PT97800A
Other languages
English (en)
Other versions
PT97800B (pt
Inventor
Bernd-Wieland Krueger
Guenther Nentwig
Klaus Stroech
Peter Hoever
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of PT97800A publication Critical patent/PT97800A/pt
Publication of PT97800B publication Critical patent/PT97800B/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
    • C07D295/205—Radicals derived from carbonic acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
    • C07D295/215—Radicals derived from nitrogen analogues of carbonic acid
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A01N47/38—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the group >N—CO—N< where at least one nitrogen atom is part of a heterocyclic ring; Thio analogues thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14—The ring being saturated

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Veterinary Medicine (AREA)
  • Pest Control & Pesticides (AREA)
  • Animal Behavior & Ethology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
PT97800A 1990-06-06 1991-05-29 Processo para a preparacao duma composicao repelente de insectos e acaros contendo derivados de morfolino-ureia PT97800B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4018070A DE4018070A1 (de) 1990-06-06 1990-06-06 Morpholinoharnstoff-derivate

Publications (2)

Publication Number Publication Date
PT97800A true PT97800A (pt) 1992-03-31
PT97800B PT97800B (pt) 1998-10-30

Family

ID=6407857

Family Applications (1)

Application Number Title Priority Date Filing Date
PT97800A PT97800B (pt) 1990-06-06 1991-05-29 Processo para a preparacao duma composicao repelente de insectos e acaros contendo derivados de morfolino-ureia

Country Status (18)

Country Link
US (1) US5218002A (pt)
EP (1) EP0467045B1 (pt)
JP (1) JPH04235978A (pt)
KR (1) KR920000741A (pt)
AT (1) ATE163644T1 (pt)
AU (1) AU644438B2 (pt)
BR (1) BR9102322A (pt)
CA (1) CA2043797A1 (pt)
DE (2) DE4018070A1 (pt)
EG (1) EG19884A (pt)
ES (1) ES2112845T3 (pt)
HU (1) HU216891B (pt)
IL (1) IL98340A0 (pt)
NZ (1) NZ238351A (pt)
PT (1) PT97800B (pt)
TR (1) TR26723A (pt)
TW (1) TW198028B (pt)
ZA (1) ZA914278B (pt)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT400566B (de) * 1993-01-22 1996-01-25 Chemie Linz Gmbh Verwendung und verfahren zur herstellung von n-cyclischen und n,n'-dicyclischen harnstoffen
DE4302860A1 (de) * 1993-01-22 1994-08-04 Chemie Linz Deutschland N-Cyclische und N,N'dicyclische Harnstoffe
JPH09510184A (ja) * 1993-12-23 1997-10-14 ツッチ アソシエイツ,インコーポレイティド 徐放性昆虫忌避製剤及びその利用
US6015570A (en) * 1993-12-23 2000-01-18 Tucci Associates, Inc. Slow-release insect-repellent compositions and uses
EP0850222B1 (en) * 1996-06-29 2003-05-28 Samjin Pharmaceutical Co., Ltd. Piperazine derivatives and process for the preparation thereof
DK1087952T3 (da) 1998-06-18 2004-10-04 Novartis Ag Banzazolforbindelser samt deres anvendelse
DE10032877A1 (de) * 2000-07-06 2002-02-07 Bayer Ag Anthelmintika zur Verhinderung von parasitären Infektionen bei Mensch und Tier III
BRPI0516132A (pt) * 2004-10-07 2007-12-04 Vitae Pharmaceuticals Inc compostos, composição destes, método de antagonização de uma ou mais proteases aspárticas e método para tratar ou melhorar um distúrbio mediado por protease aspártica
TWI411607B (zh) * 2005-11-14 2013-10-11 Vitae Pharmaceuticals Inc 天門冬胺酸蛋白酶抑制劑
JP2010503682A (ja) * 2006-09-18 2010-02-04 ビテ ファーマシューティカルズ, インコーポレイテッド レニン阻害剤としてのピペリジン誘導体
CL2007002689A1 (es) 2006-09-18 2008-04-18 Vitae Pharmaceuticals Inc Compuestos derivados de piperidin-1-carboxamida, inhibidores de la renina; compuestos intermediarios; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como hipertension, insuficiencia cardiaca, fibrosis cardiaca, entre otras.
WO2009096996A1 (en) * 2007-06-20 2009-08-06 Smithkline Beecham Corporation Renin inhibitors
US20100160424A1 (en) * 2007-06-20 2010-06-24 Baldwin John J Renin inhibitors
US8741874B2 (en) * 2007-11-07 2014-06-03 Bayer Cropscience Lp Insecticidal compositions with disinfectant
WO2009154766A1 (en) * 2008-06-20 2009-12-23 Vitae Pharmaceuticals, Inc. Renin inhibitors and method of use thereof
CN102088850A (zh) * 2008-06-26 2011-06-08 生命医药公司 甲基2-((r)-(3-氯苯基)((r)-1-((s)-2-(甲氨基)-3((r)-四氢-2h-吡喃-3-基)丙基氨甲酰基)哌啶-3-基)甲氧基)氨基甲酸乙酯的盐
AR077692A1 (es) * 2009-08-06 2011-09-14 Vitae Pharmaceuticals Inc Sales de 2-((r)-(3-clorofenil) ((r)-1-((s) -2-(metilamino)-3-((r)-tetrahidro-2h-piran-3-il) propilcarbamoil) piperidin -3-il) metoxi) etilcarbamato de metilo
WO2012104865A1 (en) * 2011-01-28 2012-08-09 Director General, Defence Research & Development Organisation (Drdo) N, n- dialkyl -morpholin- 4 - carboxamide compounds as insect repelling agents and a process for their preparation
WO2013065059A1 (en) * 2011-11-04 2013-05-10 Director General, Defence Research & Development Organisation Process for preparation of n,n-di substituted carboxamides
GB201603581D0 (en) 2016-03-01 2016-04-13 Spts Technologies Ltd Plasma processing apparatus

