SE9801990D0 - New 3-aryl propionic acid derivatives and analogs - Google Patents

New 3-aryl propionic acid derivatives and analogs

Info

Publication number
SE9801990D0
SE9801990D0 SE9801990A SE9801990A SE9801990D0 SE 9801990 D0 SE9801990 D0 SE 9801990D0 SE 9801990 A SE9801990 A SE 9801990A SE 9801990 A SE9801990 A SE 9801990A SE 9801990 D0 SE9801990 D0 SE 9801990D0
Authority
SE
Sweden
Prior art keywords
analogs
new
propionic acid
acid derivatives
aryl propionic
Prior art date
Application number
SE9801990A
Other languages
English (en)
Swedish (sv)
Inventor
Kjell Andersson
Maria Boije
Johan Gottfries
Tord Inghardt
Lanna Li
Eva-Lotte Lindstedt
Original Assignee
Astra Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astra Ab filed Critical Astra Ab
Priority to SE9801990A priority Critical patent/SE9801990D0/xx
Publication of SE9801990D0 publication Critical patent/SE9801990D0/xx
Priority to MA25591A priority patent/MA26634A1/fr
Priority to DZ990099A priority patent/DZ2799A1/xx
Priority to TW088108577A priority patent/TW548263B/zh
Priority to TW088108575A priority patent/TW446694B/zh
Priority to MA25601A priority patent/MA26637A1/fr
Priority to IDW20002669A priority patent/ID29457A/id
Priority to ES99930058T priority patent/ES2216527T3/es
Priority to CN99809354A priority patent/CN1312795A/zh
Priority to NZ508453A priority patent/NZ508453A/xx
Priority to JP2000552083A priority patent/JP3568897B2/ja
Priority to PCT/SE1999/000942 priority patent/WO1999062871A1/en
Priority to UA2000116620A priority patent/UA66852C2/uk
Priority to SI9930576T priority patent/SI1084101T1/xx
Priority to RU2000130191/04A priority patent/RU2243214C2/ru
Priority to HK01105768.8A priority patent/HK1034957B/en
Priority to DE69915470T priority patent/DE69915470T2/de
Priority to HU0103226A priority patent/HUP0103226A3/hu
Priority to SK1769-2000A priority patent/SK284849B6/sk
Priority to JP2000552084A priority patent/JP3723739B2/ja
Priority to PT99930058T priority patent/PT1084101E/pt
Priority to US09/341,931 priority patent/US6630600B1/en
Priority to TR2000/03583T priority patent/TR200003583T2/xx
Priority to AT99930060T priority patent/ATE251130T1/de
Priority to KR1020007013663A priority patent/KR20010052522A/ko
Priority to EP99930058A priority patent/EP1084101B1/en
Priority to KR1020007013673A priority patent/KR20010052529A/ko
Priority to IDW20002584A priority patent/ID28164A/id
Priority to EEP200000725A priority patent/EE04463B1/xx
Priority to ES99930060T priority patent/ES2209457T3/es
Priority to DK99930060T priority patent/DK1084102T3/da
Priority to US09/341,935 priority patent/US6362360B1/en
Priority to PL99344681A priority patent/PL344681A1/xx
Priority to AU46672/99A priority patent/AU752262B2/en
Priority to SK1767-2000A priority patent/SK17672000A3/sk
Priority to DE69911770T priority patent/DE69911770T2/de
Priority to DK99930058T priority patent/DK1084101T3/da
Priority to CA002334374A priority patent/CA2334374A1/en
Priority to CA002334107A priority patent/CA2334107A1/en
Priority to TR2000/03543T priority patent/TR200003543T2/xx
Priority to PCT/SE1999/000940 priority patent/WO1999062870A1/en
Priority to SI9930452T priority patent/SI1084102T1/xx
Priority to PL99344682A priority patent/PL344682A1/xx
Priority to AT99930058T priority patent/ATE261429T1/de
Priority to EEP200000717A priority patent/EE200000717A/xx
Priority to BR9910921-2A priority patent/BR9910921A/pt
Priority to AU46670/99A priority patent/AU4667099A/en
Priority to EP99930060A priority patent/EP1084102B1/en
Priority to IL13994299A priority patent/IL139942A0/xx
Priority to CN99809355A priority patent/CN1311769A/zh
Priority to IL13963599A priority patent/IL139635A0/xx
Priority to PT99930060T priority patent/PT1084102E/pt
Priority to BR9910913-1A priority patent/BR9910913A/pt
Priority to TNTNSN99103A priority patent/TNSN99103A1/fr
Priority to MYPI99002185A priority patent/MY129581A/en
Priority to TNTNSN99107A priority patent/TNSN99107A1/fr
Priority to ARP990102636A priority patent/AR019853A1/es
Priority to ARP990102634A priority patent/AR035305A1/es
Priority to ZA200006773A priority patent/ZA200006773B/en
Priority to ZA200006771A priority patent/ZA200006771B/en
Priority to IS5735A priority patent/IS5735A/is
Priority to IS5744A priority patent/IS5744A/is
Priority to NO20006114A priority patent/NO20006114L/no
Priority to NO20006116A priority patent/NO20006116L/no
Priority to US10/678,739 priority patent/US20040229949A1/en
Priority to JP2004118663A priority patent/JP2004256548A/ja
Priority to JP2004183263A priority patent/JP2004346079A/ja
Priority to US11/388,942 priority patent/US20060173204A1/en

