SE8003821L - Nya 3-aminovinylcefalosporiner och forfarande for framstellning derav - Google Patents

Nya 3-aminovinylcefalosporiner och forfarande for framstellning derav

Info

Publication number: SE8003821L
Authority: SE; Sweden
Prior art keywords: radical; protective; protective radical; bicyclooct; vinyl
Prior art date: 1979-05-23

Application number

SE8003821A

Other languages

Unknown language ( )

English (en)

Other versions

SE451072B (sv

Inventor

D Farge

Roy P Le

C Moutonnier

J-F Peyronel

Original Assignee

Rhone Poulenc Ind

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1979-05-23

Filing date

1980-05-21

Publication date

1980-11-24

1980-05-21 Application filed by Rhone Poulenc Ind filed Critical Rhone Poulenc Ind

1980-11-24 Publication of SE8003821L publication Critical patent/SE8003821L/sv

1987-08-31 Publication of SE451072B publication Critical patent/SE451072B/sv

Links

238000000034 method Methods 0.000 title 1
230000001681 protective effect Effects 0.000 abstract 5
125000000217 alkyl group Chemical group 0.000 abstract 2
239000001257 hydrogen Substances 0.000 abstract 2
229910052739 hydrogen Inorganic materials 0.000 abstract 2
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
125000002373 5 membered heterocyclic group Chemical group 0.000 abstract 1
125000004070 6 membered heterocyclic group Chemical group 0.000 abstract 1
229930186147 Cephalosporin Natural products 0.000 abstract 1
125000003545 alkoxy group Chemical group 0.000 abstract 1
125000003282 alkyl amino group Chemical group 0.000 abstract 1
239000003242 anti bacterial agent Substances 0.000 abstract 1
229940124587 cephalosporin Drugs 0.000 abstract 1
150000001780 cephalosporins Chemical class 0.000 abstract 1
-1 cyanomethyl Chemical group 0.000 abstract 1
125000004663 dialkyl amino group Chemical group 0.000 abstract 1
125000005842 heteroatom Chemical group 0.000 abstract 1
125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
239000000543 intermediate Substances 0.000 abstract 1
239000000203 mixture Substances 0.000 abstract 1
229910052757 nitrogen Inorganic materials 0.000 abstract 1
125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
125000001424 substituent group Chemical group 0.000 abstract 1
125000000391 vinyl group Chemical group [H]C([*])=C([H])[H] 0.000 abstract 1
229920002554 vinyl polymer Chemical group 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/02—Nutrients, e.g. vitamins, minerals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Diabetes (AREA)
Bioinformatics & Cheminformatics (AREA)
Obesity (AREA)
Hematology (AREA)
Nutrition Science (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Cephalosporin Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

SE8003821A 1979-05-23 1980-05-21 Nya 3-aminovinylcefalosporiner och forfarande for framstellning derav SE451072B (sv)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR7913096A FR2457296A1 (fr)	1979-05-23	1979-05-23	Nouveaux derives de vinyl-3 cephalosporines et leur preparation

Publications (2)

Publication Number	Publication Date
SE8003821L true SE8003821L (sv)	1980-11-24
SE451072B SE451072B (sv)	1987-08-31

Family

ID=9225762

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SE8003821A SE451072B (sv)	1979-05-23	1980-05-21	Nya 3-aminovinylcefalosporiner och forfarande for framstellning derav

Country Status (31)

