RS52304B - Supstituisani indolil alkil amino derivati kao novi inhibitori histon deacetilaze - Google Patents

Supstituisani indolil alkil amino derivati kao novi inhibitori histon deacetilaze

Info

Publication number
RS52304B
RS52304B RS20120165A RSP20120165A RS52304B RS 52304 B RS52304 B RS 52304B RS 20120165 A RS20120165 A RS 20120165A RS P20120165 A RSP20120165 A RS P20120165A RS 52304 B RS52304 B RS 52304B
Authority
RS
Serbia
Prior art keywords
formula
alkyl
mol
compound
hydrogen
Prior art date
Application number
RS20120165A
Other languages
English (en)
Serbian (sr)
Inventor
Marc Gustaaf C. Verdonck
Patrick René ANGIBAUD
Bruno Roux
Isabelle Noëlle Constance PILATTE
Peter Ten Holte
Janine Arts
Kristof Van Emelen
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Priority claimed from PCT/EP2005/053612 external-priority patent/WO2006010750A1/fr
Publication of RS52304B publication Critical patent/RS52304B/sr

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
RS20120165A 2004-07-28 2005-07-25 Supstituisani indolil alkil amino derivati kao novi inhibitori histon deacetilaze RS52304B (sr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP04077172 2004-07-28
US59218204P 2004-07-29 2004-07-29
PCT/EP2005/053612 WO2006010750A1 (fr) 2004-07-28 2005-07-25 Derives d'indolyl alkyl amine substitues utilises en tant que nouveaux inhibiteurs d'histone deacetylase

Publications (1)

Publication Number Publication Date
RS52304B true RS52304B (sr) 2012-12-31

Family

ID=34928411

Family Applications (1)

Application Number Title Priority Date Filing Date
RS20120165A RS52304B (sr) 2004-07-28 2005-07-25 Supstituisani indolil alkil amino derivati kao novi inhibitori histon deacetilaze

Country Status (10)

Country Link
CN (1) CN1993353B (fr)
AT (1) ATE542812T1 (fr)
DK (1) DK1781639T3 (fr)
ES (1) ES2381117T3 (fr)
ME (1) ME01444B (fr)
PT (1) PT1781639E (fr)
RS (1) RS52304B (fr)
SI (1) SI1781639T1 (fr)
UA (1) UA93352C2 (fr)
ZA (1) ZA200700764B (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN107095871A (zh) * 2016-02-22 2017-08-29 中国科学院上海巴斯德研究所 Quisinostat,一种新型的高效抗疟药物
CN107721980B (zh) * 2017-08-25 2019-07-12 南京医科大学 一类氟尿嘧啶和Quisinosta的乏氧靶向前药及其应用
CN112485233B (zh) * 2020-11-03 2022-08-26 山东师范大学 一种检测去乙酰化酶用纳米传感器及其检测方法和应用

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7446109B2 (en) * 2002-03-13 2008-11-04 Janssen Pharmaceutica N.V. Carbonylamino-derivatives as novel inhibitors of histone deacetylase

Also Published As

Publication number Publication date
CN1993353B (zh) 2010-12-01
DK1781639T3 (da) 2012-05-14
ES2381117T3 (es) 2012-05-23
ME01444B (fr) 2013-12-20
PT1781639E (pt) 2012-05-02
SI1781639T1 (sl) 2012-06-29
ZA200700764B (en) 2008-09-25
UA93352C2 (ru) 2011-02-10
ATE542812T1 (de) 2012-02-15
CN1993353A (zh) 2007-07-04

Similar Documents

Publication Publication Date Title
CA2572833C (fr) Derives d'indolyl alkyl amine substitues utilises en tant que nouveaux inhibiteurs d'histone deacetylase
EP1981874B1 (fr) Dérivés d'aminophényle en tant que nouveaux inibiteurs d'histone désacétylase
CN101370791B (zh) 作为组蛋白脱乙酰基酶抑制剂的吡啶和嘧啶衍生物
AU2007206941B2 (en) Heterocyclylalkyl derivatives as novel inhibitors of histone deacetylase
US7947830B2 (en) Substituted propenyl piperazine derivatives as novel inhibitors of histone deacetylase
EP1776358B1 (fr) Derivés substitués de propenyl piperazine comme nouveaux inhibiteurs de histone deacetylase
RS52304B (sr) Supstituisani indolil alkil amino derivati kao novi inhibitori histon deacetilaze
HK1128281A1 (zh) 作为组蛋白去乙酰化酶抑制剂的吡啶和嘧啶衍生物