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3161676A (en) * 1962-05-21 1964-12-15 Berkeley Chemical Corp Preparation of substituted alkyl ureas
US3296306A (en) * 1965-03-04 1967-01-03 Upjohn Co Process for 2, 2-diaryl-nu-substituted acetamides
FR2050522A5 (en) * 1969-06-17 1971-04-02 Aries Robert Pesticidal carbamoyl morpholines
DE2206366C3 (de) * 1971-02-16 1980-10-23 Ciba-Geigy Ag, Basel (Schweiz) Verfahren zur Herstellung von substituierten Diaminocarbonylderivaten
US4025652A (en) * 1975-03-31 1977-05-24 William H. Rorer, Inc. Amidinoureas
US4052385A (en) * 1975-10-21 1977-10-04 The Dow Chemical Company Certain n-(2-hydroxyethyl)heteroiminocarboxamides
US4400512A (en) * 1976-12-17 1983-08-23 Rohm And Haas Company Azaspiro compounds
US4356180A (en) * 1979-02-02 1982-10-26 The United States Of America As Represented By The Secretary Of Agriculture Insect repellants
US4389401A (en) * 1979-07-10 1983-06-21 Rohm And Haas Company Arthropod repellents
EP0085286B1 (en) * 1981-12-17 1986-04-30 Aktiebolaget Hässle Para-substituted 3-phenoxy-1-carbonylaminoalkylamino-propan-2-ols having beta receptor blocking properties
DE3314435A1 (de) * 1983-04-21 1984-10-25 Basf Ag, 6700 Ludwigshafen Verfahren zur herstellung von 1,1-disubstituierten thioharnstoffen
JPS61215381A (ja) * 1985-03-22 1986-09-25 Ube Ind Ltd ベンゾオキサジン誘導体および除草剤
DE3539994A1 (de) * 1985-11-12 1987-05-14 Bayer Ag Herbizide mittel enthaltend photosynthesehemmer-herbizide in kombination mit harnstoffderivaten

Also Published As

Publication number Publication date
TW198028B (pt) 1993-01-11
EP0467045A2 (de) 1992-01-22
EP0467045B1 (de) 1998-03-04
AU644438B2 (en) 1993-12-09
EG19884A (en) 1996-10-31
KR920000741A (ko) 1992-01-29
DE4018070A1 (de) 1991-12-12
IL98340A0 (en) 1992-07-15
PT97800B (pt) 1998-10-30
ZA914278B (en) 1992-03-25
NZ238351A (en) 1992-06-25
ATE163644T1 (de) 1998-03-15
HU216891B (hu) 1999-10-28
EP0467045A3 (en) 1992-02-05
US5218002A (en) 1993-06-08
BR9102322A (pt) 1992-01-07
TR26723A (tr) 1995-05-15
ES2112845T3 (es) 1998-04-16
CA2043797A1 (en) 1991-12-07
DE59108943D1 (de) 1998-04-09
HUT57548A (en) 1991-12-30
JPH04235978A (ja) 1992-08-25
AU7806491A (en) 1991-12-12

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Legal Events

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BB1A Laying open of patent application

Effective date: 19911122

FG3A Patent granted, date of granting

Effective date: 19980721

MM3A Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 20010131