Country	Link
US (1)	US4307233A (sv)
JP (1)	JPS55154981A (sv)
AT (1)	AT369375B (sv)
AU (1)	AU534806B2 (sv)
BE (1)	BE883416A (sv)
CA (1)	CA1144919A (sv)
CH (1)	CH645379A5 (sv)
CS (1)	CS244405B2 (sv)
DD (1)	DD150899A5 (sv)
DE (1)	DE3019462A1 (sv)
DK (1)	DK222080A (sv)
ES (1)	ES491687A0 (sv)
FI (1)	FI801641A7 (sv)
FR (1)	FR2457296A1 (sv)
GB (1)	GB2051062B (sv)
GR (1)	GR68426B (sv)
HU (1)	HU185890B (sv)
IE (1)	IE49814B1 (sv)
IL (1)	IL60139A (sv)
IT (1)	IT1140974B (sv)
LU (1)	LU82477A1 (sv)
NL (1)	NL8003023A (sv)
NO (1)	NO801502L (sv)
NZ (1)	NZ193799A (sv)
PH (1)	PH15946A (sv)
PL (1)	PL126481B1 (sv)
PT (1)	PT71276A (sv)
SE (1)	SE451072B (sv)
SU (1)	SU1031409A3 (sv)
YU (1)	YU136880A (sv)
ZA (1)	ZA803038B (sv)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ES485938A1 (es) *	1978-11-15	1980-07-01	Glaxo Group Ltd	Un procedimiento para la preparacion de antibioticos de ce- falosporina
FR2494279A1 (fr) *	1980-11-20	1982-05-21	Rhone Poulenc Ind	Nouvelles oxacephalosporines, leur preparation et les medicaments qui les contiennent
FR2494275A2 (fr) *	1980-11-20	1982-05-21	Rhone Poulenc Ind	Nouveaux derives de vinyl-3 cephalosporines et leur preparation
FR2494280A1 (fr) *	1980-11-20	1982-05-21	Rhone Poulenc Ind	Nouveaux derives de la cephalosporine et leur preparation
FR2505334A1 (fr) *	1981-05-11	1982-11-12	Rhone Poulenc Sante	Nouvelles oxacephalosporines et leur preparation
FR2511372A1 (fr) *	1981-08-17	1983-02-18	Rhone Poulenc Sante	Nouveaux derives de la cephalosporine et leur preparation
US4486586A (en) *	1983-02-10	1984-12-04	Bristol-Myers Company	Cephalosporin derivatives
US4560749A (en) *	1983-11-18	1985-12-24	Eli Lilly And Company	Cephem-3-imidates and 3-amidines
US4708955A (en) *	1985-06-24	1987-11-24	Bristol-Myers Company	3-(substituted)propenyl-7-aminothiazol-ylcephalosporanic acids and esters thereof
US4874856A (en) *	1985-06-24	1989-10-17	Bristol-Myers Company	3-(substituted)propenyl-7-(aminothiazolylacetamido) ceph-3-em-4-carboxylic acids and esters thereof
EP0346465B1 (en) *	1986-04-14	1993-08-11	Banyu Pharmaceutical Co., Ltd.	1-carboxy-1-vyniloxyiminoaminothiazole cephalosporing derivatives and process for their preparation
ATE354577T1 (de)	1996-11-06	2007-03-15	Basilea Pharmaceutica Ag	Vinylpyrrolidinon-cephalosporin-derivate
CA2702257C (en)	2007-10-09	2016-07-12	Sopharmia, Inc.	Broad spectrum beta-lactamase inhibitors
US9975905B2 (en)	2013-03-12	2018-05-22	Gladius Pharmaceuticals Corporation	Derivatized 3-styryl-cephalosporins

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4065620A (en) *	1971-06-14	1977-12-27	Eli Lilly And Company	3-(Substituted) vinyl cephalosporins
GB1463077A (en) *	1973-04-19	1977-02-02	Glaxo Lab Ltd	7-substituted-ethyl-cephalosporin derivatives
ES433226A1 (es) *	1973-12-21	1977-07-01	Glaxo Lab Ltd	Un procedimiento para la preparación de compuestos antibióticos de cefalosporina.
US4144393A (en) *	1973-12-21	1979-03-13	Glaxo Laboratories Limited	3-Acetoxymethyl cephalosporins having at position-7 a carboxy substituted α-etherified hydroxyiminoarylacetamido group
JPS5129492A (en) *	1974-09-04	1976-03-12	Sankyo Co	Sefuarosuhorinjudotai no seiho
DK154939C (da) *	1974-12-19	1989-06-12	Takeda Chemical Industries Ltd	Analogifremgangsmaade til fremstilling af thiazolylacetamido-cephemforbindelser eller farmaceutisk acceptable salte eller estere deraf
JPS5253890A (en) *	1975-10-14	1977-04-30	Syntex Inc	Production of cephalosporin type compound
PT71652B (en) *	1979-08-15	1982-01-21	Merck & Co Inc	Process for preparing allysulfoxide enzyme inhibitor