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SE9801990A 1998-06-04 1998-06-04 New 3-aryl propionic acid derivatives and analogs SE9801990D0 (sv)

Priority Applications (68)

Application Number Priority Date Filing Date Title
SE9801990A SE9801990D0 (sv) 1998-06-04 1998-06-04 New 3-aryl propionic acid derivatives and analogs
MA25591A MA26634A1 (fr) 1998-06-04 1999-05-20 Nouveaux derives de l'acide 3-aryl propionique et analogues
DZ990099A DZ2799A1 (fr) 1998-06-04 1999-05-23 Nouveaux dérivés de l'acide 3-aryl propionique et analogues.
TW088108577A TW548263B (en) 1998-06-04 1999-05-25 New 3-aryl propionic acid derivatives and analogs
TW088108575A TW446694B (en) 1998-06-04 1999-05-25 Novel 3-aryl-2-hydroxypropionic acid derivative for use in conditions associated with insulin resistance and pharmaceutical composition containing same
MA25601A MA26637A1 (fr) 1998-06-04 1999-05-28 Nouveau derive iii de l'acide 3-aryl-2-hydroxypropionique.
IDW20002669A ID29457A (id) 1998-06-04 1999-05-31 Turunan dan analog asam 3-aril propionat
ES99930058T ES2216527T3 (es) 1998-06-04 1999-05-31 Nuevo derivado (iii) de acido 3-aril-2-hidroxipropionico.
CN99809354A CN1312795A (zh) 1998-06-04 1999-05-31 新的3－芳基丙酸衍生物和其类似物
NZ508453A NZ508453A (en) 1998-06-04 1999-05-31 New 3-aryl propionic acid derivatives and analogs and their use in the treatment of insulin resistance
JP2000552083A JP3568897B2 (ja) 1998-06-04 1999-05-31 新規な３−アリール−２−ヒドロキシプロピオン酸誘導体ｉｉｉ
PCT/SE1999/000942 WO1999062871A1 (en) 1998-06-04 1999-05-31 New 3-aryl propionic acid derivatives and analogs
UA2000116620A UA66852C2 (uk) 1998-06-04 1999-05-31 Похідні та аналоги 3-арилпропіонової кислоти, спосіб їх отримання, фармацевтична композиція (варіанти) та спосіб профілактики та/або лікування асоційованих з резистентністю до інсуліну клінічних станів
SI9930576T SI1084101T1 (en) 1998-06-04 1999-05-31 New 3-aryl-2-hydroxypropionic acid derivative iii
RU2000130191/04A RU2243214C2 (ru) 1998-06-04 1999-05-31 Новые производные и аналоги 3-арилпропионовой кислоты
HK01105768.8A HK1034957B (en) 1998-06-04 1999-05-31 New 3-aryl propionic acid derivatives and analogs
DE69915470T DE69915470T2 (de) 1998-06-04 1999-05-31 Neue 3-aryl-2-hydroxypropionsäure-derivate iii
HU0103226A HUP0103226A3 (en) 1998-06-04 1999-05-31 New 3-aryl propionic acid derivatives and analogs
SK1769-2000A SK284849B6 (sk) 1998-06-04 1999-05-31 Deriváty a analógy kyseliny 3-arylpropiónovej, spôsob ich prípravy, farmaceutické formulácie s ich obsahom a ich použitie
JP2000552084A JP3723739B2 (ja) 1998-06-04 1999-05-31 新規３−アリールプロピオン酸誘導体および類似体
PT99930058T PT1084101E (pt) 1998-06-04 1999-05-31 Novo derivado do acido 3-aril-2-hidroxipropionico (iii)
US09/341,931 US6630600B1 (en) 1998-06-04 1999-05-31 3-aryl propionic acid derivatives and analogs
