SK10752003A3 - Použitie inverzných agonistov GABAA v kombinácii s parciálnymi agonistami receptora nikotínu, estrogénom, selektívnymi modulátormi estrogénu alebo vitamínom E pri liečení kognitívnych porúch - Google Patents

Použitie inverzných agonistov GABAA v kombinácii s parciálnymi agonistami receptora nikotínu, estrogénom, selektívnymi modulátormi estrogénu alebo vitamínom E pri liečení kognitívnych porúch Download PDF

Info

Publication number: SK10752003A3
Authority: SK; Slovakia
Prior art keywords: triene; hexahydro; diazocin; methano; pyrido
Prior art date: 2001-03-01

Application number

SK1075-2003A

Other languages

English (en)

Slovak (sk)

Inventor

Anabella Villalobos

Original Assignee

Pfizer Products Inc.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-03-01

Filing date

2002-02-20

Publication date

2004-08-03

2002-02-20 Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.

2004-08-03 Publication of SK10752003A3 publication Critical patent/SK10752003A3/sk

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- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A—HUMAN NECESSITIES
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SK1075-2003A 2001-03-01 2002-02-20 Použitie inverzných agonistov GABAA v kombinácii s parciálnymi agonistami receptora nikotínu, estrogénom, selektívnymi modulátormi estrogénu alebo vitamínom E pri liečení kognitívnych porúch SK10752003A3 (sk)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US27256601P	2001-03-01	2001-03-01
PCT/IB2002/000515 WO2002069948A1 (en)	2001-03-01	2002-02-20	Use of gabaa inverse agonists in combination with nicotine receptor partial agonists, estrogen, selective estrogen modulators, or vitamin e for the treatment of cognitive disorders

Publications (1)

Publication Number	Publication Date
SK10752003A3 true SK10752003A3 (sk)	2004-08-03

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SK1075-2003A SK10752003A3 (sk)	2001-03-01	2002-02-20	Použitie inverzných agonistov GABAA v kombinácii s parciálnymi agonistami receptora nikotínu, estrogénom, selektívnymi modulátormi estrogénu alebo vitamínom E pri liečení kognitívnych porúch

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Country	Link
US (2)	US20020193360A1 (cs)
EP (1)	EP1363606A1 (cs)
JP (1)	JP2004527500A (cs)
KR (1)	KR20030076717A (cs)
CN (1)	CN1494422A (cs)
AP (1)	AP2002002465A0 (cs)
AR (1)	AR033425A1 (cs)
BG (1)	BG108131A (cs)
BR (1)	BR0207802A (cs)
CA (1)	CA2439581A1 (cs)
CR (1)	CR7059A (cs)
CZ (1)	CZ20032338A3 (cs)
DO (1)	DOP2002000345A (cs)
EA (1)	EA200300854A1 (cs)
EC (1)	ECSP034759A (cs)
EE (1)	EE200300422A (cs)
GT (1)	GT200200039A (cs)
HU (1)	HUP0303448A3 (cs)
IL (1)	IL157465A0 (cs)
IS (1)	IS6905A (cs)
MA (1)	MA26999A1 (cs)
MX (1)	MXPA03007834A (cs)
NO (1)	NO20033821L (cs)
NZ (1)	NZ527397A (cs)
OA (1)	OA12554A (cs)
PA (1)	PA8540701A1 (cs)
PE (1)	PE20020927A1 (cs)
PL (1)	PL364081A1 (cs)
SK (1)	SK10752003A3 (cs)
TN (1)	TNSN02018A1 (cs)
UY (1)	UY27188A1 (cs)
WO (1)	WO2002069948A1 (cs)
ZA (1)	ZA200306193B (cs)