1979
- 1979-05-23 FR FR7913096A patent/FR2457296A1/fr active Granted
1980
- 1980-05-21 CH CH398980A patent/CH645379A5/fr not_active IP Right Cessation
- 1980-05-21 NZ NZ193799A patent/NZ193799A/xx unknown
- 1980-05-21 CS CS803543A patent/CS244405B2/cs unknown
- 1980-05-21 SU SU802926697A patent/SU1031409A3/ru active
- 1980-05-21 GR GR62015A patent/GR68426B/el unknown
- 1980-05-21 YU YU01368/80A patent/YU136880A/xx unknown
- 1980-05-21 HU HU801278A patent/HU185890B/hu unknown
- 1980-05-21 FI FI801641A patent/FI801641A7/fi not_active Application Discontinuation
- 1980-05-21 AT AT0270980A patent/AT369375B/de active
- 1980-05-21 NO NO801502A patent/NO801502L/no unknown
- 1980-05-21 LU LU82477A patent/LU82477A1/fr unknown
- 1980-05-21 DE DE19803019462 patent/DE3019462A1/de not_active Ceased
- 1980-05-21 PL PL1980224391A patent/PL126481B1/pl unknown
- 1980-05-21 BE BE0/200707A patent/BE883416A/fr not_active IP Right Cessation
- 1980-05-21 DD DD80221272A patent/DD150899A5/de unknown
- 1980-05-21 IT IT22243/80A patent/IT1140974B/it active
- 1980-05-21 SE SE8003821A patent/SE451072B/sv not_active IP Right Cessation
- 1980-05-21 CA CA000352324A patent/CA1144919A/fr not_active Expired
- 1980-05-21 IE IE1062/80A patent/IE49814B1/en unknown
- 1980-05-21 ZA ZA00803038A patent/ZA803038B/xx unknown
- 1980-05-21 US US06/152,085 patent/US4307233A/en not_active Expired - Lifetime
- 1980-05-21 DK DK222080A patent/DK222080A/da not_active Application Discontinuation
- 1980-05-21 GB GB8016727A patent/GB2051062B/en not_active Expired
- 1980-05-21 AU AU58595/80A patent/AU534806B2/en not_active Ceased
- 1980-05-21 PT PT71276A patent/PT71276A/pt unknown
- 1980-05-21 ES ES491687A patent/ES491687A0/es active Granted
- 1980-05-22 IL IL60139A patent/IL60139A/xx unknown
- 1980-05-22 PH PH24056A patent/PH15946A/en unknown
- 1980-05-23 JP JP6800980A patent/JPS55154981A/ja active Granted
- 1980-05-23 NL NL8003023A patent/NL8003023A/nl not_active Application Discontinuation

Also Published As

Publication number	Publication date
LU82477A1 (fr)	1980-12-16
FR2457296A1 (fr)	1980-12-19
ATA270980A (de)	1982-05-15
CA1144919A (fr)	1983-04-19
IT8022243A0 (it)	1980-05-21
GR68426B (sv)	1981-12-30
IE801062L (en)	1980-11-23
PH15946A (en)	1983-04-29
PT71276A (fr)	1980-06-01
AU5859580A (en)	1980-11-27
AT369375B (de)	1982-12-27
ES8102136A1 (es)	1980-12-16
IT1140974B (it)	1986-10-10
PL224391A1 (sv)	1981-02-13
SU1031409A3 (ru)	1983-07-23
NZ193799A (en)	1983-03-15
FI801641A7 (fi)	1981-01-01
FR2457296B1 (sv)	1982-02-05
IL60139A0 (en)	1980-07-31
ES491687A0 (es)	1980-12-16
CS244405B2 (en)	1986-07-17
DK222080A (da)	1980-11-24
IE49814B1 (en)	1985-12-25
HU185890B (en)	1985-04-28
US4307233A (en)	1981-12-22
GB2051062B (en)	1983-10-12
DD150899A5 (de)	1981-09-23
YU136880A (en)	1983-04-30
JPS55154981A (en)	1980-12-02
ZA803038B (en)	1981-05-27
JPH0246595B2 (sv)	1990-10-16
BE883416A (fr)	1980-11-21
IL60139A (en)	1984-04-30
SE451072B (sv)	1987-08-31
CS354380A2 (sv)	1985-09-17
AU534806B2 (en)	1984-02-16
CH645379A5 (fr)	1984-09-28
PL126481B1 (en)	1983-08-31
NL8003023A (nl)	1980-11-25
NO801502L (no)	1980-11-24
DE3019462A1 (de)	1980-12-04
GB2051062A (en)	1981-01-14