TR2000/03583T TR200003583T2 (tr) 1998-06-04 1999-05-31 Yeni 3-aril propiyonik asit türevleri ve benzerleri.
AT99930060T ATE251130T1 (de) 1998-06-04 1999-05-31 Neue 3-aryl-propionsäurederivate und analoge
KR1020007013663A KR20010052522A (ko) 1998-06-04 1999-05-31 신규한 3-아릴-2-히드록시프로피온산 유도체 ⅲ
EP99930058A EP1084101B1 (en) 1998-06-04 1999-05-31 New 3-aryl-2-hydroxypropionic acid derivative iii
KR1020007013673A KR20010052529A (ko) 1998-06-04 1999-05-31 신규한 3-아릴 프로피온산 유도체 및 동족체
IDW20002584A ID28164A (id) 1998-06-04 1999-05-31 Turunan iii asam 3-aril-2-hidroksipropionat baru
EEP200000725A EE04463B1 (et) 1998-06-04 1999-05-31 3-arüülpropaanhappe derivaadid ja nende analoogid, nende valmistamise meetod, neid sisaldavad ravimkoostised ja ühendid kasutamiseks ravis
ES99930060T ES2209457T3 (es) 1998-06-04 1999-05-31 Nuevos derivados del acido 3-aril-propionico, y analogos.
DK99930060T DK1084102T3 (da) 1998-06-04 1999-05-31 Nye 3-arylpropionsyrederivater og analoge
US09/341,935 US6362360B1 (en) 1998-06-04 1999-05-31 3-aryl-2-hydroxypropionic acid derivative III
PL99344681A PL344681A1 (en) 1998-06-04 1999-05-31 New 3-aryl propionic acid derivatives and analogs
AU46672/99A AU752262B2 (en) 1998-06-04 1999-05-31 New 3-aryl propionic acid derivatives and analogs
SK1767-2000A SK17672000A3 (sk) 1998-06-04 1999-05-31 Derivát kyseliny 3-aryl-2-hydroxypropiónovej
DE69911770T DE69911770T2 (de) 1998-06-04 1999-05-31 Neue 3-aryl-propionsäurederivate und analoge
DK99930058T DK1084101T3 (da) 1998-06-04 1999-05-31 Nyt 3-aryl-2-hydroxypropionsyrederivat (III)
CA002334374A CA2334374A1 (en) 1998-06-04 1999-05-31 New 3-aryl propionic acid derivatives and analogs
CA002334107A CA2334107A1 (en) 1998-06-04 1999-05-31 New 3-aryl-2-hydroxypropionic acid derivative iii
TR2000/03543T TR200003543T2 (tr) 1998-06-04 1999-05-31 Yeni 3-aril-2-hidroksipropiyonik asit türevi III.
PCT/SE1999/000940 WO1999062870A1 (en) 1998-06-04 1999-05-31 New 3-aryl-2-hydroxypropionic acid derivative iii
SI9930452T SI1084102T1 (en) 1998-06-04 1999-05-31 New 3-aryl propionic acid derivatives and analogs
PL99344682A PL344682A1 (en) 1998-06-04 1999-05-31 New 3-aryl-2-hydroxypropionic acid derivative iii
AT99930058T ATE261429T1 (de) 1998-06-04 1999-05-31 Neue 3-aryl-2-hydroxypropionsäure-derivate iii
EEP200000717A EE200000717A (et) 1998-06-04 1999-05-31 Uus 3-arüül-2-hüdroksüpropaanhappe derivaat III
BR9910921-2A BR9910921A (pt) 1998-06-04 1999-05-31 Composto, processo para preparar o mesmo, formulação farmacêutica, uso de um composto, e, processo para a profilaxia e/ou tratamento de condições clìnicas associadas com a resistência à insulina
AU46670/99A AU4667099A (en) 1998-06-04 1999-05-31 New 3-aryl-2-hydroxypropionic acid derivative iii
