SK12032003A3 - Farmaceutická formulácia obsahujúca 4'-kyano-alfa', alfa', alfa'-trifluór-3-(4-fluórfenylsulfonyl)-2-hydroxy-2- metylpropiono-m-toluidín a PVP - Google Patents

Farmaceutická formulácia obsahujúca 4'-kyano-alfa', alfa', alfa'-trifluór-3-(4-fluórfenylsulfonyl)-2-hydroxy-2- metylpropiono-m-toluidín a PVP Download PDF

Info

Publication number: SK12032003A3
Authority: SK; Slovakia
Prior art keywords: hydroxy; trifluoro; cyano; fluorophenylsulfonyl; toluidine
Prior art date: 2001-04-02

Application number

SK1203-2003A

Other languages

English (en)

Slovak (sk)

Inventor

Julie Kay Cahill

Nicola Frances Bateman

Original Assignee

Astrazeneca Ab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-04-02

Filing date

2002-03-27

Publication date

2004-03-02

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27354679&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SK12032003(A3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2001-04-02 Priority claimed from SE0101171A external-priority patent/SE0101171D0/xx

2001-09-04 Priority claimed from SE0102957A external-priority patent/SE0102957D0/xx

2001-10-25 Priority claimed from SE0103565A external-priority patent/SE0103565D0/xx

2002-03-27 Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab

2004-03-02 Publication of SK12032003A3 publication Critical patent/SK12032003A3/sk

Links

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Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/275—Nitriles; Isonitriles
- A61K31/277—Nitriles; Isonitriles having a ring, e.g. verapamil
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
- A61K9/146—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents

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General Health & Medical Sciences (AREA)
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Medicinal Chemistry (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Epidemiology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

SK1203-2003A 2001-04-02 2002-03-27 Farmaceutická formulácia obsahujúca 4'-kyano-alfa', alfa', alfa'-trifluór-3-(4-fluórfenylsulfonyl)-2-hydroxy-2- metylpropiono-m-toluidín a PVP SK12032003A3 (sk)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
SE0101171A SE0101171D0 (sv)	2001-04-02	2001-04-02	Pharmaceutical formulation
SE0102957A SE0102957D0 (sv)	2001-09-04	2001-09-04	Pharmaceutical formulation
SE0103565A SE0103565D0 (sv)	2001-10-25	2001-10-25	Pharmaceutical formulation
PCT/GB2002/001439 WO2002080902A1 (en)	2001-04-02	2002-03-27	Solid pharmaceutical composition comprising 4 -cyano-trifluoro-3-(4-fluorophenylsulphonyl)-2-hydroxy-2-methylpropiono- m toluidide and pvp

Publications (1)

Publication Number	Publication Date
SK12032003A3 true SK12032003A3 (sk)	2004-03-02

Family

ID=27354679

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SK1203-2003A SK12032003A3 (sk)	2001-04-02	2002-03-27	Farmaceutická formulácia obsahujúca 4'-kyano-alfa', alfa', alfa'-trifluór-3-(4-fluórfenylsulfonyl)-2-hydroxy-2- metylpropiono-m-toluidín a PVP

Country Status (21)

Country	Link
US (1)	US20040138299A1 (cs)
EP (1)	EP1381358B1 (cs)
JP (1)	JP2004525164A (cs)
KR (1)	KR20030087048A (cs)
CN (1)	CN1536993A (cs)
AT (1)	ATE324886T1 (cs)
BR (1)	BR0208421A (cs)
CA (1)	CA2443040A1 (cs)
CZ (1)	CZ20032647A3 (cs)
DE (1)	DE60211139T2 (cs)
EE (1)	EE200300476A (cs)
ES (1)	ES2261655T3 (cs)
HU (1)	HUP0303454A3 (cs)
IL (1)	IL157955A0 (cs)
IS (1)	IS6970A (cs)
MX (1)	MXPA03008999A (cs)
NO (1)	NO20034386L (cs)
NZ (1)	NZ528284A (cs)
PL (1)	PL365330A1 (cs)
SK (1)	SK12032003A3 (cs)
WO (1)	WO2002080902A1 (cs)