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TW201206425A (en)	2004-05-18	2012-02-16	Brni Neurosciences Inst	Treatment of depressive disorders
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US8510055B2 (en)	2005-08-03	2013-08-13	The Johns Hopkins University	Methods for characterizing and treating cognitive impairment in aging and disease
EP2032987B1 (en) *	2006-05-22	2016-02-24	The Board of Trustees of The Leland Stanford Junior University	Pharmacological treatment of cognitive impairment
NZ576036A (en)	2006-10-16	2010-10-29	Bionomics Ltd	Naphthyridine containing compounds for treating anxiety disorders
AU2013202426B2 (en) *	2006-10-16	2015-08-06	Bionomics Limited	Novel anxiolytic compounds
US10954231B2 (en)	2006-10-16	2021-03-23	Bionomics Limited	Anxiolytic compounds
EP3332797A3 (en)	2007-02-09	2018-08-01	Blanchette Rockefeller Neurosciences Institute	Therapeutic effects of bryostatins, bryologs and other related substances on head trauma-induced memory impairment and brain injury
US8039620B2 (en) *	2008-05-22	2011-10-18	Teva Pharmaceutical Industries Ltd.	Varenicline tosylate, an intermediate in the preparation process of varenicline L-tartrate
US20090318695A1 (en) *	2008-06-19	2009-12-24	Vinod Kumar Kansal	Processes for the preparation of varenicline and intermediates thereof
WO2010005643A1 (en) *	2008-07-10	2010-01-14	Teva Pharmaceutical Industries Ltd.	Processes for purifying varenicline l-tartrate salt and preparing crystalline forms of varenicline l-tartrate salt
US10206921B2 (en) *	2009-06-03	2019-02-19	The Regents Of The University Of California	Methods and compositions for treating a subject for central nervous system (CNS) injury
EP2438054A1 (en) *	2009-06-22	2012-04-11	Teva Pharmaceutical Industries Ltd.	Solid states forms of varenicline salts and processes for preparation thereof
EP3034079B1 (en)	2010-11-15	2018-01-10	Agenebio, Inc.	Pyridazine derivatives, compositions and methods for treating cognitive impairment
US20140051701A1 (en) *	2011-03-02	2014-02-20	Bionomics Limited	Methods of treating a disease or condition of the central nervous system
US9023848B2 (en)	2011-03-02	2015-05-05	Bionomics Limited	Small-molecules as therapeutics
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US20180170941A1 (en)	2016-12-19	2018-06-21	Agenebio, Inc.	Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment
US11505555B2 (en)	2016-12-19	2022-11-22	Agenebio, Inc.	Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment
CN112601749B (zh)	2018-06-19	2024-03-26	艾吉因生物股份有限公司	用于治疗认知损害的苯并二氮杂环庚三烯衍生物，组合物和方法
CN116008442B (zh) *	2023-03-27	2023-06-30	上海赛默罗生物科技有限公司	α5-GABAA受体调节剂的合成中间体的杂质检测方法
CN116077459B (zh) *	2023-04-10	2023-07-07	上海赛默罗生物科技有限公司	α5-GABAA受体调节剂的胶囊剂及其制备方法

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WO2000071528A1 (en) *	1999-05-25	2000-11-30	Neurogen Corporation	4h-1,4-benzothiazine-2-carboxamides and their use as gaba brain receptor ligands

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- 2002-02-20 CZ CZ20032338A patent/CZ20032338A3/cs unknown
- 2002-02-20 EE EEP200300422A patent/EE200300422A/xx unknown
- 2002-02-20 KR KR10-2003-7011366A patent/KR20030076717A/ko not_active Ceased
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- 2002-02-20 SK SK1075-2003A patent/SK10752003A3/sk not_active Application Discontinuation
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- 2002-02-20 EP EP02700509A patent/EP1363606A1/en not_active Withdrawn
- 2002-02-26 PE PE2002000157A patent/PE20020927A1/es not_active Application Discontinuation
- 2002-02-26 DO DO2002000345A patent/DOP2002000345A/es unknown
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- 2002-02-27 UY UY27188A patent/UY27188A1/es not_active Application Discontinuation
- 2002-02-28 TN TNTNSN02018A patent/TNSN02018A1/fr unknown
- 2002-02-28 AP APAP/P/2002/002465A patent/AP2002002465A0/en unknown
- 2002-02-28 PA PA20028540701A patent/PA8540701A1/es unknown
2003
- 2003-08-07 IS IS6905A patent/IS6905A/is unknown
- 2003-08-11 ZA ZA200306193A patent/ZA200306193B/en unknown
- 2003-08-19 MA MA27286A patent/MA26999A1/fr unknown
- 2003-08-25 BG BG108131A patent/BG108131A/xx unknown
- 2003-08-25 CR CR7059A patent/CR7059A/es not_active Application Discontinuation
- 2003-08-28 NO NO20033821A patent/NO20033821L/no not_active Application Discontinuation
- 2003-09-01 EC EC2003004759A patent/ECSP034759A/es unknown
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Also Published As