EP99930060A EP1084102B1 (en) 1998-06-04 1999-05-31 New 3-aryl propionic acid derivatives and analogs
IL13994299A IL139942A0 (en) 1998-06-04 1999-05-31 New 3-aryl-2-hydroxypropionic acid derivative iii
CN99809355A CN1311769A (zh) 1998-06-04 1999-05-31 新的3－芳基－2－羟基丙酸衍生物iii
IL13963599A IL139635A0 (en) 1998-06-04 1999-05-31 New 3-aryl propionic acid derivatives and analogs
PT99930060T PT1084102E (pt) 1998-06-04 1999-05-31 Novos derivados do acido 3-aril-propionico e analogos
BR9910913-1A BR9910913A (pt) 1998-06-04 1999-05-31 Composto, processo para a preparação de um composto, formulação farmacêutica, uso de um composto, e, processo para a profilaxia e/ou tratamento de condições clìnicas associadas com resistência a insulina
TNTNSN99103A TNSN99103A1 (fr) 1998-06-04 1999-06-02 Nouveaux derives de l'acide 3-aryl propionique et analogues
MYPI99002185A MY129581A (en) 1998-06-04 1999-06-02 New 3-aryl propionic acid derivatives and analogs
TNTNSN99107A TNSN99107A1 (fr) 1998-06-04 1999-06-02 Nouveau derive iii de l'acide 3-aryl-2-hydroxypropionique
ARP990102636A AR019853A1 (es) 1998-06-04 1999-06-03 Derivado del acido 3-aril-2-hidroxipropionico, proceso e intermediario para su preparacion, formulaciones farmaceuticas, uso de dicho compuesto en laelaboracion de un medicamento, metodo para la profilaxis y/o tratamiento de trastornos clinicos asociados con la resistencia a la insulina, y formulaci
ARP990102634A AR035305A1 (es) 1998-06-04 1999-06-03 Derivados y analogos del acido 3-arilpropionico, proceso para su preparacion, formulaciones farmaceuticas, uso de los mismos en la elaboracion de medicamentos, y formulacion farmaceutica para usar en la profilaxis y/o tratamiento de trastornos clinicos asociados con la resistencia a la insulina
ZA200006773A ZA200006773B (en) 1998-06-04 2000-11-20 New 3-aryl-2-hydroxypropionic acid derivative III.
ZA200006771A ZA200006771B (en) 1998-06-04 2000-11-20 New 3-aryl propionic acid derivatives and analogs.
IS5735A IS5735A (is) 1998-06-04 2000-11-28 Ný 3-arýl-2-hýdroxýprópínsýruafleiða III
IS5744A IS5744A (is) 1998-06-04 2000-11-29 Nýjar 3-arýl-própíónsýruafleiður og -hliðstæður
NO20006114A NO20006114L (no) 1998-06-04 2000-12-01 Nytt 3-aryl-2-hydroksypropionsyrederivat III
NO20006116A NO20006116L (no) 1998-06-04 2000-12-01 Nye 3-arylpropionsyrederivater og -analoger
US10/678,739 US20040229949A1 (en) 1998-06-04 2003-10-02 New 3-aryl propionic acid derivatives and analogs
JP2004118663A JP2004256548A (ja) 1998-06-04 2004-04-14 新規な３−アリール−２−ヒドロキシプロピオン酸誘導体ｉｉｉ
JP2004183263A JP2004346079A (ja) 1998-06-04 2004-06-22 新規３−アリールプロピオン酸誘導体および類似体
US11/388,942 US20060173204A1 (en) 1998-06-04 2006-03-24 New 3-aryl propionic acid derivatives and analogs