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CZ20032225A3 (cs) *	2001-02-27	2003-11-12	Astrazeneca Ab	Farmaceutická formulace
SE0103424D0 (sv) *	2001-10-15	2001-10-15	Astrazeneca Ab	Pharmaceutical formulation
SE0103838D0 (sv) *	2001-11-16	2001-11-16	Astrazeneca Ab	Pharmaceutical formulation & product
US20050008691A1 (en) *	2003-05-14	2005-01-13	Arturo Siles Ortega	Bicalutamide compositions
KR20070085465A (ko) *	2004-11-29	2007-08-27	노파르티스 아게	Ｓ１ｐ 수용체 효능제의 투여 용법
WO2006090129A2 (en) *	2005-02-23	2006-08-31	Astrazeneca Ab	Bicalutamide for delivering increasing steady state plasma levels
US7785629B2 (en) *	2005-06-21	2010-08-31	Helm Ag	Bicalutamide-adsorbates, process for preparing same, and pharmaceutical compositions thereof
US20070026073A1 (en) *	2005-07-28	2007-02-01	Doney John A	Amorphous efavirenz and the production thereof
US20080045600A1 (en) *	2006-08-17	2008-02-21	Gawande Rahul S	Bicalutamide compositions
US20080152717A1 (en) *	2006-12-14	2008-06-26	Isp Investments, Inc.	Amorphous valsartan and the production thereof
JP5508859B2 (ja) *	2007-01-26	2014-06-04	アイエスピーインヴェストメンツインコーポレイテッド	噴霧乾燥製品を製造するための調剤処理方法
PL2278960T5 (pl)	2008-03-17	2020-06-29	Actelion Pharmaceuticals Ltd.	Schemat dawkowania dla selektywnego agonisty receptora sip1
US9018253B2 (en)	2010-07-02	2015-04-28	Bio-Pharm Solutions Co., Ltd.	Phenylcarbamate compound and muscle relaxant containing the same
CA2815460C (en)	2011-01-13	2017-04-18	Bio-Pharm Solutions Co., Ltd.	Process for preparation of phenyl carbamate derivatives
EP2797880B1 (en)	2011-12-27	2017-03-01	Bio-Pharm Solutions Co., Ltd.	Phenyl carbamate compounds for use in preventing or treating epilepsy
TW201431570A (zh)	2012-11-22	2014-08-16	Ucb Pharma Gmbh	用於經皮投服羅替戈汀（Ｒｏｔｉｇｏｔｉｎｅ）之多天式貼片
JP6726096B2 (ja)	2013-07-03	2020-07-22	エルテーエスローマンテラピー−システメアーゲー	電子部品を有する経皮治療システム
CA2948219C (en)	2014-05-20	2023-04-04	Lts Lohmann Therapie-Systeme Ag	Method for adjusting the release of active agent in a transdermal delivery system
CN106456566B (zh) *	2014-05-20	2020-06-16	Lts勒曼治疗系统股份公司	含罗替戈汀的经皮递送系统
US11752110B2 (en)	2014-05-20	2023-09-12	Lts Lohmann Therapie-Systeme Ag	Transdermal delivery system including an interface mediator
LT3226842T (lt)	2014-12-05	2021-03-25	Aragon Pharmaceuticals, Inc.	Priešvėžinės kompozicijos
HUE054935T2 (hu)	2014-12-05	2021-10-28	Aragon Pharmaceuticals Inc	Rákellenes készítmények
SG11201704267VA (en)	2014-12-05	2017-06-29	Aragon Pharmaceuticals Inc	Anticancer compositions

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AU1687395A (en) *	1994-01-21	1995-08-08	Sepracor, Inc.	Methods and compositions for treating androgen-dependent diseases using optically pure r-(-)-casodex
ATE400252T1 (de) *	1999-02-10	2008-07-15	Pfizer Prod Inc	Pharmazeutische feste dispersionen
GB9930839D0 (en) *	1999-12-30	2000-02-16	Pharmacia & Upjohn Spa	Process for treating gynecomastia