Legal Events

Date

Code

Title

Description

1995-01-31

NUG

Patent has lapsed

Ref document number: 8003821-9

Effective date: 19911209

Format of ref document f/p: F

Publication	Publication Date	Title
FI823923L (fi)	1983-05-18	Antifibrinolytiskt aktiva foereningar
SE7714592L (sv)	1978-06-24	Cyklopentan-1-aminer, forfarande for framstellning derav och medel innehallande dessa foreningar
ES8102136A1 (es)	1980-12-16	Procedimiento para la obtencion de derivados de vinil-3 ce- falosporina
SE8003823L (sv)	1980-11-24	Nya 3-formylmetylcefalosporiner och forfarande for framstellning derav
ES466366A1 (es)	1978-10-01	Un procedimiento para preparar derivados de metasulfonamido-benzamida.
AU536912B2 (en)	1984-05-31	Benzothiazole derivatives
IE782502L (en)	1979-06-20	Cephalosporins
SE7706655L (sv)	1977-12-10	Nya bensylcyanoacetaler och sett att framstella dessa
SE8000367L (sv)	1980-07-17	Fenoxi- och tiofenoxintriler och anvendning derav
AU538591B2 (en)	1984-08-23	3h-naphtho(1,2-d)imidazole derivatives
FI890187A0 (fi)	1989-01-13	Foerfarande foer framstaellning av hydroxialkylerande foereningar, saolunda erhaollna nya foereningar och deras anvaendning.
ES457197A1 (es)	1978-08-16	Procedimiento para preparar carbamatos de oxima.
DK392579A (da)	1980-03-22	Fremgangsmaade til fremstilling af 4,5-methano-bufadienolid-rhamnosider
ATE8633T1 (de)	1984-08-15	Vinyl-3-cephalosporinverbindungen und ihre herstellung.
FI841408A0 (fi)	1984-04-10	Foerfarande foer framstaellning av 4- acetyl-2-substituerade-imidazoler och i foerfarandet anvaenda mellanproduk mellanprodukter.
ES515047A0 (es)	1983-05-01	Procedimiento para la obtencion de derivados de cefalosporina.
ES455841A1 (es)	1978-06-16	Procedimiento para preparar composiciones insecticidas a ba-se de ditiofo-fatos-(-fonatos) de formamidina.
DK160051C (da)	1991-06-10	N-methyl-n-silylcarbamat, fremgangsmaade til bekaempelse af skadedyr under anvendelse deraf samt skadedyrsbekaempelsesmiddel indeholdende forbindelsen
SE8000298L (sv)	1980-07-16	Karbamatderivat av merkaptoacylhydroxiproliner
IE43116L (en)	1976-12-09	Oxadiazolidine derivatives
ES451217A1 (es)	1977-12-01	Procedimiento para la obtencion de fenilureas de actividad herbicida.
JPS53112887A (en)	1978-10-02	Production of n-substituted trialkoxybenzylpiperazine derivative
ES454090A1 (es)	1978-01-16	Un metodo para preparar compuestos heterociclicos.
SE8306048L (sv)	1984-05-06	Nya heterocykliska ettiksyror och forfarande for framstellning derav
DK320582A (da)	1983-01-19	Substituerede phenyl-cyclopropancarboxylsyreestere,fremgangsmaade til fremstilling deraf samt deres anvendelse som midler til bekaempelse af skadelige organismer