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EP (1) EP1084101B1 (pt)
JP (2) JP3568897B2 (pt)
KR (1) KR20010052522A (pt)
CN (1) CN1311769A (pt)
AR (1) AR019853A1 (pt)
AT (1) ATE261429T1 (pt)
AU (1) AU4667099A (pt)
BR (1) BR9910913A (pt)
CA (1) CA2334107A1 (pt)
DE (1) DE69915470T2 (pt)
DK (1) DK1084101T3 (pt)
EE (1) EE200000717A (pt)
ES (1) ES2216527T3 (pt)
ID (1) ID28164A (pt)
IL (1) IL139942A0 (pt)
IS (1) IS5735A (pt)
MA (1) MA26637A1 (pt)
NO (1) NO20006114L (pt)
PL (1) PL344682A1 (pt)
PT (1) PT1084101E (pt)
SE (1) SE9801990D0 (pt)
SK (1) SK17672000A3 (pt)
TN (1) TNSN99107A1 (pt)
TR (1) TR200003543T2 (pt)
TW (1) TW446694B (pt)
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ZA (2) ZA200006771B (pt)

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CN1280574A (zh) * 1997-10-27 2001-01-17 雷迪研究基金会 新的杂环化合物及其在医药中的应用、它们的制备方法和含有它们的药物组合物
MA26634A1 (fr) 1998-06-04 2004-12-20 Astra Ab Nouveaux derives de l'acide 3-aryl propionique et analogues
SE9801992D0 (sv) * 1998-06-04 1998-06-04 Astra Ab New 3-aryl-2-hydroxypropionic acid derivative I
SE9904415D0 (sv) * 1999-12-03 1999-12-03 Astra Ab New process
CA2392038A1 (en) * 1999-12-03 2001-06-07 Astrazeneca Ab Crystalline form of (s)-2 ethoxy-3-[4-(2-{4-methanesulfonyloxyphenyl} ethoxy) phenyl] propanoic acid
WO2001040165A1 (en) * 1999-12-03 2001-06-07 Astrazeneca Ab Crystalline form of 3-{4-[2-(4-tert-butoxycarbonylaminophenyl)ethoxy]phenyl}-(s)-2-ethoxy propanoic acid
SE9904412D0 (sv) * 1999-12-03 1999-12-03 Astra Ab Comminuted form
TW574193B (en) 1999-12-03 2004-02-01 Astrazeneca Ab Novel phenalkyloxy-phenyl derivatives, pharmaceutical composition containing the same and their uses
SE9904421D0 (sv) * 1999-12-03 1999-12-03 Astra Ab New compounds
US6559335B2 (en) 2000-09-22 2003-05-06 Dr. Reddy's Laboratories Limited Process for the preparation of 3-aryl-2-hydroxy propanoic acid
SE0101386D0 (sv) 2001-04-20 2001-04-20 Astrazeneca Ab New compounds
SE0101980D0 (sv) * 2001-06-01 2001-06-01 Astrazeneca Ab Pharmaceutical combination
SE0101978D0 (sv) 2001-06-01 2001-06-01 Astrazeneca Ab New compounds
SE0101982D0 (sv) * 2001-06-01 2001-06-01 Astrazeneca Ab Pharmaceutical combination
SE0101981D0 (sv) * 2001-06-01 2001-06-01 Astrazeneca Ab Pharmaceutical combination
CZ20033309A3 (cs) 2001-06-07 2004-05-12 Eliálillyáandácompany Modulátory receptorů aktivovaných peroxizomálními proliferátory }PPARB
WO2003008362A1 (en) * 2001-06-28 2003-01-30 Dr. Reddy's Laboratories Ltd Novel 3-aryl-2-hydroxy propanol derivatives and a process for their preparation
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FR2872159B1 (fr) * 2004-06-28 2007-10-05 Merck Sante Soc Par Actions Si Nouveaux derives acides carboxyliques phenyliques et leur utilisation dans le traitement du diabete
FR2917086B1 (fr) * 2007-06-05 2009-07-17 Galderma Res & Dev Nouveaux derives d'acide 3-phenyl acrylique activateurs des recepteurs de type ppar, leur methode de preparation et leur utilisation dans des compositions cosmetiques ou pharmaceutiques.
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DK2637646T3 (en) 2010-11-08 2016-08-29 Albireo Ab PHARMACEUTICAL COMBINATION CONTAINING AN IBAT inhibitor and a bile acid binder
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PL344682A1 (en) 2001-11-19
ZA200006773B (en) 2002-02-20
JP3568897B2 (ja) 2004-09-22
EP1084101A1 (en) 2001-03-21
TNSN99107A1 (fr) 2005-11-10
MA26637A1 (fr) 2004-12-20
SK17672000A3 (sk) 2001-08-06
ZA200006771B (en) 2002-05-20
TR200003543T2 (tr) 2001-04-20
DE69915470T2 (de) 2005-02-24
CA2334107A1 (en) 1999-12-09
US6362360B1 (en) 2002-03-26
ID28164A (id) 2001-05-10
JP2002516898A (ja) 2002-06-11
NO20006114L (no) 2001-02-02
DE69915470D1 (en) 2004-04-15
NO20006114D0 (no) 2000-12-01
EP1084101B1 (en) 2004-03-10
TW446694B (en) 2001-07-21
AU4667099A (en) 1999-12-20
EE200000717A (et) 2001-08-15
AR019853A1 (es) 2002-03-20
ES2216527T3 (es) 2004-10-16
IL139942A0 (en) 2002-02-10
BR9910913A (pt) 2001-03-06
CN1311769A (zh) 2001-09-05
ATE261429T1 (de) 2004-03-15
WO1999062870A1 (en) 1999-12-09
JP2004256548A (ja) 2004-09-16
DK1084101T3 (da) 2004-06-14
IS5735A (is) 2000-11-28
PT1084101E (pt) 2004-07-30
KR20010052522A (ko) 2001-06-25

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