2002
- 2002-03-27 EP EP02718317A patent/EP1381358B1/en not_active Revoked
- 2002-03-27 IL IL15795502A patent/IL157955A0/xx unknown
- 2002-03-27 CA CA002443040A patent/CA2443040A1/en not_active Abandoned
- 2002-03-27 BR BR0208421-0A patent/BR0208421A/pt not_active IP Right Cessation
- 2002-03-27 EE EEP200300476A patent/EE200300476A/xx unknown
- 2002-03-27 ES ES02718317T patent/ES2261655T3/es not_active Expired - Lifetime
- 2002-03-27 CN CNA028077474A patent/CN1536993A/zh active Pending
- 2002-03-27 MX MXPA03008999A patent/MXPA03008999A/es unknown
- 2002-03-27 HU HU0303454A patent/HUP0303454A3/hu unknown
- 2002-03-27 DE DE60211139T patent/DE60211139T2/de not_active Expired - Fee Related
- 2002-03-27 NZ NZ528284A patent/NZ528284A/en unknown
- 2002-03-27 WO PCT/GB2002/001439 patent/WO2002080902A1/en not_active Ceased
- 2002-03-27 KR KR10-2003-7012900A patent/KR20030087048A/ko not_active Withdrawn
- 2002-03-27 PL PL02365330A patent/PL365330A1/xx not_active Application Discontinuation
- 2002-03-27 JP JP2002578941A patent/JP2004525164A/ja active Pending
- 2002-03-27 US US10/473,709 patent/US20040138299A1/en not_active Abandoned
- 2002-03-27 SK SK1203-2003A patent/SK12032003A3/sk unknown
- 2002-03-27 AT AT02718317T patent/ATE324886T1/de not_active IP Right Cessation
- 2002-03-27 CZ CZ20032647A patent/CZ20032647A3/cs unknown
2003
- 2003-09-29 IS IS6970A patent/IS6970A/is unknown
- 2003-10-01 NO NO20034386A patent/NO20034386L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
NO20034386L (no)	2003-11-28
DE60211139T2 (de)	2007-03-01
PL365330A1 (en)	2004-12-27
HUP0303454A3 (en)	2005-12-28
CA2443040A1 (en)	2002-10-17
CN1536993A (zh)	2004-10-13
IL157955A0 (en)	2004-03-28
WO2002080902A1 (en)	2002-10-17
ATE324886T1 (de)	2006-06-15
DE60211139D1 (de)	2006-06-08
CZ20032647A3 (cs)	2004-09-15
NZ528284A (en)	2005-04-29
BR0208421A (pt)	2004-03-30
EE200300476A (et)	2003-12-15
JP2004525164A (ja)	2004-08-19
KR20030087048A (ko)	2003-11-12
NO20034386D0 (no)	2003-10-01
EP1381358B1 (en)	2006-05-03
EP1381358A1 (en)	2004-01-21
MXPA03008999A (es)	2004-02-12
HUP0303454A2 (hu)	2004-01-28
US20040138299A1 (en)	2004-07-15
ES2261655T3 (es)	2006-11-16
IS6970A (is)	2003-09-29

Publication	Publication Date	Title
SK12032003A3 (sk)	2004-03-02	Farmaceutická formulácia obsahujúca 4'-kyano-alfa', alfa', alfa'-trifluór-3-(4-fluórfenylsulfonyl)-2-hydroxy-2- metylpropiono-m-toluidín a PVP
EP2259777A2 (en)	2010-12-15	Pharmaceutical composition for poorly soluble drugs
HUE031177T2 (hu)	2017-07-28	Rivaroxabant tartalmazó szilárd gyógyszerkészítmény
US20110097414A1 (en)	2011-04-28	Pharmaceutical compositions comprising adsorbate of fenofibrate
KR20210125994A (ko)	2021-10-19	비정질 스파르센탄 조성물
KR100209201B1 (ko)	1999-07-15	1,4-디히드로피리딘 유도체를 함유하는 고체 분산 정제 및 그의 제조방법
US20050038111A1 (en)	2005-02-17	Pharmaceutical formulation comprising bicalutamide
JP3639587B2 (ja)	2005-04-20	医薬製剤
EA017553B1 (ru)	2013-01-30	Гидробромид ивабрадина
KR20040101437A (ko)	2004-12-02	고체 분산체 조성물
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WO2003043630A1 (en)	2003-05-30	Solid pharmaceutical composition comprising 4-cyano-trifluoro-3-(4-fluorophenyl sulphonyl)-2-hydroxy-2-methylpropiono- m toluidide, pvp, an anti-oestrogen and/or an aromatase inhibitor
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ZA200307579B (en)	2005-03-17	Solid pharmaceutical composition comprising 4 -cyano-trifluoro-3-(4-fluorophenylsulphonyl)-2-hydroxyl-2-methylpropiono-m-toluidide and PVP.
AU2002249387A1 (en)	2002-10-21	Solid pharmaceutical composition comprising 4-cyano-trifluoro-3-(4-fluorophenylsulphonyl)-2-hydroxy-2-methylpropiono-M toluidide and PVP
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