Publication number	Publication date
BG108131A (en)	2004-09-30
EE200300422A (et)	2004-02-16
CN1494422A (zh)	2004-05-05
AP2002002465A0 (en)	2002-06-30
ECSP034759A (es)	2003-10-28
UY27188A1 (es)	2002-10-31
WO2002069948A1 (en)	2002-09-12
US20040082555A1 (en)	2004-04-29
CA2439581A1 (en)	2002-09-12
KR20030076717A (ko)	2003-09-26
US20020193360A1 (en)	2002-12-19
PE20020927A1 (es)	2002-10-30
IL157465A0 (en)	2004-03-28
OA12554A (en)	2006-06-07
AR033425A1 (es)	2003-12-17
HUP0303448A2 (hu)	2004-01-28
MXPA03007834A (es)	2003-12-08
PL364081A1 (en)	2004-12-13
NZ527397A (en)	2005-05-27
TNSN02018A1 (fr)	2005-12-23
EA200300854A1 (ru)	2004-02-26
PA8540701A1 (es)	2002-09-30
MA26999A1 (fr)	2004-12-20
DOP2002000345A (es)	2002-12-15
NO20033821L (no)	2003-09-10
EP1363606A1 (en)	2003-11-26
GT200200039A (es)	2002-11-21
BR0207802A (pt)	2004-03-09
ZA200306193B (en)	2004-08-11
IS6905A (is)	2003-08-07
NO20033821D0 (no)	2003-08-28
HUP0303448A3 (en)	2005-05-30
CZ20032338A3 (cs)	2004-08-18
JP2004527500A (ja)	2004-09-09
CR7059A (es)	2004-03-10

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Publication	Publication Date	Title
SK10752003A3 (sk)	2004-08-03	Použitie inverzných agonistov GABAA v kombinácii s parciálnymi agonistami receptora nikotínu, estrogénom, selektívnymi modulátormi estrogénu alebo vitamínom E pri liečení kognitívnych porúch
JP6675688B2 (ja)	2020-04-01	５−ｈｔ２ｃ受容体アゴニストおよび組成物ならびに使用方法
JP7514534B2 (ja)	2024-07-11	認知障害を処置するためのベンゾジアゼピン誘導体、組成物および方法
JP2018519251A5 (cs)	2019-05-30
US11608339B2 (en)	2023-03-21	5-HT2C receptor agonists and compositions and methods of use
JP5666910B2 (ja)	2015-02-12	認知機能障害を治療するためのキット、組成物、製品もしくは医薬
JP6789578B2 (ja)	2020-11-25	５−ｈｔ２ｃ受容体アゴニストおよび組成物、ならびに使用方法
WO2008013556A1 (en)	2008-01-31	Combination 5-ht7 receptor antagonist and serotonin reuptake inhibitor therapy
CA2640223A1 (en)	2007-08-02	Methods and compositions for treating schizophrenia
KR20200133259A (ko)	2020-11-26	Kv7 채널 활성화제 조성물 및 이의 사용 방법
TW201605856A (zh)	2016-02-16	５－ＨＴｃ受體促效劑
CZ2004524A3 (cs)	2004-07-14	Agonisté nikotinového acetylcholinového receptoru v léčbě syndromu neklidných nohou
CN102365269A (zh)	2012-02-29	用于治疗认知缺损的新药物
AU2002233585A1 (en)	2002-09-19	Use of GABAA inverse agonists in combination with nicotine receptor partial agonisits, estrogen, selective estrogen modulators, or vitamin E for the treatment of cognitive disorders
NZ739883B2 (en)	2021-06-29	5-ht2c receptor agonists and compositions and methods of use
HK40010293A (en)	2020-07-03	5-ht2c receptor agonists and compositions and methods of use
HK40010293B (en)	2022-12-23	5-ht2c receptor agonists and compositions and methods of use